| Compound ID |
Compound Name |
Compound Formula |
|
CP0503845
|
2-N-[[1-[4-bromo-2-(trifluoromethoxy)phenyl]sulfonylpiperidin-4-yl]methyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C23H25BrF3N5O3S
|
1
|
| 1 |
IC50 = 5.6 nM
|
|
|
|
CP0871069
|
4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-2-trifluoromethoxy-benzenesulfonamide hydrochloride
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|
C25H30BrClF3N5O3S
|
1
|
| 1 |
IC50 = 7.7 nM
|
|
|
|
CP0404808
|
4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-2-trifluoromethoxy-benzenesulfonamide
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|
C25H29BrF3N5O3S
|
1
|
| 1 |
IC50 = 7.7 nM
|
|
|
|
CP0500756
|
4-bromo-N-[[4-[[[4-(dimethylamino)quinazolin-2-yl]amino]methyl]cyclohexyl]methyl]-2-(trifluoromethoxy)benzamide
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|
C26H29BrF3N5O2
|
1
|
| 1 |
IC50 = 9.9 nM
|
|
|
|
CP0404813
|
4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexyl}-2-trifluoromethoxy-benzenesulfonamide
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|
C24H27BrF3N5O3S
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0464467
|
2-N-[[4-[[[4-bromo-2-(trifluoromethoxy)phenyl]methylamino]methyl]cyclohexyl]methyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C26H31BrF3N5O
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0494619
|
4-bromo-N-[[4-[[[4-(dimethylamino)quinazolin-2-yl]amino]methyl]cyclohexyl]methyl]-N-methyl-2-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C26H31BrF3N5O3S
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0392533
|
2-N-[[4-[[[4-bromo-2-(trifluoromethoxy)phenyl]methyl-methylamino]methyl]cyclohexyl]methyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C27H33BrF3N5O
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0475855
|
3,4-Dichloro-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-benzamide
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|
C23H25Cl2N5O
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0495240
|
4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C23H25BrF3N5O3S
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0392292
|
4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C23H25BrF3N5O3S
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0409351
|
4-Bromo-N-[4-(quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C21H20BrF3N4O3S
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0466919
|
Butane-1-sulfonic acid {4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-amide
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|
C22H35N5O2S
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0496862
|
N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-3-(trifluoromethyl)benzamide
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|
C24H26F3N5O
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0449373
|
3-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-benzamide
Show/Hide
|
C23H26BrN5O
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0497065
|
N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-3,5-dimethoxybenzamide
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|
C25H31N5O3
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0431375
|
3-Chloro-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-benzamide
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|
C23H26ClN5O
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0493156
|
N-[[4-[[[4-(dimethylamino)quinazolin-2-yl]amino]methyl]cyclohexyl]methyl]methanesulfonamide
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|
C19H29N5O2S
|
1
|
| 1 |
IC50 = 86 nM
|
|
|
|
CP0424979
|
N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-3-nitrobenzamide
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|
C23H26N6O3
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
|
CP0039984
|
CGP 71683
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|
C26H29N5O2S
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
|
CP0431012
|
N-[[4-[[(4-aminoquinazolin-2-yl)amino]methyl]cyclohexyl]methyl]-4-bromo-2-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C23H25BrF3N5O3S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0404697
|
N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-3-methylbenzamide
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|
C24H29N5O
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0431015
|
4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C24H27BrF3N5O3S
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0378340
|
4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C24H27BrF3N5O3S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0424928
|
N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-3-fluorobenzamide
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|
C23H26FN5O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0409350
|
4-Bromo-N-[4-(quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C22H22BrF3N4O3S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0404811
|
4-Bromo-N-[4-(quinazolin-2-ylaminomethyl)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide
Show/Hide
|
C23H24BrF3N4O3S
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0378311
|
N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-4-fluorobenzamide
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|
C23H26FN5O
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0392541
|
3-Cyano-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-benzamide
Show/Hide
|
C24H26N6O
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0379328
|
2-N-[4-[[4-bromo-2-(trifluoromethoxy)phenyl]methylamino]cyclohexyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
Show/Hide
|
C24H27BrF3N5O
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0440289
|
2-N-[1-[4-bromo-2-(trifluoromethoxy)phenyl]sulfonylpiperidin-4-yl]-4-N,4-N-dimethylquinazoline-2,4-diamine
Show/Hide
|
C22H23BrF3N5O3S
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0480696
|
N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-2,3,4-trifluorobenzamide
Show/Hide
|
C23H24F3N5O
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0043469
|
ATC0175
Show/Hide
|
C23H25F2N5O
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0431371
|
2-N-[4-[[[4-bromo-2-(trifluoromethoxy)phenyl]methylamino]methyl]cyclohexyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
Show/Hide
|
C25H29BrF3N5O
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0392299
|
4-bromo-N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-2-(trifluoromethoxy)benzamide
Show/Hide
|
C24H25BrF3N5O2
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0424935
|
2-N-[1-[[4-bromo-2-(trifluoromethoxy)phenyl]methyl]piperidin-4-yl]-4-N,4-N-dimethylquinazoline-2,4-diamine
Show/Hide
|
C23H25BrF3N5O
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0436964
|
4-bromo-N-[[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]methyl]-2-(trifluoromethoxy)benzamide
Show/Hide
|
C25H27BrF3N5O2
|
1
|
| 1 |
IC50 = 570 nM
|
|
|
