| Compound ID |
Compound Name |
Compound Formula |
|
CP0536515
|
1-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
|
C20H15F3N6O2S2
|
1
|
| 1 |
IC50 = 63.7 nM
|
|
|
|
CP0432103
|
1-(2-methoxy-5-methylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O3S2
|
1
|
| 1 |
IC50 = 358.6 nM
|
|
|
|
CP0437861
|
1-(5-chloro-2,4-dimethoxyphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C26H27ClN4O3
|
1
|
| 1 |
IC50 = 423.2 nM
|
|
|
|
CP0415956
|
1-(3-chloro-4-methylphenyl)-3-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H17ClN6O2S2
|
1
|
| 1 |
IC50 = 771 nM
|
|
|
|
CP0462272
|
1-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]-3-(2-methoxy-5-methylphenyl)urea
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|
C26H28N4O2
|
1
|
| 1 |
IC50 = 778 nM
|
|
|
|
CP0411046
|
1-(3-chlorophenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
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|
C24H23ClN4O
|
1
|
| 1 |
IC50 = 1196.8 nM
|
|
|
|
CP0536522
|
1-(3-chlorophenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C19H15ClN6O2S2
|
1
|
| 1 |
IC50 = 1340.8 nM
|
|
|
|
CP0439911
|
1-(4-ethylphenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O2S2
|
1
|
| 1 |
IC50 = 2027.5 nM
|
|
|
|
CP0562562
|
1-(2,5-dimethylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O2S2
|
1
|
| 1 |
IC50 = 2138.5 nM
|
|
|
|
CP0455623
|
1-(2,5-dimethoxyphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O4S2
|
1
|
| 1 |
IC50 = 2497.3 nM
|
|
|
|
CP0471908
|
1-(2-ethoxyphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C26H28N4O2
|
1
|
| 1 |
IC50 = 2594.4 nM
|
|
|
|
CP0455624
|
1-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]-3-(3-methylphenyl)urea
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|
C25H26N4O
|
1
|
| 1 |
IC50 = 2843.4 nM
|
|
|
|
CP0455620
|
1-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]-3-(3-methoxyphenyl)urea
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|
C25H26N4O2
|
1
|
| 1 |
IC50 = 3224.9 nM
|
|
|
|
CP0439918
|
1-(3,5-dimethoxyphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H26N4O3
|
1
|
| 1 |
IC50 = 3575.6 nM
|
|
|
|
CP0462271
|
1-(2,4-dimethoxyphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H26N4O3
|
1
|
| 1 |
IC50 = 3886.6 nM
|
|
|
|
CP0459228
|
1-(3-fluoro-4-methylphenyl)-3-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H17FN6O2S2
|
1
|
| 1 |
IC50 = 4615.5 nM
|
|
|
|
CP0543741
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(5-chloro-2-methoxyphenyl)urea
Show/Hide
|
C23H21ClN4O2
|
1
|
| 1 |
IC50 = 5460.3 nM
|
|
|
|
CP0415961
|
1-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(3-methylsulfanylphenyl)urea
Show/Hide
|
C20H18N6O2S3
|
1
|
| 1 |
IC50 = 6706 nM
|
|
|
|
CP0569559
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(2,5-dimethoxyphenyl)urea
Show/Hide
|
C24H24N4O3
|
1
|
| 1 |
IC50 = 9064.5 nM
|
|
|
|
CP0230588
|
1-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
|
C20H15F3N6O2S2
|
1
|
| 1 |
IC50 = 9280 nM
|
|
|
|
CP0553533
|
1-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(3-methylphenyl)urea
Show/Hide
|
C20H18N6O2S2
|
1
|
| 1 |
IC50 = 9792.4 nM
|
|
|
|
CP0391172
|
1-(2-methoxyphenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H18N6O3S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0391175
|
1-(3,5-dimethoxyphenyl)-3-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O4S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0411050
|
1-(5-chloro-2-methylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H17ClN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0411052
|
1-(2,3-dimethylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0421264
|
1-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(3-methylsulfanylphenyl)urea
Show/Hide
|
C20H18N6O2S3
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0426413
|
1-(3,4-dimethoxyphenyl)-3-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O4S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0432129
|
1-(3-fluorophenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C19H15FN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0455616
|
1-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)urea
Show/Hide
|
C20H18N6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0455626
|
1-[5-[(7-chloro-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(3,4-dimethylphenyl)urea
Show/Hide
|
C20H17ClN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0459233
|
1-(3-chloro-4-fluorophenyl)-3-[5-[(3-oxo-4H-quinoxalin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C18H12ClFN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0459237
|
1-(2-fluorophenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C19H15FN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0462277
|
1-(2,4-difluorophenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C19H14F2N6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0468986
|
1-(2-chloro-4-methylphenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H17ClN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0471905
|
1-(3,5-dimethylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0471909
|
1-(2-fluorophenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C19H15FN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0471910
|
methyl 2-[[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]carbamoylamino]benzoate
Show/Hide
|
C21H18N6O4S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0477367
|
1-(3-chloro-4-methylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H17ClN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0479251
|
ethyl 2-[[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]carbamoylamino]benzoate
Show/Hide
|
C22H20N6O4S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0533430
|
1-(3,4-dimethoxyphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O4S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0536505
|
1-(3-fluoro-4-methylphenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H17FN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0538075
|
1-(3-methoxyphenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H18N6O3S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0554853
|
1-(2-fluorophenyl)-3-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C19H15FN6O2S2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0426131
|
[2-(4-butan-2-ylanilino)-2-oxoethyl] 1,3-benzothiazole-6-carboxylate
Show/Hide
|
C20H20N2O3S
|
1
|
| 1 |
IC50 = 10461.4 nM
|
|
|
|
CP0391054
|
1-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]-3-[2-(trifluoromethyl)phenyl]urea
Show/Hide
|
C24H21F3N4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0391170
|
1-(2-methylphenyl)-3-[5-[(4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C19H16N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0391171
|
1-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)urea
Show/Hide
|
C20H18N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0391174
|
1-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-phenylurea
Show/Hide
|
C19H16N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0411047
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(3-fluoro-4-methylphenyl)urea
Show/Hide
|
C23H21FN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0411048
|
1-(4-ethylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0411051
|
1-(3,4-dimethylphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C26H28N4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0415957
|
1-(5-chloro-2-methoxyphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C24H23ClN4O2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0415958
|
1-(3,5-dimethylphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C26H28N4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0415959
|
1-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]-3-(3-methylsulfanylphenyl)urea
Show/Hide
|
C25H26N4OS
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0415975
|
1-(4-fluorophenyl)-3-[5-[(4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C18H13FN6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0420975
|
1-(2-chlorophenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C23H21ClN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0421263
|
1-(2,5-dimethylphenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0421265
|
1-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[2-(trifluoromethyl)phenyl]urea
Show/Hide
|
C20H15F3N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0421268
|
1-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]-3-(2-fluorophenyl)urea
Show/Hide
|
C24H23FN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0426409
|
1-(3-chloro-4-fluorophenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C23H20ClFN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0426412
|
1-(2-ethoxyphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O3S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0426416
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(3-methylphenyl)urea
Show/Hide
|
C23H22N4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0426417
|
1-(3-chlorophenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C23H21ClN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0426418
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(3-chloro-4-methylphenyl)urea
Show/Hide
|
C23H21ClN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0432097
|
1-(3-chloro-4-methylphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C24H23ClN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0432100
|
methyl 2-[[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]carbamoylamino]benzoate
Show/Hide
|
C21H18N6O4S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0432105
|
1-(2,5-dimethoxyphenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O4S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0432107
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(3-chlorophenyl)urea
Show/Hide
|
C22H19ClN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0432109
|
1-(3,4-dimethylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0432111
|
1-(5-chloro-2-methoxyphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H25ClN4O2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0432113
|
1-(5-chloro-2,4-dimethoxyphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H25ClN4O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
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CP0433952
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1-(2-chloro-4-methylphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
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C20H17ClN6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0433953
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1-(3,5-dimethoxyphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
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C26H28N4O3
|
1
|
| 1 |
IC50 = 20000 nM
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CP0433958
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1-[5-[(3-oxo-4H-quinoxalin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
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C19H13F3N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0437856
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ethyl 2-[[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]carbamoylamino]benzoate
Show/Hide
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C22H20N6O4S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0437862
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1-(4-ethylphenyl)-3-[5-[(3-oxo-4H-quinoxalin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
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C20H18N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0439912
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1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(2-methoxy-5-methylphenyl)urea
Show/Hide
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C24H24N4O2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0455613
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1-[5-[(3-oxo-4H-quinoxalin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-phenylurea
Show/Hide
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C18H14N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0455618
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1-(2-ethoxyphenyl)-3-[4-[2-(1-phenylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
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C30H28N4O2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0455625
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1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(3-methylsulfanylphenyl)urea
Show/Hide
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C23H22N4OS
|
1
|
| 1 |
IC50 = 20000 nM
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CP0459231
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1-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
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C24H21F3N4O
|
1
|
| 1 |
IC50 = 20000 nM
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CP0459232
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1-(3-bromophenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
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C23H21BrN4O
|
1
|
| 1 |
IC50 = 20000 nM
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CP0459235
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1-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]-3-(4-methylphenyl)urea
Show/Hide
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C25H26N4O
|
1
|
| 1 |
IC50 = 20000 nM
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CP0462262
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1-(4-methylphenyl)-3-[5-[(3-oxo-4H-quinoxalin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
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C19H16N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0462269
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1-(3-chlorophenyl)-3-[5-[(3-oxo-4H-quinoxalin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C18H13ClN6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0462270
|
1-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(2-methylphenyl)urea
Show/Hide
|
C20H18N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0462275
|
1-(4-methylphenyl)-3-[4-[2-(1-phenylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C29H26N4O
|
1
|
| 1 |
IC50 = 20000 nM
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|
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CP0468975
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(2,4-dimethoxyphenyl)urea
Show/Hide
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C24H24N4O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
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CP0468978
|
1-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(3-methylphenyl)urea
Show/Hide
|
C20H18N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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|
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CP0468979
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(3-bromophenyl)urea
Show/Hide
|
C22H19BrN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
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CP0468984
|
1-[5-[(7-chloro-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(3-fluoro-4-methylphenyl)urea
Show/Hide
|
C19H14ClFN6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0468985
|
1-(2,5-dimethylphenyl)-3-[5-[(4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H18N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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|
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CP0468987
|
1-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[2-(trifluoromethyl)phenyl]urea
Show/Hide
|
C20H15F3N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0471907
|
1-(2-ethoxyphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H26N4O2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
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CP0471911
|
1-(2-methoxyphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H18N6O3S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0477368
|
1-(3,5-dimethylphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H26N4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0477380
|
1-(2,3-dimethylphenyl)-3-[5-[(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
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CP0479252
|
1-(2,4-dimethylphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C26H28N4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0479253
|
1-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]-3-(3-methylsulfanylphenyl)urea
Show/Hide
|
C24H24N4OS
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0479284
|
1-(2,5-dimethoxyphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H26N4O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0533431
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(3,4,5-trimethoxyphenyl)urea
Show/Hide
|
C25H26N4O4
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0533432
|
1-(2,5-dimethoxyphenyl)-3-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C21H20N6O4S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0533434
|
1-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
|
C20H15F3N6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0536514
|
1-(1,3-benzodioxol-5-yl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H24N4O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0536521
|
1-(2,5-dimethoxyphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C26H28N4O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0536523
|
1-(2-methoxyphenyl)-3-[5-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H18N6O3S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0536525
|
1-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]-3-(3,4,5-trimethoxyphenyl)urea
Show/Hide
|
C27H30N4O4
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0536534
|
1-(4-fluorophenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C19H15FN6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0543743
|
1-(2-chlorophenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C24H23ClN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0543744
|
1-(3-acetylphenyl)-3-[4-[2-(1-ethylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C26H26N4O2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0543756
|
1-[5-[(7-chloro-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]-3-(4-fluorophenyl)urea
Show/Hide
|
C18H12ClFN6O2S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0554852
|
1-(2,5-dimethylphenyl)-3-[4-[2-(1-methylbenzimidazol-2-yl)ethyl]phenyl]urea
Show/Hide
|
C25H26N4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0567468
|
1-(3-methoxyphenyl)-3-[5-[(9-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-1,3,4-thiadiazol-2-yl]urea
Show/Hide
|
C20H18N6O3S2
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0569544
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-[3-(trifluoromethyl)phenyl]urea
Show/Hide
|
C23H19F3N4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0569549
|
1-[4-[2-(1H-benzimidazol-2-yl)ethyl]phenyl]-3-(4-bromophenyl)urea
Show/Hide
|
C22H19BrN4O
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0412964
|
2-[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanyl-N-[5-methyl-2-(4-methylphenyl)pyrazol-3-yl]acetamide
Show/Hide
|
C20H19N7O2S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0412965
|
[2-(3,4-dimethoxyanilino)-2-oxoethyl] 1H-indazole-3-carboxylate
Show/Hide
|
C18H17N3O5
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0412966
|
[2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 4-(tetrazol-1-yl)benzoate
Show/Hide
|
C23H23N7O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0412967
|
N-(5-tert-butyl-2-phenylpyrazol-3-yl)-2-[(4-cyclopropyl-5-pyridin-3-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
Show/Hide
|
C25H27N7OS
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0412968
|
[2-(naphthalen-2-ylamino)-2-oxoethyl] 4-(tetrazol-1-yl)benzoate
Show/Hide
|
C20H15N5O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0412969
|
[2-oxo-2-[3-(trifluoromethyl)anilino]ethyl] 4-(hydroxymethyl)benzoate
Show/Hide
|
C17H14F3NO4
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0426132
|
[2-[(3-carbamoyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)amino]-2-oxoethyl] 4-(1H-indol-3-yl)butanoate
Show/Hide
|
C22H23N3O4S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0426133
|
[2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 5,6-dichloropyridine-3-carboxylate
Show/Hide
|
C21H20Cl2N4O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0528229
|
N-(5-tert-butyl-2-phenylpyrazol-3-yl)-2-[1-(2-ethoxyphenyl)tetrazol-5-yl]sulfanylacetamide
Show/Hide
|
C24H27N7O2S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0542725
|
N-(5-tert-butyl-2-phenylpyrazol-3-yl)-2-(1-phenyltetrazol-5-yl)sulfanylacetamide
Show/Hide
|
C22H23N7OS
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
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CP0543678
|
[2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 4-acetamidobenzoate
Show/Hide
|
C24H26N4O4
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0552758
|
[2-(naphthalen-2-ylamino)-2-oxoethyl] 1,3-benzothiazole-6-carboxylate
Show/Hide
|
C20H14N2O3S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0554216
|
[2-(4-tert-butylanilino)-2-oxoethyl] 1,3-benzothiazole-6-carboxylate
Show/Hide
|
C20H20N2O3S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0559579
|
[2-[(3-carbamoyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)amino]-2-oxoethyl] 4-(4-chlorophenyl)-4-oxobutanoate
Show/Hide
|
C20H19ClN2O5S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0559597
|
N-(5-tert-butyl-2-phenylpyrazol-3-yl)-2-[1-(4-methoxyphenyl)tetrazol-5-yl]sulfanylacetamide
Show/Hide
|
C23H25N7O2S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0559598
|
[2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl] 1,3-benzothiazole-6-carboxylate
Show/Hide
|
C17H11F3N2O4S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0559599
|
[2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 4-cyanobenzoate
Show/Hide
|
C23H22N4O3
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0560648
|
[2-oxo-2-[4-(trifluoromethyl)anilino]ethyl] 1,3-benzothiazole-6-carboxylate
Show/Hide
|
C17H11F3N2O3S
|
1
|
| 1 |
IC50 = 20000 nM
|
|
|
|
CP0573027
|
[2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 9-oxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-b]quinazoline-6-carboxylate
Show/Hide
|
C27H29N5O4
|
1
|
| 1 |
IC50 = 20000 nM
|
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