| Compound ID |
Compound Name |
Compound Formula |
|
CP0268743
|
4-[[(6R)-7-cyano-6-ethyl-5-propan-2-yl-6H-imidazo[1,5-f]pteridin-3-yl]amino]-N-(1-ethylpiperidin-4-yl)-2-fluoro-5-methoxybenzamide
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|
C29H36FN9O2
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0196606
|
4-[[(6R)-7-cyano-5-cyclohexyl-6-ethyl-6H-imidazo[1,5-f]pteridin-3-yl]amino]-2-fluoro-5-methoxy-N-(1-methylpiperidin-4-yl)benzamide
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|
C31H38FN9O2
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0447608
|
(6R)-5-cyclopentyl-6-ethyl-3-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-6H-imidazo[1,5-f]pteridine-7-carboxylic acid
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|
C30H38N8O4
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0244570
|
4-[[(6R)-7-cyano-5-cyclopentyl-6-ethyl-6H-imidazo[1,5-f]pteridin-3-yl]amino]-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide
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|
C30H37N9O2
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0575521
|
4-[[(6R)-7-cyano-6-ethyl-5-propan-2-yl-6H-imidazo[1,5-f]pteridin-3-yl]amino]-2-fluoro-5-methoxy-N-(1-methylazetidin-3-yl)benzamide
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|
C26H30FN9O2
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0483568
|
4-[[(6R)-7-cyano-6-ethyl-5-propan-2-yl-6H-imidazo[1,5-f]pteridin-3-yl]amino]-2-fluoro-5-methoxy-N-(1-methylpiperidin-4-yl)benzamide
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|
C28H34FN9O2
|
1
|
| 1 |
IC50 = 1.9 nM
|
|
|
|
CP0492736
|
(6R)-5-cyclopentyl-6-ethyl-3-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-6H-imidazo[1,5-f]pteridine-7-carboxamide
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|
C30H39N9O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0410308
|
ethyl (6R)-5-cyclopentyl-6-ethyl-3-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-6H-imidazo[1,5-f]pteridine-7-carboxylate
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|
C32H42N8O4
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0268742
|
4-[[(6R)-7-cyano-5-cyclopentyl-6-ethyl-6H-imidazo[1,5-f]pteridin-3-yl]amino]-2-fluoro-5-methoxy-N-(1-methylpiperidin-4-yl)benzamide
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|
C30H36FN9O2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0558960
|
4-[[(6R)-5-cyclopentyl-6-ethyl-7-(hydroxymethyl)-6H-imidazo[1,5-f]pteridin-3-yl]amino]-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide
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|
C30H40N8O3
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0483569
|
4-[[(6R)-7-cyano-6-ethyl-5-propan-2-yl-6H-imidazo[1,5-f]pteridin-3-yl]amino]-N-[4-[4-(cyclopropylmethyl)piperazin-1-yl]cyclohexyl]-2-fluoro-5-methoxybenzamide
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|
C36H47FN10O2
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0575901
|
(6R)-5-cyclopentyl-6-ethyl-N-hydroxy-3-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-N-methyl-6H-imidazo[1,5-f]pteridine-7-carboxamide
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|
C31H41N9O4
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0492738
|
4-[[(6R)-7-cyano-6-ethyl-5-propan-2-yl-6H-imidazo[1,5-f]pteridin-3-yl]amino]-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide
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|
C28H35N9O2
|
1
|
| 1 |
IC50 = 8.6 nM
|
|
|
|
CP0492737
|
(6R)-5-cyclopentyl-N,6-diethyl-3-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-6H-imidazo[1,5-f]pteridine-7-carboxamide
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|
C32H43N9O3
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0072678
|
5-(1,3-benzodioxol-5-yl)-7-[[(2R)-1-ethenylsulfonylpyrrolidin-2-yl]methyl]pyrrolo[2,3-d]pyrimidin-4-amine
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|
C20H21N5O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0012721
|
[3-[4-[(4-cyclopropylphenyl)methoxy]-3-methoxyphenyl]azetidin-1-yl]-[4-[[(2S)-2,3-dihydroxypropoxy]methyl]pyridin-2-yl]methanone
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|
C30H34N2O6
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
