Brief Information of the Compound and Protein
Compound Name
(6R)-5-cyclopentyl-6-ethyl-N-hydroxy-3-[2-methoxy-4-[(1-methylpiperidin-4-yl)carbamoyl]anilino]-N-methyl-6H-imidazo[1,5-f]pteridine-7-carboxamide
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PubChem ID
CID: 137653047
Canonical SMILES
CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2-n2cnc(C(=O)N(C)O)c12
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Compound Formula C31H41N9O4
Compound Structure
Protein Name
Serine/threonine-protein kinase PLK1
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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Other protein kinase group
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Other protein kinase PLK family
Uniprot ID
P53350
Gene Name
PLK1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000012 Sf21 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 7 nM
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