All Bioactivity

Brief Information of the Cell Line and Protein

Cell Line ID: CL000009 , LLC-PK1

Cell Line Info

Synonyms	LLC-PK(1) LLC-PK-1 LLC PK-1 LLc-PK1 LLC PK1 LLCPK1 Lilly Laboratories Culture-Porcine Kidney 1
Category	Spontaneously immortalized cell line
Organism	Sus scrofa (Pig)
Cellosaurus ID	CVCL_0391

Protein ID: PT01155 , Growth hormone secretagogue receptor type 1

Protein Info

Gene Name	GHSR
Organism	Homo sapiens, Human
Protein Classification	Membrane receptor
Uniprot ID	Q92847

Table of Molecular Bioactivities Related to the Cell Line and Protein

Cell Line ID: CL000009

Cell Line Info

Protein ID: PT01155

Protein Info

Compound ID	Compound Name	Compound Formula
CP0454969 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]ethyl]piperidine-4-carboxamide Show/Hide	C36H39N7O2	2
1	IC50 = 0.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 0.6 nM Bioactivity Info	TI LI LO TS
CP0134612 Compound Info	GHRELIN Show/Hide	C147H245N45O42	1
1	IC50 = 0.39 nM Bioactivity Info	TI LI LO TS
CP0454974 Compound Info	N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-4-carboxamide Show/Hide	C37H41N7O3	1
1	IC50 = 0.5 nM Bioactivity Info	TI LI LO TS
CP0870851 Compound Info	(R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide Show/Hide	C34H40N6O2	1
1	IC50 = 0.6 nM Bioactivity Info	TI LI LO TS
CP0455084 Compound Info	(R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)picolinamide Show/Hide	C33H30N6O2	1
1	IC50 = 0.7 nM Bioactivity Info	TI LI LO TS
CP0154574 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide Show/Hide	C34H32N6O2	1
1	IC50 = 0.7 nM Bioactivity Info	TI LI LO TS
CP0037119 Compound Info	1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-1-oxopropan-2-yl]carbamoyl}-1-methylethan-1-aminium Show/Hide	C27H36N4O5S	1
1	IC50 = 0.76 nM Bioactivity Info	TI LI LO TS
CP0910551 Compound Info	(R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide Show/Hide	C35H42N6O3	1
1	IC50 = 0.9 nM Bioactivity Info	TI LI LO TS
CP0075872 Compound Info	(R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)picolinamide Show/Hide	C34H32N6O3	1
1	IC50 = 1.1 nM Bioactivity Info	TI LI LO TS
CP0316950 Compound Info	N-[(2R)-1-[[(1R)-1-formamido-2-(1H-indol-3-yl)ethyl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]piperidine-4-carboxamide Show/Hide	C28H32N6O3	1
1	IC50 = 1.155 nM Bioactivity Info	TI LI LO TS
CP0428229 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)picolinamide Show/Hide	C36H33N7O3	1
1	IC50 = 1.8 nM Bioactivity Info	TI LI LO TS
CP0459859 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)picolinamide Show/Hide	C35H31N7O2	1
1	IC50 = 1.9 nM Bioactivity Info	TI LI LO TS
CP0489341 Compound Info	(R)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethylcarbamate Show/Hide	C36H33N7O3	1
1	IC50 = 1.9 nM Bioactivity Info	TI LI LO TS
CP0432520 Compound Info	6-fluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide Show/Hide	C34H31FN6O2	1
1	IC50 = 2 nM Bioactivity Info	TI LI LO TS
CP0850992 Compound Info	(R)-N-(2-(1H-indol-3-yl)-1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)ethyl)-6-methoxypicolinamide Show/Hide	C35H34N6O3	1
1	IC50 = 2 nM Bioactivity Info	TI LI LO TS
CP0421892 Compound Info	(R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-2-yl)acetamide Show/Hide	C34H32N6O2	1
1	IC50 = 3 nM Bioactivity Info	TI LI LO TS
CP0395265 Compound Info	3-fluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide Show/Hide	C34H31FN6O2	1
1	IC50 = 3 nM Bioactivity Info	TI LI LO TS
CP0491423 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-6-methylpyridine-2-carboxamide Show/Hide	C35H34N6O2	1
1	IC50 = 3.4 nM Bioactivity Info	TI LI LO TS
CP0219009 Compound Info	US9708370, GHRP-6 Show/Hide	C46H56N12O6	2
1	IC50 = 3.65 nM Bioactivity Info	TI LI LO TS
2	IC50 = 6.08 nM Bioactivity Info	TI LI LO TS
CP0385058 Compound Info	3,5-difluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide Show/Hide	C34H30F2N6O2	1
1	IC50 = 4 nM Bioactivity Info	TI LI LO TS
CP0462505 Compound Info	(R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)pyrazine-2-carboxamide Show/Hide	C33H31N7O3	1
1	IC50 = 5 nM Bioactivity Info	TI LI LO TS
CP0421812 Compound Info	(2S)-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]pyrrolidine-2-carboxamide Show/Hide	C36H39N7O3	1
1	IC50 = 5.6 nM Bioactivity Info	TI LI LO TS
CP0420542 Compound Info	2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazol-3-yl}ethyl]-2-methylpropanamide Show/Hide	C34H37N7O2	1
1	IC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0876615 Compound Info	N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)tetrahydro-2H-pyran-4-carboxamide Show/Hide	C34H39N5O3	1
1	IC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0501203 Compound Info	6-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide Show/Hide	C34H33N7O2	1
1	IC50 = 6 nM Bioactivity Info	TI LI LO TS
CP0510818 Compound Info	N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-3-carboxamide Show/Hide	C37H41N7O3	1
1	IC50 = 6.5 nM Bioactivity Info	TI LI LO TS
CP0454975 Compound Info	(3R)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}ethyl]piperidine-3-carboxamide Show/Hide	C34H38N6O2	1
1	IC50 = 7 nM Bioactivity Info	TI LI LO TS
CP0489342 Compound Info	(S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide Show/Hide	C36H39N7O2	1
1	IC50 = 7 nM Bioactivity Info	TI LI LO TS
CP0459855 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-2-yl)acetamide Show/Hide	C36H33N7O2	1
1	IC50 = 7.9 nM Bioactivity Info	TI LI LO TS
CP0457704 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)picolinamide Show/Hide	C36H33N7O2	1
1	IC50 = 8 nM Bioactivity Info	TI LI LO TS
CP0424338 Compound Info	(2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazol-3-yl}ethyl]pyrrolidine-2-carboxamide Show/Hide	C35H37N7O2	1
1	IC50 = 9 nM Bioactivity Info	TI LI LO TS
CP0890892 Compound Info	(S)-N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)pyrrolidine-2-carboxamide Show/Hide	C33H38N6O2	1
1	IC50 = 9.5 nM Bioactivity Info	TI LI LO TS
CP0454970 Compound Info	(3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazol-3-yl}ethyl]piperidine-3-carboxamide Show/Hide	C36H39N7O2	1
1	IC50 = 10 nM Bioactivity Info	TI LI LO TS
CP0435194 Compound Info	(2R)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}ethyl]piperidine-2-carboxamide Show/Hide	C34H38N6O2	1
1	IC50 = 11 nM Bioactivity Info	TI LI LO TS
CP0461127 Compound Info	2-amino-N-[(R)-1H-indol-3-yl-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]methyl]-2-methylpropanamide Show/Hide	C31H34N6O2	1
1	IC50 = 11 nM Bioactivity Info	TI LI LO TS
CP0424823 Compound Info	(R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O2	1
1	IC50 = 11 nM Bioactivity Info	TI LI LO TS
CP0378569 Compound Info	(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C35H39N7O	1
1	IC50 = 11 nM Bioactivity Info	TI LI LO TS
CP0403076 Compound Info	(R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)benzamide Show/Hide	C35H33N5O3	1
1	IC50 = 11.8 nM Bioactivity Info	TI LI LO TS
CP0424824 Compound Info	(R)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H38N6O2	1
1	IC50 = 12 nM Bioactivity Info	TI LI LO TS
CP0454971 Compound Info	N-[(1R)-1-{4-benzyl-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-3-carboxamide Show/Hide	C35H37N7O	1
1	IC50 = 13 nM Bioactivity Info	TI LI LO TS
CP0496602 Compound Info	(R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)pyrazine-2-carboxamide Show/Hide	C32H29N7O2	1
1	IC50 = 14 nM Bioactivity Info	TI LI LO TS
CP0378566 Compound Info	(R)-N-(1-(4-(2-(1H-indol-3-yl)ethyl)-5-(3-(1H-indol-3-yl)propyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C37H40N8O	1
1	IC50 = 14 nM Bioactivity Info	TI LI LO TS
CP0467750 Compound Info	(R)-N-(1-(5-(2-(1H-Indol-3-yl)ethyl)-4-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H35N7O	1
1	IC50 = 15 nM Bioactivity Info	TI LI LO TS
CP0310354 Compound Info	Examorelin Show/Hide	C47H58N12O6	1
1	IC50 = 15.9 nM Bioactivity Info	TI LI LO TS
CP0522237 Compound Info	(3S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}ethyl]piperidine-3-carboxamide Show/Hide	C34H38N6O2	1
1	IC50 = 16 nM Bioactivity Info	TI LI LO TS
CP0882982 Compound Info	(R,S)-N-((R)-1-(5-((1H-indol-3-yl)methyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide Show/Hide	C35H40N8O2	1
1	IC50 = 18 nM Bioactivity Info	TI LI LO TS
CP0906075 Compound Info	N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)cyclohexanecarboxamide Show/Hide	C35H41N5O2	1
1	IC50 = 18 nM Bioactivity Info	TI LI LO TS
CP0420539 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C34H37N7O2	1
1	IC50 = 18 nM Bioactivity Info	TI LI LO TS
CP0493357 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)pyrazine-2-carboxamide Show/Hide	C35H32N8O3	1
1	IC50 = 18.5 nM Bioactivity Info	TI LI LO TS
CP0434205 Compound Info	N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-4-carboxamide Show/Hide	C35H40N6O	1
1	IC50 = 19 nM Bioactivity Info	TI LI LO TS
CP0378565 Compound Info	(R)-N-(1-(4-(4-methylbenzyl)-5-(3-phenylpropyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H38N6O	1
1	IC50 = 21 nM Bioactivity Info	TI LI LO TS
CP0475200 Compound Info	(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(3-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C35H39N7O2	1
1	IC50 = 22 nM Bioactivity Info	TI LI LO TS
CP0112161 Compound Info	N-[(2R)-1-[[(1R)-1-formamido-2-(1H-indol-3-yl)ethyl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-methyl-2-(methylamino)propanamide Show/Hide	C27H32N6O3	1
1	IC50 = 22.7 nM Bioactivity Info	TI LI LO TS
CP0477945 Compound Info	(2S)-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}ethyl]piperidine-2-carboxamide Show/Hide	C34H38N6O2	1
1	IC50 = 23 nM Bioactivity Info	TI LI LO TS
CP0454973 Compound Info	N-[(1R)-1-{4-benzyl-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-4-carboxamide Show/Hide	C35H37N7O	1
1	IC50 = 24 nM Bioactivity Info	TI LI LO TS
CP0454978 Compound Info	(2R)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazol-3-yl}ethyl]pyrrolidine-2-carboxamide Show/Hide	C35H37N7O2	1
1	IC50 = 28 nM Bioactivity Info	TI LI LO TS
CP0511871 Compound Info	(R)-N-(1-(5-(2-(1H-indol-2-yl)ethyl)-4-(4-methylbenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C34H37N7O	1
1	IC50 = 28 nM Bioactivity Info	TI LI LO TS
CP0485812 Compound Info	(2R)-N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazol-3-yl}ethyl]piperidine-2-carboxamide Show/Hide	C36H39N7O2	1
1	IC50 = 29 nM Bioactivity Info	TI LI LO TS
CP0427676 Compound Info	(R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-3-yl)acetamide Show/Hide	C34H32N6O2	1
1	IC50 = 29 nM Bioactivity Info	TI LI LO TS
CP0102070 Compound Info	N-[(2R)-1-[[(1R)-1-acetamido-2-(1H-indol-3-yl)ethyl]-methylamino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-methyl-2-(methylamino)propanamide Show/Hide	C29H36N6O3	1
1	IC50 = 29.5 nM Bioactivity Info	TI LI LO TS
CP0385963 Compound Info	2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}ethyl]acetamide Show/Hide	C30H32N6O2	1
1	IC50 = 32 nM Bioactivity Info	TI LI LO TS
CP0890895 Compound Info	(R,S)-N-((R)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide Show/Hide	C36H42N8O3	1
1	IC50 = 32 nM Bioactivity Info	TI LI LO TS
CP0910549 Compound Info	(R)-N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)pyrrolidine-2-carboxamide Show/Hide	C33H38N6O2	1
1	IC50 = 32 nM Bioactivity Info	TI LI LO TS
CP0421832 Compound Info	N-[(R)-[4-(2,4-dimethoxyphenyl)-5-(2-phenylethyl)-1,2,4-triazol-3-yl]-(1H-indol-3-yl)methyl]pyridine-2-carboxamide Show/Hide	C33H30N6O3	1
1	IC50 = 33 nM Bioactivity Info	TI LI LO TS
CP0378570 Compound Info	(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C34H37N7O	1
1	IC50 = 33 nM Bioactivity Info	TI LI LO TS
CP0464178 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-2-yl)acetamide Show/Hide	C37H35N7O3	1
1	IC50 = 34 nM Bioactivity Info	TI LI LO TS
CP0877433 Compound Info	N-((R)-1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide Show/Hide	C34H41N7O3	1
1	IC50 = 35 nM Bioactivity Info	TI LI LO TS
CP0434204 Compound Info	2-amino-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]acetamide Show/Hide	C33H35N7O3	1
1	IC50 = 38 nM Bioactivity Info	TI LI LO TS
CP0484685 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-1-oxidopyridin-1-ium-2-carboxamide Show/Hide	C34H32N6O3	1
1	IC50 = 42 nM Bioactivity Info	TI LI LO TS
CP0911147 Compound Info	(S)-N-((R)-1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)pyrrolidine-2-carboxamide Show/Hide	C34H40N6O3	1
1	IC50 = 44 nM Bioactivity Info	TI LI LO TS
CP0428458 Compound Info	(R)-N-(1-(4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H38N6O	1
1	IC50 = 44 nM Bioactivity Info	TI LI LO TS
CP0486752 Compound Info	(R)-tetrahydro-2H-pyran-4-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethylcarbamate Show/Hide	C36H38N6O4	1
1	IC50 = 45 nM Bioactivity Info	TI LI LO TS
CP0461142 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-ethylphenyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)picolinamide Show/Hide	C35H31N7O	1
1	IC50 = 49 nM Bioactivity Info	TI LI LO TS
CP0393028 Compound Info	(R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-2-yl)acetamide Show/Hide	C35H34N6O	1
1	IC50 = 51 nM Bioactivity Info	TI LI LO TS
CP0890896 Compound Info	N-((R)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-2-carboxamide Show/Hide	C36H39N7O2	1
1	IC50 = 53 nM Bioactivity Info	TI LI LO TS
CP0890894 Compound Info	N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide Show/Hide	C33H39N7O2	1
1	IC50 = 54 nM Bioactivity Info	TI LI LO TS
CP0441883 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3,4-dichlorobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H33Cl2N7O	1
1	IC50 = 55 nM Bioactivity Info	TI LI LO TS
CP0436918 Compound Info	(R)-N-(1-(4-(2-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O2	1
1	IC50 = 56 nM Bioactivity Info	TI LI LO TS
CP0160317 Compound Info	N-[(2R)-1-[[(1R)-1-acetamido-2-(1H-indol-3-yl)ethyl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-methyl-2-(methylamino)propanamide Show/Hide	C28H34N6O3	1
1	IC50 = 58 nM Bioactivity Info	TI LI LO TS
CP0464204 Compound Info	(R)-N-((4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)isonicotinamide Show/Hide	C34H32N6O3	1
1	IC50 = 58 nM Bioactivity Info	TI LI LO TS
CP0906077 Compound Info	(R)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-3-aminopropanamide Show/Hide	C31H36N6O2	1
1	IC50 = 59 nM Bioactivity Info	TI LI LO TS
CP0393030 Compound Info	2-amino-N-[(R)-[4-[(2,4-dimethoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]-(1H-indol-3-yl)methyl]-2-methylpropanamide Show/Hide	C32H36N6O3	1
1	IC50 = 60 nM Bioactivity Info	TI LI LO TS
CP0454074 Compound Info	(R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H38N6O3	2
1	IC50 = 60 nM Bioactivity Info	TI LI LO TS
2	IC50 = 62 nM Bioactivity Info	TI LI LO TS
CP0454088 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-benzyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-2-yl)acetamide Show/Hide	C35H31N7O	1
1	IC50 = 61 nM Bioactivity Info	TI LI LO TS
CP0513888 Compound Info	2-amino-N-[(2R)-1-[[(2R)-1-amino-3-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]-2-methylpropanamide Show/Hide	C28H34N6O3	1
1	IC50 = 62.9 nM Bioactivity Info	TI LI LO TS
CP0879905 Compound Info	N-((R)-1-(4-(2,4-dimethoxyphenyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide Show/Hide	C34H40N6O3	1
1	IC50 = 63 nM Bioactivity Info	TI LI LO TS
CP0425157 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-5-pyrrolidin-1-ylpyridine-2-carboxamide Show/Hide	C38H39N7O2	1
1	IC50 = 65 nM Bioactivity Info	TI LI LO TS
CP0495967 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-fluorobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H34FN7O	1
1	IC50 = 66 nM Bioactivity Info	TI LI LO TS
CP0449132 Compound Info	(R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)picolinamide Show/Hide	C34H32N6O	1
1	IC50 = 67 nM Bioactivity Info	TI LI LO TS
CP0454968 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-{5-[2-(1H-indol-3-yl)ethyl]-4-phenyl-4H-1,2,4-triazol-3-yl}ethyl]piperidine-4-carboxamide Show/Hide	C34H35N7O	1
1	IC50 = 70 nM Bioactivity Info	TI LI LO TS
CP0530462 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-4-yl)acetamide Show/Hide	C36H33N7O2	1
1	IC50 = 76 nM Bioactivity Info	TI LI LO TS
CP0419726 Compound Info	(R)-N-(1-(4-(3-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O2	1
1	IC50 = 78 nM Bioactivity Info	TI LI LO TS
CP0449111 Compound Info	(R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)benzamide Show/Hide	C34H31N5O2	1
1	IC50 = 80 nM Bioactivity Info	TI LI LO TS
CP0475199 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C34H37N7O	1
1	IC50 = 80 nM Bioactivity Info	TI LI LO TS
CP0455042 Compound Info	(S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C35H39N7O3	1
1	IC50 = 83 nM Bioactivity Info	TI LI LO TS
CP0406403 Compound Info	5-bromo-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide Show/Hide	C34H31BrN6O2	1
1	IC50 = 84 nM Bioactivity Info	TI LI LO TS
CP0454087 Compound Info	(R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)pyrazine-2-carboxamide Show/Hide	C33H31N7O	1
1	IC50 = 89 nM Bioactivity Info	TI LI LO TS
CP0485811 Compound Info	N-[(1R)-1-[4-(4-ethylphenyl)-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]piperidine-4-carboxamide Show/Hide	C36H39N7O	1
1	IC50 = 96 nM Bioactivity Info	TI LI LO TS
CP0433215 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(4-ethylphenyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-2-yl)acetamide Show/Hide	C36H33N7O	1
1	IC50 = 96 nM Bioactivity Info	TI LI LO TS
CP0378572 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2-methoxy)benzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C34H37N7O2	1
1	IC50 = 96 nM Bioactivity Info	TI LI LO TS
CP0436927 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-bromobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H34BrN7O	1
1	IC50 = 100 nM Bioactivity Info	TI LI LO TS
CP0388314 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]isoquinoline-3-carboxamide Show/Hide	C38H34N6O2	1
1	IC50 = 100 nM Bioactivity Info	TI LI LO TS
CP0428227 Compound Info	(R)-N-((1H-indol-3-yl)(5-phenethyl-4-phenyl-4H-1,2,4-triazol-3-yl)methyl)picolinamide Show/Hide	C31H26N6O	1
1	IC50 = 105 nM Bioactivity Info	TI LI LO TS
CP0510581 Compound Info	2-amino-N-[(R)-[4-[(2,4-dimethoxyphenyl)methyl]-5-[2-(1H-indol-3-yl)ethyl]-1,2,4-triazol-3-yl]-(1H-indol-3-yl)methyl]-2-methylpropanamide Show/Hide	C34H37N7O3	1
1	IC50 = 108 nM Bioactivity Info	TI LI LO TS
CP0454068 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C35H39N7O3	1
1	IC50 = 108 nM Bioactivity Info	TI LI LO TS
CP0424822 Compound Info	(R)-N-(1-(4-(3,5-dimethoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O3	1
1	IC50 = 110 nM Bioactivity Info	TI LI LO TS
CP0464203 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-aminobenzamide Show/Hide	C37H35N7O3	1
1	IC50 = 112 nM Bioactivity Info	TI LI LO TS
CP0906079 Compound Info	(S)-N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-aminopropanamide Show/Hide	C31H36N6O2	1
1	IC50 = 113 nM Bioactivity Info	TI LI LO TS
CP0235411 Compound Info	N-[(1R)-1-[[(2R)-2-[(2-amino-2-methylpropanoyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-2-(1H-indol-3-yl)ethyl]piperidine-2-carboxamide Show/Hide	C31H39N7O3	1
1	IC50 = 116 nM Bioactivity Info	TI LI LO TS
CP0428225 Compound Info	N-[(R)-[4-(2,4-dimethoxyphenyl)-5-(2-phenylethyl)-1,2,4-triazol-3-yl]-(1H-indol-3-yl)methyl]-2-pyridin-2-ylacetamide Show/Hide	C34H32N6O3	1
1	IC50 = 120 nM Bioactivity Info	TI LI LO TS
CP0455074 Compound Info	(R)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C31H34N6O2	2
1	IC50 = 120 nM Bioactivity Info	TI LI LO TS
2	IC50 = 121 nM Bioactivity Info	TI LI LO TS
CP0495992 Compound Info	(R)-N-(1-(4-(3-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C31H34N6O2	1
1	IC50 = 120 nM Bioactivity Info	TI LI LO TS
CP0112074 Compound Info	ethyl N-[(1S)-1-[[(2R)-2-[(2-amino-2-methylpropanoyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-2-(1H-indol-3-yl)ethyl]carbamate Show/Hide	C28H34N6O4	1
1	IC50 = 122 nM Bioactivity Info	TI LI LO TS
CP0380801 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide Show/Hide	C34H32N6O2	1
1	IC50 = 122 nM Bioactivity Info	TI LI LO TS
CP0303771 Compound Info	2-Amino-N-{(R)-1-[(R)-1-formylamino-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-1H-indol-3-yl-ethyl}-2-methyl-propionamide Show/Hide	C26H30N6O3	1
1	IC50 = 123 nM Bioactivity Info	TI LI LO TS
CP0439499 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(naphthalen-1-ylmethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C37H37N7O	1
1	IC50 = 125 nM Bioactivity Info	TI LI LO TS
CP0435195 Compound Info	(3S)-N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]piperidine-3-carboxamide Show/Hide	C35H40N6O	1
1	IC50 = 130 nM Bioactivity Info	TI LI LO TS
CP0441466 Compound Info	(R)-N-(2-(1H-indol-3-yl)-1-(4-(naphthalen-1-ylmethyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C35H36N6O	1
1	IC50 = 130 nM Bioactivity Info	TI LI LO TS
CP0386294 Compound Info	6-chloro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide Show/Hide	C34H31ClN6O2	1
1	IC50 = 130 nM Bioactivity Info	TI LI LO TS
CP0916143 Compound Info	(S)-N-((R)-1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-2-carboxamide Show/Hide	C35H40N6O3	1
1	IC50 = 134 nM Bioactivity Info	TI LI LO TS
CP0906078 Compound Info	N-((R)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-aminoacetamide Show/Hide	C32H33N7O2	1
1	IC50 = 138 nM Bioactivity Info	TI LI LO TS
CP0421826 Compound Info	(1S,2R)-N-((R)-(5-(2-(1H-indol-3-yl)ethyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-aminocyclohexanecarboxamide Show/Hide	C37H41N7O3	1
1	IC50 = 140 nM Bioactivity Info	TI LI LO TS
CP0462522 Compound Info	(S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C34H37N7O2	1
1	IC50 = 140 nM Bioactivity Info	TI LI LO TS
CP0378577 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-phenyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H33N7O	1
1	IC50 = 140 nM Bioactivity Info	TI LI LO TS
CP0378583 Compound Info	(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(naphthalen-1-ylmethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C38H39N7O	1
1	IC50 = 140 nM Bioactivity Info	TI LI LO TS
CP0424813 Compound Info	(R)-N-(1-(4-(4-methylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O	1
1	IC50 = 140 nM Bioactivity Info	TI LI LO TS
CP0383401 Compound Info	(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C35H39N7O2	1
1	IC50 = 145 nM Bioactivity Info	TI LI LO TS
CP0432708 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(3,5-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C35H39N7O3	1
1	IC50 = 150 nM Bioactivity Info	TI LI LO TS
CP0441882 Compound Info	(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(4-bromobenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C34H36BrN7O	1
1	IC50 = 150 nM Bioactivity Info	TI LI LO TS
CP0495988 Compound Info	(R)-N-(1-(4,5-bis(2-(1H-indol-3-yl)ethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C36H38N8O	1
1	IC50 = 150 nM Bioactivity Info	TI LI LO TS
CP0432522 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]isoquinoline-1-carboxamide Show/Hide	C38H34N6O2	1
1	IC50 = 150 nM Bioactivity Info	TI LI LO TS
CP0454972 Compound Info	2-amino-N-[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]acetamide Show/Hide	C31H34N6O3	1
1	IC50 = 154 nM Bioactivity Info	TI LI LO TS
CP0393029 Compound Info	(R)-N-((5-(2-(1H-indol-3-yl)ethyl)-4-phenyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)picolinamide Show/Hide	C33H27N7O	1
1	IC50 = 160 nM Bioactivity Info	TI LI LO TS
CP0310947 Compound Info	2-Amino-N-[1-[(R)-(S)-1-(3-ethyl-ureido)-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-(1H-indol-3-yl)-ethyl]-2-methyl-propionamide Show/Hide	C28H35N7O3	1
1	IC50 = 162 nM Bioactivity Info	TI LI LO TS
CP0272419 Compound Info	N-[(2R)-3-(1H-indol-3-yl)-1-[[(1R)-2-(1H-indol-3-yl)-1-(propanoylamino)ethyl]amino]-1-oxopropan-2-yl]-2-methyl-2-(methylamino)propanamide Show/Hide	C29H36N6O3	1
1	IC50 = 167 nM Bioactivity Info	TI LI LO TS
CP0433469 Compound Info	(R)-N-(1-(4-(4-fluorobenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C30H31FN6O	1
1	IC50 = 170 nM Bioactivity Info	TI LI LO TS
CP0477946 Compound Info	(2S,4R)-4-hydroxy-N-[(1R)-2-(1H-indol-3-yl)-1-{4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}ethyl]pyrrolidine-2-carboxamide Show/Hide	C33H36N6O3	1
1	IC50 = 173 nM Bioactivity Info	TI LI LO TS
CP0890893 Compound Info	(R)-N-((R)-1-(4-(4-methoxybenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-3-phenylpropanamide Show/Hide	C37H40N6O2	1
1	IC50 = 175 nM Bioactivity Info	TI LI LO TS
CP0455070 Compound Info	(S)-pyridin-2-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethylcarbamate Show/Hide	C36H33N7O3	1
1	IC50 = 175 nM Bioactivity Info	TI LI LO TS
CP0428223 Compound Info	(R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-3-(pyridin-3-yl)propanamide Show/Hide	C35H34N6O2	1
1	IC50 = 177 nM Bioactivity Info	TI LI LO TS
CP0906073 Compound Info	N-((R)-1-(4-(4-ethylbenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperazine-2-carboxamide Show/Hide	C34H41N7O	1
1	IC50 = 178 nM Bioactivity Info	TI LI LO TS
CP0454976 Compound Info	(2-aminoethyl)[(1R)-1-{4-[(2,4-dimethoxyphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]amine Show/Hide	C31H36N6O2	1
1	IC50 = 190 nM Bioactivity Info	TI LI LO TS
CP0475201 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-hexyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H41N7O	1
1	IC50 = 195 nM Bioactivity Info	TI LI LO TS
CP0461205 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-phenylethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O2	1
1	IC50 = 200 nM Bioactivity Info	TI LI LO TS
CP0421829 Compound Info	(R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)isonicotinamide Show/Hide	C33H30N6O2	1
1	IC50 = 220 nM Bioactivity Info	TI LI LO TS
CP0378584 Compound Info	(R)-2-amino-N-(1-(5-benzyl-4-(naphthalen-1-ylmethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide Show/Hide	C34H34N6O	1
1	IC50 = 220 nM Bioactivity Info	TI LI LO TS
CP0388828 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-4-carboxamide Show/Hide	C34H32N6O2	1
1	IC50 = 220 nM Bioactivity Info	TI LI LO TS
CP0302498 Compound Info	N-[(2R)-1-[[(1R)-1-acetamido-2-(1H-indol-3-yl)ethyl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-amino-2-methylpropanamide Show/Hide	C27H32N6O3	1
1	IC50 = 228 nM Bioactivity Info	TI LI LO TS
CP0428146 Compound Info	(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-hexyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H43N7O	1
1	IC50 = 240 nM Bioactivity Info	TI LI LO TS
CP0386295 Compound Info	3-hydroxy-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide Show/Hide	C34H32N6O3	1
1	IC50 = 240 nM Bioactivity Info	TI LI LO TS
CP0395264 Compound Info	3-benzoyl-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide Show/Hide	C41H36N6O3	1
1	IC50 = 240 nM Bioactivity Info	TI LI LO TS
CP0380802 Compound Info	2-bromo-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide Show/Hide	C34H31BrN6O2	1
1	IC50 = 250 nM Bioactivity Info	TI LI LO TS
CP0916574 Compound Info	N-((R)-2-(1H-indol-3-yl)-1-(5-phenethyl-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl)piperidine-4-carboxamide Show/Hide	C31H36N6OS	1
1	IC50 = 255 nM Bioactivity Info	TI LI LO TS
CP0428224 Compound Info	(R)-N-((4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-4-yl)acetamide Show/Hide	C34H32N6O2	1
1	IC50 = 270 nM Bioactivity Info	TI LI LO TS
CP0879904 Compound Info	(2S)-N-((R)-1-(4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-aminopropanamide Show/Hide	C32H38N6O	1
1	IC50 = 275 nM Bioactivity Info	TI LI LO TS
CP0702454 Compound Info	Tyr-Ala-hexarelin Show/Hide	C59H72N14O9	1
1	IC50 = 286 nM Bioactivity Info	TI LI LO TS
CP0421824 Compound Info	N-[(R)-[4-(2,4-dimethoxyphenyl)-5-(2-phenylethyl)-1,2,4-triazol-3-yl]-(1H-indol-3-yl)methyl]pyrazine-2-carboxamide Show/Hide	C32H29N7O3	1
1	IC50 = 300 nM Bioactivity Info	TI LI LO TS
CP0459826 Compound Info	2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[5-(1H-indol-3-ylmethyl)-4-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-2-methylpropanamide Show/Hide	C33H35N7O	1
1	IC50 = 300 nM Bioactivity Info	TI LI LO TS
CP0495968 Compound Info	2-amino-N-[(1R)-1-[4,5-bis(2-phenylethyl)-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C32H36N6O	1
1	IC50 = 310 nM Bioactivity Info	TI LI LO TS
CP0270411 Compound Info	4-Amino-piperidine-4-carboxylic acid [1-[(R)-(R)-1-formylamino-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-(1H-indol-3-yl)-ethyl]-amide Show/Hide	C28H33N7O3	1
1	IC50 = 337 nM Bioactivity Info	TI LI LO TS
CP0426995 Compound Info	(2S)-N-[(1R)-1-[4-(4-ethylphenyl)-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyrrolidine-2-carboxamide Show/Hide	C35H37N7O	1
1	IC50 = 350 nM Bioactivity Info	TI LI LO TS
CP0910550 Compound Info	(R)-N-((R)-1-(4-(4-ethylbenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-2-carboxamide Show/Hide	C35H42N6O	1
1	IC50 = 375 nM Bioactivity Info	TI LI LO TS
CP0432521 Compound Info	2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide Show/Hide	C34H33N7O2	1
1	IC50 = 380 nM Bioactivity Info	TI LI LO TS
CP0509277 Compound Info	N-[(1R)-2-(1H-indol-3-yl)-1-[[(2R)-3-(1H-indol-3-yl)-2-[[2-methyl-2-(methylamino)propanoyl]amino]propanoyl]amino]ethyl]-3-methylbutanamide Show/Hide	C31H40N6O3	1
1	IC50 = 397 nM Bioactivity Info	TI LI LO TS
CP0419723 Compound Info	2-amino-N-[(1R)-1-[4-[(4-fluorophenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C31H33FN6O	1
1	IC50 = 400 nM Bioactivity Info	TI LI LO TS
CP0441879 Compound Info	(R)-N-(1-(4-(2-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C31H34N6O2	1
1	IC50 = 410 nM Bioactivity Info	TI LI LO TS
CP0378563 Compound Info	(R)-2-amino-N-(1-(4-(furan-2-ylmethyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide Show/Hide	C29H32N6O2	1
1	IC50 = 420 nM Bioactivity Info	TI LI LO TS
CP0268289 Compound Info	N-[(2R)-1-[[(1R)-1-acetamido-2-(1H-indol-3-yl)ethyl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-(dimethylamino)-2-methylpropanamide Show/Hide	C29H36N6O3	1
1	IC50 = 440 nM Bioactivity Info	TI LI LO TS
CP0378574 Compound Info	2-amino-N-[(1R)-1-[5-benzyl-4-[(4-bromophenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C30H31BrN6O	1
1	IC50 = 440 nM Bioactivity Info	TI LI LO TS
CP0464261 Compound Info	(S)-N-(1-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H38N6O3	1
1	IC50 = 450 nM Bioactivity Info	TI LI LO TS
CP0486728 Compound Info	(R)-benzyl 3-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-3-(2-amino-2-methylpropanamido)propanoate Show/Hide	C34H38N6O4	1
1	IC50 = 450 nM Bioactivity Info	TI LI LO TS
CP0193125 Compound Info	2-Amino-N-{2-(1H-indol-3-yl)-1-[(R)-(R)-2-(1H-indol-3-yl)-1-propionylamino-ethylcarbamoyl]-ethyl}-2-methyl-propionamide Show/Hide	C28H34N6O3	1
1	IC50 = 460 nM Bioactivity Info	TI LI LO TS
CP0526050 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-(naphthalen-1-ylmethyl)carbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C47H56N12O6	1
1	IC50 = 465 nM Bioactivity Info	TI LI LO TS
CP0957155 Compound Info	2-((S)-2-amino-3-(1H-imidazol-5-yl)propanoyl)-N-((S)-1-((S)-1-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-1-(naphthalen-1-ylmethyl)hydrazinecarboxamide Show/Hide	C47H56N12O6	1
1	IC50 = 465 nM Bioactivity Info	TI LI LO TS
CP0920117 Compound Info	N-((R)-2-(1H-indol-3-yl)-1-(5-phenethyl-4-phenyl-4H-1,2,4-triazol-3-yl)ethyl)piperidine-4-carboxamide Show/Hide	C32H36N6O	1
1	IC50 = 468 nM Bioactivity Info	TI LI LO TS
CP0441894 Compound Info	2-amino-N-((R)-1-(5-benzyl-4-hexyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide Show/Hide	C29H38N6O	1
1	IC50 = 470 nM Bioactivity Info	TI LI LO TS
CP0393046 Compound Info	(R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)-2-(pyridin-3-yl)acetamide Show/Hide	C35H34N6O	1
1	IC50 = 480 nM Bioactivity Info	TI LI LO TS
CP0890891 Compound Info	(S)-N-((R)-1-(4-(4-ethylbenzyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)pyrrolidine-2-carboxamide Show/Hide	C34H40N6O	1
1	IC50 = 490 nM Bioactivity Info	TI LI LO TS
CP0378575 Compound Info	2-amino-N-((R)-1-(4,5-dibenzyl-4H-1,2,4-triazol-3-yl)-2-(1Hindol-3-yl)ethyl)-2-methylpropanamide Show/Hide	C30H32N6O	1
1	IC50 = 500 nM Bioactivity Info	TI LI LO TS
CP0420540 Compound Info	2-amino-N-[(1R)-1-[5-benzyl-4-(3,4-dichlorophenyl)-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C29H28Cl2N6O	1
1	IC50 = 520 nM Bioactivity Info	TI LI LO TS
CP0090232 Compound Info	N-[(1R)-1-[[(2R)-2-[(2-amino-2-methylpropanoyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-2-(1H-indol-3-yl)ethyl]-3-methylbutanamide Show/Hide	C30H38N6O3	1
1	IC50 = 535 nM Bioactivity Info	TI LI LO TS
CP0378580 Compound Info	2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[2-(4-methoxyphenyl)ethyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-2-methylpropanamide Show/Hide	C33H38N6O2	1
1	IC50 = 550 nM Bioactivity Info	TI LI LO TS
CP0879903 Compound Info	N-((R)-1-(4-(furan-2-ylmethyl)-5-phenethyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)piperidine-4-carboxamide Show/Hide	C31H36N6O2	1
1	IC50 = 560 nM Bioactivity Info	TI LI LO TS
CP0419722 Compound Info	(R)-N-(1-(4-(2,4-dimethoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O3	1
1	IC50 = 560 nM Bioactivity Info	TI LI LO TS
CP0553631 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[(2R)-2-[[(2S)-2-aminopropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]carbamoylamino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C41H51N11O6	1
1	IC50 = 568 nM Bioactivity Info	TI LI LO TS
CP0378579 Compound Info	(R)-N-(2-(1H-indol-3-yl)-1-(5-phenethyl-4-(thiophen-2-ylmethyl)-4H-1,2,4-triazol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C29H32N6OS	1
1	IC50 = 570 nM Bioactivity Info	TI LI LO TS
CP0433471 Compound Info	(R)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-methyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C27H31N7O	1
1	IC50 = 580 nM Bioactivity Info	TI LI LO TS
CP0433470 Compound Info	2-amino-N-[(1R)-1-[4-(2,2-diphenylethyl)-5-[2-(1H-indol-3-yl)ethyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C40H41N7O	1
1	IC50 = 640 nM Bioactivity Info	TI LI LO TS
CP0495989 Compound Info	2-amino-N-[(1R)-1-[4-[(3,4-dichlorophenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C31H32Cl2N6O	1
1	IC50 = 640 nM Bioactivity Info	TI LI LO TS
CP0897607 Compound Info	(S)-N-((S)-1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)pyrrolidine-2-carboxamide Show/Hide	C35H37N7O2	1
1	IC50 = 650 nM Bioactivity Info	TI LI LO TS
CP0419721 Compound Info	(R)-N-(1-(5-((1H-indol-3-yl)methyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H35N7O2	1
1	IC50 = 660 nM Bioactivity Info	TI LI LO TS
CP0421828 Compound Info	(R)-N-((1H-indol-3-yl)(5-phenethyl-4-phenyl-4H-1,2,4-triazol-3-yl)methyl)-2-(pyridin-2-yl)acetamide Show/Hide	C32H28N6O	1
1	IC50 = 700 nM Bioactivity Info	TI LI LO TS
CP0495969 Compound Info	2-amino-N-[(1R)-1-[5-benzyl-4-[2-(1H-indol-3-yl)ethyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C33H35N7O	1
1	IC50 = 700 nM Bioactivity Info	TI LI LO TS
CP0521164 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-(naphthalen-1-ylmethyl)carbamoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C47H56N12O6	1
1	IC50 = 723 nM Bioactivity Info	TI LI LO TS
CP0546578 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-(2-phenylethyl)carbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C44H56N12O6	1
1	IC50 = 729 nM Bioactivity Info	TI LI LO TS
CP0907447 Compound Info	2-((S)-2-amino-3-(1H-imidazol-5-yl)propanoyl)-N-((S)-1-((S)-1-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-1-phenethylhydrazinecarboxamide Show/Hide	C44H56N12O6	1
1	IC50 = 729 nM Bioactivity Info	TI LI LO TS
CP0378562 Compound Info	(R)-N-(1-(5-(3-(1H-indol-3-yl)propyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C36H41N7O3	1
1	IC50 = 750 nM Bioactivity Info	TI LI LO TS
CP0527424 Compound Info	(2S,11S)-11-amino-N-[(2R)-1-[[(2R)-6-amino-1-[[(2S)-1-[[(2R)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]-12-oxo-1-azatricyclo[6.4.1.04,13]trideca-4,6,8(13)-triene-2-carboxamide Show/Hide	C57H70N12O7	1
1	IC50 = 750 nM Bioactivity Info	TI LI LO TS
CP0434203 Compound Info	2-amino-N-[(1R)-1-{4-[(4-ethylphenyl)methyl]-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl}-2-(1H-indol-3-yl)ethyl]acetamide Show/Hide	C31H34N6O	1
1	IC50 = 759 nM Bioactivity Info	TI LI LO TS
CP0499991 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C44H55N11O7	1
1	IC50 = 771 nM Bioactivity Info	TI LI LO TS
CP0454071 Compound Info	(S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(benzyloxy)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H38N6O3	1
1	IC50 = 800 nM Bioactivity Info	TI LI LO TS
CP0258518 Compound Info	N-[(2R)-1-[[(1R)-1-acetamido-2-(1H-indol-3-yl)ethyl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]piperidine-4-carboxamide Show/Hide	C29H34N6O3	1
1	IC50 = 807 nM Bioactivity Info	TI LI LO TS
CP0378818 Compound Info	4-Amino-piperidine-4-carboxylic acid [1-[(R)-(R)-1-acetylamino-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-(1H-indol-3-yl)-ethyl]-amide Show/Hide	C29H35N7O3	1
1	IC50 = 807 nM Bioactivity Info	TI LI LO TS
CP0513891 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]carbamoylamino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C44H53N13O6	1
1	IC50 = 808 nM Bioactivity Info	TI LI LO TS
CP0464296 Compound Info	(S)-N-(1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)picolinamide Show/Hide	C36H33N7O2	1
1	IC50 = 820 nM Bioactivity Info	TI LI LO TS
CP0378582 Compound Info	(R)-N-(1-(4-(4-methylbenzyl)-5-(3-benzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C31H34N6O	1
1	IC50 = 840 nM Bioactivity Info	TI LI LO TS
CP0475202 Compound Info	(R)-N-(1-(4-(2-(1H-indol-3-yl)ethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C26H29N7O	1
1	IC50 = 850 nM Bioactivity Info	TI LI LO TS
CP0552413 Compound Info	(R)-N-(1-(5-((1H-indol-3-yl)methyl)-4-(2,4-dimethoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C34H37N7O3	1
1	IC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0553630 Compound Info	(2S)-N-[(2R)-1-[2-[[(2S)-1-[[(2R)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]carbamoyl]-2-(2-methylpropyl)hydrazinyl]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]pyrrolidine-2-carboxamide Show/Hide	C47H61N11O6	1
1	IC50 = 1170 nM Bioactivity Info	TI LI LO TS
CP0453467 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C48H61N13O6	1
1	IC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0486754 Compound Info	(S)-tetrahydro-2H-pyran-4-yl 1-(5-(2-(1H-indol-3-yl)ethyl)-4-(4-methoxybenzyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethylcarbamate Show/Hide	C36H38N6O4	1
1	IC50 = 1300 nM Bioactivity Info	TI LI LO TS
CP0488660 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-[(4-phenylphenyl)methyl]carbamoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C49H58N12O6	1
1	IC50 = 1340 nM Bioactivity Info	TI LI LO TS
CP0526049 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-[(4-phenylphenyl)methyl]carbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C49H58N12O6	1
1	IC50 = 1640 nM Bioactivity Info	TI LI LO TS
CP0958469 Compound Info	2-((S)-2-amino-3-(1H-imidazol-5-yl)propanoyl)-1-(biphenyl-4-ylmethyl)-N-((S)-1-((S)-1-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)hydrazinecarboxamide Show/Hide	C49H58N12O6	1
1	IC50 = 1640 nM Bioactivity Info	TI LI LO TS
CP0427139 Compound Info	(R)-N-(1-(5-((1H-indol-3-yl)methyl)-4-methyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C26H29N7O	1
1	IC50 = 1700 nM Bioactivity Info	TI LI LO TS
CP0424830 Compound Info	(R)-N-(1-(5-((1H-indol-3-yl)methyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C25H27N7O	1
1	IC50 = 2200 nM Bioactivity Info	TI LI LO TS
CP0455304 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-benzylcarbamoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C43H54N12O6	1
1	IC50 = 2770 nM Bioactivity Info	TI LI LO TS
CP0526047 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2R)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C44H55N11O7	1
1	IC50 = 3250 nM Bioactivity Info	TI LI LO TS
CP0546576 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[[(2R)-2-[[(2R)-2-aminopropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C45H59N11O6	1
1	IC50 = 3610 nM Bioactivity Info	TI LI LO TS
CP0413909 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-(2-phenylethyl)carbamoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C44H56N12O6	1
1	IC50 = 3740 nM Bioactivity Info	TI LI LO TS
CP0546577 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-3-(1H-indol-3-yl)-2-[[[[(2R)-3-(1H-indol-3-yl)-2-(propanoylamino)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C45H58N10O6	1
1	IC50 = 3860 nM Bioactivity Info	TI LI LO TS
CP0966456 Compound Info	2-((S)-2-((R)-2-((S)-2-amino-3-(1H-imidazol-5-yl)propanamido)-3-(1H-indol-3-yl)propanamido)propanoyl)-1-(cyclohexylmethyl)-N-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)hydrazinecarboxamide Show/Hide	C43H60N12O6	1
1	IC50 = 4280 nM Bioactivity Info	TI LI LO TS
CP0565972 Compound Info	(2R)-2-[[(2S)-2-[[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanamide Show/Hide	C42H49N11O5	1
1	IC50 = 4550 nM Bioactivity Info	TI LI LO TS
CP0565973 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[[(2R)-2-[(2-aminoacetyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C44H57N11O6	1
1	IC50 = 5410 nM Bioactivity Info	TI LI LO TS
CP0897006 Compound Info	2-((S)-2-amino-3-(1H-imidazol-5-yl)propanoyl)-1-(cyclohexylmethyl)-N-((S)-1-((S)-1-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)hydrazinecarboxamide Show/Hide	C43H60N12O6	1
1	IC50 = 5490 nM Bioactivity Info	TI LI LO TS
CP0453607 Compound Info	(2R)-2-[[(2S)-2-[[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-N-[(2S)-1-amino-1-oxopropan-2-yl]-3-phenylpropanamide Show/Hide	C45H54N12O6	1
1	IC50 = 8170 nM Bioactivity Info	TI LI LO TS
CP0441032 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-[(4-hydroxyphenyl)methyl]carbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C43H54N12O7	1
1	IC50 = 8530 nM Bioactivity Info	TI LI LO TS
CP0962126 Compound Info	2-((S)-2-amino-3-(1H-imidazol-5-yl)propanoyl)-N-((S)-1-((S)-1-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-1-(4-hydroxybenzyl)hydrazinecarboxamide Show/Hide	C43H54N12O7	1
1	IC50 = 8530 nM Bioactivity Info	TI LI LO TS
CP0397561 Compound Info	2-[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]-N-[(2S)-1-[[(2R)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]pyrazolidine-1-carboxamide Show/Hide	C47H57N13O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0397563 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-aminopropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-benzylcarbamoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C40H52N10O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0397565 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[(2S)-2-aminopropanoyl]amino]-benzylcarbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C40H52N10O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0413906 Compound Info	2-[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]-N-[(2S)-1,6-diamino-1-oxohexan-2-yl]pyrazolidine-1-carboxamide Show/Hide	C41H53N13O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0431200 Compound Info	(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-benzylcarbamoyl]amino]-N-[(2S)-1-amino-1-oxopropan-2-yl]-3-phenylpropanamide Show/Hide	C40H47N11O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0453608 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-benzylcarbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]hexanamide Show/Hide	C37H50N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0463511 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C40H56N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0463512 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]propanoyl]amino]-benzylcarbamoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C35H49N11O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0463514 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]carbamoylamino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]hexanamide Show/Hide	C38H49N13O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0463515 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-benzylcarbamoyl]amino]propanoyl]amino]hexanamide Show/Hide	C37H50N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0473935 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C40H56N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0476936 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-benzylcarbamoyl]amino]propanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C35H49N11O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0480292 Compound Info	2-[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]-N-[(2R)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrazolidine-1-carboxamide Show/Hide	C39H52N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0483294 Compound Info	(2R)-2-[[(2S)-2-[[(2S)-2-[[[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-[(4-hydroxyphenyl)methyl]carbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-N-[(2S)-1-amino-1-oxopropan-2-yl]-3-phenylpropanamide Show/Hide	C40H47N11O7	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0483296 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[(2S)-2-aminopropanoyl]amino]-[(4-hydroxyphenyl)methyl]carbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C40H52N10O7	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0488659 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]hexanamide Show/Hide	C42H57N13O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0499989 Compound Info	(2S)-1-[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]carbamoyl]-N-[(2R)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide Show/Hide	C38H50N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0499990 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-[(4-hydroxyphenyl)methyl]carbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]hexanamide Show/Hide	C37H50N12O7	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0513889 Compound Info	2-[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]-N-[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]pyrazolidine-1-carboxamide Show/Hide	C39H52N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0513890 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]carbamoylamino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C36H48N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0526046 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]carbamoylamino]propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C36H48N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0546575 Compound Info	(2S)-2-[[[[(2R)-2-amino-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanamide Show/Hide	C27H33N7O3	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0553632 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-[(4-hydroxyphenyl)methyl]carbamoyl]amino]propanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C35H49N11O7	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0413908 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[[[(2R)-2-[[(2S)-2-aminopropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C45H59N11O6	2
1	IC50 >= 10000 nM Bioactivity Info	TI LI LO TS
2	IC50 = 11200 nM Bioactivity Info	TI LI LO TS
CP0535726 Compound Info	(2R)-2-[[(2S)-2-[[(2S)-2-[[[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-benzylcarbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-N-[(2S)-1-amino-1-oxopropan-2-yl]-3-phenylpropanamide Show/Hide	C40H47N11O6	2
1	IC50 >= 10000 nM Bioactivity Info	TI LI LO TS
2	IC50 = 51000 nM Bioactivity Info	TI LI LO TS
CP0897007 Compound Info	2-((S)-2-((R)-2-((S)-2-amino-3-phenylpropanamido)-3-(1H-indol-3-yl)propanamido)propanoyl)-N-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-(4-hydroxybenzyl)hydrazinecarboxamide Show/Hide	C46H56N10O7	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0897008 Compound Info	H-Ala-D-Trp-Ala-azaTyr-D-Phe-Lys-NH2 Show/Hide	C40H52N10O7	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0955466 Compound Info	1-(2-((R)-2-((S)-2-amino-3-(1H-imidazol-5-yl)propanamido)-3-(1H-indol-3-yl)propanoyl)hydrazinecarbonyl)-N-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)pyrrolidine-2-carboxamide Show/Hide	C38H50N12O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0955467 Compound Info	2-((S)-2-((R)-3-(1H-indol-3-yl)-2-(3-phenylpropanamido)propanamido)propanoyl)-N-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-1-(4-hydroxybenzyl)hydrazinecarboxamide Show/Hide	C46H55N9O7	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0958470 Compound Info	2-((S)-2-amino-3-(1H-imidazol-5-yl)propanoyl)-1-benzyl-N-((S)-1-((S)-1-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)hydrazinecarboxamide Show/Hide	C35H49N11O6	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0962127 Compound Info	2-((S)-2-amino-3-(1H-imidazol-5-yl)propanoyl)-N-((S)-1-((S)-1-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-1-(4-hydroxybenzyl)hydrazinecarboxamide Show/Hide	C35H49N11O7	1
1	IC50 > 10000 nM Bioactivity Info	TI LI LO TS
CP0448680 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-[(4-hydroxyphenyl)methyl]carbamoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C43H54N12O7	1
1	IC50 = 15700 nM Bioactivity Info	TI LI LO TS
CP0544543 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[[[2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-benzylcarbamoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C43H54N12O6	1
1	IC50 = 16100 nM Bioactivity Info	TI LI LO TS
CP0970125 Compound Info	2-((S)-2-amino-3-(1H-imidazol-5-yl)propanoyl)-1-benzyl-N-((S)-1-((S)-1-((R)-1-((S)-1,6-diamino-1-oxohexan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)hydrazinecarboxamide Show/Hide	C43H54N12O6	1
1	IC50 = 16100 nM Bioactivity Info	TI LI LO TS
CP0526048 Compound Info	(2S)-6-amino-2-[[(2R)-2-[[[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-phenylpropanoyl]amino]hexanamide Show/Hide	C40H56N12O6	1
1	IC50 = 19500 nM Bioactivity Info	TI LI LO TS
CP0463513 Compound Info	(2R)-2-[[(2S)-2-[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]carbamoylamino]-3-(1H-indol-3-yl)propanoyl]amino]-N-[(2S)-1-amino-1-oxopropan-2-yl]-3-phenylpropanamide Show/Hide	C41H46N12O6	1
1	IC50 = 45000 nM Bioactivity Info	TI LI LO TS
CP0453606 Compound Info	(2S)-2-[[[[(2R)-2-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-(2-methylpropyl)carbamoyl]amino]-3-(1H-indol-3-yl)propanamide Show/Hide	C33H40N10O4	1
1	IC50 = 85600 nM Bioactivity Info	TI LI LO TS
CP0435197 Compound Info	2-amino-N-[(1R)-1-[4-(2,4-dimethoxyphenyl)-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]acetamide Show/Hide	C30H32N6O3	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0505415 Compound Info	2-amino-N-[(1R)-1-[4-(4-ethylphenyl)-5-[2-(1H-indol-3-yl)ethyl]-4H-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]acetamide Show/Hide	C32H33N7O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0505417 Compound Info	2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-phenyl-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]ethyl]acetamide Show/Hide	C28H28N6O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0877434 Compound Info	(2S)-N-((R)-2-(1H-indol-3-yl)-1-(5-phenethyl-4-phenyl-4H-1,2,4-triazol-3-yl)ethyl)pyrrolidine-2-carboxamide Show/Hide	C31H34N6O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0902723 Compound Info	piperidine-4-carboxylic acid [(R)-1-[5-benzyl-4-(2-methyl-pyridin-1-yl)-4,5-dihydro-1H-[1,2,4]triazol-3-yl]-2-(1H-indol-3-yl)-ethyl]-amide Show/Hide	C32H35N7O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0906076 Compound Info	(S)-piperidine-3-carboxylic acid {(R)-2-(1H-indol-3-yl)-1-[4-(2-methyl-pyridin-1-yl)-5-phenethyl-4H-[1,2,4]triazol-3-yl]-ethyl}-amide Show/Hide	C32H35N7O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0421831 Compound Info	(R)-N-((4-(4-ethylbenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)(1H-indol-3-yl)methyl)isonicotinamide Show/Hide	C34H32N6O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0454009 Compound Info	(R)-(4-(2,4-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-N-benzyl(1H-indol-3-yl)methanamine Show/Hide	C35H35N5O2	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0455073 Compound Info	(S)-N-(1-(4-(2,4-dimethoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O3	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0464305 Compound Info	(S)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C31H34N6O2	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0486779 Compound Info	(S)-N-(1-(4-(4-methoxybenzyl)-5-(3-phenylpropyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H38N6O2	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0501238 Compound Info	(R)-N-(1-(4-(4-methoxybenzyl)-5-benzyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl)-2-amino-2-methylpropanamide Show/Hide	C29H33N5O2	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0522341 Compound Info	(S)-N-(1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C32H36N6O2	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0378564 Compound Info	(R)-2-amino-N-(1-(5-benzyl-4-(pyridin-2-ylmethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide Show/Hide	C29H31N7O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0378568 Compound Info	(R)-2-amino-N-(1-(5-benzyl-4-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide Show/Hide	C31H34N6O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0378581 Compound Info	(R)-2-amino-N-(1-(5-phenethyl-4-(pyridin-2-ylmethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide Show/Hide	C30H33N7O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0378586 Compound Info	(R)-N-(1-(4-(3,5-dimethoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-amino-2-methylpropanamide Show/Hide	C33H38N6O3	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0419728 Compound Info	2-amino-N-((R)-1-(5-benzyl-4-(2,2-diphenylethyl)-4H-1,2,4-triazol-3-yl)-2-(1H-indol-3-yl)ethyl)-2-methylpropanamide Show/Hide	C37H38N6O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0428144 Compound Info	2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-nitrophenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-2-methylpropanamide Show/Hide	C31H33N7O3	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0388313 Compound Info	(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethanamine;hydrochloride Show/Hide	C28H30ClN5O	1
1	IC50 > 1000 nM Bioactivity Info	TI LI LO TS
CP0229128 Compound Info	US8546435, 6 Show/Hide	C32H34N6O4	1
1	Ki = 0.8 nM Bioactivity Info	TI LI LO TS
CP0475496 Compound Info	US8546435, 7 Show/Hide	C35H39N7O4	1
1	Ki = 2 nM Bioactivity Info	TI LI LO TS
CP0475559 Compound Info	N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3-fluoropyridine-2-carboxamide Show/Hide	C36H34FN7O3	1
1	Ki = 4 nM Bioactivity Info	TI LI LO TS
CP0126988 Compound Info	US8546435, 5 Show/Hide	C35H33N7O3	1
1	Ki = 8 nM Bioactivity Info	TI LI LO TS
CP0419825 Compound Info	US8546435, 3 Show/Hide	C38H36N8O3	1
1	Ki = 9 nM Bioactivity Info	TI LI LO TS
CP0475492 Compound Info	N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide Show/Hide	C36H38N6O4	1
1	Ki = 9 nM Bioactivity Info	TI LI LO TS
CP0284845 Compound Info	US8546435, 4 Show/Hide	C36H35N7O3	1
1	Ki = 10 nM Bioactivity Info	TI LI LO TS
CP0475493 Compound Info	N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-4,6-difluoropyridine-2-carboxamide Show/Hide	C36H33F2N7O3	1
1	Ki = 11 nM Bioactivity Info	TI LI LO TS
CP0510760 Compound Info	US8546435, 8 Show/Hide	C36H40N8O3	1
1	Ki = 12 nM Bioactivity Info	TI LI LO TS
CP0475494 Compound Info	N-[(1R)-1-[5-[(1S)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide Show/Hide	C36H35N7O3	1
1	Ki = 17 nM Bioactivity Info	TI LI LO TS
CP0455241 Compound Info	N-[(1R)-1-[5-[(1R)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide Show/Hide	C34H33N7O2	1
1	Ki = 18 nM Bioactivity Info	TI LI LO TS
CP0327955 Compound Info	US8546435, 9 Show/Hide	C35H38N8O3	1
1	Ki = 46 nM Bioactivity Info	TI LI LO TS
CP0475560 Compound Info	N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide Show/Hide	C34H39N7O3	1
1	Ki = 46 nM Bioactivity Info	TI LI LO TS
CP0475747 Compound Info	2-amino-N-[(1R)-1-[5-[(1R)-1-formamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C33H37N7O3	1
1	Ki = 59 nM Bioactivity Info	TI LI LO TS
CP0414782 Compound Info	N-[(1R)-1-[5-[(1S)-1-acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide Show/Hide	C38H36N8O3	1
1	Ki = 62 nM Bioactivity Info	TI LI LO TS
CP0475749 Compound Info	N-[(1R)-1-[5-[(1S)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide Show/Hide	C34H33N7O2	1
1	Ki = 62 nM Bioactivity Info	TI LI LO TS
CP0475562 Compound Info	2-amino-N-[(1R)-1-[5-[(1R)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C34H38N8O2	1
1	Ki = 131 nM Bioactivity Info	TI LI LO TS
CP0447867 Compound Info	2-amino-N-[(1R)-1-[5-[(1R)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C32H37N7O2	1
1	Ki = 154 nM Bioactivity Info	TI LI LO TS
CP0475561 Compound Info	N-[(1R)-1-[5-[(1S)-1-formamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide Show/Hide	C37H34N8O3	1
1	Ki = 154 nM Bioactivity Info	TI LI LO TS
CP0379866 Compound Info	N-[(1R)-1-[5-[(1S)-1-acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide Show/Hide	C36H40N8O3	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0385352 Compound Info	N-[(1R)-1-[5-[(1S)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide Show/Hide	C34H39N7O3	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0419823 Compound Info	2-amino-N-[(1R)-1-[5-[(1S)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C32H37N7O2	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS
CP0561894 Compound Info	2-amino-N-[(1R)-1-[5-[(1S)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide Show/Hide	C34H38N8O2	1
1	Ki > 1000 nM Bioactivity Info	TI LI LO TS

Cite

About MolBiC

Correspondence

Prof. Feng ZHU

Prof. Leo, Lianyi Han