| Compound ID |
Compound Name |
Compound Formula |
|
CP0074934
|
6-[2-(4-fluoro-2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-8-methyl-4H-1,4-benzoxazin-3-one
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|
C20H15F4N3O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
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CP0428030
|
6-[1-(3,3-difluorobutyl)-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C22H20F3N3O2
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
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CP0418726
|
6-[5-(4-fluorophenyl)-3-methyl-1-(4,4,4-trifluorobutyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C22H19F4N3O2
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
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CP0418805
|
6-[5-(4-fluorophenyl)-3-methyl-1-(pyridin-3-ylmethyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C24H19FN4O2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0236141
|
6-[2-(4-fluoro-2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one
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|
C19H13F4N3O2
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
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CP0428029
|
6-[1-butyl-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C22H22FN3O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0379928
|
6-[5-(4-fluorophenyl)-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C22H22FN3O2
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0035175
|
2',15'-dimethyl-5,5'-dioxo-(9'R)-spiro[tetrahydrofuran-2,14'-tetracyclo[8.7.0.02,7.011,15]heptadec-6'-ene]-9-yl ethanethioate
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|
C24H32O4S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0428028
|
6-[1-benzyl-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C25H20FN3O2
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0093885
|
8-chloro-6-[2-(4-fluoro-2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one
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|
C19H12ClF4N3O2
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
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CP0418792
|
6-[1-(2,2-difluoro-3-hydroxypropyl)-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C21H18F3N3O3
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0397446
|
6-[4-(4-fluorophenyl)-2-methyl-5-oxo-1,2-dihydropyrrol-3-yl]-8-methyl-4H-1,4-benzoxazin-3-one
Show/Hide
|
C20H17FN2O3
|
1
|
| 1 |
IC50 = 83 nM
|
|
|
|
CP0268314
|
8-fluoro-6-[2-(4-fluoro-2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one
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|
C19H12F5N3O2
|
1
|
| 1 |
IC50 = 85 nM
|
|
|
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CP0418725
|
6-[5-(4-fluorophenyl)-1-(4-hydroxybutyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C22H22FN3O3
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0275206
|
6-[2-(2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C19H14F3N3O2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
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CP0379342
|
6-[5-(4-fluorophenyl)-1,3-dimethylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C19H16FN3O2
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0428026
|
6-[5-(4-fluorophenyl)-1-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C18H14FN3O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
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CP0418804
|
6-[5-(4-fluorophenyl)-3-methyl-1-propylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
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|
C21H20FN3O2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
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CP0428025
|
6-[1-(3,3-difluoro-4-hydroxybutyl)-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C22H20F3N3O3
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
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CP0379930
|
6-[5-(4-fluorophenyl)-1,3-dimethylpyrazol-4-yl]-8-methyl-4H-1,4-benzoxazin-3-one
Show/Hide
|
C20H18FN3O2
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
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CP0418723
|
6-[5-(4-fluorophenyl)-3-methyl-1-(pyridin-4-ylmethyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C24H19FN4O2
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0498692
|
3-[5-(4-fluorophenyl)-3-methyl-4-(3-oxo-4H-1,4-benzoxazin-6-yl)pyrazol-1-yl]propanenitrile
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|
C21H17FN4O2
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
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CP0379885
|
6-[1-(2,2-difluoro-4-hydroxybutyl)-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C22H20F3N3O3
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
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CP0428027
|
6-[5-(2,4-difluorophenyl)-1,3-dimethylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C19H15F2N3O2
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
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CP0418959
|
6-[5-(4-fluorophenyl)-1-(3-hydroxypropyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C21H20FN3O3
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
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CP0459594
|
6-[1-ethyl-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C20H18FN3O2
|
1
|
| 1 |
IC50 = 950 nM
|
|
|
|
CP0418955
|
6-[5-(4-fluorophenyl)-3-methyl-1-(pyridin-2-ylmethyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C24H19FN4O2
|
1
|
| 1 |
IC50 = 990 nM
|
|
|
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CP0100868
|
methyl (1R,2S,9R,10R,11S,14R,15S,17R)-2,15-dimethyl-5,5'-dioxospiro[18-oxapentacyclo[8.8.0.01,17.02,7.011,15]octadec-6-ene-14,2'-oxolane]-9-carboxylate
Show/Hide
|
C24H30O6
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
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CP0379889
|
6-[4-(4-fluorophenyl)-5-methyl-1,2-oxazol-3-yl]-4H-1,4-benzoxazin-3-one
Show/Hide
|
C18H13FN2O3
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
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CP0418729
|
N-[2-[5-(4-fluorophenyl)-3-methyl-4-(3-oxo-4H-1,4-benzoxazin-6-yl)pyrazol-1-yl]ethyl]methanesulfonamide
Show/Hide
|
C21H21FN4O4S
|
1
|
| 1 |
IC50 = 2000 nM
|
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|
