4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cycloheptyl-N-methylpiperidine-1-carboxamide

N-(2-adamantyl)-4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-methylpiperidine-1-carboxamide

(3beta,20beta)-20-carboxy-11-oxo-30-norolean-12-en-3-yl-2-O-beta-D-glucopyranuronosyl-alpha-D-glucopyranosiduronic acid

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cycloheptyl-N-cyclopropylpiperidine-1-carboxamide

N-(1-adamantyl)-4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]benzamide

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cycloheptylpiperidine-1-carboxamide

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cyclohexyl-N-cyclopropylpiperidine-1-carboxamide

N-(1-adamantyl)-4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-methylbenzamide

3-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cyclohexyl-N-cyclopropylbenzamide

N-(2-adamantyl)-3-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-methylbenzamide

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cycloheptyl-N-cyclopropylbenzamide

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cycloheptylbenzamide

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cyclooctylbenzamide

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cyclohexyl-N-cyclopropylbenzamide

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cycloheptyl-N-methylbenzamide

3-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cycloheptyl-N-cyclopropylbenzamide

3-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cycloheptyl-N-methylbenzamide

4-[(7-chloro-1,1,3-trioxo-4H-1lambda6,2,4-benzothiadiazin-2-yl)methyl]-N-cyclohexylbenzamide

4-[(3-Chlorophenylsulfonamido)methyl]-N-cycloheptyl-N-methylbenzamide

4-[(3-Chlorophenylsulfonamido)methyl]-N-cycloheptyl-N-propylbenzamide

N-butyl-4-[[(3-chlorophenyl)sulfonylamino]methyl]-N-cycloheptylbenzamide

18beta-glycyrrhetic acid

5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-1-(3-methylphenyl)-6,7-dihydropyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-1-(2-methylphenyl)-6,7-dihydropyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-1-phenyl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

4-[(3-Chlorophenylsulfonamido)methyl]-N-(1-adamantyl)benzamide

CHEMBL2338263

4-[(3-Chlorophenylsulfonamido)methyl]-N-cycloheptylbenzamide

1-(3-chlorophenyl)-5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-1-(2-methoxyphenyl)-8,8-dimethyl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

1-cyclohexyl-5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

1-cyclohexyl-5-(5-hydroxy-2-adamantyl)-7,8-dihydro-6H-pyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-1-[3-(trifluoromethyl)phenyl]-6,7-dihydropyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-1-phenyl-7,8-dihydro-6H-pyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-1-[4-(trifluoromethyl)phenyl]-6,7-dihydropyrazolo[4,3-c]azepin-4-one

1-(3-fluorophenyl)-5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-1-(4-methylphenyl)-6,7-dihydropyrazolo[4,3-c]azepin-4-one

1-(4-fluorophenyl)-5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

CHEMBL2338253

CHEMBL2338266

5-(5-hydroxy-2-adamantyl)-1-pyridin-2-yl-7,8-dihydro-6H-pyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-7-methyl-1-phenyl-7,8-dihydro-6H-pyrazolo[4,3-c]azepin-4-one

CHEMBL2338258

arylsulfonylpiperazine, 2

3-Chloro-N-[4-(piperidine-1-carbonyl)benzyl]benzenesulfonamide

4-[(3-Chlorophenylsulfonamido)methyl]-N-cyclohexylbenzamide

4-[(3-Chlorophenylsulfonamido)methyl]-N,N-diethylbenzamide

N-[(5-hydroxy-1,3,3-trimethylcyclohexyl)methyl]dibenzofuran-2-sulfonamide

3-Chloro-N-[4-(pyrrolidine-1-carbonyl)benzyl]benzenesulfonamide

3-{4-{2-Amino-6-[4-(4-propyl-benzoyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid

3-chloro-N-(4-((2R,6S)-2,6-dimethylmorpholine-4-carbonyl)benzyl)benzenesulfonamide

BMS-823778

(5R,9R,10R,13R,14R,17R)-17-[(2S,4R)-4-[(2S)-3,3-dimethyloxiran-2-yl]-4-hydroxybutan-2-yl]-4,4,10,13,14-pentamethyl-1,2,5,6,9,11,12,15,16,17-decahydrocyclopenta[a]phenanthren-3-one

3-{4-[2-Amino-6-(4-benzyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid

4-[(3-Chlorophenylsulfonamido)methyl]-N-cyclopentylbenzamide

3-{4-{2-Amino-6-[4-(4-tert-butyl-benzyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid

(5R,9R,10R,13S,14S,17S)-4,4,10,13,14-pentamethyl-17-[(1S,3R,4S)-3,4,5-trihydroxy-1,5-dimethyl-hexyl]-1,2,5,6,9,11,12,15,16,17-decahydrocyclopenta[a]phenanthren-3-one

3-Chloro-N-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]benzyl}-4-fluorobenzenesulfonamide

3-{4-{2-Amino-6-[4-(3-trifluoromethyl-benzyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid

3-[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]-3-methylbutan-1-ol

1-[(2R,3S)-3-[(1R)-1-[(3R,5R,9R,10R,13S,14S,17S)-3-hydroxy-4,4,10,13,14-pentamethyl-2,3,5,6,9,11,12,15,16,17-decahydro-1H-cyclopenta[a]phenanthren-17-yl]ethyl]oxiran-2-yl]-2-methylpropane-1,2-diol

3-Chloro-N-[4-(4-methylpiperazine-1-carbonyl)benzyl]benzenesulfonamide

3-{4-[2-Amino-6-(4-cyclohexylmethyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid

4-Chloro-N-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]benzyl}benzenesulfonmide

3-{4-{2-Amino-6-[4-(3-chloro-phenyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid

3-{4-[2-Amino-6-(4-phenyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid

3-{4-[2-Amino-6-(4-(naphthalen-1-ylmethyl)-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxypropionic acid

3-{4-{2-Amino-6-[4-(3-methyl-benzyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid

(3S,5R,8R,9R,10R,12R,13R,14R,17R)-3,12-dihydroxy-17-methoxy-4,4,8,10,14-pentamethyl-1,2,3,5,6,7,9,11,12,13,16,17-dodecahydrocyclopenta[a]phenanthren-15-one

(3S,5R,8R,9R,10R,12R,13R,14R)-3,12-dihydroxy-4,4,8,10,14-pentamethyl-1,2,3,5,6,7,9,11,12,13-decahydrocyclopenta[a]phenanthren-15-one

(E)-N'-(2,4-dihydroxy-6-methylbenzylidene)-2,3-dihydrobenzo[b][1,4]dioxine-2-carbohydrazide

3-{4-[2-Amino-6-(4-benzoyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid

[(3S,5R,8R,9R,10R,12R,13S,14R,17R)-3-hydroxy-17-methoxy-4,4,8,10,14-pentamethyl-15-oxo-1,2,3,5,6,7,9,11,12,13,16,17-dodecahydrocyclopenta[a]phenanthren-12-yl] acetate

3-Chloro-N-[4-(morpholine-4-carbonyl)benzyl]benzenesulfonamide

4-chloro-2-[(furan-2-ylmethyl)amino]-5-sulfamoylbenzoic acid

[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]methanol

(3S,5R,9R,10R,13R,14R,17R)-17-[(2S,4R)-4-[(2S)-3,3-dimethyloxiran-2-yl]-4-hydroxybutan-2-yl]-4,4,10,13,14-pentamethyl-2,3,5,6,9,11,12,15,16,17-decahydro-1H-cyclopenta[a]phenanthren-3-ol

[(3S,5R,8R,9R,10R,12R,13S,14R,17R)-3,17-dihydroxy-4,4,8,10,14-pentamethyl-15-oxo-1,2,3,5,6,7,9,11,12,13,16,17-dodecahydrocyclopenta[a]phenanthren-12-yl] acetate

N-[[4-[(2S,6R)-2,6-dimethylmorpholine-4-carbonyl]phenyl]methyl]-3-(trifluoromethyl)benzenesulfonamide

3-[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]propan-1-ol

2-Chloro-N-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]benzyl}benzenesulfonmide

ethyl 5-[(2,5-dimethylphenyl)sulfonylamino]-2-propyl-1-benzofuran-3-carboxylate

N-Adamantan-1-yl-3-{[2-(4-bromo-3-methyl-phenoxy)-acetyl]-hydrazono}-butyramide

[(3S,5R,8R,9R,10R,12R,13R,14R)-3-hydroxy-4,4,8,10,14-pentamethyl-15-oxo-1,2,3,5,6,7,9,11,12,13-decahydrocyclopenta[a]phenanthren-12-yl] acetate

[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]-cyclopropylmethanol

4-(4-butoxy-3-methylbenzoyl)-3-hydroxy-1-(pyridin-3-ylmethyl)-5-p-tolyl-1H-pyrrol-2(5H)-one

N-(3-chloro-4-hydroxynaphthalen-1-yl)-2,4-dimethylbenzenesulfonamide

2-(2,4-dibromophenoxy)-N-(3-(1-hydroxyethyl)phenyl)propanamide

4-(benzofuran-2-carbonyl)-5-(2-fluorophenyl)-3-hydroxy-1-(5-(4-methylbenzylthio)-1,3,4-thiadiazol-2-yl)-1H-pyrrol-2(5H)-one

N'-(2,4-dihydroxy-6-methylbenzylidene)-2-(m-tolyloxy)acetohydrazide

2-(4-allyl-5-((phenylamino)methyl)-4H-1,2,4-triazol-3-ylthio)-N'-(5-bromo-2-hydroxybenzylidene)propanehydrazide

3-{4-[2-Amino-6-(4-furan-2-ylmethyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid

3-{4-[2-Amino-6-(4-pyrimidin-2-yl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid

3-{4-{2-Amino-6-[4-(2-methoxy-benzoyl)-piperazin-1-yl]-pyrimidin-4-yloxy}-phenyl}-2-methyl-2-phenoxy-propionic acid

3-{4-[2-Amino-6-(4-pyridin-2-ylmethyl-piperazin-1-yl)-pyrimidin-4-yloxy]-phenyl}-2-methyl-2-phenoxy-propionic acid

3-(4-(2-Amino-6-(4-(furan-2-carbonyl)piperazin-1-yl)pyrimidin-4-yloxy)phenyl)-2-methyl-2-phenoxypropanoic acid

4-[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]-2-methylbutan-2-ol

1-[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]ethane-1,2-diol

2-[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]-2-methylpropanoic acid

5-(5-hydroxy-2-adamantyl)-8,8-dimethyl-1-pyridin-2-yl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-1-(4-methoxyphenyl)-8,8-dimethyl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

5-(5-hydroxy-2-adamantyl)-1,8,8-trimethyl-6,7-dihydropyrazolo[4,3-c]azepin-4-one

CHEMBL2338256

1-ethyl-5-(5-hydroxy-2-adamantyl)-7,8-dihydro-6H-pyrazolo[4,3-c]azepin-4-one