Brief Information of the Cell Line and Protein
Cell Line ID: CL000044 , CV-1
Synonyms
Cv-1
CV 1
CV-1.K
CV1
Category Finite cell line
Organism
Chlorocebus aethiops (Green monkey)
Cellosaurus ID
CVCL_0229
Protein ID: PT01018 , Thyroid hormone receptor beta
Gene Name THRB
Organism Homo sapiens, Human
Protein Classification Transcription factor
Uniprot ID P10828
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000044  Protein ID: PT01018
 
Compound ID Compound Name Compound Formula
CP0026502
(2R)-2-amino-3-[4-(4-hydroxy-3-iodophenoxy)-3,5-diiodophenyl]propanoic acid
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C15H12I3NO4
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0076899
3-[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-2-methylindol-3-yl]propanoic acid
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C22H25NO3
 1
1
EC50 = 37 nM
   TI
   LI
   LO
   TS
CP0262114
4-[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-2-methylindol-3-yl]butanoic acid
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C23H27NO3
 1
1
EC50 = 37 nM
   TI
   LI
   LO
   TS
CP0154335
5-[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-2-methylindol-3-yl]pentanoic acid
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C24H29NO3
 1
1
EC50 = 62 nM
   TI
   LI
   LO
   TS
CP0476565
2-[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-2-methylindol-3-yl]acetic acid
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C21H23NO3
 1
1
EC50 = 150 nM
   TI
   LI
   LO
   TS
CP0363634
2-[[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-7-methylindol-4-yl]amino]-2-oxoacetic acid
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C21H22N2O4
 1
1
EC50 = 500 nM
   TI
   LI
   LO
   TS
CP0154337
2-[[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-2-methylindol-4-yl]amino]-2-oxoacetic acid
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C21H22N2O4
 1
1
EC50 = 590 nM
   TI
   LI
   LO
   TS
CP0363635
3-[[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-2-methylindol-4-yl]amino]-3-oxopropanoic acid
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C22H24N2O4
 1
1
EC50 = 1700 nM
   TI
   LI
   LO
   TS
CP0076900
2-[[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]indol-4-yl]amino]-2-oxoacetic acid
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C20H20N2O4
 1
1
EC50 = 1900 nM
   TI
   LI
   LO
   TS
CP0476563
3-[[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-7-methylindol-4-yl]amino]-3-oxopropanoic acid
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C22H24N2O4
 1
1
EC50 = 3100 nM
   TI
   LI
   LO
   TS