| Compound ID |
Compound Name |
Compound Formula |
|
CP0032546
|
4-(9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-benzo[c]pyrimido[4,5-e]azepin-2-ylamino)-2-methoxybenzoic acid
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|
C27H20ClFN4O4
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0108599
|
4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid
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|
C26H18ClFN4O3
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0270630
|
4-[[6-chloro-2-(1,3-dimethylpyrazol-4-yl)-1H-imidazo[4,5-b]pyridin-7-yl]oxy]-N-phenylbenzamide
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|
C24H19ClN6O2
|
4
|
| 1 |
IC50 = 27 nM
|
|
|
| 2 |
IC50 = 29 nM
|
|
|
| 3 |
IC50 = 65 nM
|
|
|
| 4 |
IC50 = 960 nM
|
|
|
|
CP0017774
|
4-[[7-[2,6-bis(fluoranyl)phenyl]-9-chloranyl-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid
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|
C25H15ClF2N4O2
|
3
|
| 1 |
IC50 = 34 nM
|
|
|
| 2 |
IC50 = 160 nM
|
|
|
| 3 |
IC50 = 310 nM
|
|
|
|
CP0075920
|
4-[[6-chloro-2-(1,3-dimethylpyrazol-4-yl)-1H-imidazo[4,5-b]pyridin-7-yl]oxy]-N-cyclobutylbenzamide
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|
C22H21ClN6O2
|
4
|
| 1 |
IC50 = 36 nM
|
|
|
| 2 |
IC50 = 42 nM
|
|
|
| 3 |
IC50 = 43 nM
|
|
|
| 4 |
IC50 = 2290 nM
|
|
|
|
CP0482155
|
1-[4-[2-[(5-chloro-6-phenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl]phenyl]-3-[3-[(dimethylamino)methyl]phenyl]urea
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|
C30H29ClN6O2
|
1
|
| 1 |
IC50 = 59.9 nM
|
|
|
|
CP0481968
|
1-[4-[2-[(5-chloro-6-phenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl]phenyl]-3-[2-[(dimethylamino)methyl]phenyl]urea
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|
C30H29ClN6O2
|
1
|
| 1 |
IC50 = 73.4 nM
|
|
|
|
CP0296124
|
4-[[6-chloro-2-(1,3-dimethylpyrazol-4-yl)-1H-imidazo[4,5-b]pyridin-7-yl]oxy]-N-(3-methyl-1,2-oxazol-5-yl)benzamide
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|
C22H18ClN7O3
|
1
|
| 1 |
IC50 = 95 nM
|
|
|
|
CP0476941
|
1-[4-[2-[(5-chloro-6-phenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl]phenyl]-3-[3-[[ethyl(methyl)amino]methyl]phenyl]urea
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|
C31H31ClN6O2
|
1
|
| 1 |
IC50 = 132.2 nM
|
|
|
|
CP0385532
|
4-[[9-chloro-7-(2-fluorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid
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|
C25H16ClFN4O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0432163
|
1-[4-[2-[(5-chloro-6-phenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl]phenyl]-3-phenylurea
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|
C27H22ClN5O2
|
1
|
| 1 |
IC50 = 389.6 nM
|
|
|
|
CP0037005
|
2,4-Bisanilinopyrimidine, 10
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|
C31H31ClFN7O2
|
2
|
| 1 |
IC50 = 390 nM
|
|
|
| 2 |
IC50 = 2500 nM
|
|
|
|
CP0457859
|
1-[4-[2-[(5-chloro-6-phenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl]phenyl]-3-[2-[(4-hydroxypiperidin-1-yl)methyl]phenyl]urea
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|
C33H33ClN6O3
|
1
|
| 1 |
IC50 = 1513 nM
|
|
|
|
CP0020413
|
2,4-Bisanilinopyrimidine, 9
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|
C31H29ClFN7O3
|
2
|
| 1 |
IC50 = 1600 nM
|
|
|
| 2 |
IC50 = 2500 nM
|
|
|
|
CP0024021
|
2,4-Bisanilinopyrimidine, 13
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|
C23H17ClFN5O2
|
2
|
| 1 |
IC50 = 1600 nM
|
|
|
| 2 |
IC50 = 5000 nM
|
|
|
|
CP0298941
|
2,4-Bisanilinopyrimidine, 5
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|
C23H17ClFN5O2
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0395997
|
9-chloro-7-(2-fluorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-amine
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|
C18H12ClFN4
|
1
|
| 1 |
IC50 = 6000 nM
|
|
|
|
CP0253748
|
2,4-Bisanilinopyrimidine, 14
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|
C20H18FN5O2
|
1
|
| 1 |
IC50 = 6300 nM
|
|
|
