| Compound ID |
Compound Name |
Compound Formula |
|
CP0170580
|
5-(2,3-difluorophenyl)-N-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1H-indazole-3-carboxamide
Show/Hide
|
C23H26F2N4O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0103229
|
6-(4-hydroxy-4-phenylpiperidin-1-yl)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C21H22N4O2
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0170578
|
N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(6-methoxypyridin-3- yl)-1H-indazole-3-carboxamide
Show/Hide
|
C23H29N5O3
|
1
|
| 1 |
IC50 = 790 nM
|
|
|
|
CP0321228
|
6-(2-methoxyphenethylamino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C19H20N4O2
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0366365
|
N-{[1-(2-methoxyethyl)piperidin-4- yl]methyl}-5-(5-methoxypyridin-3- yl)-1H-indazole-3-carboxamide
Show/Hide
|
C23H29N5O3
|
1
|
| 1 |
IC50 = 800 nM
|
|
|
|
CP0076763
|
US9163013, 14
Show/Hide
|
C22H26N4O5
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0238538
|
(S)-6-(2-(2-methoxyphenyl)morpholino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C21H22N4O3
|
1
|
| 1 |
IC50 = 840 nM
|
|
|
|
CP0463173
|
US9163013, 3
Show/Hide
|
C22H24Cl2N4O2
|
1
|
| 1 |
IC50 = 1390 nM
|
|
|
|
CP0436285
|
(R)-6-(2-(2-methoxyphenyl)morpholino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C21H22N4O3
|
1
|
| 1 |
IC50 = 1530 nM
|
|
|
|
CP0405084
|
6-((2-methoxyphenethyl)(methyl)amino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C20H22N4O2
|
1
|
| 1 |
IC50 = 1690 nM
|
|
|
|
CP0550808
|
US9163013, 7
Show/Hide
|
C21H25N5O4S
|
1
|
| 1 |
IC50 = 2130 nM
|
|
|
|
CP0503473
|
6-(diethylamino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C14H18N4O
|
1
|
| 1 |
IC50 = 2210 nM
|
|
|
|
CP0405085
|
6-(3-(2-methoxyphenyl)piperidin-1-yl)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C22H24N4O2
|
1
|
| 1 |
IC50 = 2320 nM
|
|
|
|
CP0404987
|
6-(4-(2-methoxyphenyl)piperidin-1-yl)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C22H24N4O2
|
1
|
| 1 |
IC50 = 3210 nM
|
|
|
|
CP0528380
|
1-methyl-6-(3-phenylpiperidin-1-yl)-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C21H22N4O
|
1
|
| 1 |
IC50 = 4640 nM
|
|
|
|
CP0066138
|
US9163013, 9
Show/Hide
|
C21H25N5O5
|
1
|
| 1 |
IC50 = 5170 nM
|
|
|
|
CP0409853
|
6-(3-(2-methoxyphenyl)propylamino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C20H22N4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0437010
|
1-methyl-6-(phenethylamino)-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C18H18N4O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0437011
|
6-(4-methoxyphenethylamino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C19H20N4O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0471854
|
1-methyl-6-phenyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C16H13N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0273974
|
US9163013, 17
Show/Hide
|
C26H27N5O5
|
1
|
| 1 |
IC50 = 70800 nM
|
|
|
|
CP0066186
|
US9163013, 12
Show/Hide
|
C25H23F2N5O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0476593
|
1-methyl-6-(piperidin-1-yl)-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C15H18N4O
|
1
|
| 1 |
IC50 > 910 nM
|
|
|
|
CP0471856
|
1-methyl-6-morpholino-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C14H16N4O2
|
1
|
| 1 |
IC50 > 5040 nM
|
|
|
|
CP0028728
|
4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(1H)-one
Show/Hide
|
C17H14N2O2
|
1
|
| 1 |
IC50 > 5280 nM
|
|
|
|
CP0409852
|
6-(2-methoxybenzylamino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C18H18N4O2
|
1
|
| 1 |
IC50 > 9000 nM
|
|
|
|
CP0476594
|
6-(3-methoxyphenethylamino)-1-methyl-4-(pyrimidin-4-yl)pyridin-2(1H)-one
Show/Hide
|
C19H20N4O2
|
1
|
| 1 |
IC50 > 9000 nM
|
|
|
