General Information of the Compound
Compound ID
CP0916136
Compound Name
1-(4-(1-cyclobutylpiperidin-4-yloxy)phenyl)-4-(2,4-difluorobenzoyl)piperazin-2-one formic acid
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Structure
Formula
C27H31F2N3O5
Molecular Weight
515.557
Canonical SMILES
O=C(c1ccc(F)cc1F)N1CCN(c2ccc(OC3CCN(C4CCC4)CC3)cc2)C(=O)C1.O=CO
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InChI
InChI=1S/C26H29F2N3O3.CH2O2/c27-18-4-9-23(24(28)16-18)26(33)30-14-15-31(25(32)17-30)20-5-7-21(8-6-20)34-22-10-12-29(13-11-22)19-2-1-3-19;2-1-3/h4-9,16,19,22H,1-3,10-15,17H2;1H,(H,2,3)
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InChIKey
VDZPNNUVDOABNY-UHFFFAOYSA-N
Physicochemical Property
logP
3.5503
Rotatable Bonds
5
Heavy Atom Count
37
Polar Areas
90.39
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 24749291
SID: 49651411
ChEMBL ID
CHEMBL239321
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01206, Histamine H1 receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki < 2511.89 nM
   TI
   LI
   LO
   TS
Protein ID: PT01194, Histamine H3 receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1.585 nM
   TI
   LI
   LO
   TS
Protein ID: PT00897, Potassium voltage-gated channel subfamily H member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 < 63095.73 nM
   TI
   LI
   LO
   TS