General Information of the Compound
Compound ID
CP0451771
Compound Name
(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-N-[(4R)-1-methylsulfonyl-6-(quinolin-3-ylmethyl)-3,4-dihydro-2H-quinolin-4-yl]propanamide;2,2,2-trifluoroacetic acid
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Structure
Formula
C33H35F3N4O6S
Molecular Weight
672.726
Canonical SMILES
OC(=O)C(F)(F)F.Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N[C@@H]1CCN(c2ccc(Cc3cnc4ccccc4c3)cc12)S(C)(=O)=O
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InChI
InChI=1S/C31H34N4O4S.C2HF3O2/c1-19-12-24(36)13-20(2)25(19)17-27(32)31(37)34-29-10-11-35(40(3,38)39)30-9-8-21(16-26(29)30)14-22-15-23-6-4-5-7-28(23)33-18-22;3-2(4,5)1(6)7/h4-9,12-13,15-16,18,27,29,36H,10-11,14,17,32H2,1-3H3,(H,34,37);(H,6,7)/t27-,29+;/m0./s1
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InChIKey
VPNKUJITOSCPPY-RGJHRIFYSA-N
Physicochemical Property
logP
4.67834
Rotatable Bonds
7
Heavy Atom Count
47
Polar Areas
162.92
Hydrogen Bond Donor Count
4
Hydrogen Bond Acceptor Count
7
Complexity
47

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 155535193
ChEMBL ID
CHEMBL4471560
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01526, Delta-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000049 C6 Rattus norvegicus (Rat)  1
1
Ki = 0.64 nM
   TI
   LI
   LO
   TS
Protein ID: PT00983, Kappa-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 7 nM
   TI
   LI
   LO
   TS
Protein ID: PT01549, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000049 C6 Rattus norvegicus (Rat)  2
1
EC50 = 0.26 nM
   TI
   LI
   LO
   TS
2
Ki = 0.23 nM
   TI
   LI
   LO
   TS