General Information of the Compound
Compound ID
CP0036566
Compound Name
5-L-isoleucineangiotensin II
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Synonyms
1-8-Angiotensin I
4474-91-3
5-Isoleucine-angiotensin II
5-L-Isoleucineangiotensin II
ANGIOTENSIN II
Ang II
Angiotensin II (human)
Angiotensin II (mouse)
Angiotensin II human
Angiotensin II, ile(5)-
Angiotensin ii [INN:JAN]
Giapreza
Human angiotensin II
Ile(5)-angiotensin II
Isoleucine5-angiotensin II
isoleucine(5)-angiotensin II;Angiotensin II, human
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Structure
Formula
C50H71N13O12
Molecular Weight
1046.197
Canonical SMILES
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](N)CC(O)=O)C(C)C)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(O)=O
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InChI
InChI=1S/C50H71N13O12/c1-5-28(4)41(47(72)59-36(23-31-25-54-26-56-31)48(73)63-20-10-14-38(63)45(70)60-37(49(74)75)22-29-11-7-6-8-12-29)62-44(69)35(21-30-15-17-32(64)18-16-30)58-46(71)40(27(2)3)61-43(68)34(13-9-19-55-50(52)53)57-42(67)33(51)24-39(65)66/h6-8,11-12,15-18,25-28,33-38,40-41,64H,5,9-10,13-14,19-24,51H2,1-4H3,(H,54,56)(H,57,67)(H,58,71)(H,59,72)(H,60,70)(H,61,68)(H,62,69)(H,65,66)(H,74,75)(H4,52,53,55)/t28-,33-,34-,35-,36-,37-,38-,40-,41-/m0/s1
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InChIKey
CZGUSIXMZVURDU-JZXHSEFVSA-N
CAS
11128-99-7
1407-47-2
Physicochemical Property
logP
-1.3147
Rotatable Bonds
29
Heavy Atom Count
75
Polar Areas
408.84
Hydrogen Bond Donor Count
13
Hydrogen Bond Acceptor Count
13
Complexity
75

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 172198
SID: 14816795
ChEMBL ID
CHEMBL408403
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01197, Type-1 angiotensin II receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  3
1
EC50 = 2.6 nM
   TI
   LI
   LO
   TS
2
EC50 = 9.7 nM
   TI
   LI
   LO
   TS
3
IC50 = 10.2 nM
   TI
   LI
   LO
   TS
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
Ki = 0.5 nM
   TI
   LI
   LO
   TS
2
Ki = 0.9 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Kd = 2 nM
Protein ID: PT04214, Type-1 angiotensin II receptor A
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 1.3 nM
   TI
   LI
   LO
   TS
2
EC50 = 6.8 nM
   TI
   LI
   LO
   TS
Protein ID: PT01553, Type-2 angiotensin II receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 0.08 nM
   TI
   LI
   LO
   TS
2
IC50 = 0.617 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 2.5 nM
2 Ki = 0.2 nM
3 Ki = 0.23 nM
4 Ki = 1.2 nM
Clinical Information about the Compound
Drug 1 ( ANGIOTENSIN II )
Drug Name ANGIOTENSIN II
Company La Jolla Pharmaceutical Company
Indication
Increase blood pressure
Approved
Target(s)
Angiotensin II receptor type-1 (AGTR1)
Inhibitor
Angiotensin II receptor type-2 (AGTR2)
Inhibitor