General Information of the Cell Line
Cell Line ID
CL000826
Cell Line Name
C127
Synonyms
C-127
Category
Cancer cell line
Organism
Mus musculus (Mouse)
Tissue Information
Mammary gland
Disease
Malignant neoplasms of the mouse mammary gland (NCIt: C21678)
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT02042, ATP-binding cassette sub-family C member 7
Compound ID Compound Name Compound Formula
CP0441881
(S)-2-(3-Isopropoxy-4-methoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C32H38N2O4
 1
1
EC50 = 3.5 nM
   TI
   LI
   LO
   TS
CP0408605
(S)-2-(4-Isopropoxy-pyridine-2-carbonyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C30H35N3O3
 1
1
EC50 = 6 nM
   TI
   LI
   LO
   TS
CP0378111
(S)-2-(3-Isopropoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C31H36N2O3
 1
1
EC50 = 6.3 nM
   TI
   LI
   LO
   TS
CP0382250
(S)-2-(4-Cyclohexyloxy-pyridine-2-carbonyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C33H39N3O3
 1
1
EC50 = 9.4 nM
   TI
   LI
   LO
   TS
CP0495229
(S)-2-(3-Isobutoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C32H38N2O3
 1
1
EC50 = 10 nM
   TI
   LI
   LO
   TS
CP0486014
(S)-2-(2-Isopropoxy-pyridine-4-carbonyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C30H35N3O3
 1
1
EC50 = 11 nM
   TI
   LI
   LO
   TS
CP0408603
(S)-2-(4-Methoxy-3-phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C35H36N2O4
 1
1
EC50 = 12 nM
   TI
   LI
   LO
   TS
CP0495230
(S)-2-(3-Cyclopentyloxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C33H38N2O3
 1
1
EC50 = 15 nM
   TI
   LI
   LO
   TS
CP0451716
(S)-2-(5-Isopropoxy-pyridine-3-carbonyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C30H35N3O3
 1
1
EC50 = 16 nM
   TI
   LI
   LO
   TS
CP0378112
(S)-2-(3-Cyclohexyloxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C34H40N2O3
 1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
CP0408604
(S)-2-(4-Phenoxy-pyridine-2-carbonyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C33H33N3O3
 1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
CP0502580
(S)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C34H34N2O3
 1
1
EC50 = 23 nM
   TI
   LI
   LO
   TS
CP0494429
(S)-2-(3-Ethoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C30H34N2O3
 1
1
EC50 = 26 nM
   TI
   LI
   LO
   TS
CP0502587
(S)-2-(5-Cyclohexyloxy-pyridine-3-carbonyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C33H39N3O3
 1
1
EC50 = 35 nM
   TI
   LI
   LO
   TS
CP0486022
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid pyridin-3-ylamide
   Show/Hide
C28H23N3O3
 1
1
EC50 = 41 nM
   TI
   LI
   LO
   TS
CP0403131
(S)-2-(3-Chloro-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C28H29ClN2O2
 1
1
EC50 = 51 nM
   TI
   LI
   LO
   TS
CP0441832
(S)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (6-pentyl-pyridin-3-yl)-amide
   Show/Hide
C33H33N3O3
 1
1
EC50 = 53 nM
   TI
   LI
   LO
   TS
CP0540210
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C34H34N2O3
 1
1
EC50 = 61 nM
   TI
   LI
   LO
   TS
CP0508768
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid [4-(acetyl-butyl-amino)-phenyl]-amide
   Show/Hide
C35H35N3O4
 1
1
EC50 = 66 nM
   TI
   LI
   LO
   TS
CP0540211
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (6-chloro-pyridin-3-yl)-amide
   Show/Hide
C28H22ClN3O3
 1
1
EC50 = 66 nM
   TI
   LI
   LO
   TS
CP0508769
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid [4-(acetyl-pentyl-amino)-phenyl]-amide
   Show/Hide
C36H37N3O4
 1
1
EC50 = 71 nM
   TI
   LI
   LO
   TS
CP0378113
(S)-2-(4-Chloro-pyridine-2-carbonyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C27H28ClN3O2
 1
1
EC50 = 79 nM
   TI
   LI
   LO
   TS
CP0403132
(S)-2-(3,4-Dichloro-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C28H28Cl2N2O2
 1
1
EC50 = 82 nM
   TI
   LI
   LO
   TS
CP0514258
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-hexyl-phenyl)-amide
   Show/Hide
C35H36N2O3
 1
1
EC50 = 100 nM
   TI
   LI
   LO
   TS
CP0378105
(S)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C29H23ClN2O3
 1
1
EC50 = 119 nM
   TI
   LI
   LO
   TS
CP0378107
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-butoxy-phenyl)-amide
   Show/Hide
C33H32N2O4
 1
1
EC50 = 145 nM
   TI
   LI
   LO
   TS
CP0508767
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid [4-(4-methyl-pentyl)-phenyl]-amide
   Show/Hide
C35H36N2O3
 1
1
EC50 = 160 nM
   TI
   LI
   LO
   TS
CP0378109
(R)-2-[3-(4-Methoxy-phenoxy)-benzoyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C30H25ClN2O4
 1
1
EC50 = 167 nM
   TI
   LI
   LO
   TS
CP0382246
(S)-2-(3-Methoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-pentyl-phenyl)-amide
   Show/Hide
C29H32N2O3
 1
1
EC50 = 176 nM
   TI
   LI
   LO
   TS
CP0498234
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-fluoro-phenyl)-amide
   Show/Hide
C29H23FN2O3
 1
1
EC50 = 202 nM
   TI
   LI
   LO
   TS
CP0508766
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-butyl-phenyl)-amide
   Show/Hide
C33H32N2O3
 1
1
EC50 = 202 nM
   TI
   LI
   LO
   TS
CP0408779
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-heptyl-phenyl)-amide
   Show/Hide
C36H38N2O3
 1
1
EC50 = 230 nM
   TI
   LI
   LO
   TS
CP0394808
(R)-2-[3-(Pyridin-2-yloxy)-benzoyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C28H22ClN3O3
 1
1
EC50 = 268 nM
   TI
   LI
   LO
   TS
CP0445612
(R)-2-[3-(4-Trifluoromethyl-phenoxy)-benzoyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C30H22ClF3N2O3
 1
1
EC50 = 282 nM
   TI
   LI
   LO
   TS
CP0449076
(R)-2-(3-Benzyl-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C30H25ClN2O2
 1
1
EC50 = 291 nM
   TI
   LI
   LO
   TS
CP0378106
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-bromo-phenyl)-amide
   Show/Hide
C29H23BrN2O3
 1
1
EC50 = 292 nM
   TI
   LI
   LO
   TS
CP0408778
2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C29H23ClN2O3
 1
1
EC50 = 294 nM
   TI
   LI
   LO
   TS
CP0502579
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-iodo-phenyl)-amide
   Show/Hide
C29H23IN2O3
 1
1
EC50 = 314 nM
   TI
   LI
   LO
   TS
CP0441874
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C29H23ClN2O3
 1
1
EC50 = 336 nM
   TI
   LI
   LO
   TS
CP0378108
(R)-2-(2-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C29H23ClN2O3
 1
1
EC50 = 338 nM
   TI
   LI
   LO
   TS
CP0449077
(R)-2-(3-Phenylsulfanyl-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C29H23ClN2O2S
 1
1
EC50 = 394 nM
   TI
   LI
   LO
   TS
CP0499882
(R)-2-(3-Phenoxy-benzoyl)-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-ethoxy-phenyl)-amide
   Show/Hide
C31H28N2O4
 1
1
EC50 = 420 nM
   TI
   LI
   LO
   TS
CP0495228
(R)-2-[3-(4-Fluoro-phenoxy)-benzoyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (4-chloro-phenyl)-amide
   Show/Hide
C29H22ClFN2O3
 1
1
EC50 = 590 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Mammary gland)
Cell Line Name Organism Disease
4T1 Mus musculus (Mouse) Malignant neoplasms of the mouse mammary gland
SC-3 Mus musculus (Mouse) Malignant neoplasms of the mouse mammary gland
EMT6 Mus musculus (Mouse) Malignant neoplasms of the mouse mammary gland
SC-115 Mus musculus (Mouse) Malignant neoplasms of the mouse mammary gland
NMU Rattus norvegicus (Rat) Adenocarcinoma of the rat mammary gland
HC11 Mus musculus (Mouse) -