| Compound ID |
Compound Name |
Compound Formula |
|
CP0421187
|
3-[(1E)-1-[3-fluoro-8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C29H25FN4O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0468897
|
3-[(1E)-1-[8-[[7-chloro-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C28H22ClFN4O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0421190
|
3-[(1E)-1-[8-[(7-chloro-2-cyclopropylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C29H22ClFN4O3
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0391625
|
3-[(1E)-1-[8-[(2-cyclopropyl-7-fluoroimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C29H22F2N4O3
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0421189
|
3-[(1E)-1-[8-[(6-chloro-2-cyclopropylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C29H22ClFN4O3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0472427
|
3-[(1E)-1-[8-[(8-chloro-2-cyclopropylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C29H22ClFN4O3
|
1
|
| 1 |
EC50 = 2.5 nM
|
|
|
|
CP0391624
|
3-[(1E)-1-[8-[(2-cyclopropylthieno[3,4-d]imidazol-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C27H21FN4O3S
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0416268
|
3-[(1E)-1-[8-[(4-methyl-2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C30H28N4O3
|
1
|
| 1 |
EC50 = 3.3 nM
|
|
|
|
CP0457474
|
3-[(1E)-1-[4-fluoro-8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C29H25FN4O3
|
1
|
| 1 |
EC50 = 3.8 nM
|
|
|
|
CP0391626
|
3-[(1E)-1-[8-[[8-chloro-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C28H22ClFN4O4
|
1
|
| 1 |
EC50 = 4.5 nM
|
|
|
|
CP0468896
|
3-[(1E)-1-[8-[(2-cyclopropylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C29H23FN4O3
|
1
|
| 1 |
EC50 = 5.3 nM
|
|
|
|
CP0421186
|
3-[(1E)-1-[2-fluoro-8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C29H25FN4O3
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0411178
|
3-[(1E)-1-[8-[(4-cyclopropyl-10-oxa-3,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-5-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C31H25FN4O4
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0457475
|
3-[(1E)-1-[8-[(4-chloro-2-cyclopropylimidazo[4,5-c]pyridin-1-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C28H21ClFN5O3
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0421188
|
3-[(1E)-1-[8-[(7-chloro-2-cyclopropylimidazo[4,5-b]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
Show/Hide
|
C28H21ClFN5O3
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0158747
|
2,4-dichloro-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide
Show/Hide
|
C21H12Cl4N2O3S
|
1
|
| 1 |
EC50 > 500 nM
|
|
|
|
CP0416271
|
ATx08-001
Show/Hide
|
C21H23Cl2N3O3S
|
1
|
| 1 |
EC50 > 500 nM
|
|
|
|
CP0876439
|
ARHALOFENATE
Show/Hide
|
C19H17ClF3NO4
|
1
|
| 1 |
EC50 > 500 nM
|
|
|
