| Compound ID |
Compound Name |
Compound Formula |
|
CP0037621
|
(oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyrrolidin-2-one
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|
C12H18N2O
|
1
|
| 1 |
EC50 = 270 nM
|
|
|
|
CP0848677
|
SID50106828
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|
C11H19IN2O
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0845687
|
5-(3-Methyl-[1,2,4]oxadiazol-5-yl)-1,4,5,6-tetrahydro-pyrimidine TFA
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|
C9H11F3N4O3
|
4
|
| 1 |
EC50 = 5400 nM
|
|
|
| 2 |
Ki = 2.31 nM
|
|
|
| 3 |
Ki = 2.5 nM
|
|
|
| 4 |
Ki = 21.1 nM
|
|
|
|
CP0371787
|
5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine; oxalic acid
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|
C14H23N3OS
|
1
|
| 1 |
EC50 = 5700 nM
|
|
|
|
CP0089021
|
(+)-pilocarpine
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|
C11H16N2O2
|
1
|
| 1 |
EC50 = 6900 nM
|
|
|
|
CP0374204
|
1-Methyl-5-(3-methyl-[1,2,4]oxadiazol-5-yl)-1,2,3,6-tetrahydro-pyridine
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|
C9H13N3O
|
3
|
| 1 |
EC50 = 12000 nM
|
|
|
| 2 |
Ki = 0.589 nM
|
|
|
| 3 |
Ki = 1.05 nM
|
|
|
|
CP0847680
|
5-(3-Ethyl-[1,2,4]oxadiazol-5-yl)-1,4,5,6-tetrahydro-pyrimidine TFA
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|
C10H13F3N4O3
|
1
|
| 1 |
EC50 = 12000 nM
|
|
|
|
CP0847223
|
5-(3-Methylsulfanylmethyl-[1,2,4]oxadiazol-5-yl)-1,4,5,6-tetrahydro-pyrimidine TFA
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|
C10H13F3N4O3S
|
1
|
| 1 |
EC50 = 14000 nM
|
|
|
|
CP0018455
|
1-methyl-3,6-dihydro-2H-pyridine-5-carboxylic acid methyl ester;hydrobromide
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|
C8H13NO2
|
3
|
| 1 |
EC50 = 27000 nM
|
|
|
| 2 |
Ki = 3.33 nM
|
|
|
| 3 |
Ki = 5.45 nM
|
|
|
|
CP0875146
|
1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid prop-2-ynyl ester hydrochloride
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|
C8H11ClN2O2
|
3
|
| 1 |
EC50 = 33000 nM
|
|
|
| 2 |
Ki = 2.88 nM
|
|
|
| 3 |
Ki = 41.7 nM
|
|
|
|
CP0635477
|
(2-Carbamoyloxy-ethyl)-trimethyl-ammonium chloride
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|
C6H15ClN2O2
|
4
|
| 1 |
EC50 = 40000 nM
|
|
|
| 2 |
Ki = 19.9 nM
|
|
|
| 3 |
Ki = 37.1 nM
|
|
|
| 4 |
Ki = 739 nM
|
|
|
|
CP0879042
|
6-Amino-2,3,4,5-tetrahydro-pyridine-3-carboxylic acid methyl ester hydrochloride
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|
C7H13ClN2O2
|
1
|
| 1 |
EC50 = 41000 nM
|
|
|
|
CP0859779
|
1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid ethyl ester hydrochloride
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|
C7H13ClN2O2
|
1
|
| 1 |
EC50 = 44000 nM
|
|
|
|
CP0861321
|
1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid but-2-ynyl ester hydrochloride
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|
C9H13ClN2O2
|
3
|
| 1 |
EC50 = 50000 nM
|
|
|
| 2 |
Ki = 9.01 nM
|
|
|
| 3 |
Ki = 14 nM
|
|
|
|
CP0888198
|
1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid (E)-3-methyl-pent-2-en-4-ynyl ester hydrochloride
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|
C11H15ClN2O2
|
1
|
| 1 |
EC50 = 80000 nM
|
|
|
|
CP0863249
|
1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid but-3-ynyl ester hydrochloride
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|
C9H13ClN2O2
|
2
|
| 1 |
Ki = 15.5 nM
|
|
|
| 2 |
Ki = 30.9 nM
|
|
|
|
CP0882900
|
5-(3-Pent-1-ynyl-[1,2,4]oxadiazol-5-yl)-1,4,5,6-tetrahydro-pyrimidine TFA
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|
C13H15F3N4O3
|
2
|
| 1 |
Ki = 17.4 nM
|
|
|
| 2 |
Ki = 138 nM
|
|
|
|
CP0856374
|
1,4,5,6-Tetrahydro-pyrimidine-5-carboxylic acid methyl ester hydrochloride
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|
C6H11ClN2O2
|
3
|
| 1 |
Ki = 23.6 nM
|
|
|
| 2 |
Ki = 26.8 nM
|
|
|
| 3 |
Ki = 359 nM
|
|
|
