Compound ID |
Compound Name |
Compound Formula |
CP0477949
|
US9315518, 34-3
Show/Hide
|
C17H23F2N3O3S
|
1
|
1 |
EC50 = 14.38 nM
|
|
|
CP0561520
|
US9315518, 8-38
Show/Hide
|
C23H27N5O3
|
1
|
1 |
EC50 = 17.91 nM
|
|
|
CP0560900
|
US9315518, 2-34
Show/Hide
|
C23H27N5O3
|
1
|
1 |
EC50 = 22.79 nM
|
|
|
CP0545810
|
US9315518, 2-8
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|
C22H26N6O2S
|
1
|
1 |
EC50 = 28.14 nM
|
|
|
CP0560901
|
US9315518, 6-4
Show/Hide
|
C22H21F2N5O3
|
1
|
1 |
EC50 = 28.96 nM
|
|
|
CP0560903
|
US9315518, 18-200
Show/Hide
|
C23H32N6O2S
|
1
|
1 |
EC50 = 43.24 nM
|
|
|
CP0575884
|
US9315518, 24-7
Show/Hide
|
C21H26F2N4O4S
|
1
|
1 |
EC50 = 48.5 nM
|
|
|
CP0556492
|
US9315518, 2-22
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|
C23H29N7O2
|
1
|
1 |
EC50 = 56.06 nM
|
|
|
CP0518496
|
US9315518, 2-16
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|
C23H30N4O2
|
1
|
1 |
EC50 = 64.1 nM
|
|
|
CP0478027
|
US9315518, 2-9
Show/Hide
|
C25H29N5O2
|
1
|
1 |
EC50 = 100.1 nM
|
|
|
CP0560904
|
US9315518, 19-62
Show/Hide
|
C27H38N4O3S
|
1
|
1 |
EC50 = 116.3 nM
|
|
|
CP0545811
|
US9315518, 14-6
Show/Hide
|
C22H21F2N5O3
|
1
|
1 |
EC50 = 123.3 nM
|
|
|
CP0563408
|
US9315518, 8-14
Show/Hide
|
C24H32N4O3
|
1
|
1 |
EC50 = 134.2 nM
|
|
|
CP0477948
|
US9315518, 24-20
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|
C18H17F2N5O4S
|
1
|
1 |
EC50 = 177.4 nM
|
|
|
CP0536942
|
US9315518, 8-9
Show/Hide
|
C21H28N4O3
|
1
|
1 |
EC50 = 269.9 nM
|
|
|
CP0560876
|
US9315518, 17-20
Show/Hide
|
C23H32N4O3
|
1
|
1 |
EC50 = 332.7 nM
|
|
|
CP0536943
|
US9315518, 25-5
Show/Hide
|
C15H20F2N4O2S
|
1
|
1 |
EC50 = 359.2 nM
|
|
|
CP0560902
|
US9315518, 11-5
Show/Hide
|
C23H29N5O3
|
1
|
1 |
EC50 = 390.7 nM
|
|
|
CP0565717
|
US9315518, 8-6
Show/Hide
|
C29H41N5O5
|
1
|
1 |
EC50 = 512.7 nM
|
|
|
CP0478028
|
US9315518, 17-15
Show/Hide
|
C23H29N5O3
|
1
|
1 |
EC50 = 594.1 nM
|
|
|
CP0413561
|
US9315518, 19-4
Show/Hide
|
C21H30N6O3S
|
1
|
1 |
EC50 = 951.1 nM
|
|
|
CP0565728
|
US9315518, 18-42
Show/Hide
|
C28H35F3N4O3
|
1
|
1 |
EC50 = 985.5 nM
|
|
|
CP0519501
|
US9315518, 38-5
Show/Hide
|
C21H30N6O2
|
1
|
1 |
EC50 = 1178 nM
|
|
|
CP0561588
|
US9315518, 18-10
Show/Hide
|
C25H37N7O2
|
1
|
1 |
EC50 = 2189 nM
|
|
|
CP0544342
|
US9278960, 8-50
Show/Hide
|
C24H21FN4O2
|
1
|
1 |
IC50 = 4 nM
|
|
|
CP0530613
|
US9278960, 8-51
Show/Hide
|
C24H20F2N4O2
|
1
|
1 |
IC50 = 5 nM
|
|
|
CP0550635
|
US9278960, 2-29
Show/Hide
|
C22H19N3O3
|
1
|
1 |
IC50 = 5 nM
|
|
|
CP0238235
|
US9278960, 8-29
Show/Hide
|
C24H21FN4O2
|
1
|
1 |
IC50 = 6 nM
|
|
|
CP0478034
|
US9278960, 8-33
Show/Hide
|
C24H18FN5O2
|
1
|
1 |
IC50 = 6 nM
|
|
|
CP0567635
|
US9278960, 6-21
Show/Hide
|
C21H16F3N5O
|
1
|
1 |
IC50 = 6 nM
|
|
|
CP0414567
|
US9278960, 8-15
Show/Hide
|
C22H17FN4O
|
1
|
1 |
IC50 = 7 nM
|
|
|
CP0414571
|
US9278960, 8-32
Show/Hide
|
C24H19N5O2
|
1
|
1 |
IC50 = 7 nM
|
|
|
CP0537472
|
US9278960, 6-25
Show/Hide
|
C21H15ClF3N5O
|
1
|
1 |
IC50 = 7 nM
|
|
|
CP0545115
|
US9278960, 2-27
Show/Hide
|
C22H23N3O3
|
1
|
1 |
IC50 = 7 nM
|
|
|
CP0574036
|
US9278960, 8-35
Show/Hide
|
C23H21N5O2
|
1
|
1 |
IC50 = 7 nM
|
|
|
CP0379773
|
US9278960, 7-29
Show/Hide
|
C25H21F5N4O3
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0413602
|
US9278960, 8-34
Show/Hide
|
C25H21N5O2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0414449
|
US9278960, 2-39
Show/Hide
|
C22H18FN3O4
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0537019
|
US9278960, 6-7
Show/Hide
|
C23H18FN3O2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0567632
|
US9278960, 4-135
Show/Hide
|
C22H24F3N5O2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0570551
|
US9278960, 4-91
Show/Hide
|
C21H22F3N5O2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0576899
|
US9278960, 4-90
Show/Hide
|
C21H22F3N5O2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0576900
|
US9278960, 4-96
Show/Hide
|
C22H24F3N5O2
|
1
|
1 |
IC50 = 8 nM
|
|
|
CP0068843
|
US9278960, 2-7
Show/Hide
|
C21H16FN3O3
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0480096
|
US9278960, 4-86
Show/Hide
|
C20H19F4N5O2
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0516444
|
US9278960, 8-30
Show/Hide
|
C24H22N4O2
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0555385
|
US9278960, 8-31
Show/Hide
|
C24H21FN4O2
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0556048
|
US9278960, 4-51
Show/Hide
|
C20H19F3N4O2S
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0414566
|
US9278960, 8-1
Show/Hide
|
C23H17ClFN3O2
|
1
|
1 |
IC50 = 10 nM
|
|
|
CP0535539
|
US9278960, 3-51
Show/Hide
|
C25H23F3N4O3
|
1
|
1 |
IC50 = 10 nM
|
|
|
CP0544339
|
US9278960, 7-28
Show/Hide
|
C25H21F5N4O3
|
1
|
1 |
IC50 = 10 nM
|
|
|
CP0560719
|
US9278960, 7-23
Show/Hide
|
C22H16F2N4O2
|
1
|
1 |
IC50 = 10 nM
|
|
|
CP0567637
|
US9278960, 8-16
Show/Hide
|
C23H18FN3O
|
1
|
1 |
IC50 = 10 nM
|
|
|
CP0477812
|
US9278960, 4-84
Show/Hide
|
C20H18F5N5O2
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0480097
|
US9278960, 4-95
Show/Hide
|
C22H24F3N5O2
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0515283
|
US9278960, 8-54
Show/Hide
|
C24H20F2N4O2
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0554181
|
US9278960, 4-9
Show/Hide
|
C21H22F3N5O2
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0477810
|
US9278960, 2-24
Show/Hide
|
C21H15ClFN3O3
|
1
|
1 |
IC50 = 12 nM
|
|
|
CP0511951
|
US9278960, 4-54
Show/Hide
|
C20H20F3N5O2
|
1
|
1 |
IC50 = 12 nM
|
|
|
CP0544365
|
US9278960, 6-26
Show/Hide
|
C24H20F3N5O
|
1
|
1 |
IC50 = 12 nM
|
|
|
CP0419162
|
US9278960, 4-118
Show/Hide
|
C21H20F5N5O2
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0419593
|
US9278960, 4-126
Show/Hide
|
C21H21F3N4O2S
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0480093
|
US9278960, 4-16
Show/Hide
|
C22H25N5OS
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0529275
|
US9278960, 7-13
Show/Hide
|
C22H16F2N2O4
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0539876
|
US9278960, 6-6
Show/Hide
|
C23H15FN4O
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0550651
|
US9278960, 7-36
Show/Hide
|
C21H21F4N5O
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0555384
|
US9278960, 8-7
Show/Hide
|
C25H19FN4O2
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0515281
|
US9278960, 7-35
Show/Hide
|
C22H20FN5O2
|
1
|
1 |
IC50 = 14 nM
|
|
|
CP0567723
|
US9278960, 7-20-A
Show/Hide
|
C21H20F4N4O3
|
1
|
1 |
IC50 = 14 nM
|
|
|
CP0578555
|
US9278960, 4-116
Show/Hide
|
C21H20F4N4O2S
|
1
|
1 |
IC50 = 14 nM
|
|
|
CP0477942
|
US9278960, 4-80
Show/Hide
|
C20H19F4N5O2
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0535537
|
US9278960, 3-44
Show/Hide
|
C24H20F4N4O2
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0550648
|
US9278960, 6-20
Show/Hide
|
C21H16N6O
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0550649
|
US9278960, 7-26
Show/Hide
|
C23H17F2N3O2
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0567636
|
US9278960, 8-2
Show/Hide
|
C23H17ClFN3O2
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0570549
|
US9278960, 4-77
Show/Hide
|
C21H22F3N5O2
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0574084
|
US9278960, 4-85
Show/Hide
|
C20H19F4N5O2
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0479671
|
US9278960, 4-66
Show/Hide
|
C21H22F3N5O2
|
1
|
1 |
IC50 = 16 nM
|
|
|
CP0544360
|
US9278960, 3-49
Show/Hide
|
C25H22F4N4O3
|
1
|
1 |
IC50 = 16 nM
|
|
|
CP0576395
|
US9278960, 2-25
Show/Hide
|
C21H21N3O3
|
1
|
1 |
IC50 = 16 nM
|
|
|
CP0379831
|
US9278960, 7-24
Show/Hide
|
C24H19F5N4O2
|
1
|
1 |
IC50 = 17 nM
|
|
|
CP0516400
|
US9278960, 4-65
Show/Hide
|
C21H22F3N5O2
|
1
|
1 |
IC50 = 17 nM
|
|
|
CP0560709
|
US9278960, 2-28
Show/Hide
|
C22H25N3O3
|
1
|
1 |
IC50 = 17 nM
|
|
|
CP0574085
|
US9278960, 4-92
Show/Hide
|
C21H22F3N5O2
|
1
|
1 |
IC50 = 17 nM
|
|
|
CP0550646
|
US9278960, 6-14
Show/Hide
|
C23H18FN3O2
|
1
|
1 |
IC50 = 18 nM
|
|
|
CP0576903
|
US9278960, 4-119
Show/Hide
|
C20H20F3N5OS
|
1
|
1 |
IC50 = 18 nM
|
|
|
CP0322665
|
US9278960, 3-45
Show/Hide
|
C24H20F4N4O2
|
1
|
1 |
IC50 = 19 nM
|
|
|
CP0478032
|
US9278960, 7-25
Show/Hide
|
C24H18F2N4O
|
1
|
1 |
IC50 = 20 nM
|
|
|
CP0134841
|
US9278960, 3-16
Show/Hide
|
C22H18F4N6O2
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0414552
|
US9278960, 2-10
Show/Hide
|
C24H22FN3O3
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0419155
|
US9278960, 2-3
Show/Hide
|
C21H17FN4O3
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0516382
|
US9278960, 7-30
Show/Hide
|
C21H18FN5O2
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0518185
|
US9278960, 7-20-B
Show/Hide
|
C21H20F4N4O3
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0544367
|
US9278960, 7-21
Show/Hide
|
C21H15F2N3O3
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0545122
|
US9278960, 3-20
Show/Hide
|
C23H19ClF3N5O2
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0556056
|
US9278960, 6-2
Show/Hide
|
C22H20N6O
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0576893
|
US9278960, 3-6
Show/Hide
|
C22H18F4N6O2
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0413601
|
US9278960, 8-19
Show/Hide
|
C24H22N4O2
|
1
|
1 |
IC50 = 22 nM
|
|
|
CP0367697
|
US9278960, 2-21
Show/Hide
|
C22H18FN3O3
|
1
|
1 |
IC50 = 23 nM
|
|
|
CP0419156
|
US9278960, 3-27
Show/Hide
|
C22H17FN4O3
|
1
|
1 |
IC50 = 23 nM
|
|
|
CP0535535
|
US9278960, 3-32
Show/Hide
|
C20H14ClFN4O
|
1
|
1 |
IC50 = 23 nM
|
|
|
CP0512333
|
US9278960, 4-100
Show/Hide
|
C23H29N5O2
|
1
|
1 |
IC50 = 24 nM
|
|
|
CP0556042
|
US9278960, 3-38
Show/Hide
|
C26H18F4N4O
|
1
|
1 |
IC50 = 24 nM
|
|
|
CP0570548
|
US9278960, 4-46
Show/Hide
|
C22H19F4N3O2
|
1
|
1 |
IC50 = 24 nM
|
|
|
CP0577279
|
US9278960, 3-7
Show/Hide
|
C22H18F4N6O2
|
1
|
1 |
IC50 = 24 nM
|
|
|
CP0414452
|
US9278960, 3-26
Show/Hide
|
C22H17FN4O3
|
1
|
1 |
IC50 = 25 nM
|
|
|
CP0419158
|
US9278960, 4-71
Show/Hide
|
C21H22F3N5O
|
1
|
1 |
IC50 = 25 nM
|
|
|
CP0556034
|
US9278960, 2-11
Show/Hide
|
C22H18FN3O4
|
1
|
1 |
IC50 = 25 nM
|
|
|
CP0567719
|
US9278960, 4-53
Show/Hide
|
C20H20F3N5O2
|
1
|
1 |
IC50 = 25 nM
|
|
|
CP0567722
|
US9278960, 6-24
Show/Hide
|
C22H21N5O
|
1
|
1 |
IC50 = 25 nM
|
|
|
CP0535536
|
US9278960, 3-35
Show/Hide
|
C24H17FN4O4S
|
1
|
1 |
IC50 = 27 nM
|
|
|
CP0556037
|
US9278960, 2-20
Show/Hide
|
C23H20FN3O3
|
1
|
1 |
IC50 = 27 nM
|
|
|
CP0556058
|
US9278960, 8-52
Show/Hide
|
C25H24N4O2
|
1
|
1 |
IC50 = 27 nM
|
|
|
CP0576396
|
US9278960, 2-38
Show/Hide
|
C22H19N3O4
|
1
|
1 |
IC50 = 27 nM
|
|
|
CP0414460
|
US9278960, 6-23
Show/Hide
|
C21H16F3N5O
|
1
|
1 |
IC50 = 28 nM
|
|
|
CP0518186
|
US9278960, 7-31
Show/Hide
|
C21H15F4N5O
|
1
|
1 |
IC50 = 28 nM
|
|
|
CP0578091
|
US9278960, 2-18
Show/Hide
|
C25H22FN3O3
|
1
|
1 |
IC50 = 28 nM
|
|
|
CP0567623
|
US9278960, 2-26
Show/Hide
|
C21H23N3O3
|
1
|
1 |
IC50 = 29 nM
|
|
|
CP0414565
|
US9278960, 7-37
Show/Hide
|
C23H20FN5O
|
1
|
1 |
IC50 = 30 nM
|
|
|
CP0477811
|
US9278960, 4-73
Show/Hide
|
C20H21F2N5O
|
1
|
1 |
IC50 = 30 nM
|
|
|
CP0556036
|
US9278960, 2-14
Show/Hide
|
C24H22FN3O3
|
1
|
1 |
IC50 = 30 nM
|
|
|
CP0545116
|
US9278960, 3-24
Show/Hide
|
C22H17FN4O3
|
1
|
1 |
IC50 = 31 nM
|
|
|
CP0545117
|
US9278960, 3-30
Show/Hide
|
C23H21FN4O
|
1
|
1 |
IC50 = 31 nM
|
|
|
CP0567624
|
US9278960, 3-11
Show/Hide
|
C24H19FN4O2
|
1
|
1 |
IC50 = 31 nM
|
|
|
CP0567633
|
US9278960, 6-12
Show/Hide
|
C23H18FN3O2
|
1
|
1 |
IC50 = 31 nM
|
|
|
CP0567721
|
US9278960, 6-10
Show/Hide
|
C23H18FN3O
|
1
|
1 |
IC50 = 31 nM
|
|
|
CP0480095
|
US9278960, 4-55
Show/Hide
|
C20H19F3N4O3S
|
1
|
1 |
IC50 = 33 nM
|
|
|
CP0544364
|
US9278960, 6-15
Show/Hide
|
C19H15ClN6O
|
1
|
1 |
IC50 = 34 nM
|
|
|
CP0570552
|
US9278960, 6-18
Show/Hide
|
C22H16F4N4O
|
1
|
1 |
IC50 = 35 nM
|
|
|
CP0544340
|
US9278960, 7-33
Show/Hide
|
C22H19FN6O
|
1
|
1 |
IC50 = 36 nM
|
|
|
CP0567625
|
US9278960, 3-18
Show/Hide
|
C23H19F4N5O2
|
1
|
1 |
IC50 = 36 nM
|
|
|
CP0554176
|
US9278960, 2-8
Show/Hide
|
C20H15FN4O3
|
1
|
1 |
IC50 = 38 nM
|
|
|
CP0556047
|
US9278960, 4-49
Show/Hide
|
C24H19F4N5O
|
1
|
1 |
IC50 = 38 nM
|
|
|
CP0530612
|
US9278960, 7-34
Show/Hide
|
C22H20FN5O
|
1
|
1 |
IC50 = 39 nM
|
|
|
CP0548013
|
US9278960, 7-38
Show/Hide
|
C21H18FN5O2
|
1
|
1 |
IC50 = 39 nM
|
|
|
CP0515269
|
US9278960, 3-21
Show/Hide
|
C23H19FN4O3
|
1
|
1 |
IC50 = 40 nM
|
|
|
CP0550647
|
US9278960, 6-19
Show/Hide
|
C20H18N6O2
|
1
|
1 |
IC50 = 41 nM
|
|
|
CP0479667
|
US9278960, 4-39
Show/Hide
|
C22H22FN3O2
|
1
|
1 |
IC50 = 42 nM
|
|
|
CP0537020
|
US9278960, 6-22
Show/Hide
|
C21H16F3N5O
|
1
|
1 |
IC50 = 42 nM
|
|
|
CP0544942
|
US9278960, 2-33
Show/Hide
|
C21H20FN3O3S
|
1
|
1 |
IC50 = 42 nM
|
|
|
CP0545118
|
US9278960, 3-37
Show/Hide
|
C29H20FN5O
|
1
|
1 |
IC50 = 42 nM
|
|
|
CP0574079
|
US9278960, 3-25
Show/Hide
|
C20H14BrFN4O
|
1
|
1 |
IC50 = 43 nM
|
|
|
CP0550653
|
US9278960, 8-14
Show/Hide
|
C23H18FN3O
|
1
|
1 |
IC50 = 44 nM
|
|
|
CP0379770
|
US9278960, 4-63
Show/Hide
|
C21H25N5O2
|
1
|
1 |
IC50 = 46 nM
|
|
|
CP0489700
|
US9278960, 3-2
Show/Hide
|
C24H17FN4O
|
1
|
1 |
IC50 = 46 nM
|
|
|
CP0545127
|
US9278960, 4-69
Show/Hide
|
C20H21F2N5O
|
1
|
1 |
IC50 = 46 nM
|
|
|
CP0578094
|
US9278960, 3-42
Show/Hide
|
C25H19FN4O
|
1
|
1 |
IC50 = 46 nM
|
|
|
CP0512335
|
US9278960, 6-5
Show/Hide
|
C22H16FN3O
|
1
|
1 |
IC50 = 47 nM
|
|
|
CP0544351
|
US9278960, 2-22
Show/Hide
|
C24H22FN3O3
|
1
|
1 |
IC50 = 47 nM
|
|
|
CP0567626
|
US9278960, 3-22
Show/Hide
|
C24H18F4N4O3
|
1
|
1 |
IC50 = 47 nM
|
|
|
CP0556057
|
US9278960, 6-17
Show/Hide
|
C21H19N5O2
|
1
|
1 |
IC50 = 48 nM
|
|
|
CP0544354
|
US9278960, 4-98
Show/Hide
|
C21H22F3N5O2
|
1
|
1 |
IC50 = 52 nM
|
|
|
CP0567638
|
US9278960, 8-53
Show/Hide
|
C26H26N4O2
|
1
|
1 |
IC50 = 52 nM
|
|
|
CP0479668
|
US9278960, 4-48
Show/Hide
|
C24H23FN6O
|
1
|
1 |
IC50 = 53 nM
|
|
|
CP0556053
|
US9278960, 4-117
Show/Hide
|
C21H19F5N4O2S
|
1
|
1 |
IC50 = 53 nM
|
|
|
CP0556041
|
US9278960, 3-31
Show/Hide
|
C21H17FN4O
|
1
|
1 |
IC50 = 54 nM
|
|
|
CP0515266
|
US9278960, 3-34
Show/Hide
|
C23H16FN5O
|
1
|
1 |
IC50 = 55 nM
|
|
|
CP0544337
|
US9278960, 6-3
Show/Hide
|
C21H15FN4O
|
1
|
1 |
IC50 = 55 nM
|
|
|
CP0544362
|
US9278960, 4-99
Show/Hide
|
C21H25N5O2
|
1
|
1 |
IC50 = 55 nM
|
|
|
CP0578095
|
US9278960, 4-37
Show/Hide
|
C23H24FN3O2
|
1
|
1 |
IC50 = 55 nM
|
|
|
CP0511954
|
US9278960, 6-8
Show/Hide
|
C23H17ClFN3O2
|
1
|
1 |
IC50 = 56 nM
|
|
|
CP0550639
|
US9278960, 4-42
Show/Hide
|
C21H20FN3O3S
|
1
|
1 |
IC50 = 56 nM
|
|
|
CP0544355
|
US9278960, 4-38
Show/Hide
|
C22H22FN3O2
|
1
|
1 |
IC50 = 57 nM
|
|
|
CP0567717
|
US9278960, 1-18
Show/Hide
|
C16H10ClFN2O
|
1
|
1 |
IC50 = 58 nM
|
|
|
CP0489699
|
US9278960, 2-37
Show/Hide
|
C22H20FN3O2
|
1
|
1 |
IC50 = 59 nM
|
|
|
CP0544350
|
US9278960, 2-16
Show/Hide
|
C22H19FN4O3
|
1
|
1 |
IC50 = 59 nM
|
|
|
CP0576400
|
US9278960, 4-25
Show/Hide
|
C21H18F3N3O
|
1
|
1 |
IC50 = 61 nM
|
|
|
CP0409359
|
US9278960, 4-94
Show/Hide
|
C23H22F4N4O
|
1
|
1 |
IC50 = 63 nM
|
|
|
CP0576397
|
US9278960, 3-10
Show/Hide
|
C24H21FN4O2
|
1
|
1 |
IC50 = 63 nM
|
|
|
CP0489701
|
US9278960, 3-29
Show/Hide
|
C20H15FN4O
|
1
|
1 |
IC50 = 64 nM
|
|
|
CP0501508
|
US9278960, 2-15
Show/Hide
|
C23H21FN4O3
|
1
|
1 |
IC50 = 64 nM
|
|
|
CP0560714
|
US9278960, 4-93
Show/Hide
|
C24H24F4N4O
|
1
|
1 |
IC50 = 66 nM
|
|
|
CP0567627
|
US9278960, 3-43
Show/Hide
|
C27H23FN4O
|
1
|
1 |
IC50 = 66 nM
|
|
|
CP0574090
|
US9278960, 3-47
Show/Hide
|
C26H25F3N4O3
|
1
|
1 |
IC50 = 67 nM
|
|
|
CP0516377
|
US9278960, 3-33
Show/Hide
|
C23H16FN5O
|
1
|
1 |
IC50 = 69 nM
|
|
|
CP0577277
|
US9278960, 2-13
Show/Hide
|
C28H22FN3O3
|
1
|
1 |
IC50 = 71 nM
|
|
|
CP0550637
|
US9278960, 3-39
Show/Hide
|
C27H21FN4O
|
1
|
1 |
IC50 = 73 nM
|
|
|
CP0556050
|
US9278960, 4-64
Show/Hide
|
C23H29N5O2
|
1
|
1 |
IC50 = 73 nM
|
|
|
CP0544338
|
US9278960, 7-22
Show/Hide
|
C21H15F2N3O3
|
1
|
1 |
IC50 = 74 nM
|
|
|
CP0550636
|
US9278960, 3-17
Show/Hide
|
C22H18F4N6O2
|
1
|
1 |
IC50 = 74 nM
|
|
|
CP0419594
|
US9278960, 6-13
Show/Hide
|
C24H19FN2O2
|
1
|
1 |
IC50 = 76 nM
|
|
|
CP0560715
|
US9278960, 4-125
Show/Hide
|
C21H21F3N4O2S
|
1
|
1 |
IC50 = 76 nM
|
|
|
CP0567634
|
US9278960, 6-16
Show/Hide
|
C19H15FN6O
|
1
|
1 |
IC50 = 76 nM
|
|
|
CP0526138
|
US9278960, 4-24
Show/Hide
|
C22H21FN4O2
|
1
|
1 |
IC50 = 78 nM
|
|
|
CP0576902
|
US9278960, 4-111
Show/Hide
|
C22H22F2N4O
|
1
|
1 |
IC50 = 80 nM
|
|
|
CP0574089
|
US9278960, 3-40
Show/Hide
|
C28H23FN4O
|
1
|
1 |
IC50 = 81 nM
|
|
|
CP0578096
|
US9278960, 4-78
Show/Hide
|
C22H24F3N5O2
|
1
|
1 |
IC50 = 81 nM
|
|
|
CP0550638
|
US9278960, 4-28
Show/Hide
|
C21H19FN4O2
|
1
|
1 |
IC50 = 82 nM
|
|
|
CP0567628
|
US9278960, 4-29
Show/Hide
|
C19H18FN3O2
|
1
|
1 |
IC50 = 82 nM
|
|
|
CP0515270
|
US9278960, 3-28
Show/Hide
|
C20H14FN5O3
|
1
|
1 |
IC50 = 84 nM
|
|
|
CP0577719
|
US9278960, 4-31
Show/Hide
|
C20H19FN4O2
|
1
|
1 |
IC50 = 84 nM
|
|
|
CP0560712
|
US9278960, 3-15
Show/Hide
|
C24H22F3N5O2
|
1
|
1 |
IC50 = 85 nM
|
|
|
CP0548014
|
US9278960, 8-12
Show/Hide
|
C23H18FN3O
|
1
|
1 |
IC50 = 86 nM
|
|
|
CP0574091
|
US9278960, 4-134
Show/Hide
|
C23H26F3N5O2
|
1
|
1 |
IC50 = 86 nM
|
|
|
CP0516399
|
US9278960, 4-56
Show/Hide
|
C21H25N5O2
|
1
|
1 |
IC50 = 88 nM
|
|
|
CP0576399
|
US9278960, 3-41
Show/Hide
|
C29H25FN4O
|
1
|
1 |
IC50 = 89 nM
|
|
|
CP0550644
|
US9278960, 4-110
Show/Hide
|
C24H25FN4O
|
1
|
1 |
IC50 = 90 nM
|
|
|
CP0512332
|
US9278960, 4-74
Show/Hide
|
C21H21F3N4O2S
|
1
|
1 |
IC50 = 91 nM
|
|
|
CP0576894
|
US9278960, 4-52
Show/Hide
|
C25H26FN3O2
|
1
|
1 |
IC50 = 93 nM
|
|
|
CP0560720
|
US9278960, 8-55
Show/Hide
|
C25H24N4O3
|
1
|
1 |
IC50 = 96 nM
|
|
|
CP0414458
|
US9278960, 4-127
Show/Hide
|
C22H25N5O3S
|
1
|
1 |
IC50 = 97 nM
|
|
|
CP0550634
|
US9278960, 1-19
Show/Hide
|
C16H10ClFN2O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0560711
|
US9278960, 2-34
Show/Hide
|
C20H18FN3O3S
|
1
|
1 |
IC50 = 105 nM
|
|
|
CP0518171
|
US9278960, 2-31
Show/Hide
|
C21H19FN4O2
|
1
|
1 |
IC50 = 109 nM
|
|
|
CP0537471
|
US9278960, 4-131
Show/Hide
|
C21H24FN5O
|
1
|
1 |
IC50 = 112 nM
|
|
|
CP0576398
|
US9278960, 3-19
Show/Hide
|
C22H18F4N6O2
|
1
|
1 |
IC50 = 112 nM
|
|
|
CP0526139
|
US9278960, 4-70
Show/Hide
|
C21H22F3N5O
|
1
|
1 |
IC50 = 114 nM
|
|
|
CP0550642
|
US9278960, 4-103
Show/Hide
|
C22H23FN4O
|
1
|
1 |
IC50 = 114 nM
|
|
|
CP0576901
|
US9278960, 4-109
Show/Hide
|
C24H27FN4O
|
1
|
1 |
IC50 = 116 nM
|
|
|
CP0516379
|
US9278960, 4-41
Show/Hide
|
C22H22FN3O3
|
1
|
1 |
IC50 = 118 nM
|
|
|
CP0518181
|
US9278960, 4-26
Show/Hide
|
C21H19F2N3O
|
1
|
1 |
IC50 = 118 nM
|
|
|
CP0550643
|
US9278960, 4-104
Show/Hide
|
C22H23FN4O
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0560710
|
US9278960, 2-30
Show/Hide
|
C20H16FN3O3
|
1
|
1 |
IC50 = 123 nM
|
|
|
CP0570543
|
US9278960, 1-21
Show/Hide
|
C17H13FN2O
|
1
|
1 |
IC50 = 124 nM
|
|
|
CP0545144
|
US9278960, 5-5
Show/Hide
|
C22H20FN3O2
|
1
|
1 |
IC50 = 125 nM
|
|
|
CP0535534
|
US9278960, 2-32
Show/Hide
|
C22H22FN3O3
|
1
|
1 |
IC50 = 129 nM
|
|
|
CP0570544
|
US9278960, 1-23
Show/Hide
|
C18H13N3O
|
1
|
1 |
IC50 = 135 nM
|
|
|
CP0570547
|
US9278960, 4-45
Show/Hide
|
C21H21FN4O
|
1
|
1 |
IC50 = 136 nM
|
|
|
CP0480073
|
US9278960, 4-23
Show/Hide
|
C23H22FN3O3
|
1
|
1 |
IC50 = 137 nM
|
|
|
CP0545141
|
US9278960, 4-33
Show/Hide
|
C22H22FN3O2
|
1
|
1 |
IC50 = 138 nM
|
|
|
CP0515268
|
US9278960, 1-20
Show/Hide
|
C17H13FN2O2
|
1
|
1 |
IC50 = 139 nM
|
|
|
CP0550645
|
US9278960, 4-128
Show/Hide
|
C20H20F3N5O2S
|
1
|
1 |
IC50 = 142 nM
|
|
|
CP0512334
|
US9278960, 6-4
Show/Hide
|
C21H14F3N5
|
1
|
1 |
IC50 = 145 nM
|
|
|
CP0550641
|
US9278960, 4-68
Show/Hide
|
C20H22FN5O
|
1
|
1 |
IC50 = 149 nM
|
|
|
CP0560716
|
US9278960, 4-132
Show/Hide
|
C22H25N5O
|
1
|
1 |
IC50 = 149 nM
|
|
|
CP0567716
|
US9278960, 1-7
Show/Hide
|
C17H13FN2O
|
1
|
1 |
IC50 = 159 nM
|
|
|
CP0570550
|
US9278960, 4-79
Show/Hide
|
C21H19F6N5O2
|
1
|
1 |
IC50 = 159 nM
|
|
|
CP0419161
|
US9278960, 4-108
Show/Hide
|
C25H29FN4O
|
1
|
1 |
IC50 = 161 nM
|
|
|
CP0419157
|
US9278960, 4-1
Show/Hide
|
C21H20FN3O2
|
1
|
1 |
IC50 = 163 nM
|
|
|
CP0576895
|
US9278960, 4-58
Show/Hide
|
C21H25N5O3
|
1
|
1 |
IC50 = 163 nM
|
|
|
CP0556049
|
US9278960, 4-61
Show/Hide
|
C20H23N5O2
|
1
|
1 |
IC50 = 166 nM
|
|
|
CP0367698
|
US9278960, 1-24
Show/Hide
|
C16H11FN2O
|
1
|
1 |
IC50 = 169 nM
|
|
|
CP0550633
|
US9278960, 1-15
Show/Hide
|
C16H11BrN2O
|
1
|
1 |
IC50 = 169 nM
|
|
|
CP0550650
|
US9278960, 7-27
Show/Hide
|
C20H21F2N5O
|
1
|
1 |
IC50 = 169 nM
|
|
|
CP0544341
|
US9278960, 8-13
Show/Hide
|
C22H15FN4
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0544353
|
US9278960, 4-47
Show/Hide
|
C26H26FN5O
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0560708
|
US9278960, 1-9
Show/Hide
|
C16H9ClF2N2O
|
1
|
1 |
IC50 = 171 nM
|
|
|
CP0414456
|
US9278960, 4-105
Show/Hide
|
C24H25FN4O
|
1
|
1 |
IC50 = 172 nM
|
|
|
CP0545140
|
US9278960, 4-27
Show/Hide
|
C22H19F4N3O
|
1
|
1 |
IC50 = 183 nM
|
|
|
CP0567629
|
US9278960, 4-35
Show/Hide
|
C23H23FN4O2
|
1
|
1 |
IC50 = 187 nM
|
|
|
CP0379771
|
US9278960, 4-82
Show/Hide
|
C22H22F3N5O2
|
1
|
1 |
IC50 = 188 nM
|
|
|
CP0577718
|
US9278960, 3-36
Show/Hide
|
C29H20FN5O
|
1
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1 |
IC50 = 189 nM
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|
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CP0574077
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US9278960, 1-29
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C18H13N3O
|
1
|
1 |
IC50 = 190 nM
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|
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CP0414450
|
US9278960, 3-23
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C26H25FN4O2
|
1
|
1 |
IC50 = 192 nM
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|
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CP0578550
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US9278960, 4-60
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C20H23N5O2
|
1
|
1 |
IC50 = 196 nM
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|
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CP0535538
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US9278960, 3-46
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C26H25F3N4O4
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1
|
1 |
IC50 = 206 nM
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|
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CP0413600
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US9278960, 7-32
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C20H19FN6O3
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1
|
1 |
IC50 = 214 nM
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|
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CP0554175
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US9278960, 1-26
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C18H16N2O2
|
1
|
1 |
IC50 = 217 nM
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|
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CP0576892
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US9278960, 2-35
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C21H16FN3O4
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1
|
1 |
IC50 = 228 nM
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|
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CP0379772
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US9278960, 4-89
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C22H20F4N4O
|
1
|
1 |
IC50 = 235 nM
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|
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CP0379769
|
US9278960, 4-57
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C21H25N5O2
|
1
|
1 |
IC50 = 237 nM
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|
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CP0545143
|
US9278960, 4-120
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C22H25N5O
|
1
|
1 |
IC50 = 238 nM
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|
|
CP0409358
|
US9278960, 4-30
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|
C21H22FN3O2
|
1
|
1 |
IC50 = 241 nM
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|
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CP0512331
|
US9278960, 4-72
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C20H22FN5O
|
1
|
1 |
IC50 = 243 nM
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|
|
CP0537017
|
US9278960, 4-130
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|
C22H25N5O
|
1
|
1 |
IC50 = 245 nM
|
|
|
CP0550640
|
US9278960, 4-43
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|
C22H23FN4O
|
1
|
1 |
IC50 = 252 nM
|
|
|
CP0567631
|
US9278960, 4-62
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|
C20H23N5O2
|
1
|
1 |
IC50 = 252 nM
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|
|
CP0945246
|
US9278960, 4-97
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|
C20H20F3N5O2
|
1
|
1 |
IC50 = 260 nM
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|
|
CP0576897
|
US9278960, 4-76
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|
C22H21F3N4O2S
|
1
|
1 |
IC50 = 261 nM
|
|
|
CP0560717
|
US9278960, 4-133
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|
C22H24F3N5O2
|
1
|
1 |
IC50 = 272 nM
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|
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CP0560713
|
US9278960, 4-36
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|
C22H21FN4O3
|
1
|
1 |
IC50 = 274 nM
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|
|
CP0518183
|
US9278960, 5-4
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|
C21H18FN3O2
|
1
|
1 |
IC50 = 299 nM
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|
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CP0577720
|
US9278960, 4-34
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C23H25FN4O
|
1
|
1 |
IC50 = 330 nM
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|
|
CP0544366
|
US9278960, 7-5
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|
C16H10F2N2O
|
1
|
1 |
IC50 = 338 nM
|
|
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CP0379830
|
US9278960, 1-17
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C17H13ClN2O
|
1
|
1 |
IC50 = 368 nM
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|
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CP0567718
|
US9278960, 1-27
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C17H13ClN2O
|
1
|
1 |
IC50 = 377 nM
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|
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CP0479670
|
US9278960, 4-50
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C22H23FN4O
|
1
|
1 |
IC50 = 381 nM
|
|
|
CP0567630
|
US9278960, 4-40
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|
C22H22FN3O2
|
1
|
1 |
IC50 = 392 nM
|
|
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CP0483718
|
US9278960, 1-28
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C17H13FN2O
|
1
|
1 |
IC50 = 393 nM
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|
|
CP0576896
|
US9278960, 4-59
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|
C20H23N5O2
|
1
|
1 |
IC50 = 394 nM
|
|
|
CP0545119
|
US9278960, 2-17
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|
C20H12FN3O3
|
1
|
1 |
IC50 = 398 nM
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|
|
CP0578547
|
US9278960, 1-25
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|
C18H16N2O
|
1
|
1 |
IC50 = 407 nM
|
|
|
CP0414551
|
US9278960, 2-9
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|
C21H14FN3O2
|
1
|
1 |
IC50 = 416 nM
|
|
|
CP0490085
|
US9278960, 2-23
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|
C27H30FN3O5
|
1
|
1 |
IC50 = 456 nM
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|
|
CP0518170
|
US9278960, 2-12
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|
C24H20FN3O2
|
1
|
1 |
IC50 = 475 nM
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|
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CP0414454
|
US9278960, 4-32
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C22H19FN4O
|
1
|
1 |
IC50 = 478 nM
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|
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CP0516380
|
US9278960, 1-22
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C19H14N4O
|
1
|
1 |
IC50 = 505 nM
|
|
|
CP0868629
|
US9278960, 4-83
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|
C19H18F3N5O2
|
1
|
1 |
IC50 = 513 nM
|
|
|
CP0414553
|
US9278960, 2-19
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|
C21H15FN4O2
|
1
|
1 |
IC50 = 588 nM
|
|
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CP0546961
|
US9278960, 1-13
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|
C15H12N2OS
|
1
|
1 |
IC50 = 641 nM
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|
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CP0546960
|
US9278960, 1-10
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C17H12F2N2O2
|
1
|
1 |
IC50 = 660 nM
|
|
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CP0550632
|
US9278960, 1-14
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C20H16N4O
|
1
|
1 |
IC50 = 667 nM
|
|
|
CP0483726
|
US9278960, 1-12
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|
C14H12N4O
|
1
|
1 |
IC50 = 678 nM
|
|
|
CP0512328
|
US9278960, 1-16
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|
C16H11BrN2O
|
1
|
1 |
IC50 = 681 nM
|
|
|
CP0576394
|
US9278960, 1-11
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|
C15H14N2O
|
1
|
1 |
IC50 = 822 nM
|
|
|
CP0556055
|
US9278960, 4-122
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|
C20H23N5O2
|
1
|
1 |
IC50 = 931 nM
|
|
|
CP0545145
|
US9278960, 5-6
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|
C21H18FN3O3
|
1
|
1 |
IC50 = 987 nM
|
|
|
CP0477941
|
US9278960, 4-75
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|
C22H23F3N4O2S
|
1
|
1 |
IC50 = 1090 nM
|
|
|
CP0969344
|
US9278960, 4-67
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|
C19H18F3N5O2
|
1
|
1 |
IC50 = 1153 nM
|
|
|
CP0537485
|
US9278960, 4-81
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|
C20H19F3N4O3
|
1
|
1 |
IC50 = 1629 nM
|
|
|
CP0518172
|
US9278960, 2-36
Show/Hide
|
C21H16FN3O
|
1
|
1 |
IC50 = 3059 nM
|
|
|
CP0544363
|
US9278960, 4-129
Show/Hide
|
C20H20F3N5O2S
|
1
|
1 |
IC50 > 1000 nM
|
|
|
CP0576904
|
US9278960, 4-121
Show/Hide
|
C20H23N5O2
|
1
|
1 |
IC50 > 1000 nM
|
|
|