Compound ID |
Compound Name |
Compound Formula |
CP0071243
|
3,4,5,6-Tetrahydro-2H-[1,2']bipyridinyl-4'-carboxylic acid [4'-(cyclopropylmethyl-carbamoyl)-6-methyl-biphenyl-3-yl]-amide
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|
C29H32N4O2
|
1
|
1 |
IC50 = 2 nM
|
|
|
CP0019121
|
N-[3-[4-(cyclopropylmethylcarbamoyl)phenyl]-4-methylphenyl]-2-morpholin-4-ylpyridine-4-carboxamide
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|
C28H30N4O3
|
1
|
1 |
IC50 = 6 nM
|
|
|
CP0019162
|
N-[3-[4-(cyclopropylmethylcarbamoyl)phenyl]-4-methylphenyl]furan-3-carboxamide
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|
C23H22N2O3
|
1
|
1 |
IC50 = 16 nM
|
|
|
CP0035439
|
6-Methyl-biphenyl-3,4'-dicarboxylic acid 3-cyclopropylamide 4'-cyclopropylmethyl-amide
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|
C22H24N2O2
|
1
|
1 |
IC50 = 18 nM
|
|
|
CP0018897
|
1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]urea
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|
C31H37N5O3
|
1
|
1 |
IC50 = 47 nM
|
|
|
CP0060853
|
4-[4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-imidazol-5-yl]-2-methoxypyrimidine
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|
C19H20FN5O
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0935339
|
N-(3,3-dimethylbutan-2-yl)-4-(2-fluorobenzoyl)-1H-pyrrole-2-carboxamide
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|
C18H21FN2O2
|
1
|
1 |
IC50 = 158.49 nM
|
|
|
CP0091055
|
N-(furan-2-ylmethyl)-4-(2-methylbenzoyl)-1H-pyrrole-2-carboxamide
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|
C18H16N2O3
|
1
|
1 |
IC50 = 630.96 nM
|
|
|
CP0904685
|
4-(2-fluorobenzoyl)-N-(2-hydroxybenzyl)-1H-pyrrole-2-carboxamide
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|
C19H15FN2O3
|
1
|
1 |
IC50 = 794.33 nM
|
|
|
CP0920270
|
4-(2,4-difluorobenzoyl)-N-(2-hydroxybenzyl)-1H-pyrrole-2-carboxamide
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|
C19H14F2N2O3
|
1
|
1 |
IC50 = 1258.93 nM
|
|
|
CP0903358
|
N-(2,6-difluorobenzyl)-4-(2-fluorobenzoyl)-1H-pyrrole-2-carboxamide
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|
C19H13F3N2O2
|
1
|
1 |
IC50 = 1584.89 nM
|
|
|
CP0935340
|
GSK1326180
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|
C18H11F3N2O2
|
1
|
1 |
IC50 = 1584.89 nM
|
|
|
CP0921632
|
4-(2-fluorobenzoyl)-N-(3-(4-methylpiperazin-1-yl)benzyl)-1H-pyrrole-2-carboxamide
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|
C24H25FN4O2
|
1
|
1 |
IC50 = 1995.26 nM
|
|
|
CP0916036
|
N-(2,6-difluorobenzyl)-4-(2-methylbenzoyl)-1H-pyrrole-2-carboxamide
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|
C20H16F2N2O2
|
1
|
1 |
IC50 = 3162.28 nM
|
|
|
CP0920269
|
N-(2,6-difluorobenzyl)-4-(4-fluoro-2-methylbenzoyl)-1H-pyrrole-2-carboxamide
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|
C20H15F3N2O2
|
1
|
1 |
IC50 = 3981.07 nM
|
|
|