| Compound ID |
Compound Name |
Compound Formula |
|
CP0082712
|
4-Guanidino-benzoic acid 6-carbamimidoyl-naphthalen-2-yl ester
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|
C19H17N5O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0065004
|
(2R)-N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]-2-phenylacetamide
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|
C22H22N4O3S
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0234575
|
US9199927, camostat
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|
C20H22N4O5
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0064994
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-methylphenyl)sulfonylamino]acetamide
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|
C22H28N4O3S
|
2
|
| 1 |
IC50 = 33 nM
|
|
|
| 2 |
IC50 = 38 nM
|
|
|
|
CP0099151
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-fluorophenyl)sulfonylamino]acetamide
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|
C21H25FN4O3S
|
2
|
| 1 |
IC50 = 90 nM
|
|
|
| 2 |
IC50 = 190 nM
|
|
|
|
CP0549822
|
(2R)-N-(4-carbamimidoylphenyl)-2-[(4-chlorophenyl)sulfonylamino]-2-cyclohexylacetamide
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|
C21H25ClN4O3S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0548646
|
(2S)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-methylphenyl)sulfonylamino]acetamide
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|
C22H28N4O3S
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0548644
|
N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]-2-phenylacetamide
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|
C22H22N4O3S
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0067298
|
(E,E)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-one
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|
C23H24N4O
|
1
|
| 1 |
IC50 = 272 nM
|
|
|
|
CP0485679
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-methoxyphenyl)sulfonylamino]acetamide
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|
C22H28N4O4S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0326107
|
1-[(2S)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)propanoyl]-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
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|
C31H33N5O4S2
|
2
|
| 1 |
IC50 = 330 nM
|
|
|
| 2 |
IC50 = 676 nM
|
|
|
|
CP0267175
|
4-(6-Guanidino-hexanoyloxy)-benzoic acid ethyl ester
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|
C16H23N3O4
|
1
|
| 1 |
IC50 = 383 nM
|
|
|
|
CP0521053
|
N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide
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|
C20H26N4O3S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0513704
|
N-(4-carbamimidoylphenyl)-4-methyl-2-[(4-methylphenyl)sulfonylamino]pentanamide
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|
C20H26N4O3S
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0521056
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[[4-(trifluoromethyl)phenyl]sulfonylamino]acetamide
Show/Hide
|
C22H25F3N4O3S
|
2
|
| 1 |
IC50 = 680 nM
|
|
|
| 2 |
IC50 = 850 nM
|
|
|
|
CP0558969
|
N-(4-carbamimidoylphenyl)-3-cyclopentyl-2-[(4-methylphenyl)sulfonylamino]propanamide
Show/Hide
|
C22H28N4O3S
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
|
CP0521054
|
N-(4-carbamimidoylphenyl)-2-cyclopentyl-2-[(4-methylphenyl)sulfonylamino]acetamide
Show/Hide
|
C21H26N4O3S
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0417006
|
N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]-4-phenylbutanamide
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|
C24H26N4O3S
|
2
|
| 1 |
IC50 = 870 nM
|
|
|
| 2 |
IC50 = 1130 nM
|
|
|
|
CP0513705
|
N-(4-carbamimidoyl-2-fluorophenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide
Show/Hide
|
C20H25FN4O3S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0549821
|
(2R)-2-(benzenesulfonamido)-N-(4-carbamimidoylphenyl)-2-cyclohexylacetamide
Show/Hide
|
C21H26N4O3S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0558972
|
N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]-2-(oxan-4-yl)acetamide
Show/Hide
|
C21H26N4O4S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0558973
|
N-(4-carbamimidoylphenyl)-1-(4-methylphenyl)sulfonylpyrrolidine-2-carboxamide
Show/Hide
|
C19H22N4O3S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0521796
|
N-(4-carbamimidoylphenyl)-3-methyl-2-[(4-methylphenyl)sulfonylamino]butanamide
Show/Hide
|
C19H24N4O3S
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0485687
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-methylphenyl)carbamoylamino]acetamide
Show/Hide
|
C23H29N5O2
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0548645
|
2-benzyl-N-(4-carbamimidoylphenyl)-3-[(4-methylphenyl)sulfonylamino]propanamide
Show/Hide
|
C24H26N4O3S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0216665
|
3-(3-Carbamimidoyl-phenyl)-2-[2-(toluene-4-sulfonylamino)-acetylamino]-propionic acid methyl ester
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|
C20H24N4O5S
|
1
|
| 1 |
IC50 = 3140 nM
|
|
|
|
CP0384876
|
ethyl 4-[(2R)-3-(3-carbamimidoylphenyl)-2-[[2,4,6-tri(propan-2-yl)phenyl]sulfonylamino]propanoyl]piperazine-1-carboxylate
Show/Hide
|
C32H47N5O5S
|
1
|
| 1 |
IC50 = 3350 nM
|
|
|
|
CP0513703
|
2-[[(1R)-1-cyclohexyl-2-[(2S)-2-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]azetidin-1-yl]-2-oxoethyl]amino]acetic acid
Show/Hide
|
C22H32N6O4
|
1
|
| 1 |
IC50 = 4020 nM
|
|
|
|
CP0047129
|
1-[N-(naphthalen-2-ylsulfonyl)glycyl-4-carbamimidoyl-D-phenylalanyl]piperidine
Show/Hide
|
C27H31N5O4S
|
1
|
| 1 |
IC50 = 4460 nM
|
|
|
|
CP0521055
|
N-[(1R)-2-(4-carbamimidoylanilino)-1-cyclohexyl-2-oxoethyl]-4-methylbenzamide
Show/Hide
|
C23H28N4O2
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0084261
|
methyl 4-[(2S)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)propanoyl]piperazine-1-carboxylate
Show/Hide
|
C26H29N5O5S
|
1
|
| 1 |
IC50 = 6190 nM
|
|
|
|
CP0044338
|
4-[(R)-3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sulfonylamino)-propionyl]-piperazine-1-carboxylic acid dimethylamide
Show/Hide
|
C27H32N6O4S
|
1
|
| 1 |
IC50 = 6550 nM
|
|
|
|
CP0521051
|
(2R)-1-[(2R)-5-(diaminomethylideneamino)-2-[(1-hydroxynaphthalene-2-carbonyl)amino]pentanoyl]pyrrolidine-2-carboxamide
Show/Hide
|
C22H28N6O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0560438
|
(4S)-1-[(2S)-5-(diaminomethylideneamino)-2-[(3-methyl-1,2,3,4-tetrahydroquinolin-8-yl)sulfonylamino]pentanoyl]-4-methylpiperidine-2-carboxylic acid
Show/Hide
|
C23H36N6O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0558970
|
N-(4-carbamimidoylphenyl)-3-cyclohexyl-3-[(4-methylphenyl)sulfonylamino]propanamide
Show/Hide
|
C23H30N4O3S
|
1
|
| 1 |
IC50 = 11000 nM
|
|
|
|
CP0558971
|
N-(4-carbamimidoylphenyl)-4-methyl-2-[methyl-(4-methylphenyl)sulfonylamino]pentanamide
Show/Hide
|
C21H28N4O3S
|
1
|
| 1 |
IC50 > 19000 nM
|
|
|
|
CP0537151
|
N-(4-bromophenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide
Show/Hide
|
C19H23BrN2O3S
|
1
|
| 1 |
IC50 = 58000 nM
|
|
|
|
CP0560431
|
N-(3-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide
Show/Hide
|
C20H26N4O3S
|
1
|
| 1 |
IC50 = 73000 nM
|
|
|
