Brief Information of the Cell Line and Protein
Cell Line ID: CL000237 , 22Rv1
 Cell Line Info 
Synonyms
22RV1
22Rv-1
22rV1
CWR-22rv1
CWR22-Rv1
CWR22R-V1
CWR22-R1
CWR22Rv1
CWR22R
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_1045
Protein ID: PT01566 , Histone-lysine N-methyltransferase EHMT2
 Protein Info 
Gene Name EHMT2
Organism Homo sapiens, Human
Protein Classification Epigenetic regulator
Uniprot ID Q96KQ7
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000237
 Cell Line Info 
 Protein ID: PT01566
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0042224
 Compound Info 
N-(1-cyclohexylpiperidin-4-yl)-6-methoxy-7-(3-piperidin-1-ylpropoxy)-2-(4-propan-2-yl-1,4-diazepan-1-yl)quinazolin-4-amine
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C36H59N7O2
  1
1
IC50 = 14 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0341308
 Compound Info 
N-[1-(cyclohexylmethyl)piperidin-4-yl]-6-methoxy-7-(3-piperidin-1-ylpropoxy)-2-(4-propan-2-yl-1,4-diazepan-1-yl)quinazolin-4-amine
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C37H61N7O2
  1
1
IC50 = 24 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0046275
 Compound Info 
2-cyclohexyl-6-methoxy-N-(1-propan-2-ylpiperidin-4-yl)-7-(3-pyrrolidin-1-ylpropoxy)quinazolin-4-amine
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C30H47N5O2
  1
1
IC50 = 48 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS