| Compound ID |
Compound Name |
Compound Formula |
|
CP0115062
|
8-nitroindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C15H7N3O4
|
2
|
| 1 |
IC50 = 446 nM
|
|
|
| 2 |
IC50 = 450 nM
|
|
|
|
CP0210843
|
8-fluoranylindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C15H7FN2O2
|
2
|
| 1 |
IC50 = 1200 nM
|
|
|
| 2 |
IC50 = 1230 nM
|
|
|
|
CP0075092
|
8-Bromotryptanthrin
Show/Hide
|
C15H7BrN2O2
|
2
|
| 1 |
IC50 = 3200 nM
|
|
|
| 2 |
IC50 = 3220 nM
|
|
|
|
CP0420665
|
8-fluoro-2-(piperazin-1-ylmethyl)indolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C20H17FN4O2
|
1
|
| 1 |
IC50 = 3580 nM
|
|
|
|
CP0492024
|
2-[(dimethylamino)methyl]-8-fluoroindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C18H14FN3O2
|
1
|
| 1 |
IC50 = 3810 nM
|
|
|
|
CP0075091
|
indolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C15H8N2O2
|
2
|
| 1 |
IC50 = 5000 nM
|
|
|
| 2 |
IC50 = 5010 nM
|
|
|
|
CP0420666
|
tert-butyl 4-[(8-fluoro-6,12-dioxoindolo[2,1-b]quinazolin-2-yl)methyl]piperazine-1-carboxylate
Show/Hide
|
C25H25FN4O4
|
1
|
| 1 |
IC50 = 8050 nM
|
|
|
|
CP0070605
|
2,8-difluoroindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C15H6F2N2O2
|
2
|
| 1 |
IC50 = 8190 nM
|
|
|
| 2 |
IC50 = 8200 nM
|
|
|
|
CP0447827
|
8-fluoro-2-(morpholin-4-ylmethyl)indolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C20H16FN3O3
|
1
|
| 1 |
IC50 = 16540 nM
|
|
|
|
CP0489554
|
8-fluoro-2-piperazin-1-ylindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C19H15FN4O2
|
1
|
| 1 |
IC50 = 17760 nM
|
|
|
|
CP0212292
|
9-chloroindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C15H7ClN2O2
|
2
|
| 1 |
IC50 = 18370 nM
|
|
|
| 2 |
IC50 = 18400 nM
|
|
|
|
CP0159403
|
8-fluoro-2-[(4-methylpiperazin-1-yl)methyl]indolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C21H19FN4O2
|
1
|
| 1 |
IC50 = 18660 nM
|
|
|
|
CP0210794
|
7-chloroindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C15H7ClN2O2
|
2
|
| 1 |
IC50 = 19450 nM
|
|
|
| 2 |
IC50 = 19500 nM
|
|
|
|
CP0431573
|
2-morpholin-4-ylindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C19H15N3O3
|
1
|
| 1 |
IC50 = 20320 nM
|
|
|
|
CP0115133
|
8-methylindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C16H10N2O2
|
2
|
| 1 |
IC50 = 21800 nM
|
|
|
| 2 |
IC50 = 21810 nM
|
|
|
|
CP0482370
|
8-fluoro-2-piperidin-1-ylindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C20H16FN3O2
|
1
|
| 1 |
IC50 = 22220 nM
|
|
|
|
CP0431572
|
2-[(4-methylpiperazin-1-yl)methyl]indolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C21H20N4O2
|
1
|
| 1 |
IC50 = 23290 nM
|
|
|
|
CP0245009
|
2-fluoroindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C15H7FN2O2
|
2
|
| 1 |
IC50 = 37780 nM
|
|
|
| 2 |
IC50 = 37800 nM
|
|
|
|
CP0482369
|
2-(4-methylpiperazin-1-yl)indolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 = 48670 nM
|
|
|
|
CP0071950
|
(S)-2-amino-3-(1-methyl-1H-indol-3-yl)propanoic acid
Show/Hide
|
C12H14N2O2
|
2
|
| 1 |
IC50 = 56900 nM
|
|
|
| 2 |
IC50 = 82530 nM
|
|
|
|
CP0431574
|
8-fluoro-2-(4-methylpiperazin-1-yl)indolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C20H17FN4O2
|
1
|
| 1 |
IC50 = 79000 nM
|
|
|
|
CP0438462
|
2-(dimethylamino)-8-fluoroindolo[2,1-b]quinazoline-6,12-dione
Show/Hide
|
C17H12FN3O2
|
1
|
| 1 |
IC50 = 90900 nM
|
|
|
