| Compound ID |
Compound Name |
Compound Formula |
|
CP0422909
|
[2-[(2-chlorobenzoyl)amino]-6-(4-methoxyphenyl)-3-thiophen-2-yl-1-benzofuran-4-yl] acetate
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|
C28H20ClNO5S
|
12
|
| 1 |
IC50 = 0.82 nM
|
|
|
| 2 |
IC50 = 0.88 nM
|
|
|
| 3 |
IC50 = 6.3 nM
|
|
|
| 4 |
IC50 = 6.4 nM
|
|
|
| 5 |
IC50 = 9.2 nM
|
|
|
| 6 |
IC50 = 72.9 nM
|
|
|
| 7 |
IC50 = 76.6 nM
|
|
|
| 8 |
IC50 = 90.9 nM
|
|
|
| 9 |
IC50 = 114 nM
|
|
|
| 10 |
IC50 = 502 nM
|
|
|
| 11 |
IC50 = 564 nM
|
|
|
| 12 |
IC50 = 602 nM
|
|
|
|
CP0422908
|
[6-(4-methoxyphenyl)-2-[(2-methylbenzoyl)amino]-3-thiophen-2-yl-1-benzofuran-4-yl] acetate
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|
C29H23NO5S
|
12
|
| 1 |
IC50 = 0.83 nM
|
|
|
| 2 |
IC50 = 0.88 nM
|
|
|
| 3 |
IC50 = 7.2 nM
|
|
|
| 4 |
IC50 = 8.9 nM
|
|
|
| 5 |
IC50 = 9.1 nM
|
|
|
| 6 |
IC50 = 55.4 nM
|
|
|
| 7 |
IC50 = 81.8 nM
|
|
|
| 8 |
IC50 = 83.5 nM
|
|
|
| 9 |
IC50 = 89.2 nM
|
|
|
| 10 |
IC50 = 109 nM
|
|
|
| 11 |
IC50 = 478 nM
|
|
|
| 12 |
IC50 = 525 nM
|
|
|
|
CP0418685
|
[2-[(3-fluorobenzoyl)amino]-6-(4-methoxyphenyl)-3-thiophen-2-yl-1-benzofuran-4-yl] acetate
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|
C28H20FNO5S
|
12
|
| 1 |
IC50 = 3.7 nM
|
|
|
| 2 |
IC50 = 5.3 nM
|
|
|
| 3 |
IC50 = 6.3 nM
|
|
|
| 4 |
IC50 = 6.6 nM
|
|
|
| 5 |
IC50 = 24.6 nM
|
|
|
| 6 |
IC50 = 76.8 nM
|
|
|
| 7 |
IC50 = 80.6 nM
|
|
|
| 8 |
IC50 = 81.8 nM
|
|
|
| 9 |
IC50 = 96.2 nM
|
|
|
| 10 |
IC50 = 504 nM
|
|
|
| 11 |
IC50 = 559 nM
|
|
|
| 12 |
IC50 = 621 nM
|
|
|
|
CP0422913
|
[2-(diacetylamino)-6-(4-methoxyphenyl)-3-thiophen-2-yl-1-benzofuran-4-yl] acetate
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|
C25H21NO6S
|
12
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 4.5 nM
|
|
|
| 3 |
IC50 = 10 nM
|
|
|
| 4 |
IC50 = 10.5 nM
|
|
|
| 5 |
IC50 = 82.3 nM
|
|
|
| 6 |
IC50 = 87.2 nM
|
|
|
| 7 |
IC50 = 582 nM
|
|
|
| 8 |
IC50 = 645 nM
|
|
|
| 9 |
IC50 = 647 nM
|
|
|
| 10 |
IC50 = 663 nM
|
|
|
| 11 |
IC50 = 677 nM
|
|
|
| 12 |
IC50 = 874 nM
|
|
|
|
CP0036382
|
CAS_52-53-9
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|
C27H38N2O4
|
6
|
| 1 |
IC50 = 6.7 nM
|
|
|
| 2 |
IC50 = 8.6 nM
|
|
|
| 3 |
IC50 = 76.4 nM
|
|
|
| 4 |
IC50 = 412 nM
|
|
|
| 5 |
IC50 = 456 nM
|
|
|
| 6 |
IC50 = 522 nM
|
|
|
