| Compound ID |
Compound Name |
Compound Formula |
|
CP0573403
|
(1R,3R)-3-[[3-bromo-1-[3-(2-methylsulfonylethyl)-4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C25H29BrN8O3S2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0033806
|
(1R,3R)-3-[[3-bromo-1-[4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C22H23BrN8OS
|
2
|
| 1 |
IC50 = 16 nM
|
|
|
| 2 |
IC50 = 1310 nM
|
|
|
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CP0273097
|
(1R,3R)-3-[[3-bromo-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C22H23BrN8O2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0549848
|
(1R,3R)-3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N-(2-methoxyethyl)cyclopentane-1-carboxamide
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|
C23H24BrN7O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0578440
|
(1R,3R)-3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C22H22BrN7O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0343899
|
(1R,3R)-3-[[3-bromo-1-[3-(2-hydroxyethyl)-4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C24H27BrN8O2S
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0542833
|
(1R,3R)-3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N-methylcyclopentane-1-carboxamide
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|
C21H20BrN7O
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0273098
|
(1R,3R)-3-[[3-bromo-1-[3-(2-cyanoethyl)-4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C25H26BrN9OS
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0495023
|
(1R,3R)-3-[[3-bromo-1-[3-fluoro-4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C22H22BrFN8OS
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0527890
|
(1R,3R)-3-[[3-bromo-1-[3-cyano-4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C23H22BrN9OS
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0579445
|
3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N-(2-methoxyethyl)cyclobutane-1-carboxamide
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|
C22H22BrN7O2
|
1
|
| 1 |
IC50 = 86 nM
|
|
|
|
CP0573500
|
(1R,3R)-3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N-methylcyclopentane-1-sulfonamide
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|
C20H20BrN7O2S
|
1
|
| 1 |
IC50 = 106 nM
|
|
|
|
CP0579446
|
(1S,3R)-3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N-(2-methoxyethyl)cyclopentane-1-carboxamide
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|
C23H24BrN7O2
|
1
|
| 1 |
IC50 = 156 nM
|
|
|
|
CP0578439
|
N-[(1R,3R)-3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]cyclopentyl]-3-methoxypropanamide
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|
C23H24BrN7O2
|
1
|
| 1 |
IC50 = 159 nM
|
|
|
|
CP0561384
|
(1S,3S)-3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N-(2-methoxyethyl)cyclopentane-1-carboxamide
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|
C23H24BrN7O2
|
1
|
| 1 |
IC50 = 183 nM
|
|
|
|
CP0495024
|
(1R,3R)-3-[[1-[3-(2-aminoethyl)-4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-3-bromopyrazolo[3,4-d]pyrimidin-6-yl]amino]-N,1-dimethylcyclopentane-1-carboxamide
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|
C24H28BrN9OS
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0495022
|
N-[(1R,3R)-3-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]cyclopentyl]-2-methoxyethanesulfonamide
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|
C22H24BrN7O3S
|
1
|
| 1 |
IC50 = 262 nM
|
|
|
|
CP0564480
|
3-bromo-N-[(3R)-1-methylsulfonylpyrrolidin-3-yl]-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-amine
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|
C19H18BrN7O2S
|
1
|
| 1 |
IC50 = 378 nM
|
|
|
|
CP0966519
|
Trans-3-Bromo-N-(3-(1H-imidazol-2-yl)cyclopentyl)-1-(6-quinolyl)pyrazolo[3,4-d]pyrimidin-6-amine
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|
C22H19BrN8
|
1
|
| 1 |
IC50 = 545 nM
|
|
|
|
CP0572008
|
3-bromo-N-(1-piperidin-4-ylpyrazol-4-yl)-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-amine
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|
C22H20BrN9
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0572009
|
4-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N-(2-methoxyethyl)cyclohexane-1-carboxamide
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|
C24H26BrN7O2
|
1
|
| 1 |
IC50 = 628 nM
|
|
|
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CP0545400
|
4-[(3-bromo-1-quinolin-6-ylpyrazolo[3,4-d]pyrimidin-6-yl)amino]-N-(2-methoxyethyl)cyclohexane-1-carboxamide
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|
C24H26BrN7O2
|
1
|
| 1 |
IC50 = 763 nM
|
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