| Compound ID |
Compound Name |
Compound Formula |
|
CP0559154
|
3-fluoro-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C20H15FN4O4S
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0540714
|
2,4-difluoro-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C20H14F2N4O4S
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0479150
|
3,5-difluoro-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C20H14F2N4O4S
|
1
|
| 1 |
IC50 = 77.2 nM
|
|
|
|
CP0022562
|
N-[5-(3-chloro-4-oxopyrido[1,2-a]pyrimidin-7-yl)-2-methoxypyridin-3-yl]-2,4-difluorobenzenesulfonamide
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|
C20H13ClF2N4O4S
|
1
|
| 1 |
IC50 = 89.2 nM
|
|
|
|
CP0530599
|
4-fluoro-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C20H15FN4O4S
|
1
|
| 1 |
IC50 = 105.8 nM
|
|
|
|
CP0393369
|
2,5-difluoro-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C20H14F2N4O4S
|
1
|
| 1 |
IC50 = 108.5 nM
|
|
|
|
CP0405021
|
2,4-difluoro-N-[2-methoxy-5-(3-methyl-4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C21H16F2N4O4S
|
1
|
| 1 |
IC50 = 119 nM
|
|
|
|
CP0466815
|
4-methoxy-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C21H18N4O5S
|
1
|
| 1 |
IC50 = 138 nM
|
|
|
|
CP0530601
|
N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]-2-methylbenzenesulfonamide
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|
C21H18N4O4S
|
1
|
| 1 |
IC50 = 153.4 nM
|
|
|
|
CP0559153
|
N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]-4-(trifluoromethyl)benzenesulfonamide
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|
C21H15F3N4O4S
|
1
|
| 1 |
IC50 = 163.3 nM
|
|
|
|
CP0411609
|
N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C20H16N4O4S
|
1
|
| 1 |
IC50 = 197.9 nM
|
|
|
|
CP0484279
|
4-chloro-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C20H15ClN4O4S
|
1
|
| 1 |
IC50 = 223.4 nM
|
|
|
|
CP0393372
|
4-cyano-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C21H15N5O4S
|
1
|
| 1 |
IC50 = 245.7 nM
|
|
|
|
CP0013602
|
(Scheme A): Preparation of 2,2-difluoroethyl (3S)-3-{[2′-amino-5-fluoro-2-(morpholin-4-yl)-4,5′-bipyrimidin-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylate
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|
C20H25F3N8O4
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0008405
|
(2S)-1-N-[4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl]pyrrolidine-1,2-dicarboxamide
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|
C19H22F3N5O2S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0405022
|
N-[2-chloro-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]-2,4-difluorobenzenesulfonamide
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|
C19H11ClF2N4O3S
|
1
|
| 1 |
IC50 > 400 nM
|
|
|
|
CP0445672
|
N-[2-chloro-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]-2-fluorobenzenesulfonamide
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|
C19H12ClFN4O3S
|
1
|
| 1 |
IC50 > 400 nM
|
|
|
|
CP0530597
|
2-fluoro-N-[2-methoxy-5-(4-oxopyrido[1,2-a]pyrimidin-7-yl)pyridin-3-yl]benzenesulfonamide
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|
C20H15FN4O4S
|
1
|
| 1 |
IC50 > 400 nM
|
|
|
