| Compound ID |
Compound Name |
Compound Formula |
|
CP0568295
|
8-(4-chlorophenyl)-2-(ethylamino)-6-(2-methylindazol-5-yl)-1,6-naphthyridin-7-one
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|
C24H20ClN5O
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0574625
|
8-(4-chlorophenyl)-6-(2-methylindazol-5-yl)-2-(2,2,2-trifluoroethylamino)-1,6-naphthyridin-7-one
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|
C24H17ClF3N5O
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0547283
|
8-(4-chlorophenyl)-2-(2,2-difluoroethoxy)-6-(2-methylindazol-5-yl)-1,6-naphthyridin-7-one
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|
C24H17ClF2N4O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0568186
|
8-(4-chlorophenyl)-6-(2-methylindazol-5-yl)-2-(2,2,2-trifluoroethylamino)pyrido[4,3-d]pyrimidin-7-one
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|
C23H16ClF3N6O
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0569201
|
8-(4-chlorophenyl)-6-(2,3-dimethylbenzimidazol-5-yl)-2-(2,2,2-trifluoroethylamino)pyrido[4,3-d]pyrimidin-7-one
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|
C24H18ClF3N6O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0568348
|
8-(4-chlorophenyl)-2-ethoxy-6-(2-methylindazol-5-yl)-1,6-naphthyridin-7-one
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|
C24H19ClN4O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0574249
|
8-(4-chlorophenyl)-6-(3-methylbenzimidazol-5-yl)-2-(2,2,2-trifluoroethylamino)pyrido[4,3-d]pyrimidin-7-one
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|
C23H16ClF3N6O
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0547282
|
8-(4-chlorophenyl)-6-(2-methylindazol-5-yl)-2-(2,2,2-trifluoroethoxy)-1,6-naphthyridin-7-one
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|
C24H16ClF3N4O2
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0568859
|
8-(4-bromophenyl)-6-(4-methoxyphenyl)-2-(2,2,2-trifluoroethylamino)pyrido[4,3-d]pyrimidin-7-one
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|
C22H16BrF3N4O2
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0568185
|
8-(4-bromophenyl)-6-quinolin-6-yl-2-(2,2,2-trifluoroethylamino)pyrido[4,3-d]pyrimidin-7-one
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|
C24H15BrF3N5O
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0547280
|
8-(4-chlorophenyl)-6-quinolin-6-yl-2-(2,2,2-trifluoroethylamino)pyrido[4,3-d]pyrimidin-7-one
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|
C24H15ClF3N5O
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0466410
|
4-[4-(difluoromethoxy)phenyl]-2-(2-methylindazol-5-yl)-6-(2,2,2-trifluoroethoxy)pyrido[3,2-c]pyridazin-3-one
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|
C24H16F5N5O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0466411
|
6-(2,2-difluoroethoxy)-4-[4-(difluoromethoxy)phenyl]-2-(2,3-dihydro-1-benzofuran-5-yl)pyrido[3,2-c]pyridazin-3-one
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|
C24H17F4N3O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0487495
|
2-(1,3-benzothiazol-6-yl)-6-(2,2-difluoroethoxy)-4-[4-(difluoromethoxy)phenyl]pyrido[3,2-c]pyridazin-3-one
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|
C23H14F4N4O3S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0507631
|
6-(2,2-difluoroethoxy)-4-(6-methoxypyridin-3-yl)-2-(2-methylindazol-5-yl)pyrido[3,2-c]pyridazin-3-one
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|
C23H18F2N6O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0553141
|
4-(4-chlorophenyl)-2-(2-methylindazol-5-yl)-6-(2,2,2-trifluoroethoxy)pyrido[3,2-c]pyridazin-3-one
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|
C23H15ClF3N5O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0556540
|
4-[4-(difluoromethoxy)phenyl]-2-(2-methylindazol-5-yl)-6-(2,2,2-trifluoroethylsulfanyl)pyrido[3,2-c]pyridazin-3-one
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|
C24H16F5N5O2S
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0568372
|
6-(2,2-difluoroethoxy)-4-[4-(difluoromethoxy)phenyl]-2-(2-methylindazol-5-yl)pyrido[3,2-c]pyridazin-3-one
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|
C24H17F4N5O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0569312
|
6-ethoxy-4-(4-methoxyphenyl)-2-(2-methylindazol-5-yl)pyrido[3,2-c]pyridazin-3-one
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|
C24H21N5O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0569313
|
6-(2,2-difluoroethoxy)-4-[4-(difluoromethoxy)phenyl]-2-[2-methyl-3-(trideuteriomethoxy)indazol-5-yl]pyrido[3,2-c]pyridazin-3-one
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|
C25H19F4N5O4
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0547279
|
8-(4-chlorophenyl)-6-(2-methylindazol-5-yl)-2-(3,3,3-trifluoropropyl)-1,6-naphthyridin-7-one
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|
C25H18ClF3N4O
|
1
|
| 1 |
IC50 = 101 nM
|
|
|
|
CP0568184
|
8-(4-chlorophenyl)-6-(4-methoxyphenyl)-2-(2,2,2-trifluoroethylamino)pyrido[4,3-d]pyrimidin-7-one
Show/Hide
|
C22H16ClF3N4O2
|
1
|
| 1 |
IC50 = 113 nM
|
|
|
|
CP0556615
|
4-[4-(difluoromethoxy)phenyl]-2-(2-methylindazol-5-yl)-6-(3,3,3-trifluoropropoxy)pyrido[3,2-c]pyridazin-3-one
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|
C25H18F5N5O3
|
1
|
| 1 |
IC50 >= 100 nM
|
|
|
