Compound ID |
Compound Name |
Compound Formula |
CP0048984
|
(S)-4-Cyano-N-[3-(4-fluorophenyl)-3-(4-methanesulfonyl-phenyl)-propyl]-benzamide
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|
C24H21FN2O3S
|
1
|
1 |
EC50 = 0.14 nM
|
|
|
CP0166335
|
N-[(2,4-dichlorophenyl)methyl]-4-(3-methylsulfonylphenoxy)piperidine-1-carboxamide
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|
C20H22Cl2N2O4S
|
1
|
1 |
EC50 = 0.25 nM
|
|
|
CP0265634
|
N-[(2,4-dichlorophenyl)methyl]-4-[4-(methylsulfamoyl)phenoxy]piperidine-1-carboxamide
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|
C20H23Cl2N3O4S
|
1
|
1 |
EC50 = 0.29 nM
|
|
|
CP0167547
|
N-[3-(4-fluorophenyl)-3-(4-methylsulfonylphenyl)propyl]-6-(2,2,2-trifluoroethoxy)pyridine-3-carboxamide
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|
C24H22F4N2O4S
|
1
|
1 |
EC50 = 0.3 nM
|
|
|
CP0675924
|
4-cyano-N-[3-(4-fluorophenyl)-3-(4-methylsulfonylphenyl)propyl]benzamide
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|
C24H21FN2O3S
|
1
|
1 |
EC50 = 0.3 nM
|
|
|
CP0307706
|
N-[(2,4-dichlorophenyl)methyl]-4-[4-(methylcarbamoyl)phenoxy]piperidine-1-carboxamide
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|
C21H23Cl2N3O3
|
1
|
1 |
EC50 = 0.34 nM
|
|
|
CP0264731
|
N-[3-(4-fluorophenyl)-3-(4-methylsulfonylphenyl)propyl]-4-methylsulfonylbenzamide
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|
C24H24FNO5S2
|
1
|
1 |
EC50 = 0.4 nM
|
|
|
CP0316498
|
4-(2-cyanophenoxy)-N-(2,4-dichlorobenzyl)piperidine-1-carboxamide
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|
C20H19Cl2N3O2
|
1
|
1 |
EC50 = 0.44 nM
|
|
|
CP0092495
|
N-[3-(4-fluorophenyl)-3-(4-methylsulfonylphenyl)propyl]pyridine-3-carboxamide
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|
C22H21FN2O3S
|
1
|
1 |
EC50 = 0.6 nM
|
|
|
CP0307705
|
4-(3-cyanophenoxy)-N-(2,4-dichlorobenzyl)piperidine-1-carboxamide
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|
C20H19Cl2N3O2
|
1
|
1 |
EC50 = 0.63 nM
|
|
|
CP0354376
|
4-(4-cyanophenoxy)-N-(2,4-dichlorobenzyl)piperidine-1-carboxamide
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|
C20H19Cl2N3O2
|
1
|
1 |
EC50 = 0.78 nM
|
|
|
CP0298811
|
N-[(2,4-dichlorophenyl)methyl]-4-(4-methylsulfonylphenoxy)piperidine-1-carboxamide
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|
C20H22Cl2N2O4S
|
1
|
1 |
EC50 = 0.97 nM
|
|
|
CP0069782
|
N-[(2,4-dichlorophenyl)methyl]-4-(2-methylsulfonylphenoxy)piperidine-1-carboxamide
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|
C20H22Cl2N2O4S
|
1
|
1 |
EC50 = 1.65 nM
|
|
|
CP0062447
|
4-(1-(2,4-dichlorobenzylcarbamoyl)piperidin-4-yloxy)benzoic acid
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|
C20H20Cl2N2O4
|
1
|
1 |
EC50 = 1.7 nM
|
|
|
CP0362371
|
N-[(3S)-3-(4-fluorophenyl)-3-(4-methylsulfonylphenyl)propyl]-4-hydroxybenzamide
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|
C23H22FNO4S
|
1
|
1 |
EC50 = 1.7 nM
|
|
|
CP0793909
|
N-[3-(4-Fluorophenyl)-3-(4-methanesulfonyl-phenyl)-propyl]-6-hydroxy-nicotinamide
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|
C22H21FN2O4S
|
1
|
1 |
EC50 = 2.1 nM
|
|
|
CP0167548
|
(R)-4-Cyano-N-[3-(4-fluorophenyl)-3-(4-methanesulfonyl-phenyl)-propyl]-benzamide
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|
C24H21FN2O3S
|
1
|
1 |
EC50 = 2.8 nM
|
|
|
CP0353378
|
N-[(2,4-dichlorophenyl)methyl]-4-(4-fluorophenoxy)piperidine-1-carboxamide
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|
C19H19Cl2FN2O2
|
1
|
1 |
EC50 = 4.2 nM
|
|
|
CP0166334
|
4-(4-chlorophenoxy)-N-(2,4-dichlorobenzyl)piperidine-1-carboxamide
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|
C19H19Cl3N2O2
|
1
|
1 |
EC50 = 10 nM
|
|
|
CP0354375
|
N-[(2,4-dichlorophenyl)methyl]-4-[4-(trifluoromethoxy)phenoxy]piperidine-1-carboxamide
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|
C20H19Cl2F3N2O3
|
1
|
1 |
EC50 = 18 nM
|
|
|
CP0136208
|
N-[(3R)-3-(4-fluorophenyl)-3-(4-methylsulfonylphenyl)propyl]-4-hydroxybenzamide
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|
C23H22FNO4S
|
1
|
1 |
EC50 = 23 nM
|
|
|
CP0157343
|
N-[[4-bromo-2-(trifluoromethoxy)phenyl]methyl]-6-(3,3,3-trifluoropropoxy)pyridine-3-carboxamide
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|
C17H13BrF6N2O3
|
1
|
1 |
IC50 = 0.1 nM
|
|
|
CP0252290
|
4-tert-butyl-N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]benzamide
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|
C19H23ClN2O3S
|
1
|
1 |
IC50 = 1 nM
|
|
|
CP0062445
|
N-[(2,4-dichlorophenyl)methyl]-4-phenoxypiperidine-1-carboxamide
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|
C19H20Cl2N2O2
|
1
|
1 |
IC50 = 5.1 nM
|
|
|
CP0201666
|
N-[(2-chloro-4-cyanophenyl)methyl]-6-(3,3,3-trifluoropropoxy)pyridine-3-carboxamide
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|
C17H13ClF3N3O2
|
1
|
1 |
IC50 = 12 nM
|
|
|
CP0231165
|
N-(benzenesulfonyl)-4-[[5-(cyclohexylcarbamoylamino)-1-methylindol-3-yl]methyl]-3-methoxybenzamide
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|
C31H34N4O5S
|
1
|
1 |
IC50 = 14 nM
|
|
|
CP0069816
|
N-[(2,4-dichlorophenyl)methyl]-4-pyrimidin-2-yloxypiperidine-1-carboxamide
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|
C17H18Cl2N4O2
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0214723
|
N-[(2,4-dichlorophenyl)methyl]-6-(2,2,2-trifluoroethoxy)pyridine-3-carboxamide
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|
C15H11Cl2F3N2O2
|
1
|
1 |
IC50 = 18 nM
|
|
|
CP0122841
|
N-[[2-(trifluoromethoxy)phenyl]methyl]-6-(3,3,3-trifluoropropoxy)pyridine-3-carboxamide
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|
C17H14F6N2O3
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0157342
|
N-[[4-(4-methylsulfonylphenyl)phenyl]methyl]-6-(3,3,3-trifluoropropoxy)pyridine-3-carboxamide
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|
C23H21F3N2O4S
|
1
|
1 |
IC50 = 24 nM
|
|
|
CP0214722
|
N-[(2-chloro-4-methylsulfonylphenyl)methyl]-6-(3,3,3-trifluoropropoxy)pyridine-3-carboxamide
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|
C17H16ClF3N2O4S
|
1
|
1 |
IC50 = 28 nM
|
|
|
CP0226507
|
N-[[2-chloro-4-(methylsulfamoyl)phenyl]methyl]-6-(3,3,3-trifluoropropoxy)pyridine-3-carboxamide
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|
C17H17ClF3N3O4S
|
1
|
1 |
IC50 = 31 nM
|
|
|
CP0124002
|
N-[[2-chloro-4-(tetrazol-1-yl)phenyl]methyl]-6-(3,3,3-trifluoropropoxy)pyridine-3-carboxamide
Show/Hide
|
C17H14ClF3N6O2
|
1
|
1 |
IC50 = 38 nM
|
|
|