| Compound ID |
Compound Name |
Compound Formula |
|
CP0544988
|
1-(cyclopropylmethyl)-4-fluoro-5-[5-methoxy-4-oxo-3-(2-phenylpyrazol-3-yl)pyridazin-1-yl]-3,3-dimethylindol-2-one
Show/Hide
|
C28H26FN5O3
|
1
|
| 1 |
IC50 = 0.08 nM
|
|
|
|
CP0381403
|
4-fluoro-5-[5-methoxy-4-oxo-3-(2-phenylpyrazol-3-yl)pyridazin-1-yl]-3,3-dimethyl-1-propan-2-ylindol-2-one
Show/Hide
|
C27H26FN5O3
|
1
|
| 1 |
IC50 = 0.11 nM
|
|
|
|
CP0431551
|
1-cyclobutyl-4-fluoro-5-[5-methoxy-4-oxo-3-(2-phenylpyrazol-3-yl)pyridazin-1-yl]-3,3-dimethylindol-2-one
Show/Hide
|
C28H26FN5O3
|
1
|
| 1 |
IC50 = 0.12 nM
|
|
|
|
CP0544989
|
4'-fluoro-5'-[5-methoxy-4-oxo-3-(2-phenylpyrazol-3-yl)pyridazin-1-yl]-1'-methylspiro[cyclobutane-1,3'-indole]-2'-one
Show/Hide
|
C26H22FN5O3
|
1
|
| 1 |
IC50 = 0.13 nM
|
|
|
|
CP0544991
|
4-fluoro-5-[5-methoxy-4-oxo-3-(2-phenylpyrazol-3-yl)pyridazin-1-yl]-1,3,3-trimethylindol-2-one
Show/Hide
|
C25H22FN5O3
|
1
|
| 1 |
IC50 = 0.22 nM
|
|
|
|
CP0539686
|
1-(2-fluoro-4-pyrrolidin-1-ylphenyl)-5-methoxy-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C24H22FN5O2
|
1
|
| 1 |
IC50 = 0.23 nM
|
|
|
|
CP0031913
|
1-(cyclopropylmethyl)-5-[2-(1,2-dihydroimidazo[1,2-a]benzimidazol-3-yl)ethoxy]-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C28H27N7O2
|
1
|
| 1 |
IC50 = 0.76 nM
|
|
|
|
CP0468626
|
1-[2-fluoro-4-(2-oxopyrrolidin-1-yl)phenyl]-5-methoxy-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C24H20FN5O3
|
1
|
| 1 |
IC50 = 0.79 nM
|
|
|
|
CP0553095
|
1-(cyclopropylmethyl)-5-[3-(1-methylbenzimidazol-2-yl)propoxy]-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C28H28N6O2
|
1
|
| 1 |
IC50 = 0.81 nM
|
|
|
|
CP0544992
|
3-[3-fluoro-4-[5-methoxy-4-oxo-3-(2-phenylpyrazol-3-yl)pyridazin-1-yl]phenyl]-1,3-oxazolidin-2-one
Show/Hide
|
C23H18FN5O4
|
1
|
| 1 |
IC50 = 0.94 nM
|
|
|
|
CP0573808
|
1-(cyclopropylmethyl)-5-[2-(1-methylbenzimidazol-2-yl)oxyethoxy]-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C27H26N6O3
|
1
|
| 1 |
IC50 = 4.1 nM
|
|
|
|
CP0567157
|
1-(cyclopropylmethyl)-5-[2-(1-methylbenzimidazol-2-yl)ethoxy]-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C27H26N6O2
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0454948
|
1-cyclopropyl-5-methoxy-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C17H16N4O2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0558034
|
1-(cyclopropylmethyl)-5-methoxy-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C18H18N4O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0464131
|
5-methoxy-3-(2-phenylpyrazol-3-yl)-1-(2,2,2-trifluoroethyl)pyridazin-4-one
Show/Hide
|
C16H13F3N4O2
|
1
|
| 1 |
IC50 = 550 nM
|
|
|
|
CP0451863
|
1-(cyclopropylmethyl)-5-[4-(1-methylbenzimidazol-2-yl)butoxy]-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C29H30N6O2
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0454949
|
5-methoxy-1-methyl-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C15H14N4O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0456176
|
5-methoxy-3-(2-methylpyrazol-3-yl)-1-phenylpyridazin-4-one
Show/Hide
|
C15H14N4O2
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0445076
|
1-(cyclopropylmethyl)-5-[(1-methylbenzimidazol-2-yl)methoxy]-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
Show/Hide
|
C26H24N6O2
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
|
CP0474856
|
6-methyl-N-[(1R)-1-[4-(trifluoromethoxy)phenyl]propyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
Show/Hide
|
C18H17F3N4O2
|
1
|
| 1 |
IC50 = 7400 nM
|
|
|
