Brief Information of the Compound and Protein
Compound Name
1-[2-fluoro-4-(2-oxopyrrolidin-1-yl)phenyl]-5-methoxy-3-(2-phenylpyrazol-3-yl)pyridazin-4-one
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PubChem ID
CID: 46848741
SID: 99237252
Canonical SMILES
COc1cn(nc(-c2ccnn2-c2ccccc2)c1=O)-c1ccc(cc1F)N1CCCC1=O
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Compound Formula C24H20FN5O3
Compound Structure
Protein Name
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
Protein Classification
Enzyme
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Phosphodiesterase
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Phosphodiesterase 10
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Phosphodiesterase 10A
Uniprot ID
Q9Y233
Gene Name
PDE10A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000053 COS-7 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 0.79 nM
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