| Compound ID |
Compound Name |
Compound Formula |
|
CP0429946
|
Efatutazone
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|
C27H26N4O4S
|
1
|
| 1 |
EC50 = 0.038 nM
|
|
|
|
CP0108032
|
(S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid
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|
C34H30N2O5
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0077847
|
((4-Methoxy-phenoxycarbonyl)-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzyl}-amino)-acetic acid
Show/Hide
|
C29H28N2O7
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0005387
|
Avandamet
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|
C18H19N3O3S
|
6
|
| 1 |
EC50 = 4 nM
|
|
|
| 2 |
EC50 = 30 nM
|
|
|
| 3 |
EC50 = 43 nM
|
|
|
| 4 |
EC50 = 100 nM
|
|
|
| 5 |
EC50 = 144 nM
|
|
|
| 6 |
EC50 = 396 nM
|
|
|
|
CP0404238
|
3-[[6-(3-fluoro-4-methylphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
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|
C23H19FN2O4
|
1
|
| 1 |
EC50 = 4.4 nM
|
|
|
|
CP0079947
|
ethyl 3-[4-[2-[6-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxypropanoate
Show/Hide
|
C32H35NO7S
|
1
|
| 1 |
EC50 < 10 nM
|
|
|
|
CP0117013
|
3-[4-[2-[6-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxy-N-methylpropanamide
Show/Hide
|
C31H34N2O6S
|
1
|
| 1 |
EC50 < 10 nM
|
|
|
|
CP0180554
|
3-[4-[2-[6-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxypropanoic acid
Show/Hide
|
C30H31NO7S
|
1
|
| 1 |
EC50 < 10 nM
|
|
|
|
CP0246268
|
ethyl 3-[4-[2-[6-[(E)-2-(3,5-dihydroxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxypropanoate
Show/Hide
|
C30H31NO7S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0246269
|
3-[4-[2-[6-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxypropanamide
Show/Hide
|
C30H32N2O6S
|
1
|
| 1 |
EC50 < 10 nM
|
|
|
|
CP0457137
|
4-[5-chloro-1-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]indol-2-yl]butanoic acid
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|
C20H17ClN2O4S2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0863971
|
(9aS)-8-acetyl-N-[(2-ethyl-4-fluoronaphthalen-1-yl)methyl]-1,7-dihydroxy-3-methoxy-9a-methyl-9-oxo-9,9a-dihydrodibenzo[b,d]furan-4-carboxamide
Show/Hide
|
C30H26FNO7
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0486320
|
(9aS)-8-acetyl-N-[(2-ethyl-7-fluoronaphthalen-1-yl)methyl]-1,7-dihydroxy-3-methoxy-9a-methyl-9-oxodibenzofuran-4-carboxamide
Show/Hide
|
C30H26FNO7
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0458506
|
4-[5-chloro-1-[(4-methyl-2,3-dihydro-1,4-benzoxazin-6-yl)sulfonyl]indol-2-yl]butanoic acid
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|
C21H21ClN2O5S
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0235683
|
ethyl 3-[4-[2-[6-[(E)-3-(3,5-dihydroxyphenyl)prop-2-enoyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxypropanoate
Show/Hide
|
C31H31NO8S
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0241505
|
3-[4-[2-[6-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-(2,2,2-trifluoroethoxy)propanoic acid
Show/Hide
|
C30H28F3NO7S
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0101563
|
3-[[6-(2,3-dihydro-1H-inden-5-yloxy)-1-methylimidazo[4,5-c]pyridin-2-yl]methoxy]benzoic acid
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|
C24H21N3O4
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0408690
|
3-[[6-(5-chloro-3-methylpyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H18ClN3O4
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0396433
|
3-[[6-(2,3-dihydro-1-benzofuran-6-yloxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C24H20N2O5
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0404237
|
3-[[6-(3-fluoro-5-methylphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H19FN2O4
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0494049
|
3-[[6-(4-fluoro-2-methylphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H19FN2O4
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0408913
|
3-[[6-(3-chloro-5-fluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H16ClFN2O4
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0828938
|
3-({1-Methyl-6-[3-(trifluoromethyl)phenoxy]-1H-benzimidazol-2-yl}methoxy)benzoic acid Hydrochloride
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|
C23H18ClF3N2O4
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0471701
|
3-[[6-(5-chloro-3-fluoropyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H15ClFN3O4
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0352391
|
3-[[5-(2,3-dihydro-1H-inden-5-yloxy)-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C24H21N3O4
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0079948
|
ethyl 3-[4-[2-[6-[(E)-3-(3,5-dihydroxyphenyl)prop-2-enoyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-(2,2,2-trifluoroethoxy)propanoate
Show/Hide
|
C31H28F3NO8S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0456622
|
ethyl 3-[4-[2-[6-[(E)-3-(3,5-dimethoxyphenyl)prop-2-enoyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxypropanoate
Show/Hide
|
C33H35NO8S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0471671
|
3-[[6-(2,6-dimethylpyridin-3-yl)oxy-1-methyl-4-propan-2-yloxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C26H27N3O5
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0471675
|
3-[[6-(2,6-dimethylpyridin-3-yl)oxy-1-methyl-4-propoxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C26H27N3O5
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0471676
|
3-[[6-(2-methoxypyridin-4-yl)oxy-1-methyl-4-propan-2-yloxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C25H25N3O6
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0412246
|
4-(5-chloro-1-naphthalen-2-ylsulfonylindol-2-yl)butanoic acid
Show/Hide
|
C22H18ClNO4S
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0389269
|
3-[[6-(5-fluoro-2-methylphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H19FN2O4
|
1
|
| 1 |
EC50 = 39 nM
|
|
|
|
CP0101285
|
3-[[1-methyl-6-(4-methylphenoxy)benzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H20N2O4
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0111047
|
3-[[6-(3-ethoxyphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C24H22N2O5
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0479763
|
4-[1-[(2-amino-1,3-benzothiazol-6-yl)sulfonyl]-5-chloroindol-2-yl]butanoic acid
Show/Hide
|
C19H16ClN3O4S2
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0110595
|
3-[[6-(3,5-dimethylpyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O4
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0367078
|
3-[[5-(3,5-dimethylphenoxy)-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O4
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0404165
|
3-[[6-(3-fluoro-5-methylpyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H18FN3O4
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0404239
|
CS-011
Show/Hide
|
C20H19N3O4S
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0915211
|
3-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}benzonitrile dihydrochloride
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|
C24H24Cl2N4O2
|
1
|
| 1 |
EC50 = 43 nM
|
|
|
|
CP0230168
|
3-[[3-methyl-5-(4-methylphenoxy)imidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O4
|
1
|
| 1 |
EC50 = 45 nM
|
|
|
|
CP0347476
|
ethyl 3-[4-[2-[6-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-(2,2,2-trifluoroethoxy)propanoate
Show/Hide
|
C32H32F3NO7S
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0367077
|
3-[[5-(3-fluoro-4-methylphenoxy)-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H18FN3O4
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0412239
|
4-[5-chloro-1-(3-methoxyphenyl)sulfonylindol-2-yl]butanoic acid
Show/Hide
|
C19H18ClNO5S
|
1
|
| 1 |
EC50 = 55 nM
|
|
|
|
CP0101564
|
3-[[1-methyl-6-(2-methylphenoxy)benzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H20N2O4
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0426352
|
3-[[6-(2-methoxypyridin-4-yl)oxy-1,4-dimethylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O5
|
1
|
| 1 |
EC50 = 57 nM
|
|
|
|
CP0471678
|
3-[[6-(3,5-dimethylpyridin-2-yl)oxy-1-methyl-4-propan-2-yloxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C26H27N3O5
|
1
|
| 1 |
EC50 = 57 nM
|
|
|
|
CP0514759
|
3-[[4-ethoxy-6-(2-methoxypyridin-4-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C24H23N3O6
|
1
|
| 1 |
EC50 = 58 nM
|
|
|
|
CP0514760
|
3-[[6-(3,5-dimethylpyridin-2-yl)oxy-4-ethoxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C25H25N3O5
|
1
|
| 1 |
EC50 = 58 nM
|
|
|
|
CP0471672
|
3-[[7-fluoro-6-(2-methoxypyridin-4-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H18FN3O5
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0874408
|
3-{[6-(4-Fluoro-3-methylphenoxy)-1-methyl-1H-benzimidazol-2-yl]methoxy}benzoic acid Hydrochloride
Show/Hide
|
C23H20ClFN2O4
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0891653
|
3-{[6-(3-Chloro-4-fluorophenoxy)-1-methyl-1H-benzimidazol-2-yl]methoxy}benzoic acid Hydrochloride
Show/Hide
|
C22H17Cl2FN2O4
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0457134
|
4-[1-(3-methoxyphenyl)sulfonyl-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
|
C20H18F3NO5S
|
1
|
| 1 |
EC50 = 65 nM
|
|
|
|
CP0860307
|
1-(3-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}phenyl)ethanone dihydrochloride
Show/Hide
|
C25H27Cl2N3O3
|
1
|
| 1 |
EC50 = 65 nM
|
|
|
|
CP0396354
|
3-[[6-(4-chloro-3-fluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H16ClFN2O4
|
1
|
| 1 |
EC50 = 68 nM
|
|
|
|
CP0412236
|
4-[1-(1,3-benzodioxol-5-ylsulfonyl)-5-chloroindol-2-yl]butanoic acid
Show/Hide
|
C19H16ClNO6S
|
1
|
| 1 |
EC50 = 71 nM
|
|
|
|
CP0475932
|
3-[[6-(5-chloropyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H16ClN3O4
|
1
|
| 1 |
EC50 = 71 nM
|
|
|
|
CP0447392
|
4-[5-chloro-1-(4-methoxyphenyl)sulfonylindol-2-yl]butanoic acid
Show/Hide
|
C19H18ClNO5S
|
1
|
| 1 |
EC50 = 72 nM
|
|
|
|
CP0457135
|
4-[5-chloro-1-(3-methylphenyl)sulfonylindol-2-yl]butanoic acid
Show/Hide
|
C19H18ClNO4S
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
|
CP0101284
|
3-[[1-methyl-6-(3-methylphenoxy)benzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H20N2O4
|
1
|
| 1 |
EC50 = 79 nM
|
|
|
|
CP0073199
|
ethyl 3-[4-[2-[6-[(E)-2-(3,5-dihydroxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-(2,2,2-trifluoroethoxy)propanoate
Show/Hide
|
C30H28F3NO7S
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0412247
|
4-[1-(4-methoxyphenyl)sulfonyl-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
|
C20H18F3NO5S
|
1
|
| 1 |
EC50 = 82 nM
|
|
|
|
CP0007353
|
(2E,6E)-9-[(2R)-6-hydroxy-2,8-dimethyl-3,4-dihydrochromen-2-yl]-2,6-dimethylnona-2,6-dienoic acid
Show/Hide
|
C22H30O4
|
1
|
| 1 |
EC50 = 84 nM
|
|
|
|
CP0685175
|
3-{[6-(3-Chlorophenoxy)-1-methyl-1H-benzimidazol-2-yl]methoxy}benzoic acid Hydrochloride
Show/Hide
|
C22H18Cl2N2O4
|
1
|
| 1 |
EC50 = 86 nM
|
|
|
|
CP0860309
|
3-{[6-(2,3-Dihydro-1-benzofuran-5-yloxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}benzoic acid Hydrochloride
Show/Hide
|
C24H21ClN2O5
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0471698
|
3-[[6-(3,5-dichloropyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H15Cl2N3O4
|
1
|
| 1 |
EC50 = 89 nM
|
|
|
|
CP0346869
|
3-[[5-(3,4-dimethylphenoxy)-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O4
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0396434
|
3-[[6-(2-fluoro-4-methylphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H19FN2O4
|
1
|
| 1 |
EC50 = 92 nM
|
|
|
|
CP0404167
|
3-[[5-(2,3-dihydro-1-benzofuran-6-yloxy)-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H19N3O5
|
1
|
| 1 |
EC50 = 94 nM
|
|
|
|
CP0486258
|
3-[[6-(3,5-difluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H16F2N2O4
|
1
|
| 1 |
EC50 = 95 nM
|
|
|
|
CP0475934
|
3-[[6-(5-fluoro-3-methylpyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H18FN3O4
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0547492
|
3-[[6-(2-methoxy-6-methylpyridin-4-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O5
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0189356
|
3-[[5-(2,4-dimethylphenoxy)-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O4
|
1
|
| 1 |
EC50 = 101 nM
|
|
|
|
CP0471670
|
3-[[6-(2,6-dimethylpyridin-3-yl)oxy-4-ethoxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C25H25N3O5
|
1
|
| 1 |
EC50 = 104 nM
|
|
|
|
CP0230174
|
3-[[1-methyl-6-[3-(trifluoromethoxy)phenoxy]benzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H17F3N2O5
|
1
|
| 1 |
EC50 = 113 nM
|
|
|
|
CP0426355
|
3-[[6-(6-methoxypyridin-3-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O5
|
1
|
| 1 |
EC50 = 115 nM
|
|
|
|
CP0874407
|
3-((6-(3,4-difluorophenoxy)-1-methyl-1H-benzo[d]imidazol-2-yl)methoxy)benzoic acid Hydrochloride
Show/Hide
|
C22H17ClF2N2O4
|
1
|
| 1 |
EC50 = 118 nM
|
|
|
|
CP0230173
|
3-[[6-(4-fluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H17FN2O4
|
1
|
| 1 |
EC50 = 122 nM
|
|
|
|
CP0101568
|
3-[[6-(4-chlorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H17ClN2O4
|
1
|
| 1 |
EC50 = 126 nM
|
|
|
|
CP0446338
|
3-[[1-methyl-6-(5-methylpyridin-2-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O4
|
1
|
| 1 |
EC50 = 129 nM
|
|
|
|
CP0408915
|
3-[[6-(2,5-difluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H16F2N2O4
|
1
|
| 1 |
EC50 = 134 nM
|
|
|
|
CP0429947
|
3-[[6-(2-fluoro-5-methylphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H19FN2O4
|
1
|
| 1 |
EC50 = 139 nM
|
|
|
|
CP0408916
|
3-[[6-(2,4-difluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H16F2N2O4
|
1
|
| 1 |
EC50 = 143 nM
|
|
|
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CP0447366
|
4-[1-(1,3-benzothiazol-5-ylsulfonyl)-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
|
C20H15F3N2O4S2
|
1
|
| 1 |
EC50 = 147 nM
|
|
|
|
CP0408561
|
2-(2-methyl-4-(3-(2-propyl-4-(trifluoromethyl)phenoxy)propoxy)phenoxy)acetic acid
Show/Hide
|
C22H25F3O5
|
1
|
| 1 |
EC50 = 153 nM
|
|
|
|
CP0447365
|
4-[1-(2,1,3-benzothiadiazol-5-ylsulfonyl)-5-chloroindol-2-yl]butanoic acid
Show/Hide
|
C18H14ClN3O4S2
|
1
|
| 1 |
EC50 = 153 nM
|
|
|
|
CP0480048
|
3-[[5-(2-methoxy-6-methylpyridin-4-yl)oxy-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H20N4O5
|
1
|
| 1 |
EC50 = 166 nM
|
|
|
|
CP0451772
|
2-[4-[(2-heptylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
|
C28H30N2O2
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0457054
|
4-[5-chloro-1-[(2-methyl-1,3-benzothiazol-5-yl)sulfonyl]indol-2-yl]butanoic acid
Show/Hide
|
C20H17ClN2O4S2
|
1
|
| 1 |
EC50 = 175 nM
|
|
|
|
CP0404166
|
3-[[6-(5,6-dimethylpyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O4
|
1
|
| 1 |
EC50 = 176 nM
|
|
|
|
CP0471674
|
3-[[6-(2-ethoxypyridin-4-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O5
|
1
|
| 1 |
EC50 = 182 nM
|
|
|
|
CP0511702
|
3-[[6-(1-benzofuran-6-yloxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C24H18N2O5
|
1
|
| 1 |
EC50 = 188 nM
|
|
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CP0486817
|
3-[[6-(2-methoxypyridin-4-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O5
|
1
|
| 1 |
EC50 = 188 nM
|
|
|
|
CP0113760
|
2-[4-[[5-(4-chlorophenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C30H25ClN2O2
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0041219
|
Actos
Show/Hide
|
C19H20N2O3S
|
5
|
| 1 |
EC50 = 200 nM
|
|
|
| 2 |
EC50 = 300 nM
|
|
|
| 3 |
EC50 = 320 nM
|
|
|
| 4 |
EC50 = 380 nM
|
|
|
| 5 |
EC50 = 1400 nM
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CP0235682
|
ethyl 3-[4-[2-[6-[(E)-3-(3,5-dimethoxyphenyl)prop-2-enoyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-(2,2,2-trifluoroethoxy)propanoate
Show/Hide
|
C33H32F3NO8S
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0347479
|
3-[4-[2-[6-[(E)-2-(3,5-dihydroxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-(2,2,2-trifluoroethoxy)propanoic acid
Show/Hide
|
C28H24F3NO7S
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0408557
|
3-[[6-(3-chloropyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H16ClN3O4
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0507033
|
4-[1-[3-(trifluoromethoxy)phenyl]sulfonyl-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
|
C20H15F6NO5S
|
1
|
| 1 |
EC50 = 201 nM
|
|
|
|
CP0429948
|
3-[[6-(3-fluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H17FN2O4
|
1
|
| 1 |
EC50 = 201 nM
|
|
|
|
CP0261934
|
4-[1-(1,3-benzothiazol-6-ylsulfonyl)-5-chloroindol-2-yl]butanoic acid
Show/Hide
|
C19H15ClN2O4S2
|
1
|
| 1 |
EC50 = 206 nM
|
|
|
|
CP0388493
|
2-[4-[(2-hexylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
|
C27H28N2O2
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0408920
|
3-[[6-(2,3-difluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H16F2N2O4
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0426353
|
3-[[6-(5-methoxypyridin-3-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O5
|
1
|
| 1 |
EC50 = 231 nM
|
|
|
|
CP0101286
|
3-[[6-(3-methoxyphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H20N2O5
|
1
|
| 1 |
EC50 = 235 nM
|
|
|
|
CP0480049
|
3-[[6-(2,6-dimethylpyridin-3-yl)oxy-1,7-dimethylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C24H23N3O4
|
1
|
| 1 |
EC50 = 244 nM
|
|
|
|
CP0486816
|
3-[[6-(2,6-dimethylpyridin-3-yl)oxy-7-fluoro-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H20FN3O4
|
1
|
| 1 |
EC50 = 246 nM
|
|
|
|
CP0514758
|
3-[[6-(2,6-dimethylpyridin-3-yl)oxy-4-methoxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C24H23N3O5
|
1
|
| 1 |
EC50 = 249 nM
|
|
|
|
CP0514954
|
3-[[6-(6-methoxy-2-methylpyridin-3-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O5
|
1
|
| 1 |
EC50 = 255 nM
|
|
|
|
CP0412235
|
4-[1-(3-chlorophenyl)sulfonyl-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
|
C19H15ClF3NO4S
|
1
|
| 1 |
EC50 = 256 nM
|
|
|
|
CP0412237
|
4-(5-chloro-1-naphthalen-1-ylsulfonylindol-2-yl)butanoic acid
Show/Hide
|
C22H18ClNO4S
|
1
|
| 1 |
EC50 = 265 nM
|
|
|
|
CP0404164
|
3-[[5-(4-chloro-3-fluorophenoxy)-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H15ClFN3O4
|
1
|
| 1 |
EC50 = 269 nM
|
|
|
|
CP0472683
|
3-[[6-(2,6-dimethylpyridin-3-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O4
|
1
|
| 1 |
EC50 = 273 nM
|
|
|
|
CP0412241
|
4-[5-chloro-1-(4-methylphenyl)sulfonylindol-2-yl]butanoic acid
Show/Hide
|
C19H18ClNO4S
|
1
|
| 1 |
EC50 = 277 nM
|
|
|
|
CP0408701
|
3-[[6-(3-fluoropyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H16FN3O4
|
1
|
| 1 |
EC50 = 280 nM
|
|
|
|
CP0412234
|
4-[1-(benzenesulfonyl)-5-methylindol-2-yl]butanoic acid
Show/Hide
|
C19H19NO4S
|
1
|
| 1 |
EC50 = 284 nM
|
|
|
|
CP0457133
|
4-[1-(benzenesulfonyl)-5-chloroindol-2-yl]butanoic acid
Show/Hide
|
C18H16ClNO4S
|
1
|
| 1 |
EC50 = 284 nM
|
|
|
|
CP0376355
|
methyl 2-[4-[3-(4-acetyl-3-hydroxy-2-propylphenoxy)propoxy]phenoxy]acetate
Show/Hide
|
C23H28O7
|
1
|
| 1 |
EC50 = 288 nM
|
|
|
|
CP0113762
|
2-[4-[[5-(3-methoxyphenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C31H28N2O3
|
1
|
| 1 |
EC50 = 290 nM
|
|
|
|
CP0852616
|
3-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}benzoic acid dihydrochloride
Show/Hide
|
C24H25Cl2N3O4
|
1
|
| 1 |
EC50 = 299 nM
|
|
|
|
CP0223551
|
2-[[4-[(4-phenoxyphenyl)methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C25H25NO4
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0250832
|
2-[[4-[[4-methoxy-2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C21H22F3NO4
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0101287
|
3-[[6-(4-methoxyphenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H20N2O5
|
1
|
| 1 |
EC50 = 307 nM
|
|
|
|
CP0471677
|
3-[[6-(6-methoxy-5-methylpyridin-3-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O5
|
1
|
| 1 |
EC50 = 315 nM
|
|
|
|
CP0860306
|
2,6-Dimethyl-4-{[1-methyl-2-(phenoxymethyl)-1H-benzimidazol-6-yl]oxy}aniline dihydrochloride
Show/Hide
|
C23H25Cl2N3O2
|
1
|
| 1 |
EC50 = 318 nM
|
|
|
|
CP0230169
|
3-[[6-(2,3-dihydro-1-benzofuran-6-yloxy)-1-methylimidazo[4,5-c]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H19N3O5
|
1
|
| 1 |
EC50 = 335 nM
|
|
|
|
CP0860308
|
1-(4-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}phenyl)ethanone dihydrochloride
Show/Hide
|
C25H27Cl2N3O3
|
1
|
| 1 |
EC50 = 340 nM
|
|
|
|
CP0408692
|
3-[[1-methyl-6-(3-methylpyridin-2-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O4
|
1
|
| 1 |
EC50 = 351 nM
|
|
|
|
CP0874409
|
1-(2-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}phenyl)ethanone dihydrochloride
Show/Hide
|
C25H27Cl2N3O3
|
1
|
| 1 |
EC50 = 356 nM
|
|
|
|
CP0457136
|
4-[1-[(2-amino-1,3-benzoxazol-6-yl)sulfonyl]-5-chloroindol-2-yl]butanoic acid
Show/Hide
|
C19H16ClN3O5S
|
1
|
| 1 |
EC50 = 378 nM
|
|
|
|
CP0874410
|
2-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}benzonitrile dihydrochloride
Show/Hide
|
C24H24Cl2N4O2
|
1
|
| 1 |
EC50 = 391 nM
|
|
|
|
CP0915212
|
4-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}benzonitrile dihydrochloride
Show/Hide
|
C24H24Cl2N4O2
|
1
|
| 1 |
EC50 = 395 nM
|
|
|
|
CP0468275
|
2-[4-[(2-pentylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
|
C26H26N2O2
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0113819
|
2-[4-[[5-(4-methoxyphenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C31H28N2O3
|
1
|
| 1 |
EC50 = 410 nM
|
|
|
|
CP0412233
|
4-[1-(benzenesulfonyl)-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
|
C19H16F3NO4S
|
1
|
| 1 |
EC50 = 417 nM
|
|
|
|
CP0486813
|
3-[[6-(2-methoxy-6-methylpyridin-3-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O5
|
1
|
| 1 |
EC50 = 436 nM
|
|
|
|
CP0427359
|
3-[[1-methyl-6-(4-methylpyridin-2-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O4
|
1
|
| 1 |
EC50 = 458 nM
|
|
|
|
CP0685177
|
3-{[6-(2-Methoxyphenoxy)-1-methyl-1H-benzimidazol-2-yl]methoxy}benzoic acid Hydrochloride
Show/Hide
|
C23H21ClN2O5
|
1
|
| 1 |
EC50 = 474 nM
|
|
|
|
CP0480706
|
2-[4-(4-benzylanilino)-6-chloropyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C25H28ClN3O2S
|
1
|
| 1 |
EC50 = 490 nM
|
|
|
|
CP0471673
|
3-[[6-(2-ethylpyridin-4-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O4
|
1
|
| 1 |
EC50 = 509 nM
|
|
|
|
CP0204345
|
2-(4-(3-(biphenyl-4-yloxy)propoxy)phenylthio)hexanoic acid
Show/Hide
|
C27H30O4S
|
1
|
| 1 |
EC50 = 540 nM
|
|
|
|
CP0496268
|
3-[[1-methyl-6-(6-methylpyridin-3-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O4
|
1
|
| 1 |
EC50 = 543 nM
|
|
|
|
CP0766755
|
3-[(3-Methyl-5-phenoxy-3H-imidazo[4,5-b]pyridin-2-yl)methoxy]benzoic acid Dihydrochloride
Show/Hide
|
C21H19Cl2N3O4
|
1
|
| 1 |
EC50 = 550 nM
|
|
|
|
CP0447390
|
4-[1-[4-(trifluoromethoxy)phenyl]sulfonyl-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
|
C20H15F6NO5S
|
1
|
| 1 |
EC50 = 573 nM
|
|
|
|
CP0066939
|
2-[[4-[[4-fluoro-2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C20H19F4NO3
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0471700
|
3-[[6-(4-chloropyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H16ClN3O4
|
1
|
| 1 |
EC50 = 615 nM
|
|
|
|
CP0436545
|
4'-[(6-(Phenylcarbonyl)-2-propyl-1H-benzo[d]imidazol-1-yl)methyl]biphenyl-2-carboxylic acid
Show/Hide
|
C31H26N2O3
|
1
|
| 1 |
EC50 = 620 nM
|
|
|
|
CP0479762
|
4-[1-(4-chlorophenyl)sulfonyl-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
|
C19H15ClF3NO4S
|
1
|
| 1 |
EC50 = 629 nM
|
|
|
|
CP0379862
|
2-[4-(4-anilinoanilino)-6-chloropyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C24H27ClN4O2S
|
1
|
| 1 |
EC50 = 690 nM
|
|
|
|
CP0451027
|
3-[[6-(3,6-dimethylpyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C23H21N3O4
|
1
|
| 1 |
EC50 = 717 nM
|
|
|
|
CP0126725
|
(2E)-2-[[5-phenoxy-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
|
C27H25F3O4
|
1
|
| 1 |
EC50 = 720 nM
|
|
|
|
CP0471699
|
3-[[6-(6-chloropyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H16ClN3O4
|
1
|
| 1 |
EC50 = 736 nM
|
|
|
|
CP0408699
|
3-[[1-methyl-6-(4-methylphenoxy)imidazo[4,5-c]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O4
|
1
|
| 1 |
EC50 = 746 nM
|
|
|
|
CP0376354
|
methyl 2-[4-[3-(6-acetyl-5-hydroxy-4-propylpyridin-3-yl)oxypropoxy]phenoxy]acetate
Show/Hide
|
C22H27NO7
|
1
|
| 1 |
EC50 = 757 nM
|
|
|
|
CP0436543
|
2-[4-[[6-(3-chlorophenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C30H25ClN2O2
|
1
|
| 1 |
EC50 = 770 nM
|
|
|
|
CP0487368
|
3-[[1-methyl-6-(5-methylpyridin-3-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O4
|
1
|
| 1 |
EC50 = 779 nM
|
|
|
|
CP0891654
|
4-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}benzoic acid dihydrochloride
Show/Hide
|
C24H25Cl2N3O4
|
1
|
| 1 |
EC50 = 797 nM
|
|
|
|
CP0475933
|
3-[[6-(5-fluoropyridin-2-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H16FN3O4
|
1
|
| 1 |
EC50 = 808 nM
|
|
|
|
CP0535175
|
3-[[6-(2,6-dimethylpyridin-3-yl)oxy-1,4-dimethylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C24H23N3O4
|
1
|
| 1 |
EC50 = 811 nM
|
|
|
|
CP0545584
|
2-[4-[(2-heptylbenzimidazol-1-yl)methyl]phenyl]benzamide
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C28H31N3O
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1
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| 1 |
EC50 = 840 nM
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CP0725851
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3-[(1-Methyl-6-phenoxy-1H-benzimidazol-2-yl)methoxy]benzoic acid Hydrochloride
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C22H19ClN2O4
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1
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| 1 |
EC50 = 845 nM
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CP0250829
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ethyl 2-[[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]pentanoate
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C23H26F3NO3
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1
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| 1 |
EC50 = 900 nM
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CP0476179
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4-[1-(benzenesulfonyl)-5-chloroindol-2-yl]-2,2-dimethylbutanoic acid
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C20H20ClNO4S
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1
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| 1 |
EC50 = 910 nM
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CP0297475
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2-(4-(3-(p-tolyloxy)propoxy)phenylthio)hexanoic acid
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C22H28O4S
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1
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| 1 |
EC50 = 930 nM
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CP0113761
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2-[4-[[5-(2-chlorophenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
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C30H25ClN2O2
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1
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| 1 |
EC50 = 930 nM
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CP0435485
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propyl (2E,6E)-9-[(2R)-6-hydroxy-2,8-dimethyl-3,4-dihydrochromen-2-yl]-2,6-dimethylnona-2,6-dienoate
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C25H36O4
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1
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| 1 |
EC50 = 991 nM
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CP0150577
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3-[4-[2-[6-[(E)-2-(3,5-dihydroxyphenyl)ethenyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxypropanoic acid
Show/Hide
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C28H27NO7S
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1
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| 1 |
EC50 = 1000 nM
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CP0235684
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3-[4-[2-[6-[(E)-3-(3,5-dimethoxyphenyl)prop-2-enoyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-(2,2,2-trifluoroethoxy)propanoic acid
Show/Hide
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C31H28F3NO8S
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1
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| 1 |
EC50 = 1000 nM
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CP0370107
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3-[4-[2-[6-[(E)-3-(3,5-dimethoxyphenyl)prop-2-enoyl]-2-oxo-1,3-benzothiazol-3-yl]ethoxy]phenyl]-2-ethoxypropanoic acid
Show/Hide
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C31H31NO8S
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1
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| 1 |
EC50 = 1000 nM
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CP0435499
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(2E,6E)-9-[(2R)-6-methoxy-2,8-dimethyl-3,4-dihydrochromen-2-yl]-2,6-dimethylnona-2,6-dienoic acid
Show/Hide
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C23H32O4
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1
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| 1 |
EC50 = 1000 nM
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CP0484171
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2-[2,6-dimethyl-4-[[(2Z)-3-oxo-2-[(4-phenylphenyl)methylidene]-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C34H30O6
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1
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| 1 |
EC50 = 1000 nM
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CP0161201
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2-[4-[[6-(4-methoxyphenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C31H28N2O3
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1
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| 1 |
EC50 = 1010 nM
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CP0250931
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2-[4-[[5-(4-hydroxyphenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C30H26N2O3
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1
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| 1 |
EC50 = 1010 nM
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CP0388494
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2-[4-[(2-propyl-2H-1,3-benzothiazol-3-yl)methyl]phenyl]benzoic acid
Show/Hide
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C24H23NO2S
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1
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| 1 |
EC50 = 1050 nM
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CP0480705
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2-[4-(4-anilinoanilino)-6-chloropyrimidin-2-yl]sulfanylhexanoic acid
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C22H23ClN4O2S
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1
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| 1 |
EC50 = 1060 nM
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CP0367075
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3-[[5-(4-fluorophenoxy)-3-methylimidazo[4,5-b]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
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C21H16FN3O4
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1
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| 1 |
EC50 = 1060 nM
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CP0146313
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2-[[3,4-bis(2-cyclohexylethoxy)phenyl]methyl]hexanoic acid
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C29H46O4
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1
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| 1 |
EC50 = 1100 nM
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CP0408696
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3-[(1-methyl-6-pyridin-2-yloxybenzimidazol-2-yl)methoxy]benzoic acid
Show/Hide
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C21H17N3O4
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1
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| 1 |
EC50 = 1132 nM
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CP0436542
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2-[4-[[6-(4-chlorophenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C30H25ClN2O2
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1
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| 1 |
EC50 = 1150 nM
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CP0149422
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3-[[6-(4-chloro-3-fluorophenoxy)-1-methylimidazo[4,5-c]pyridin-2-yl]methoxy]benzoic acid
Show/Hide
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C21H15ClFN3O4
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1
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| 1 |
EC50 = 1174 nM
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CP0408562
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methyl 2-[4-[3-[2-propyl-4-(trifluoromethyl)phenoxy]propoxy]phenoxy]acetate
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C22H25F3O5
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1
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| 1 |
EC50 = 1185 nM
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CP0496272
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3-[[6-(2-methoxypyridin-3-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
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C22H19N3O5
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1
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| 1 |
EC50 = 1193 nM
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CP0250750
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2-(4-(3-(3-methoxyphenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
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C22H28O5S
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1
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| 1 |
EC50 = 1200 nM
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CP0433552
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2-[4-[4-(4-aminobenzoyl)anilino]-6-chloropyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C25H27ClN4O3S
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1
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| 1 |
EC50 = 1200 nM
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CP0412245
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4-[1-(2-methoxyphenyl)sulfonyl-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
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C20H18F3NO5S
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1
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| 1 |
EC50 = 1248 nM
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CP0315236
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2-[4-[[5-(3-hydroxyphenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C30H26N2O3
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1
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| 1 |
EC50 = 1250 nM
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CP0089199
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(2E)-2-[[5-(2,2-diphenylethoxy)-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C35H33F3O4
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1
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| 1 |
EC50 = 1260 nM
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CP0395321
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methyl 2-[2-methyl-4-[3-[2-propyl-4-(trifluoromethyl)phenoxy]propoxy]phenoxy]acetate
Show/Hide
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C23H27F3O5
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1
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| 1 |
EC50 = 1261 nM
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CP0140967
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2-(4-(3-(quinolin-6-yloxy)propoxy)phenylthio)hexanoic acid
Show/Hide
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C24H27NO4S
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1
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| 1 |
EC50 = 1300 nM
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CP0147938
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2-[4-chloro-6-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C25H25ClN4O2S2
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1
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| 1 |
EC50 = 1300 nM
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CP0571518
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(E)-3-[4-[[2-[3-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-1,3-thiazol-5-yl]methylsulfanyl]phenyl]prop-2-enoic acid
Show/Hide
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C21H15F4NO2S2
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1
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| 1 |
EC50 = 1300 nM
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CP0558115
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3-[[6-(2,6-difluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
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C22H16F2N2O4
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1
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| 1 |
EC50 = 1326 nM
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CP0161197
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2-[4-[[6-(3-methoxyphenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C31H28N2O3
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1
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| 1 |
EC50 = 1350 nM
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CP0238719
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2-[4-[[6-(2-chlorophenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C30H25ClN2O2
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1
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| 1 |
EC50 = 1390 nM
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CP0158254
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ethyl 2-[[4-[(4-phenoxyphenyl)methylcarbamoyl]phenyl]methyl]butanoate
Show/Hide
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C27H29NO4
|
1
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| 1 |
EC50 = 1400 nM
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CP0271211
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3-[[6-(2-fluorophenoxy)-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
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C22H17FN2O4
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1
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| 1 |
EC50 = 1434 nM
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CP0291843
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2-[[3-(2-cyclohexylethoxy)-4-(2-phenylethoxy)phenyl]methyl]hexanoic acid
Show/Hide
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C29H40O4
|
1
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| 1 |
EC50 = 1500 nM
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CP0066946
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2-[[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]pentanoic acid
Show/Hide
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C21H22F3NO3
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1
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| 1 |
EC50 = 1500 nM
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CP0457055
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3-[1-(benzenesulfonyl)-5-chloroindol-2-yl]propanoic acid
Show/Hide
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C17H14ClNO4S
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1
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| 1 |
EC50 = 1558 nM
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CP0431821
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2-(2-methyl-4-(3-(4-propyl-6-(trifluoromethyl)pyridin-3-yloxy)propoxy)phenoxy)acetic acid
Show/Hide
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C21H24F3NO5
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1
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| 1 |
EC50 = 1582 nM
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CP0206606
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2-(4-(3-(2-methoxyphenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
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C22H28O5S
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1
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| 1 |
EC50 = 1600 nM
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CP0484170
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2-[2,6-dimethyl-4-[[(2Z)-3-oxo-2-[[4-(trifluoromethylsulfanyl)phenyl]methylidene]-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C29H25F3O6S
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1
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| 1 |
EC50 = 1630 nM
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CP0435498
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(2E,6E)-9-[(2R)-2,8-dimethyl-6-propoxy-3,4-dihydrochromen-2-yl]-2,6-dimethylnona-2,6-dienoic acid
Show/Hide
|
C25H36O4
|
1
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| 1 |
EC50 = 1692 nM
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CP0432116
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2-[2,6-dimethyl-4-[[(2Z)-2-[(4-methylsulfanylphenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C29H28O6S
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1
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| 1 |
EC50 = 1720 nM
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CP0057842
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(2E)-2-[[2,5-bis(2-phenylethoxy)phenyl]methylidene]hexanoic acid
Show/Hide
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C29H32O4
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1
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| 1 |
EC50 = 1800 nM
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CP0364417
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ethyl 2-[[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoate
Show/Hide
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C22H24F3NO3
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1
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| 1 |
EC50 = 1800 nM
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CP0041706
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2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propoxy)phenoxy)acetic acid
Show/Hide
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C22H26O7
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1
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| 1 |
EC50 = 1824 nM
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CP0432146
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2-[4-[(2-propylindol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
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C25H23NO2
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1
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| 1 |
EC50 = 1860 nM
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CP0451773
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4-[4-[(2-propylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
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C24H22N2O2
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1
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| 1 |
EC50 = 1880 nM
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CP0429955
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3-[[1-methyl-6-(6-methylpyridin-2-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
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C22H19N3O4
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1
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| 1 |
EC50 = 1895 nM
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CP0396059
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3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-chlorobenzoic acid
Show/Hide
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C25H23ClN2O4
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1
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| 1 |
EC50 = 1900 nM
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CP0388785
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1-[[2-[[[4-(trifluoromethoxy)phenyl]carbamoylamino]methyl]phenyl]methyl]pyrrole-2-carboxylic acid
Show/Hide
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C21H18F3N3O4
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1
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| 1 |
EC50 = 2000 nM
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CP0109514
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ethyl 2-phenyl-3-[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]propanoate
Show/Hide
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C26H24F3NO3
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1
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| 1 |
EC50 = 2000 nM
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CP0109516
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2-[[4-[[4-(trifluoromethoxy)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
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C20H20F3NO4
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1
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| 1 |
EC50 = 2000 nM
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CP0203852
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ethyl 2-[[4-[[4-methoxy-2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoate
Show/Hide
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C23H26F3NO4
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1
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| 1 |
EC50 = 2000 nM
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CP0190521
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(2E)-2-[[5-[(3,4-dichlorophenyl)methoxy]-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C28H25Cl2F3O4
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1
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| 1 |
EC50 = 2110 nM
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CP0177524
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(2E)-2-[[5-[[4-(trifluoromethyl)cyclohexyl]methoxy]-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C29H32F6O4
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1
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| 1 |
EC50 = 2160 nM
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CP0186990
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2-[[3,4-bis(2-phenylethoxy)phenyl]methyl]hexanoic acid
Show/Hide
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C29H34O4
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1
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| 1 |
EC50 = 2200 nM
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CP0385373
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(2E)-2-[[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methylidene]butanoic acid
Show/Hide
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C20H18F3NO3
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1
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| 1 |
EC50 = 2200 nM
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CP0256752
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2-(4-(3-(o-tolyloxy)propoxy)phenylthio)hexanoic acid
Show/Hide
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C22H28O4S
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1
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| 1 |
EC50 = 2300 nM
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CP0384537
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2-[4-chloro-6-[(5-methyl-4-phenyl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C22H25ClN4O2S2
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1
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| 1 |
EC50 = 2300 nM
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CP0433551
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2-[4-chloro-6-(4-phenoxyanilino)pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
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C24H26ClN3O3S
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1
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| 1 |
EC50 = 2360 nM
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CP0218917
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2-[[4-(2-cyclohexylethoxy)-3-(2-phenylethoxy)phenyl]methyl]hexanoic acid
Show/Hide
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C29H40O4
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1
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| 1 |
EC50 = 2500 nM
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CP0318496
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(2E)-2-[[5-(pyridin-3-ylmethoxy)-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C27H26F3NO4
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1
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| 1 |
EC50 = 2560 nM
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CP0256753
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2-(4-(3-phenoxypropoxy)-phenylthio)hexanoic acid
Show/Hide
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C21H26O4S
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1
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| 1 |
EC50 = 2600 nM
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CP0387204
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2-[3-[[2-[(4-phenylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
Show/Hide
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C28H22N2O4
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1
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| 1 |
EC50 = 2600 nM
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CP0486818
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3-[[6-(2,6-dimethylpyridin-4-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
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C23H21N3O4
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1
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| 1 |
EC50 = 2745 nM
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CP0076831
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Elafibranor
Show/Hide
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C22H24O4S
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1
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| 1 |
EC50 = 2790 nM
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CP0443575
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ethyl 2-[[4-[[4-fluoro-2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoate
Show/Hide
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C22H23F4NO3
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1
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| 1 |
EC50 = 2800 nM
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CP0384532
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2-[4-chloro-6-[[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H21ClF2N4O2S2
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1
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| 1 |
EC50 = 2900 nM
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CP0113763
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2-[4-[[6-(4-hydroxyphenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C30H26N2O3
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1
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| 1 |
EC50 = 2980 nM
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CP0379834
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3-[[2-[(4-tert-butylbenzoyl)amino]-4-methoxybenzoyl]amino]benzoic acid
Show/Hide
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C26H26N2O5
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1
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| 1 |
EC50 = 2990 nM
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CP0140963
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2-(4-(3-(m-tolyloxy)propoxy)phenylthio)hexanoic acid
Show/Hide
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C22H28O4S
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1
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| 1 |
EC50 = 3000 nM
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CP0256755
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2-(4-(3-(2,3-dimethylphenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
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C23H30O4S
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1
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| 1 |
EC50 = 3000 nM
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CP0135606
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2-(4-chloro-6-(2,3-dimethylphenylamino)pyrimidin-2-ylthio)hexanoic acid
Show/Hide
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C18H22ClN3O2S
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1
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| 1 |
EC50 = 3000 nM
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CP0109418
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2-methyl-3-[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]propanoic acid
Show/Hide
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C19H18F3NO3
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1
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| 1 |
EC50 = 3000 nM
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CP0234900
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ethyl 2-[[4-[[4-(trifluoromethoxy)phenyl]methylcarbamoyl]phenyl]methyl]butanoate
Show/Hide
|
C22H24F3NO4
|
1
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| 1 |
EC50 = 3000 nM
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CP0250830
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2-phenyl-3-[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]propanoic acid
Show/Hide
|
C24H20F3NO3
|
1
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| 1 |
EC50 = 3000 nM
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CP0512465
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2-[4-[(2-hexylbenzimidazol-1-yl)methyl]phenyl]benzamide
Show/Hide
|
C27H29N3O
|
1
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| 1 |
EC50 = 3060 nM
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CP0390345
|
2-[4-[(2-propylbenzimidazol-1-yl)methyl]phenyl]benzamide
Show/Hide
|
C24H23N3O
|
1
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| 1 |
EC50 = 3150 nM
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CP0247155
|
2-[3,5-bis(2-phenylethoxy)phenyl]sulfanylhexanoic acid
Show/Hide
|
C28H32O4S
|
1
|
| 1 |
EC50 = 3400 nM
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CP0400354
|
2-[4-chloro-6-[[4-(4-nitrophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H22ClN5O4S2
|
1
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| 1 |
EC50 = 3400 nM
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CP0431418
|
2-(4-(3-(3,4-dimethylphenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
|
C23H30O4S
|
1
|
| 1 |
EC50 = 3500 nM
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CP0363438
|
ethyl 2-[[4-[[2-(trifluoromethoxy)phenyl]methylcarbamoyl]phenyl]methyl]butanoate
Show/Hide
|
C22H24F3NO4
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0477611
|
4'-[(6-(Hydroxy(phenyl)methyl)-2-propyl-1H-benzo[d]imidazol-1-yl)methyl]biphenyl-2-carboxylic acid
Show/Hide
|
C31H28N2O3
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0037112
|
2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidin-2-yl}sulfanyl)octanoic acid
Show/Hide
|
C20H26ClN3O2S
|
2
|
| 1 |
EC50 = 3600 nM
|
|
|
| 2 |
IC50 = 3600 nM
|
|
|
|
CP0379172
|
2-[4-chloro-6-[[4-(2,4-difluorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H21ClF2N4O2S2
|
1
|
| 1 |
EC50 = 3600 nM
|
|
|
|
CP0116868
|
2-(4,6-Diphenethoxypyrimidin-2-ylthio)acetic acid
Show/Hide
|
C22H22N2O4S
|
2
|
| 1 |
EC50 = 3700 nM
|
|
|
| 2 |
IC50 = 3700 nM
|
|
|
|
CP0086197
|
2-[[2,3-bis(2-phenylethoxy)phenyl]methyl]hexanoic acid
Show/Hide
|
C29H34O4
|
1
|
| 1 |
EC50 = 3700 nM
|
|
|
|
CP0379171
|
2-[4-chloro-6-[(7-methoxy-4,5-dihydrobenzo[e][1,3]benzothiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C24H27ClN4O3S2
|
1
|
| 1 |
EC50 = 3700 nM
|
|
|
|
CP0126697
|
(2E)-2-[[5-[[4-(2-morpholin-4-ylethoxy)phenyl]methoxy]-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
|
C34H38F3NO6
|
1
|
| 1 |
EC50 = 3770 nM
|
|
|
|
CP0241890
|
2-(4-(3-(2,3-dimethylphenoxy)propoxy)phenylthio)acetic acid
Show/Hide
|
C19H22O4S
|
1
|
| 1 |
EC50 = 3800 nM
|
|
|
|
CP0384541
|
2-[4-[[4-(4-bromophenyl)-5-methyl-1,3-thiazol-2-yl]amino]-6-chloropyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C22H24BrClN4O2S2
|
1
|
| 1 |
EC50 = 3800 nM
|
|
|
|
CP0256754
|
(R)-2-(4-(3-(2,3-dimethylphenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
|
C23H30O4S
|
1
|
| 1 |
EC50 = 3900 nM
|
|
|
|
CP0384539
|
2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanylbutanoic acid
Show/Hide
|
C17H14Cl2N4O2S2
|
1
|
| 1 |
EC50 = 3900 nM
|
|
|
|
CP0477280
|
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]benzoic acid
Show/Hide
|
C25H24N2O4
|
1
|
| 1 |
EC50 = 3900 nM
|
|
|
|
CP0432147
|
2-[4-[(2-pentylbenzimidazol-1-yl)methyl]phenyl]benzamide
Show/Hide
|
C26H27N3O
|
1
|
| 1 |
EC50 = 3900 nM
|
|
|
|
CP0353436
|
2-[[4-[(4-chlorophenyl)methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C19H20ClNO3
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0360414
|
2-[[4-[(2-methylphenyl)methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C20H23NO3
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0214970
|
2-[4-[[6-(3-hydroxyphenyl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C30H26N2O3
|
1
|
| 1 |
EC50 = 4090 nM
|
|
|
|
CP0140962
|
2-(4-(3-(2-isopropylphenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
|
C24H32O4S
|
1
|
| 1 |
EC50 = 4100 nM
|
|
|
|
CP0415361
|
2-[4-chloro-6-[[4-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C25H29ClN4O2S2
|
1
|
| 1 |
EC50 = 4100 nM
|
|
|
|
CP0249320
|
4'-[(2-Propyl-1H-benzo[d]imidazol-1-yl)methyl]biphenyl-2-carboxylic acid
Show/Hide
|
C24H22N2O2
|
3
|
| 1 |
EC50 = 4170 nM
|
|
|
| 2 |
EC50 = 6440 nM
|
|
|
| 3 |
EC50 = 7220 nM
|
|
|
|
CP0273341
|
2-(4-(3-(2,3-dimethylphenoxy)propoxy)benzyl)hexanoic acid
Show/Hide
|
C24H32O4
|
1
|
| 1 |
EC50 = 4200 nM
|
|
|
|
CP0223549
|
ethyl 2-[[4-[[4-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoate
Show/Hide
|
C22H24F3NO3
|
1
|
| 1 |
EC50 = 4200 nM
|
|
|
|
CP0444072
|
2-[2,6-dimethyl-4-[[(2Z)-3-oxo-2-[[4-(trifluoromethyl)phenyl]methylidene]-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C29H25F3O6
|
1
|
| 1 |
EC50 = 4220 nM
|
|
|
|
CP0083167
|
4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidazol)-1'-yl)methyl)-(1,1'-biphenyl)-2-carboxylic acid
Show/Hide
|
C33H30N4O2
|
3
|
| 1 |
EC50 = 4280 nM
|
|
|
| 2 |
EC50 = 4710 nM
|
|
|
| 3 |
EC50 = 4970 nM
|
|
|
|
CP0116866
|
2-(4,6-Bis(2-cyclopropylethoxy)pyrimidin-2-ylthio)hexanoic acid
Show/Hide
|
C20H30N2O4S
|
1
|
| 1 |
EC50 = 4300 nM
|
|
|
|
CP0396062
|
2-[3-[[2-[[4-(trifluoromethylsulfanyl)benzoyl]amino]benzoyl]amino]phenyl]acetic acid
Show/Hide
|
C23H17F3N2O4S
|
1
|
| 1 |
EC50 = 4400 nM
|
|
|
|
CP0399542
|
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methoxybenzoic acid
Show/Hide
|
C26H26N2O5
|
1
|
| 1 |
EC50 = 4400 nM
|
|
|
|
CP0447701
|
2-(4-chloro-6-(2,3-dimethylphenylamino)pyrimidin-2-ylthio)-2-(4-phenylnaphthalen-1-yl)acetic acid
Show/Hide
|
C30H24ClN3O2S
|
1
|
| 1 |
EC50 = 4500 nM
|
|
|
|
CP0379832
|
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-methoxybenzoic acid
Show/Hide
|
C26H26N2O5
|
1
|
| 1 |
EC50 = 4500 nM
|
|
|
|
CP0387232
|
3-[[2-[(4-bromobenzoyl)amino]benzoyl]amino]benzoic acid
Show/Hide
|
C21H15BrN2O4
|
1
|
| 1 |
EC50 = 4500 nM
|
|
|
|
CP0185952
|
2-(4-(3-(3-(trifluoromethyl)phenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
|
C22H25F3O4S
|
1
|
| 1 |
EC50 = 4600 nM
|
|
|
|
CP0248018
|
(2E)-2-[[5-[[3,5-bis(trifluoromethyl)phenyl]methoxy]-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
|
C30H25F9O4
|
1
|
| 1 |
EC50 = 4640 nM
|
|
|
|
CP0086195
|
2-[[3,5-bis(2-phenylethoxy)phenyl]methyl]hexanoic acid
Show/Hide
|
C29H34O4
|
1
|
| 1 |
EC50 = 4700 nM
|
|
|
|
CP0388903
|
3-[[5-chloro-2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
Show/Hide
|
C22H14ClF3N2O4
|
1
|
| 1 |
EC50 = 4700 nM
|
|
|
|
CP0179682
|
2-[3,5-bis(2-phenylethoxy)phenoxy]hexanoic acid
Show/Hide
|
C28H32O5
|
1
|
| 1 |
EC50 = 4800 nM
|
|
|
|
CP0203849
|
2-[[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C20H20F3NO3
|
1
|
| 1 |
EC50 = 4800 nM
|
|
|
|
CP0387199
|
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methylbenzoic acid
Show/Hide
|
C26H26N2O4
|
1
|
| 1 |
EC50 = 5000 nM
|
|
|
|
CP0387200
|
3-[3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]phenyl]propanoic acid
Show/Hide
|
C27H28N2O4
|
1
|
| 1 |
EC50 = 5000 nM
|
|
|
|
CP0446094
|
2-[4-[(2-propylbenzimidazol-1-yl)methyl]phenyl]benzonitrile
Show/Hide
|
C24H21N3
|
1
|
| 1 |
EC50 = 5010 nM
|
|
|
|
CP0069348
|
(2E)-2-[[5-[(4-fluorophenyl)methoxy]-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
|
C28H26F4O4
|
1
|
| 1 |
EC50 = 5170 nM
|
|
|
|
CP0486453
|
(E)-3-[4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylamino]phenyl]prop-2-enoic acid
Show/Hide
|
C21H17F3N2O2S
|
1
|
| 1 |
EC50 = 5280 nM
|
|
|
|
CP0241891
|
2-(4-(3-(3-isopropylphenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
|
C24H32O4S
|
1
|
| 1 |
EC50 = 5300 nM
|
|
|
|
CP0379835
|
3-[[2-[(4-tert-butylbenzoyl)amino]-5-chlorobenzoyl]amino]benzoic acid
Show/Hide
|
C25H23ClN2O4
|
1
|
| 1 |
EC50 = 5400 nM
|
|
|
|
CP0388902
|
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-chlorobenzoic acid
Show/Hide
|
C25H23ClN2O4
|
1
|
| 1 |
EC50 = 5400 nM
|
|
|
|
CP0387227
|
3-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]benzoic acid
Show/Hide
|
C25H18N2O4
|
1
|
| 1 |
EC50 = 5500 nM
|
|
|
|
CP0400356
|
2-[4-chloro-6-[(4-phenyl-1,3-thiazol-2-yl)amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H23ClN4O2S2
|
1
|
| 1 |
EC50 = 5700 nM
|
|
|
|
CP0379833
|
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-fluorobenzoic acid
Show/Hide
|
C25H23FN2O4
|
1
|
| 1 |
EC50 = 5800 nM
|
|
|
|
CP0480047
|
3-[[6-(2-chloropyridin-4-yl)oxy-1-methylbenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C21H16ClN3O4
|
1
|
| 1 |
EC50 = 5947 nM
|
|
|
|
CP0514762
|
3-[[1-methyl-6-(2-methylpyridin-4-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
|
C22H19N3O4
|
1
|
| 1 |
EC50 = 5947 nM
|
|
|
|
CP0256577
|
1-[[2-[(1-adamantylcarbamoylamino)methyl]phenyl]methyl]pyrrole-2-carboxylic acid
Show/Hide
|
C24H29N3O3
|
1
|
| 1 |
EC50 = 6000 nM
|
|
|
|
CP0852617
|
2-{[6-(4-Amino-3,5-dimethylphenoxy)-1-methyl-1Hbenzimidazol-2-yl]methoxy}benzoic acid dihydrochloride
Show/Hide
|
C24H25Cl2N3O4
|
1
|
| 1 |
EC50 = 6094 nM
|
|
|
|
CP0096106
|
2-(4,6-Diphenethoxypyrimidin-2-ylthio)butanoic acid
Show/Hide
|
C24H26N2O4S
|
1
|
| 1 |
EC50 = 6100 nM
|
|
|
|
CP0266724
|
2-(4-chloro-6-(2,3-dimethylphenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C24H20ClN3O2S
|
2
|
| 1 |
EC50 = 6200 nM
|
|
|
| 2 |
IC50 = 6200 nM
|
|
|
|
CP0419731
|
2-[3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
Show/Hide
|
C26H26N2O4
|
1
|
| 1 |
EC50 = 6200 nM
|
|
|
|
CP0512466
|
3-[4-[(2-propylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
|
C24H22N2O2
|
1
|
| 1 |
EC50 = 6240 nM
|
|
|
|
CP0396060
|
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-methylbenzoic acid
Show/Hide
|
C26H26N2O4
|
1
|
| 1 |
EC50 = 6300 nM
|
|
|
|
CP0398725
|
2-bromo-5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]benzoic acid
Show/Hide
|
C25H23BrN2O4
|
1
|
| 1 |
EC50 = 6300 nM
|
|
|
|
CP0234899
|
2-[[4-[[4-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C20H20F3NO3
|
1
|
| 1 |
EC50 = 6300 nM
|
|
|
|
CP0450948
|
2-[2,6-dimethyl-4-[[(2Z)-3-oxo-2-[[4-(trifluoromethoxy)phenyl]methylidene]-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C29H25F3O7
|
1
|
| 1 |
EC50 = 6360 nM
|
|
|
|
CP0474289
|
2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C21H22Cl2N4O2S2
|
1
|
| 1 |
EC50 = 6400 nM
|
|
|
|
CP0066945
|
2-[[3-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C20H20F3NO3
|
1
|
| 1 |
EC50 = 6400 nM
|
|
|
|
CP0042526
|
2-(4,6-Bis(2-cyclohexylethoxy)pyrimidin-2-ylthio)hexanoic acid
Show/Hide
|
C26H42N2O4S
|
1
|
| 1 |
EC50 = 6600 nM
|
|
|
|
CP0267796
|
2-(4-chloro-6-(2,3-dihydro-1H-inden-5-ylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C25H20ClN3O2S
|
1
|
| 1 |
EC50 = 6800 nM
|
|
|
|
CP0425684
|
3-[(1-methyl-6-pyridin-3-yloxybenzimidazol-2-yl)methoxy]benzoic acid
Show/Hide
|
C21H17N3O4
|
1
|
| 1 |
EC50 = 6831 nM
|
|
|
|
CP0245202
|
2-(4-chloro-6-(naphthalen-2-ylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C26H18ClN3O2S
|
1
|
| 1 |
EC50 = 6900 nM
|
|
|
|
CP0387068
|
3-[[2-[[3-fluoro-4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
Show/Hide
|
C22H14F4N2O4
|
1
|
| 1 |
EC50 = 6900 nM
|
|
|
|
CP0398732
|
3-[3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]phenyl]propanoic acid
Show/Hide
|
C24H19F3N2O4
|
1
|
| 1 |
EC50 = 6900 nM
|
|
|
|
CP0145378
|
2-(4,6-Bis(4-cyanophenethoxy)pyrimidin-2-ylthio)hexanoic acid
Show/Hide
|
C28H28N4O4S
|
1
|
| 1 |
EC50 = 7000 nM
|
|
|
|
CP0175041
|
2-[[4-[(4-methoxyphenyl)methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C20H23NO4
|
1
|
| 1 |
EC50 = 7000 nM
|
|
|
|
CP0120615
|
(2E)-2-[[2,5-bis[2-[4-(trifluoromethyl)phenyl]ethoxy]phenyl]methylidene]hexanoic acid
Show/Hide
|
C31H30F6O4
|
1
|
| 1 |
EC50 = 7200 nM
|
|
|
|
CP0415500
|
2-[4-chloro-6-[[4-(4-methylphenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanyloctanoic acid
Show/Hide
|
C22H25ClN4O2S2
|
1
|
| 1 |
EC50 = 7200 nM
|
|
|
|
CP0289446
|
2-(4-chloro-6-(3-chlorophenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C22H15Cl2N3O2S
|
1
|
| 1 |
EC50 = 7300 nM
|
|
|
|
CP0096107
|
2-(4,6-Bis(4-methylphenethoxy)pyrimidin-2-ylthio)-hexanoic acid
Show/Hide
|
C28H34N2O4S
|
1
|
| 1 |
EC50 = 7500 nM
|
|
|
|
CP0218346
|
2-(4-chloro-6-(4-isopropylphenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C25H22ClN3O2S
|
1
|
| 1 |
EC50 = 7600 nM
|
|
|
|
CP0400697
|
2-[4-chloro-6-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]pyrimidin-2-yl]sulfanylhexanoic acid
Show/Hide
|
C19H18Cl2N4O2S2
|
1
|
| 1 |
EC50 = 7600 nM
|
|
|
|
CP0140961
|
2-(4-(3-(4-chloro-3-(trifluoromethyl)phenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
|
C22H24ClF3O4S
|
1
|
| 1 |
EC50 = 7800 nM
|
|
|
|
CP0225016
|
2-(4-chloro-6-(3,4-dimethylphenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
|
C24H20ClN3O2S
|
1
|
| 1 |
EC50 = 7800 nM
|
|
|
|
CP0120616
|
(2E)-2-[[3,5-bis(2-phenylethoxy)phenyl]methylidene]hexanoic acid
Show/Hide
|
C29H32O4
|
1
|
| 1 |
EC50 = 7800 nM
|
|
|
|
CP0385045
|
ethyl 2-methyl-3-[4-[[2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]propanoate
Show/Hide
|
C21H22F3NO3
|
1
|
| 1 |
EC50 = 8000 nM
|
|
|
|
CP0455454
|
2-[[4-[[2-(trifluoromethoxy)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid
Show/Hide
|
C20H20F3NO4
|
1
|
| 1 |
EC50 = 8000 nM
|
|
|
|
CP0464441
|
2-[4-[(2-propylindol-1-yl)methyl]phenyl]benzonitrile
Show/Hide
|
C25H22N2
|
1
|
| 1 |
EC50 = 8030 nM
|
|
|
|
CP0217019
|
2-(4-(3-(5,6,7,8-tetrahydronaphthalen-1-yloxy)propoxy)phenylthio)hexanoic acid
Show/Hide
|
C25H32O4S
|
1
|
| 1 |
EC50 = 8100 nM
|
|
|
|
CP0476578
|
2-[4-[(4-bromo-2-propylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
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C24H21BrN2O2
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1
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| 1 |
EC50 = 8250 nM
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CP0146439
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2-(4,6-Diphenethoxypyrimidin-2-ylthio)hexanoic acid
Show/Hide
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C26H30N2O4S
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1
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| 1 |
EC50 = 8300 nM
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CP0387067
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3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
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C22H15F3N2O4
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1
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| 1 |
EC50 = 8500 nM
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CP0421689
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2-[4-[(4-fluoro-2-propylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
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C24H21FN2O2
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1
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| 1 |
EC50 = 8660 nM
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CP0476576
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2-[4-[(4-chloro-2-propylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
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C24H21ClN2O2
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1
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| 1 |
EC50 = 8670 nM
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CP0396063
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3-[[4-chloro-2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
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C22H14ClF3N2O4
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1
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| 1 |
EC50 = 8700 nM
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CP0046254
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2-(4,6-diphenethoxypyrimidin-2-ylthio)octanoic acid
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C28H34N2O4S
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1
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| 1 |
EC50 = 8800 nM
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CP0164700
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2-(4-chloro-6-(isopentylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
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C21H22ClN3O2S
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1
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| 1 |
EC50 = 8900 nM
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CP0261620
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2-(4-chloro-6-(3-phenylpropylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
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C25H22ClN3O2S
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1
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| 1 |
EC50 = 8900 nM
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CP0110708
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2-(4,6-Bis(3-phenylpropoxy)pyrimidin-2-ylthio)hexanoic acid
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C28H34N2O4S
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1
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| 1 |
EC50 = 8900 nM
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CP0267779
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2-(4-chloro-6-(4-chlorophenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
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C22H15Cl2N3O2S
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1
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| 1 |
EC50 = 9000 nM
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CP0387230
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3-[[2-[(4-tert-butylbenzoyl)amino]-4-chlorobenzoyl]amino]benzoic acid
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C25H23ClN2O4
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1
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| 1 |
EC50 = 9000 nM
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CP0445061
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2-[3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]phenyl]acetic acid
Show/Hide
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C23H17F3N2O4
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1
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| 1 |
EC50 = 9400 nM
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CP0060839
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2-[4-[[2-[3-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-1,3-thiazol-5-yl]methylsulfanyl]-2-methylphenoxy]acetic acid
Show/Hide
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C21H17F4NO3S2
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1
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| 1 |
EC50 = 9530 nM
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CP0252121
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(S)-2-(4-(3-(2,3-dimethylphenoxy)propoxy)phenylthio)hexanoic acid
Show/Hide
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C23H30O4S
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1
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| 1 |
EC50 = 9900 nM
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CP0039118
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2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy}acetic acid
Show/Hide
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C21H18F3NO3S2
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1
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| 1 |
EC50 = 10000 nM
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CP0232805
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2-(4,6-Bis(4-phenylbutoxy)pyrimidin-2-ylthio)hexanoic acid
Show/Hide
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C30H38N2O4S
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1
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| 1 |
EC50 = 10000 nM
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CP0486812
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3-[[1-methyl-6-(4-methylpyridin-3-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
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C22H19N3O4
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1
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| 1 |
EC50 > 10000 nM
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CP0514761
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3-[[1-methyl-6-(2-methylpyridin-3-yl)oxybenzimidazol-2-yl]methoxy]benzoic acid
Show/Hide
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C22H19N3O4
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1
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| 1 |
EC50 > 10000 nM
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CP0444071
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2-[4-[[(2Z)-2-[(4-ethoxyphenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxymethyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
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C30H30O7
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1
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| 1 |
EC50 > 10000 nM
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CP0450947
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2-[4-[[(2Z)-2-[(4-fluorophenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxymethyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
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C28H25FO6
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1
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| 1 |
EC50 > 10000 nM
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CP0520738
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2-[4-[[(2Z)-2-benzylidene-3-oxo-1-benzofuran-6-yl]oxymethyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
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C28H26O6
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1
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| 1 |
EC50 > 10000 nM
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CP0558901
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2-[2,6-dimethyl-4-[[(2Z)-3-oxo-2-[[2-(trifluoromethyl)phenyl]methylidene]-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C29H25F3O6
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1
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| 1 |
EC50 > 10000 nM
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CP0558902
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2-[2,6-dimethyl-4-[[(2Z)-2-(naphthalen-2-ylmethylidene)-3-oxo-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C32H28O6
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1
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| 1 |
EC50 > 10000 nM
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CP0559505
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2-[4-[[(2Z)-2-[(4-chlorophenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxymethyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
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C28H25ClO6
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1
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| 1 |
EC50 > 10000 nM
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CP0559506
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2-[4-[[(2Z)-2-[(4-bromophenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxymethyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
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C28H25BrO6
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1
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| 1 |
EC50 > 10000 nM
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CP0559507
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2-[4-[[(2Z)-2-[(4-cyanophenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxymethyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
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C29H25NO6
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1
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| 1 |
EC50 > 10000 nM
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CP0559509
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2-[4-[[(2Z)-2-[(4-methoxyphenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxymethyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
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C29H28O7
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1
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| 1 |
EC50 > 10000 nM
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CP0568632
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2-[2,6-dimethyl-4-[[(2Z)-3-oxo-2-[(4-propan-2-ylphenyl)methylidene]-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C31H32O6
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1
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| 1 |
EC50 > 10000 nM
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CP0568976
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2-[2,6-dimethyl-4-[[(2Z)-2-[(4-methylphenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxymethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C29H28O6
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1
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| 1 |
EC50 > 10000 nM
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CP0116848
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2-(4,6-Bis(4-(trifluoromethoxy)phenethoxy)pyrimidin-2-ylthio)hexanoic acid
Show/Hide
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C28H28F6N2O6S
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1
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| 1 |
EC50 = 10300 nM
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CP0093185
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(S)-2-(4,6-diphenethoxypyrimidin-2-ylthio)hexanoic acid
Show/Hide
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C26H30N2O4S
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1
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| 1 |
EC50 = 10400 nM
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CP0240939
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2-(4-chloro-6-(phenethylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
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C24H20ClN3O2S
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1
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| 1 |
EC50 = 10800 nM
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CP0169316
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2-[[2,5-bis(2-phenylethoxy)phenyl]methyl]hexanoic acid
Show/Hide
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C29H34O4
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1
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| 1 |
EC50 = 10800 nM
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CP0036764
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2-(4,6-Bis(isopentyloxy)pyrimidin-2-ylthio)hexanoic acid
Show/Hide
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C20H34N2O4S
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1
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| 1 |
EC50 = 11000 nM
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CP0147349
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2-(4,6-Bis(4-(trifluoromethyl)phenethoxy)pyrimidin-2-ylthio)-hexanoic Acid
Show/Hide
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C28H28F6N2O4S
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1
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| 1 |
EC50 = 11000 nM
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CP0451729
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3-[[2-[[3,5-bis(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
Show/Hide
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C23H14F6N2O4
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1
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| 1 |
EC50 = 11000 nM
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CP0363439
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ethyl 2-[[4-[(4-fluorophenyl)methylcarbamoyl]phenyl]methyl]butanoate
Show/Hide
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C21H24FNO3
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1
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| 1 |
EC50 = 11000 nM
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CP0390346
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2-[4-[(4-methyl-2-propylbenzimidazol-1-yl)methyl]phenyl]benzoic acid
Show/Hide
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C25H24N2O2
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1
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| 1 |
EC50 = 11100 nM
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CP0116223
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(2E)-2-[[5-phenylmethoxy-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C28H27F3O4
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1
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| 1 |
EC50 = 11700 nM
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CP0093184
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2-(4,6-Bis(2-cyclopentylethoxy)pyrimidin-2-ylthio)hexanoic acid
Show/Hide
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C24H38N2O4S
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1
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| 1 |
EC50 = 12100 nM
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CP0390347
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2-[4-[[2-propyl-4-(trifluoromethyl)benzimidazol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C25H21F3N2O2
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1
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| 1 |
EC50 = 12100 nM
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CP0473978
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2-[4-(4-anilinoanilino)-6-chloropyrimidin-2-yl]sulfanylacetic acid
Show/Hide
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C18H15ClN4O2S
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1
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| 1 |
EC50 = 12400 nM
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CP0862665
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Methyl 3-[(3-methyl-5-phenoxy-3H-imidazo[4,5-b]pyridin-2-yl)methoxy]benzoate Dihydrochloride
Show/Hide
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C22H21Cl2N3O4
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1
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| 1 |
EC50 = 12400 nM
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CP0053214
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(2E)-2-[[5-[(E)-3-phenylprop-2-enoxy]-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C30H29F3O4
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1
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| 1 |
EC50 = 12900 nM
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CP0267797
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2-(4-chloro-6-(4-fluorophenylamino)pyrimidin-2-ylthio)-2-(naphthalen-1-yl)acetic acid
Show/Hide
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C22H15ClFN3O2S
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1
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| 1 |
EC50 = 13000 nM
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CP0417149
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4-[[2-[(4-phenylbenzoyl)amino]benzoyl]amino]butanoic acid
Show/Hide
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C24H22N2O4
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1
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| 1 |
EC50 = 13000 nM
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CP0528133
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(E)-3-[4-[[2-[3-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-1,3-thiazol-5-yl]methoxy]phenyl]prop-2-enoic acid
Show/Hide
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C21H15F4NO3S
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1
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| 1 |
EC50 = 13200 nM
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CP0379495
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3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methylbenzoic acid
Show/Hide
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C26H26N2O4
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1
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| 1 |
EC50 = 13500 nM
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CP0360413
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2-[[4-(benzylcarbamoyl)phenyl]methyl]butanoic acid
Show/Hide
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C19H21NO3
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1
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| 1 |
EC50 = 13500 nM
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CP0140959
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3-(4-(3-(2,3-dimethylphenoxy)propoxy)phenyl)propanoic acid
Show/Hide
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C20H24O4
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1
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| 1 |
EC50 = 15700 nM
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CP0066948
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ethyl 2-[[4-(benzylcarbamoyl)phenyl]methyl]butanoate
Show/Hide
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C21H25NO3
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1
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| 1 |
EC50 = 16000 nM
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CP0488748
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(E)-3-[4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylsulfanyl]phenyl]prop-2-enoic acid
Show/Hide
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C21H16F3NO2S2
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1
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| 1 |
EC50 = 17000 nM
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CP0387203
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2-[3-[[2-[(4-methylsulfanylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
Show/Hide
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C23H20N2O4S
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1
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| 1 |
EC50 = 17400 nM
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CP0387205
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2-[3-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]phenyl]acetic acid
Show/Hide
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C26H20N2O4
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1
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| 1 |
EC50 = 18000 nM
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CP0385188
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4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]butanoic acid
Show/Hide
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C22H20N2O4
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1
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| 1 |
EC50 = 18100 nM
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CP0403496
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4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]benzoic acid
Show/Hide
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C25H18N2O4
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1
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| 1 |
EC50 = 21000 nM
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CP0417147
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4-[[2-[(2-phenylbenzoyl)amino]benzoyl]amino]butanoic acid
Show/Hide
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C24H22N2O4
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1
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| 1 |
EC50 = 23000 nM
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CP0540303
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(E)-3-[4-[methyl-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methyl]amino]phenyl]prop-2-enoic acid
Show/Hide
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C22H19F3N2O2S
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1
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| 1 |
EC50 = 24700 nM
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CP0398523
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3-[[2-(1,3-benzodioxole-5-carbonylamino)benzoyl]amino]benzoic acid
Show/Hide
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C22H16N2O6
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1
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| 1 |
EC50 = 25000 nM
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CP0403351
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5-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]pentanoic acid
Show/Hide
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C23H22N2O4
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1
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| 1 |
EC50 = 26000 nM
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CP0387072
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4-[[2-[(3-phenylbenzoyl)amino]benzoyl]amino]butanoic acid
Show/Hide
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C24H22N2O4
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1
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| 1 |
EC50 = 37000 nM
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CP0445072
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4-[[2-(naphthalene-1-carbonylamino)benzoyl]amino]butanoic acid
Show/Hide
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C22H20N2O4
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1
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| 1 |
EC50 = 41000 nM
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CP0012720
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2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidin-2-yl}sulfanyl)acetic acid
Show/Hide
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C14H14ClN3O2S
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2
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| 1 |
EC50 = 53700 nM
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| 2 |
IC50 = 53700 nM
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CP0014077
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2,2-Dimethyl-5-(2,5-dimethylphenoxy)valeriansaeure
Show/Hide
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C15H22O3
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1
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| 1 |
EC50 = 68400 nM
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CP0916464
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(Z)-5-(4-(3-(Piperidin-1-yl)propoxy)benzylidene)-2-thioxothiazolidin-4-one
Show/Hide
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C18H22N2O2S2
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1
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| 1 |
EC50 > 100000 nM
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CP0412244
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4-[1-(3H-benzimidazol-5-ylsulfonyl)-5-chloroindol-2-yl]butanoic acid
Show/Hide
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C19H16ClN3O4S
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1
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| 1 |
EC50 > 5000 nM
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CP0458600
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4-[1-(2-chlorophenyl)sulfonyl-5-(trifluoromethyl)indol-2-yl]butanoic acid
Show/Hide
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C19H15ClF3NO4S
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1
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| 1 |
EC50 > 5000 nM
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CP0230610
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2-(4-Chloro-6-(4'-cyanobiphenyl-4-ylamino)pyrimidin-2-ylthio)octanoic acid
Show/Hide
|
C25H25ClN4O2S
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1
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| 1 |
IC50 = 1500 nM
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CP0035851
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2-{[4-chloro-6-(quinolin-6-ylamino)pyrimidin-2-yl]sulfanyl}octanoic acid
Show/Hide
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C21H23ClN4O2S
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1
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| 1 |
IC50 = 3500 nM
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