N-pyrimidin-2-yl-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-pyridin-2-yl-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

5-methyl-4-(1H-pyrazol-4-yl)-N-pyridin-2-yl-1,3-thiazol-2-amine

N-[3-chloro-4-[(2-chlorophenyl)sulfamoyl]phenyl]pyridine-2-carboxamide

N-(4-methylpyrimidin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

4-(5-methyl-1H-pyrazol-4-yl)-N-pyridin-2-yl-1,3-thiazol-2-amine

N-pyrimidin-2-yl-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

N-(4-methoxypyrimidin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-(6-fluoropyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-(6-methylpyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

[4-(1-phenylpyrazol-4-yl)quinolin-7-yl] piperidine-1-carboxylate

N-pyridin-2-yl-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

4-(1-phenylpyrazol-4-yl)quinoline

7-methoxy-4-(1-phenylpyrazol-4-yl)quinoline

N-(4-chloro-3-methoxyphenyl)pyridine-2-carboxamide

7-(3-methoxypropoxy)-4-(1-phenylpyrazol-4-yl)quinoline

N-(6-ethoxypyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

6-N,6-N-dimethyl-2-N-(5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-yl)pyridine-2,6-diamine

N-[6-(2-methoxyethoxy)pyridin-2-yl]-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

[4-(1-phenylpyrazol-4-yl)quinolin-7-yl] N,N-diethylcarbamate

7-(2-methoxyethoxy)-4-(1-phenylpyrazol-4-yl)quinoline

4-(1H-pyrazol-4-yl)-N-pyridin-2-yl-1,3-thiazol-2-amine

4-(3-methyl-1-phenylpyrazol-4-yl)quinoline

[4-(1-phenylpyrazol-4-yl)quinolin-7-yl] pyrrolidine-1-carboxylate

7-ethoxy-4-(1-phenylpyrazol-4-yl)quinoline

4-(1-phenylpyrazol-4-yl)-7-(trifluoromethyl)quinoline

7-chloro-4-(1-phenylpyrazol-4-yl)quinoline

2-N-ethyl-6-N-(5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-yl)pyridine-2,6-diamine

7-phenylmethoxy-4-(1-phenylpyrazol-4-yl)quinoline

N-(6-methoxypyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

4-(5-methyl-1-phenylpyrazol-4-yl)quinoline

1-[4-[2-[4-(1-phenylpyrazol-4-yl)quinolin-7-yl]oxyethyl]piperazin-1-yl]ethanone

7-fluoro-4-(1-phenylpyrazol-4-yl)quinoline

(1R,2S)-2-[(3,5-dichlorophenyl)carbamoyl]cyclohexane-1-carboxylic acid

N-(5-fluoropyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

4-(3,5-dimethyl-1-phenylpyrazol-4-yl)quinoline

[4-(1-phenylpyrazol-4-yl)quinolin-7-yl] morpholine-4-carboxylate

N-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

[4-(1-phenylpyrazol-4-yl)quinolin-7-yl] N,N-dimethylcarbamate

4-((E)-styryl)-pyrimidin-2-ylamine

N-(6-chloropyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

4-[1-(2-fluorophenyl)pyrazol-4-yl]quinoline

2,3-dimethyl-4-(1-phenylpyrazol-4-yl)pyridine

N-pyrimidin-4-yl-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-cyclohexyl-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

4-((2-(3-methylquinoxalin-2-yl)hydrazono)methyl)phenol

4-[2-[4-(1-phenylpyrazol-4-yl)quinolin-7-yl]oxyethyl]morpholine

4-(1-pyridin-2-ylpyrazol-4-yl)quinoline

N-phenyl-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

4-(1-phenylpyrazol-4-yl)-6,7-dihydro-5H-cyclopenta[b]pyridine

N-(5-methyl-1H-pyrazol-3-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

3-(1-phenylpyrazol-4-yl)-1H-indazole

3-(1-phenylpyrazol-4-yl)-1H-indole

[6-(5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-ylamino)pyridin-2-yl]methanol

4-(1-phenylpyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine

4-[3-[4-(1-phenylpyrazol-4-yl)quinolin-7-yl]oxypropyl]morpholine

4-[1-(4-fluorophenyl)pyrazol-4-yl]quinoline

2-(1-phenylethyl)-3-p-tolyl-2,3-dihydroquinazolin-4(1H)-one

N-(1-methylpyrazol-3-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

(1aS,7E,7aS)-7-hydroxyimino-N-phenyl-1,7a-dihydrocyclopropa[b]chromene-1a-carboxamide

4-[1-(3-fluorophenyl)pyrazol-4-yl]quinoline

N-(1H-pyrazol-5-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-(3-methylpyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

4-(1-phenylpyrazol-4-yl)quinazoline

4-(1-thiophen-2-ylpyrazol-4-yl)quinoline

1-(3,5-dimethylphenyl)-4-(3-methylpiperidin-1-yl)pyrazolo[3,4-d]pyrimidine

6-(5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-ylamino)pyridine-2-carbonitrile

3-methyl-4-(1-phenylpyrazol-4-yl)pyridine

4-(1-phenylpyrazol-4-yl)-7-(2-piperidin-1-ylethoxy)quinoline

N-(6-methylpyridazin-3-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-pyridin-3-yl-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

5-methyl-4-(5-methyl-1H-pyrazol-4-yl)-N-pyridin-2-yl-1,3-thiazol-2-amine

N-pyrazin-2-yl-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-pyridin-3-yl-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-(4,6-dimethylpyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-(5-methylpyridin-2-yl)-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

N-(6-pyrrolidin-1-ylpyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

methyl 6-(5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-ylamino)pyridine-2-carboxylate

N-(4-methylpyridin-2-yl)-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

N-pyridin-4-yl-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

N-(4,6-dimethylpyridin-2-yl)-5,6-dihydro-4H-pyrazolo[4,3-e][1,3]benzothiazol-2-amine

N-(1,3-thiazol-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

N-(5-methylpyridin-2-yl)-5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-amine

4-(1H-pyrazol-4-yl)quinoline

4-(1-phenylpyrazol-4-yl)-7-(2-pyrrolidin-1-ylethoxy)quinoline

4-(1-phenylpyrazol-4-yl)quinolin-7-ol

3-[4-(1-phenylpyrazol-4-yl)quinolin-7-yl]oxypropan-1-ol

4-(1-phenylpyrazol-4-yl)-7-(3-piperidin-1-ylpropoxy)quinoline

1-morpholin-4-yl-2-[4-(1-phenylpyrazol-4-yl)quinolin-7-yl]oxyethanone

N,N-dimethyl-2-[4-(1-phenylpyrazol-4-yl)quinolin-7-yl]oxyacetamide

4-(1-phenylpyrazol-4-yl)-7-(3-pyrrolidin-1-ylpropoxy)quinoline

[4-(1-phenylpyrazol-4-yl)quinolin-7-yl] N-ethylcarbamate

4-(1-phenylpyrazol-4-yl)pyridine

N,N-dimethyl-2-[4-(1-phenylpyrazol-4-yl)quinolin-7-yl]oxyethanamine

(2S)-2-aminopentanedioic acid

(S)-2-amino-4-sulfobutanoic acid