Brief Information of the Compound and Protein
Compound Name
 Compound Info 
6-N,6-N-dimethyl-2-N-(5-thia-3,11,12-triazatricyclo[8.3.0.02,6]trideca-1(10),2(6),3,12-tetraen-4-yl)pyridine-2,6-diamine
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 PubChem ID
CID: 53388195
SID: 125315649
Canonical SMILES
CN(C)c1cccc(Nc2nc-3c(CCCc4[nH]ncc-34)s2)n1
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Compound Formula C16H18N6S
Compound Structure
Protein Name
 Protein Info 
Metabotropic glutamate receptor 4
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q14833
Gene Name
GRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000051 BHK-21
 Cell Line Info 
Mesocricetus auratus (Golden hamster)  1
1
EC50 = 340 nM
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