| Compound ID |
Compound Name |
Compound Formula |
|
CP0498230
|
N-(4-benzoylphenyl)-2-[4-(2-oxo-4H-3,1-benzoxazin-1-yl)piperidin-1-yl]acetamide
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|
C28H27N3O4
|
1
|
| 1 |
IC50 = 7.6 nM
|
|
|
|
CP0382307
|
2-[4-(6-Fluoro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-quinolin-6-yl-acetamide
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|
C24H23FN4O3
|
1
|
| 1 |
IC50 = 7.7 nM
|
|
|
|
CP0853661
|
2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-hydroxy-9H-fluoren-3-yl)-acetamide
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|
C28H27Cl2N3O4
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0853470
|
N-(9-Hydroxy-9H-fluoren-3-yl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
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|
C28H28ClN3O4
|
1
|
| 1 |
IC50 = 8.7 nM
|
|
|
|
CP0853768
|
N-(9-Methyl-9H-carbazol-3-yl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
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|
C28H29ClN4O3
|
1
|
| 1 |
IC50 = 9.6 nM
|
|
|
|
CP0847596
|
N-(4-Benzoyl-phenyl)-2-[4-(6-chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide hydrochloride
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|
C28H27Cl2N3O4
|
1
|
| 1 |
IC50 = 11.2 nM
|
|
|
|
CP0862685
|
N-(4-Acetyl-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
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|
C23H26ClN3O4
|
1
|
| 1 |
IC50 = 17.3 nM
|
|
|
|
CP0853767
|
2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-phenoxy-phenyl)-acetamide
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|
C27H28ClN3O4
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0914844
|
N-(4-Acetyl-phenyl)-2-[4-(6-chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
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|
C23H25Cl2N3O4
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0914843
|
2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-3-yl)-acetamide
Show/Hide
|
C28H26ClN3O4
|
1
|
| 1 |
IC50 = 23.3 nM
|
|
|
|
CP0853762
|
2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-3-yl)-acetamide
Show/Hide
|
C28H25Cl2N3O4
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0862666
|
N-(4-Acetyl-phenyl)-2-[4-(6-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
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|
C24H28ClN3O4
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0897799
|
N-(9-Hydroxy-9H-fluoren-3-yl)-2-[4-(8-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C29H30ClN3O4
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0853763
|
N-(4-Benzoyl-phenyl)-2-[4-(8-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C29H30ClN3O4
|
1
|
| 1 |
IC50 = 39.6 nM
|
|
|
|
CP0855594
|
N-(9-Ethyl-9H-carbazol-3-yl)-2-[4-(8-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C30H33ClN4O3
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0862659
|
2-[4-(8-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-3-yl)-acetamide
Show/Hide
|
C29H28ClN3O4
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0914842
|
N-(9-Ethyl-9H-carbazol-3-yl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C29H30Cl2N4O3
|
1
|
| 1 |
IC50 = 54.6 nM
|
|
|
|
CP0551253
|
N-dibenzofuran-2-yl-2-[4-(8-methoxy-2-oxo-4H-3,1-benzoxazin-1-yl)piperidin-1-yl]acetamide
Show/Hide
|
C28H27N3O5
|
1
|
| 1 |
IC50 = 55.7 nM
|
|
|
|
CP0869625
|
2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-phenoxy-phenyl)-acetamide
Show/Hide
|
C27H27Cl2N3O4
|
1
|
| 1 |
IC50 = 60.7 nM
|
|
|
|
CP0847595
|
2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-2-yl)-acetamide
Show/Hide
|
C28H25Cl2N3O4
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0873399
|
2-[4-(6-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-2-yl)-acetamide
Show/Hide
|
C29H28ClN3O4
|
1
|
| 1 |
IC50 = 86.7 nM
|
|
|
|
CP0849398
|
2-[4-(5-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-ethyl-9H-carbazol-3-yl)-acetamide
Show/Hide
|
C29H30Cl2N4O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0859973
|
2-[4-(6-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-phenoxy-phenyl)-acetamide
Show/Hide
|
C28H30ClN3O4
|
1
|
| 1 |
IC50 = 104 nM
|
|
|
|
CP0859974
|
2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-cyclohexyl-phenyl)-acetamide
Show/Hide
|
C27H33Cl2N3O3
|
1
|
| 1 |
IC50 = 112.4 nM
|
|
|
|
CP0849405
|
N-(4-Cyano-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide hydrochloride
Show/Hide
|
C22H23ClN4O3
|
1
|
| 1 |
IC50 = 132 nM
|
|
|
|
CP0849370
|
2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-4-yl)-acetamide
Show/Hide
|
C28H26ClN3O4
|
1
|
| 1 |
IC50 = 138.2 nM
|
|
|
|
CP0441489
|
2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-quinolin-6-yl-acetamide
Show/Hide
|
C24H23ClN4O3
|
1
|
| 1 |
IC50 = 148 nM
|
|
|
|
CP0859978
|
2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(4-cyano-phenyl)-acetamide hydrochloride
Show/Hide
|
C22H22Cl2N4O3
|
1
|
| 1 |
IC50 = 199 nM
|
|
|
|
CP0871297
|
N-(4-Chloro-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C21H23Cl2N3O3
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0853761
|
N-(9-Ethyl-9H-carbazol-3-yl)-2-[4-(8-methoxy-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C30H33ClN4O4
|
1
|
| 1 |
IC50 = 765.1 nM
|
|
|
|
CP0403141
|
2-{2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetylamino}-benzoic acid methyl ester
Show/Hide
|
C23H25N3O5
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0493174
|
2-{2-[4-(6-Chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetylamino}-benzoic acid methyl ester
Show/Hide
|
C23H24ClN3O5
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0515468
|
2-{2-[4-(8-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetylamino}-benzoic acid methyl ester
Show/Hide
|
C24H27N3O5
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0515469
|
2-{2-[4-(6-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetylamino}-benzoic acid methyl ester
Show/Hide
|
C24H27N3O5
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0849397
|
2-[4-(8-Methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-phenyl-acetamide
Show/Hide
|
C22H26ClN3O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0862661
|
2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-(9-oxo-9H-fluoren-2-yl)-acetamide
Show/Hide
|
C28H26ClN3O4
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0869626
|
N-(2-Benzoyl-phenyl)-2-[4-(8-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C29H30ClN3O4
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0873398
|
N-(4-Cyclohexyl-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C27H34ClN3O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0880940
|
2-[4-(2-Oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-N-phenyl-acetamide hydrochloride
Show/Hide
|
C21H24ClN3O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0915990
|
N-(4-Chloro-phenyl)-2-[4-(8-methyl-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C22H25Cl2N3O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0926670
|
N-(2-Benzoyl-phenyl)-2-[4-(2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide hydrochloride
Show/Hide
|
C28H28ClN3O4
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0957085
|
N-(2-Benzoyl-phenyl)-2-[4-(6-chloro-2-oxo-4H-benzo[d][1,3]oxazin-1-yl)-piperidin-1-yl]-acetamide
Show/Hide
|
C28H27Cl2N3O4
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
