| Compound ID |
Compound Name |
Compound Formula |
|
CP0355893
|
3-cyano-5-[2-[4-[2-(1H-indol-3-yl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
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|
C35H40N6O
|
1
|
| 1 |
EC50 = 270 nM
|
|
|
|
CP0528322
|
3-cyano-5-[2-[4-[2-(3,4-dichlorophenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
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|
C33H37Cl2N5O
|
3
|
| 1 |
EC50 = 425 nM
|
|
|
| 2 |
IC50 = 670 nM
|
|
|
| 3 |
IC50 = 5000 nM
|
|
|
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CP0344698
|
5-[2-[4-[2-(3,4-dichlorophenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
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|
C31H37Cl2N5O
|
1
|
| 1 |
EC50 = 450 nM
|
|
|
|
CP0232183
|
6-[2-[4-[2-(3,4-dichlorophenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
Show/Hide
|
C32H37Cl2N7O
|
1
|
| 1 |
EC50 = 549 nM
|
|
|
|
CP0344699
|
5-[2-[4-[2-(1H-indol-3-yl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C33H40N6O
|
3
|
| 1 |
EC50 = 1020 nM
|
|
|
| 2 |
IC50 = 2430 nM
|
|
|
| 3 |
IC50 = 13260 nM
|
|
|
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CP0224978
|
3-cyano-5-[2-[4-[2-(3-methylphenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
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|
C34H41N5O
|
1
|
| 1 |
EC50 = 1210 nM
|
|
|
|
CP0484190
|
2-[2-[4-[2-(3-methoxyphenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-4-carboxamide
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|
C32H41N5O2
|
1
|
| 1 |
EC50 = 1220 nM
|
|
|
|
CP0565951
|
2-[2-[4-[2-(4-chlorophenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-4-carboxamide
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|
C31H38ClN5O
|
1
|
| 1 |
EC50 = 1620 nM
|
|
|
|
CP0552549
|
2-[2-[4-[2-(4-methoxyphenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-4-carboxamide
Show/Hide
|
C32H41N5O2
|
1
|
| 1 |
EC50 = 2440 nM
|
|
|
|
CP0344883
|
3-cyano-5-[2-[4-[2-(3-methoxyphenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
Show/Hide
|
C34H41N5O2
|
1
|
| 1 |
EC50 = 2690 nM
|
|
|
|
CP0572983
|
3-[2-[4-[2-(4-chlorophenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
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|
C32H39ClN4O
|
1
|
| 1 |
EC50 = 3120 nM
|
|
|
|
CP0558319
|
3-[2-[4-[2-(3,4-dichlorophenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
Show/Hide
|
C32H38Cl2N4O
|
1
|
| 1 |
EC50 = 3230 nM
|
|
|
|
CP0528321
|
3-[2-[4-[2-(1H-indol-3-yl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
Show/Hide
|
C34H41N5O
|
1
|
| 1 |
EC50 = 3460 nM
|
|
|
|
CP0491817
|
3-[2-[4-[2-(3-methoxyphenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
Show/Hide
|
C33H42N4O2
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0261343
|
3-[2-[4-[2-(3-methylphenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
Show/Hide
|
C33H42N4O
|
1
|
| 1 |
EC50 = 4140 nM
|
|
|
|
CP0274376
|
3-[2-[4-(2-phenylethyl)piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
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|
C32H40N4O
|
1
|
| 1 |
EC50 = 4910 nM
|
|
|
|
CP0496391
|
2-[2-[4-[2-(3,4-dichlorophenyl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-4-carboxamide
Show/Hide
|
C31H37Cl2N5O
|
1
|
| 1 |
EC50 = 5570 nM
|
|
|
|
CP0266851
|
2-[2-[4-[2-(1H-indol-3-yl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-4-carboxamide
Show/Hide
|
C33H40N6O
|
1
|
| 1 |
EC50 = 5610 nM
|
|
|
|
CP0367033
|
5-[2-[4-[(3-methoxyphenyl)methylamino]piperidin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C32H41N5O2
|
1
|
| 1 |
EC50 = 5760 nM
|
|
|
|
CP0560912
|
5-[2-[1-[2-(3,4-dichlorophenyl)ethyl]azetidin-3-yl]oxyphenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C30H34Cl2N4O2
|
1
|
| 1 |
EC50 > 24000 nM
|
|
|
|
CP0322272
|
5-[2-[4-[2-(3,4-dichlorophenyl)acetyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C31H35Cl2N5O2
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0264631
|
5-[2-[4-[3-(3,4-dichlorophenyl)propanoyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C32H37Cl2N5O2
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0357898
|
5-[2-[1-[2-(3,4-dichlorophenyl)acetyl]azetidin-3-yl]oxyphenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C30H32Cl2N4O3
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0357896
|
5-[2-[4-[2-(1H-indol-3-yl)acetyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C33H38N6O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0218350
|
5-[2-[4-(3-methylindol-1-yl)butylcarbamoyl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C33H39N5O2
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0274462
|
5-[2-[1-[3-(3,4-dichlorophenyl)propanoyl]azetidin-3-yl]oxyphenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C31H34Cl2N4O3
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0967426
|
5-[2-[4-[2-amino-3-(1H-indol-3-yl)propanoyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C34H41N7O2
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0091740
|
3-cyano-5-[2-[4-[2-(3-methylindol-1-yl)ethyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
Show/Hide
|
C36H42N6O
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0562202
|
5-[2-(4-indol-1-ylbutylcarbamoyl)phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C32H37N5O2
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0240644
|
5-[2-[1-[2-(3,4-dichlorophenyl)acetyl]piperidin-4-yl]oxyphenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C32H36Cl2N4O3
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0357901
|
N-(3,4-dichlorophenyl)-4-[2-[5-(3-pyrrolidin-1-ylpropylcarbamoyl)pyridin-3-yl]phenyl]piperazine-1-carboxamide
Show/Hide
|
C30H34Cl2N6O2
|
1
|
| 1 |
IC50 = 522 nM
|
|
|
|
CP0357899
|
5-[2-[4-(3,4-dichlorobenzoyl)piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C30H33Cl2N5O2
|
1
|
| 1 |
IC50 = 891 nM
|
|
|
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CP0251194
|
5-[2-[4-(2-phenylacetyl)piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C31H37N5O2
|
1
|
| 1 |
IC50 = 1002 nM
|
|
|
|
CP0096816
|
[3-(4-amino-6-methylimidazo[4,5-c]pyridin-1-yl)-3-methylazetidin-1-yl]-[1-[[1-[(1R)-cyclohept-2-en-1-yl]piperidin-4-yl]methyl]pyrrol-3-yl]methanone
Show/Hide
|
C29H39N7O
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0322271
|
5-[2-[4-[(2R)-pyrrolidine-2-carbonyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C28H38N6O2
|
1
|
| 1 |
IC50 = 1469 nM
|
|
|
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CP0240645
|
5-[2-[4-(benzimidazol-1-yl)butylcarbamoyl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C31H36N6O2
|
1
|
| 1 |
IC50 = 1502 nM
|
|
|
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CP0251197
|
3-[5-[1-[2-(3,4-dichlorophenyl)ethyl]azetidin-3-yl]oxy-3-methylpyrazol-1-yl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
Show/Hide
|
C29H35Cl2N5O2
|
1
|
| 1 |
IC50 = 1699 nM
|
|
|
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CP0264628
|
5-[2-(1-propanoylazetidin-3-yl)oxyphenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C25H32N4O3
|
1
|
| 1 |
IC50 = 1914 nM
|
|
|
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CP0569756
|
5-[2-[1-(2-cyanoacetyl)azetidin-3-yl]oxyphenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C25H29N5O3
|
1
|
| 1 |
IC50 = 2415 nM
|
|
|
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CP0426271
|
3-[2-(3,4-dichlorophenyl)ethylamino]-N-[2-[2-(5-hydroxy-3-oxo-4H-1,4-benzoxazin-8-yl)ethylamino]ethyl]-N-methylpropanamide
Show/Hide
|
C24H30Cl2N4O4
|
2
|
| 1 |
IC50 = 9980 nM
|
|
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| 2 |
IC50 = 23590 nM
|
|
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CP0251196
|
5-[2-[4-[2-[4-(2-methylpropyl)phenyl]propanoyl]piperazin-1-yl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C36H47N5O2
|
1
|
| 1 |
IC50 > 2500 nM
|
|
|
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CP0218352
|
3-[1-[4-(3-methylindol-1-yl)butyl]triazol-4-yl]-N-(3-pyrrolidin-1-ylpropyl)benzamide
Show/Hide
|
C29H36N6O
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
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CP0240649
|
5-[2-[4-(cyclopropanecarbonylamino)butylcarbamoyl]phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C28H37N5O3
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
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CP0251198
|
5-[2-(octylcarbamoyl)phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C28H40N4O2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
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CP0274463
|
5-[2-(4-aminobutylcarbamoyl)phenyl]-N-(3-pyrrolidin-1-ylpropyl)pyridine-3-carboxamide
Show/Hide
|
C24H33N5O2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
