| Compound ID |
Compound Name |
Compound Formula |
|
CP0839448
|
2-((2S,3R)-2-Benzyl-3-methylpyrrolidin-1-yl)-6-morpholinopyrimidin-4(3H)-one
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|
C20H26N4O2
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0968778
|
2-((1R,2S,5S)-2-Benzyl-3-azabicyclo[3.1.0]hexan-3-yl)-6-morpholinopyrimidin-4(3H)-one
Show/Hide
|
C20H24N4O2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0953200
|
6-((1S,2S,5R)-2-Benzyl-3-azabicyclo[3.1.0]hexan-3-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C21H25N3O2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0953816
|
(R)-2-(2-Benzylazepan-1-yl)-6-morpholinopyrimidin-4(3H)-one
Show/Hide
|
C21H28N4O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0946565
|
(R)-6-(2-Benzylazepan-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C22H29N3O2
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0016003
|
2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-one
Show/Hide
|
C21H17NO3S2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0953820
|
6-((1R,2S,5S)-2-Benzyl-3-azabicyclo[3.1.0]hexan-3-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C21H25N3O2
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0965262
|
2-((1S,2S,5R)-2-Benzyl-3-azabicyclo[3.1.0]hexan-3-yl)-6-morpholinopyrimidin-4(3H)-one
Show/Hide
|
C20H24N4O2
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
|
CP0569952
|
2-[(2R)-2-benzylpyrrolidin-1-yl]-4-morpholin-4-yl-1H-pyrimidin-6-one
Show/Hide
|
C19H24N4O2
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0953819
|
6-((1S,2S,5R)-2-Benzyl-3-azabicyclo[3.1.0]hexan-3-yl)-4-((R)-2-methylmorpholino)pyridin-2(1H)-one
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0953818
|
2-((1R,2S,5S)-2-Benzyl-3-azabicyclo[3.1.0]hexan-3-yl)-6-((R)-2-methylmorpholino)pyrimidin-4(3H)-one
Show/Hide
|
C21H26N4O2
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0967579
|
2-((R)-2-Benzylazepan-1-yl)-6-((R)-2-methylmorpholino)pyrimidin-4(3H)-one
Show/Hide
|
C22H30N4O2
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0547036
|
6-(7-methoxy-9H-thioxanthen-4-yl)-4-morpholin-4-yl-1H-pyridin-2-one
Show/Hide
|
C23H22N2O3S
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
|
CP0968776
|
(S)-6-(2-Benzyl-3,3-difluoropyrrolidin-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C20H23F2N3O2
|
1
|
| 1 |
IC50 = 920 nM
|
|
|
|
CP0965944
|
6-((1R,2S,5S)-2-Benzyl-3-azabicyclo[3.1.0]hexan-3-yl)-4-((R)-2-methylmorpholino)pyridin-2(1H)-one
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0135733
|
2-(7-methoxy-9H-thioxanthen-4-yl)-6-morpholin-4-ylpyran-4-one
Show/Hide
|
C23H21NO4S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0967580
|
2-((1S,2S,5R)-2-Benzyl-3-azabicyclo[3.1.0]hexan-3-yl)-6-((R)-2-methylmorpholino)pyrimidin-4(3H)-one
Show/Hide
|
C21H26N4O2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0968777
|
6-((2S,3R)-2-Benzyl-3-fluoropyrrolidin-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C20H24FN3O2
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0839447
|
6-((R)-2-Benzylazepan-1-yl)-4-((R)-2-methylmorpholino)pyridin-2(1H)-one
Show/Hide
|
C23H31N3O2
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0955420
|
(R)-6-(2-Benzylpiperidin-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C21H27N3O2
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0953815
|
(R)-6-(2-Benzylpyrrolidin-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
IC50 = 3400 nM
|
|
|
|
CP0965110
|
6-((2S,3R)-2-Benzyl-3-methoxypyrrolidin-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C21H27N3O3
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
|
CP0839445
|
Rac-6-(2-Benzylpyrrolidin-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0363798
|
4-(7-methoxy-9H-thioxanthen-4-yl)-2-morpholin-4-yl-1H-pyrimidin-6-one
Show/Hide
|
C22H21N3O3S
|
1
|
| 1 |
IC50 = 6700 nM
|
|
|
|
CP0547037
|
4-(7-methoxy-9H-thioxanthen-4-yl)-6-morpholin-4-yl-1H-pyridin-2-one
Show/Hide
|
C23H22N2O3S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0569555
|
2-(7-methoxy-9H-thioxanthen-4-yl)-4-morpholin-4-yl-1H-pyrimidin-6-one
Show/Hide
|
C22H21N3O3S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0573590
|
4-[2-methoxy-6-(7-methoxy-9H-thioxanthen-4-yl)pyridin-4-yl]morpholine
Show/Hide
|
C24H24N2O3S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0573591
|
6-(7-methoxy-9H-thioxanthen-4-yl)-4-morpholin-4-yl-1H-pyrimidin-2-one
Show/Hide
|
C22H21N3O3S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0575457
|
6-(7-methoxy-9H-thioxanthen-4-yl)-1-methyl-4-morpholin-4-ylpyridin-2-one
Show/Hide
|
C24H24N2O3S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0575458
|
2-(7-methoxy-9H-thioxanthen-4-yl)-6-morpholin-4-yl-1H-pyridin-4-one
Show/Hide
|
C23H22N2O3S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0575459
|
4-[(2R)-2-benzylpyrrolidin-1-yl]-2-morpholin-4-yl-1H-pyrimidin-6-one
Show/Hide
|
C19H24N4O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0839446
|
6-(3-Benzylpyrrolidin-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0966210
|
(S)-6-(2-benzylpyrrolidin-1-yl)-4-morpholinopyridin-2(1H)-one
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
