| Compound ID |
Compound Name |
Compound Formula |
|
CP0538381
|
1-[3-(2-methoxyethoxy)-4-phenoxyphenyl]-3-(3-methylphenyl)-1,3,5-triazinane-2,4,6-trione
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|
C25H23N3O6
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0477098
|
1-[3-(2-methoxyethoxy)-4-phenoxyphenyl]-3-(4-methylphenyl)-1,3,5-triazinane-2,4,6-trione
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|
C25H23N3O6
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0536435
|
1-(3-chlorophenyl)-3-[3-(2-methoxyethoxy)-4-phenoxyphenyl]-1,3,5-triazinane-2,4,6-trione
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|
C24H20ClN3O6
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
|
CP0434610
|
1-(3-bromo-4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
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|
C21H14BrN3O4
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0538383
|
1-methyl-3-[3-(oxetan-3-ylmethoxy)-4-phenoxyphenyl]-1,3,5-triazinane-2,4,6-trione
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|
C20H19N3O6
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0434609
|
1-(4-chlorophenyl)-3-[3-(2-methoxyethoxy)-4-phenoxyphenyl]-1,3,5-triazinane-2,4,6-trione
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|
C24H20ClN3O6
|
1
|
| 1 |
EC50 = 330 nM
|
|
|
|
CP0455522
|
1-(4-phenoxy-3-propan-2-yloxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
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|
C24H21N3O5
|
1
|
| 1 |
EC50 = 330 nM
|
|
|
|
CP0440106
|
1-[3-(oxolan-3-yloxy)-4-phenoxyphenyl]-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C25H21N3O6
|
1
|
| 1 |
EC50 = 480 nM
|
|
|
|
CP0536434
|
1-(3-ethoxy-4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
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|
C23H19N3O5
|
1
|
| 1 |
EC50 = 510 nM
|
|
|
|
CP0545872
|
1-[3-(oxetan-3-ylmethoxy)-4-phenoxyphenyl]-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C25H21N3O6
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0485953
|
1-(4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
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|
C21H15N3O4
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0480003
|
6-(1-methylpyrazol-4-yl)-3-[(3R)-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]pyrrolidin-3-yl]oxypyridine-2-carboxamide
Show/Hide
|
C23H22F3N5O4
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0274475
|
N-[5-(4-amino-7-propan-2-ylpyrrolo[2,3-d]pyrimidine-5-carbonyl)pyridin-3-yl]-2-(4-chlorophenyl)acetamide
Show/Hide
|
C23H21ClN6O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0284251
|
US8846698, 250
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|
C23H21ClN6O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0123936
|
2-[(3R,4S)-3-fluoro-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxy-5-(1-methylimidazol-4-yl)pyridine-3-carboxamide
Show/Hide
|
C24H23F4N5O4
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0514698
|
N-[5-[2-amino-7-(1-hydroxy-2-methylpropan-2-yl)pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl]-2-(4-chlorophenyl)acetamide
Show/Hide
|
C24H23ClN6O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0198981
|
6-amino-5-[(3S)-4,4-difluoro-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]pyrrolidin-3-yl]oxy-N-methylpyridine-3-carboxamide
Show/Hide
|
C20H19F5N4O4
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0456114
|
5-(1-methylimidazol-4-yl)-2-[1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxybenzamide
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|
C25H25F3N4O4
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0188940
|
US8846698, 69
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|
C23H20ClN5O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0261329
|
PF06273340
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|
C23H22ClN7O3
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0198982
|
2-[(3R,4S)-3-fluoro-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxy-4-(2-hydroxy-2-methylpropoxy)benzamide
Show/Hide
|
C25H28F4N2O6
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0514699
|
US8846698, 253
Show/Hide
|
C23H24N8O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0540119
|
1-[4-(4-amino-7-propan-2-ylpyrrolo[2,3-d]pyrimidine-5-carbonyl)pyridin-2-yl]-3-(2,4-difluorophenyl)urea
Show/Hide
|
C22H19F2N7O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0245290
|
4-[2-carbamoyl-4-(1-methylpyrazol-4-yl)phenoxy]-N-[4-(trifluoromethoxy)phenyl]piperidine-1-carboxamide
Show/Hide
|
C24H24F3N5O4
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0322061
|
US9163021, 21
Show/Hide
|
C22H19F3N6O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0245291
|
6-(1-methylpyrazol-4-yl)-3-[1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxypyridine-2-carboxamide
Show/Hide
|
C24H24F3N5O4
|
1
|
| 1 |
IC50 = 8.4 nM
|
|
|
|
CP0415710
|
6-(1-methylpyrazol-4-yl)-3-[(3S)-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]pyrrolidin-3-yl]oxypyridine-2-carboxamide
Show/Hide
|
C23H22F3N5O4
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0535882
|
N-(pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)ethanamine
Show/Hide
|
C20H19N3S
|
1
|
| 1 |
IC50 = 25140 nM
|
|
|
|
CP0457124
|
2-(2-phenylindol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C22H19N3O
|
1
|
| 1 |
IC50 = 25960 nM
|
|
|
|
CP0538993
|
N-(pyrazin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C19H16N4OS
|
1
|
| 1 |
IC50 > 27000 nM
|
|
|
|
CP0457122
|
N-(1,3-oxazol-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C18H15N3O2S
|
1
|
| 1 |
IC50 = 38500 nM
|
|
|
|
CP0457119
|
2-(2-phenylpyrrolo[2,3-b]pyridin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C21H18N4O
|
1
|
| 1 |
IC50 = 38550 nM
|
|
|
|
CP0535880
|
2-[2-(5-methylthiophen-2-yl)indol-1-yl]-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C21H19N3OS
|
1
|
| 1 |
IC50 = 47860 nM
|
|
|
|
CP0447388
|
2-(2-phenylpyrrolo[2,3-c]pyridin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C21H18N4O
|
1
|
| 1 |
IC50 = 51000 nM
|
|
|
|
CP0476186
|
2-[2-(1,3-oxazol-2-yl)indol-1-yl]-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C19H16N4O2
|
1
|
| 1 |
IC50 = 53490 nM
|
|
|
|
CP0457115
|
N-(pyrimidin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C19H16N4OS
|
1
|
| 1 |
IC50 = 58440 nM
|
|
|
|
CP0535881
|
N-(1H-benzimidazol-2-ylmethyl)-2-[2-(1,3-oxazol-2-yl)indol-1-yl]acetamide
Show/Hide
|
C21H17N5O2
|
1
|
| 1 |
IC50 = 68160 nM
|
|
|
|
CP0476188
|
N-(1H-benzimidazol-2-ylmethyl)-2-[5-fluoro-2-(1,3-oxazol-2-yl)indol-1-yl]acetamide
Show/Hide
|
C21H16FN5O2
|
1
|
| 1 |
IC50 = 68750 nM
|
|
|
|
CP0458606
|
N-(pyridin-2-ylmethyl)-2-[2-(1,2-thiazol-5-yl)indol-1-yl]acetamide
Show/Hide
|
C19H16N4OS
|
1
|
| 1 |
IC50 = 70240 nM
|
|
|
|
CP0566086
|
N-(imidazo[1,2-a]pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C22H18N4OS
|
1
|
| 1 |
IC50 = 71720 nM
|
|
|
|
CP0457116
|
2-[2-(5-methylfuran-2-yl)indol-1-yl]-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C21H19N3O2
|
1
|
| 1 |
IC50 = 73070 nM
|
|
|
|
CP0481932
|
N-[2-(2-thiophen-2-ylindol-1-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C20H17N3OS
|
1
|
| 1 |
IC50 = 80020 nM
|
|
|
|
CP0571702
|
N-(2-pyridin-2-ylethyl)-2-thiophen-2-ylindole-1-carboxamide
Show/Hide
|
C20H17N3OS
|
1
|
| 1 |
IC50 = 80270 nM
|
|
|
|
CP0447385
|
N-(pyridin-2-ylmethyl)-2-[2-(1,2-thiazol-3-yl)indol-1-yl]acetamide
Show/Hide
|
C19H16N4OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0457117
|
N-(pyridin-2-ylmethyl)-2-[2-(1,3-thiazol-2-yl)indol-1-yl]acetamide
Show/Hide
|
C19H16N4OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0457118
|
2-(2-phenylpyrrolo[3,2-b]pyridin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C21H18N4O
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0457120
|
N-[2-(2-thiophen-2-ylindol-1-yl)ethyl]pyridine-2-sulfonamide
Show/Hide
|
C19H17N3O2S2
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0457121
|
N-(1,3-thiazol-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C18H15N3OS2
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0457123
|
N-[(2-phenyl-1H-imidazol-5-yl)methyl]-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C24H20N4OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0458601
|
2-(5-fluoro-2-phenylindol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C22H18FN3O
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0458604
|
N-(pyridin-3-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C20H17N3OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0458605
|
N-[(1-methylimidazol-2-yl)methyl]-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C19H18N4OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0458607
|
2-(2-phenylpyrrolo[3,2-c]pyridin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C21H18N4O
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0476187
|
2-(2-pyridin-3-ylindol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C21H18N4O
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0508119
|
2-(4-fluoro-2-phenylindol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C22H18FN3O
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0535794
|
N-(1H-imidazol-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C18H16N4OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0535883
|
N-(pyridin-4-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C20H17N3OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0535884
|
N-[(5-phenyl-1H-imidazol-2-yl)methyl]-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C24H20N4OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0535885
|
2-(6-fluoro-2-phenylindol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C22H18FN3O
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0544837
|
N-(pyridin-2-ylmethyl)-2-[2-(1,3-thiazol-5-yl)indol-1-yl]acetamide
Show/Hide
|
C19H16N4OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0544840
|
N-methyl-N-(pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C21H19N3OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0558663
|
N-(1H-benzimidazol-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C22H18N4OS
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0558664
|
2-(2-pyridin-2-ylindol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C21H18N4O
|
1
|
| 1 |
IC50 > 81010 nM
|
|
|
|
CP0535793
|
N-(pyridin-2-ylmethyl)-2-thiophen-2-ylindole-1-carboxamide
Show/Hide
|
C19H15N3OS
|
1
|
| 1 |
IC50 = 81160 nM
|
|
|
|
CP0540336
|
N-benzyl-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C21H18N2OS
|
1
|
| 1 |
IC50 > 3000 nM
|
|
|
|
CP0458603
|
2-(7-fluoro-2-phenylindol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
Show/Hide
|
C22H18FN3O
|
1
|
| 1 |
IC50 > 9001 nM
|
|
|
|
CP0544839
|
N-pyridin-2-yl-2-(2-thiophen-2-ylindol-1-yl)acetamide
Show/Hide
|
C19H15N3OS
|
1
|
| 1 |
IC50 > 9001 nM
|
|
|
