| Compound ID |
Compound Name |
Compound Formula |
|
CP0120450
|
N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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|
C22H30N4O3
|
2
|
| 1 |
EC50 = 17.6 nM
|
|
|
| 2 |
EC50 = 28 nM
|
|
|
|
CP0089916
|
1-(4-fluorobutyl)-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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|
C20H26FN3O2
|
2
|
| 1 |
EC50 = 20.6 nM
|
|
|
| 2 |
EC50 = 21.8 nM
|
|
|
|
CP0051374
|
1-(4-hydroxybutyl)-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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|
C20H27N3O3
|
1
|
| 1 |
EC50 = 23.7 nM
|
|
|
|
CP0051372
|
1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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|
C23H24FN3O2
|
1
|
| 1 |
EC50 = 29.6 nM
|
|
|
|
CP0048192
|
2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl)-5-(2-methyloctan-2-yl)phenol
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|
C24H40O3
|
1
|
| 1 |
EC50 = 37.15 nM
|
|
|
|
CP0382145
|
(3',5'-dichloro-2,6-dihydroxybiphenyl-4-yl)(phenyl)methanone
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|
C19H12Cl2O3
|
1
|
| 1 |
EC50 = 154.88 nM
|
|
|
|
CP0152977
|
5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1H-pyrazole-3-carboxylic acid ((1S,2S,4R)-1,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl)-amide
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|
C29H34ClN3O
|
1
|
| 1 |
EC50 = 1174.9 nM
|
|
|
|
CP0533352
|
[4-[3,5-bis(trifluoromethyl)phenyl]-3,5-dihydroxyphenyl]-thiophen-2-ylmethanone
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|
C19H10F6O3S
|
1
|
| 1 |
EC50 = 1288.25 nM
|
|
|
|
CP0424598
|
[4-[3,5-bis(trifluoromethyl)phenyl]-3,5-dihydroxyphenyl]-phenylmethanone
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|
C21H12F6O3
|
1
|
| 1 |
EC50 = 1412.54 nM
|
|
|
|
CP0507627
|
[3,5-dihydroxy-4-[3-(trifluoromethyl)phenyl]phenyl]-phenylmethanone
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|
C20H13F3O3
|
1
|
| 1 |
EC50 = 3467.37 nM
|
|
|
|
CP0517388
|
[4-(2,5-dichlorophenyl)-3,5-dihydroxyphenyl]-phenylmethanone
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|
C19H12Cl2O3
|
1
|
| 1 |
EC50 = 6025.6 nM
|
|
|
|
CP0507623
|
[3,5-dihydroxy-4-(3-methylphenyl)phenyl]-thiophen-2-ylmethanone
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|
C18H14O3S
|
1
|
| 1 |
EC50 = 6165.95 nM
|
|
|
|
CP0424594
|
[3,5-dihydroxy-4-[3-(trifluoromethyl)phenyl]phenyl]-thiophen-2-ylmethanone
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|
C18H11F3O3S
|
1
|
| 1 |
EC50 = 8511.38 nM
|
|
|
|
CP0424596
|
[4-(3,5-difluorophenyl)-3,5-dihydroxyphenyl]-phenylmethanone
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|
C19H12F2O3
|
1
|
| 1 |
EC50 = 8912.51 nM
|
|
|
|
CP0487498
|
[4-(2,5-dichlorophenyl)-3,5-dihydroxyphenyl]-thiophen-2-ylmethanone
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|
C17H10Cl2O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0562921
|
US9139546, 26
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|
C20H16O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0396544
|
(E)-3-(2-methoxyphenyl)-N-[[4-[methyl(phenyl)sulfamoyl]phenyl]carbamothioyl]prop-2-enamide
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|
C24H23N3O4S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0396545
|
MLS000569095
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|
C23H18FN5O2S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0456697
|
3-[4-(2,3-dimethylphenyl)piperazin-1-yl]carbonyl-N,N-dimethyl-4-pyrrolidin-1-yl-benzenesulfonamide
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|
C25H34N4O3S
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0051315
|
6-bromo-1-[(4-fluorophenyl)methyl]-N-(4-methylcyclohexyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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|
C23H23BrFN3O2
|
1
|
| 1 |
IC50 = 31.6 nM
|
|
|
|
CP0362820
|
6-bromo-N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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|
C22H29BrN4O3
|
2
|
| 1 |
IC50 = 32.1 nM
|
|
|
| 2 |
IC50 = 59.6 nM
|
|
|
|
CP0244993
|
6-(4-methoxyphenyl)-N-(4-methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-2-oxo-1,8-naphthyridine-3-carboxamide
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|
C29H36N4O4
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
