| Compound ID |
Compound Name |
Compound Formula |
|
CP0419825
|
US8546435, 3
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|
C38H36N8O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0475559
|
N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3-fluoropyridine-2-carboxamide
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|
C36H34FN7O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0432520
|
6-fluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide
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|
C34H31FN6O2
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
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CP0385058
|
3,5-difluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide
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|
C34H30F2N6O2
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
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CP0475492
|
N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
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|
C36H38N6O4
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0284845
|
US8546435, 4
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|
C36H35N7O3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
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CP0475493
|
N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-4,6-difluoropyridine-2-carboxamide
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|
C36H33F2N7O3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0154574
|
N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide
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|
C34H32N6O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
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CP0455241
|
N-[(1R)-1-[5-[(1R)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C34H33N7O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
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CP0491423
|
N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-6-methylpyridine-2-carboxamide
Show/Hide
|
C35H34N6O2
|
1
|
| 1 |
IC50 = 7.5 nM
|
|
|
|
CP0126988
|
US8546435, 5
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|
C35H33N7O3
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0229128
|
US8546435, 6
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|
C32H34N6O4
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0395265
|
3-fluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide
Show/Hide
|
C34H31FN6O2
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
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CP0850992
|
(R)-N-(2-(1H-indol-3-yl)-1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)ethyl)-6-methoxypicolinamide
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|
C35H34N6O3
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0475496
|
US8546435, 7
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|
C35H39N7O4
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0501203
|
6-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide
Show/Hide
|
C34H33N7O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0510760
|
US8546435, 8
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|
C36H40N8O3
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0327955
|
US8546435, 9
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|
C35H38N8O3
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
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CP0475560
|
N-[(1R)-1-[5-[(1R)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide
Show/Hide
|
C34H39N7O3
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
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CP0432522
|
N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]isoquinoline-1-carboxamide
Show/Hide
|
C38H34N6O2
|
1
|
| 1 |
IC50 = 73 nM
|
|
|
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CP0484685
|
N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-1-oxidopyridin-1-ium-2-carboxamide
Show/Hide
|
C34H32N6O3
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0414782
|
N-[(1R)-1-[5-[(1S)-1-acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C38H36N8O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0386295
|
3-hydroxy-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide
Show/Hide
|
C34H32N6O3
|
1
|
| 1 |
IC50 = 108 nM
|
|
|
|
CP0475747
|
2-amino-N-[(1R)-1-[5-[(1R)-1-formamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C33H37N7O3
|
1
|
| 1 |
IC50 = 113 nM
|
|
|
|
CP0447867
|
2-amino-N-[(1R)-1-[5-[(1R)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C32H37N7O2
|
1
|
| 1 |
IC50 = 115 nM
|
|
|
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CP0388314
|
N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]isoquinoline-3-carboxamide
Show/Hide
|
C38H34N6O2
|
1
|
| 1 |
IC50 = 126 nM
|
|
|
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CP0475562
|
2-amino-N-[(1R)-1-[5-[(1R)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C34H38N8O2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
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CP0380802
|
2-bromo-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide
Show/Hide
|
C34H31BrN6O2
|
1
|
| 1 |
IC50 = 193 nM
|
|
|
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CP0406403
|
5-bromo-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide
Show/Hide
|
C34H31BrN6O2
|
1
|
| 1 |
IC50 = 222 nM
|
|
|
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CP0395264
|
3-benzoyl-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamide
Show/Hide
|
C41H36N6O3
|
1
|
| 1 |
IC50 = 313 nM
|
|
|
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CP0475749
|
N-[(1R)-1-[5-[(1S)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C34H33N7O2
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
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CP0475494
|
N-[(1R)-1-[5-[(1S)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C36H35N7O3
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
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CP0475561
|
N-[(1R)-1-[5-[(1S)-1-formamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C37H34N8O3
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
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CP0380801
|
N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide
Show/Hide
|
C34H32N6O2
|
1
|
| 1 |
IC50 = 411 nM
|
|
|
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CP0432521
|
2-amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide
Show/Hide
|
C34H33N7O2
|
1
|
| 1 |
IC50 = 427 nM
|
|
|
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CP0386294
|
6-chloro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamide
Show/Hide
|
C34H31ClN6O2
|
1
|
| 1 |
IC50 = 771 nM
|
|
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CP0388828
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N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-4-carboxamide
Show/Hide
|
C34H32N6O2
|
1
|
| 1 |
IC50 = 828 nM
|
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CP0425157
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N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-5-pyrrolidin-1-ylpyridine-2-carboxamide
Show/Hide
|
C38H39N7O2
|
1
|
| 1 |
IC50 = 1210 nM
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CP0379866
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N-[(1R)-1-[5-[(1S)-1-acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide
Show/Hide
|
C36H40N8O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
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CP0385352
|
N-[(1R)-1-[5-[(1S)-1-acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamide
Show/Hide
|
C34H39N7O3
|
1
|
| 1 |
IC50 > 1000 nM
|
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CP0419823
|
2-amino-N-[(1R)-1-[5-[(1S)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C32H37N7O2
|
1
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| 1 |
IC50 > 1000 nM
|
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CP0561894
|
2-amino-N-[(1R)-1-[5-[(1S)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamide
Show/Hide
|
C34H38N8O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
