| Compound ID |
Compound Name |
Compound Formula |
|
CP0164458
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-methoxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,4-dimethylpyridin-3-yl)methanone
Show/Hide
|
C27H35BrN4O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0351357
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-ethoxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,4-dimethylpyridin-3-yl)methanone
Show/Hide
|
C28H37BrN4O2
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
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CP0136664
|
(Z)-(4-((4-bromophenyl)(ethoxyimino)methyl)-4'-methyl-1,4'-bipiperidin-1'-yl)(2,6-dimethylphenyl)methanone
Show/Hide
|
C29H38BrN3O2
|
1
|
| 1 |
Ki = 2 nM
|
|
|
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CP0735442
|
(4-{(4-Bromo-phenyl)-[(Z)-ethoxyimino]-methyl}-4'-methyl-[1,4']bipiperidinyl-1'-yl)-(2,4-dimethyl-1-oxy-pyridin-3-yl)-methanone
Show/Hide
|
C28H37BrN4O3
|
1
|
| 1 |
Ki = 2.1 nM
|
|
|
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CP0530346
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-ethoxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-[2-fluoro-6-(trifluoromethyl)phenyl]methanone
Show/Hide
|
C28H32BrF4N3O2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
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CP0268868
|
(2-Amino-6-chloro-phenyl)-{4-[(4-bromo-phenyl)-methoxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
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|
C26H32BrClN4O2
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
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CP0879072
|
(2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[ethoxyimino-(4-trifluoromethyl-phenyl)-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C29H37F3N4O3
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0438586
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-propan-2-yloxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C30H40BrN3O2
|
1
|
| 1 |
Ki = 4 nM
|
|
|
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CP0949924
|
(2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[ethoxyimino-(4-trifluoromethoxy-phenyl)-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C29H37F3N4O4
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
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CP0306750
|
(2-Amino-6-methyl-phenyl)-{4-[(4-bromo-phenyl)-methoxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C27H35BrN4O2
|
1
|
| 1 |
Ki = 4.5 nM
|
|
|
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CP0899348
|
(2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[methoxyimino-(4-trifluoromethyl-phenyl)-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C28H35F3N4O3
|
1
|
| 1 |
Ki = 5.3 nM
|
|
|
|
CP0942067
|
{4-[(4-Chloro-phenyl)-ethoxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-(2,4-dimethyl-1-oxy-pyridin-3-yl)-methanone
Show/Hide
|
C28H37ClN4O3
|
1
|
| 1 |
Ki = 5.6 nM
|
|
|
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CP0437459
|
5-[4-[4-[(Z)-C-(4-bromophenyl)-N-ethoxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidine-1-carbonyl]-4,6-dimethyl-1H-pyridin-2-one
Show/Hide
|
C28H37BrN4O3
|
1
|
| 1 |
Ki = 7 nM
|
|
|
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CP0860148
|
(2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[methoxyimino-(4-trifluoromethoxy-phenyl)-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C28H35F3N4O4
|
1
|
| 1 |
Ki = 7.6 nM
|
|
|
|
CP0346147
|
[4-[4-[1-(4-bromophenyl)ethenyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C28H35BrN2O
|
1
|
| 1 |
Ki = 8 nM
|
|
|
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CP0461466
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-[(2-methylpropan-2-yl)oxy]carbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C31H42BrN3O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0527493
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-(2-methoxyethoxy)carbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C30H40BrN3O3
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0467811
|
4-[(Z)-(4-Bromophenyl)(ethoxyimino)methyl]-4'-methyl-1'-[(3-methyl-2-pyridinyl)carbonyl]-1,4'-bipiperidine NOxide
Show/Hide
|
C27H35BrN4O3
|
1
|
| 1 |
Ki = 16 nM
|
|
|
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CP0241386
|
1'-(2-Hydroxy-6-methylbenzoyl)-4-[(Z)-(4-bromophenyl)-(methoxyimino)methyl]-4'-methyl-1,4'-bipiperidine
Show/Hide
|
C27H34BrN3O3
|
1
|
| 1 |
Ki = 18 nM
|
|
|
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CP0757393
|
{4-[(4-Bromo-phenyl)-methoxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-(2,4-dimethyl-1-oxy-pyridin-3-yl)-methanone
Show/Hide
|
C27H35BrN4O3
|
1
|
| 1 |
Ki = 19 nM
|
|
|
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CP0941464
|
(2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[ethoxyimino-(4-methanesulfonyl-phenyl)-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C29H40N4O5S
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0895051
|
{4-[(4-Chloro-phenyl)-methoxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-(2,4-dimethyl-1-oxy-pyridin-3-yl)-methanone
Show/Hide
|
C27H35ClN4O3
|
1
|
| 1 |
Ki = 24 nM
|
|
|
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CP0088336
|
(2,6-Dimethyl-phenyl)-[4'-methyl-4-(4-trifluoromethyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C28H35F3N2O
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0289873
|
(4-{(4-Bromo-phenyl)-[(E)-methoxyimino]-methyl}-4'-methyl-[1,4']bipiperidinyl-1'-yl)-(2,6-dimethyl-phenyl)-methanone
Show/Hide
|
C28H36BrN3O2
|
1
|
| 1 |
Ki = 25 nM
|
|
|
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CP0461318
|
4-[(Z)-(4-Bromophenyl)(ethoxyimino)methyl]-4'-methyl-1'-[(2-methyl-3-pyridinyl)carbonyl]-1,4'-bipiperidine
Show/Hide
|
C27H35BrN4O2
|
1
|
| 1 |
Ki = 26 nM
|
|
|
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CP0216375
|
[4-[4-(4-bromophenoxy)piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C26H33BrN2O2
|
1
|
| 1 |
Ki = 29 nM
|
|
|
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CP0852709
|
(2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[(4-methanesulfonyl-phenyl)-methoxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C28H38N4O5S
|
1
|
| 1 |
Ki = 30 nM
|
|
|
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CP0949925
|
(2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[ethoxyimino-(4-fluoro-phenyl)-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C28H37FN4O3
|
1
|
| 1 |
Ki = 30 nM
|
|
|
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CP0328212
|
(2,6-Dimethyl-phenyl)-[4-(4-methanesulfonyl-benzyl)-4'-methyl-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C28H38N2O3S
|
1
|
| 1 |
Ki = 33 nM
|
|
|
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CP0337666
|
(2,6-Dimethyl-phenyl)-[4-(4-iodo-benzyl)-4'-methyl-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C27H35IN2O
|
1
|
| 1 |
Ki = 33 nM
|
|
|
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CP0463536
|
2-{(4-Bromo-phenyl)-[1'-(2,6-dimethyl-benzoyl)-4'-methyl-[1,4']bipiperidinyl-4-yl]-methyleneaminooxy}-N-methyl-acetamide
Show/Hide
|
C30H39BrN4O3
|
1
|
| 1 |
Ki = 33 nM
|
|
|
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CP0467860
|
ethyl 2-[(Z)-[(4-bromophenyl)-[1-[1-(2,6-dimethylbenzoyl)-4-methylpiperidin-4-yl]piperidin-4-yl]methylidene]amino]oxyacetate
Show/Hide
|
C31H40BrN3O4
|
1
|
| 1 |
Ki = 33 nM
|
|
|
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CP0438532
|
4-[(Z)-(4-Bromophenyl)(ethoxyimino)methyl]-1'-[(2-hydroxy-4,6-dimethyl-3-pyridinyl)carbonyl]-4'-methyl-1,4'-bipiperidine
Show/Hide
|
C28H37BrN4O3
|
1
|
| 1 |
Ki = 43 nM
|
|
|
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CP0219064
|
(4-{(4-Bromo-phenyl)-[(E)-ethoxyimino]-methyl}-4'-methyl-[1,4']bipiperidinyl-1'-yl)-(2,6-dimethyl-phenyl)-methanone
Show/Hide
|
C29H38BrN3O2
|
1
|
| 1 |
Ki = 48 nM
|
|
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CP0061031
|
(4-Bromo-phenyl)-[1'-(2,6-dimethyl-benzoyl)-4'-methyl-[1,4']bipiperidinyl-4-yl]-methanone
Show/Hide
|
C27H33BrN2O2
|
1
|
| 1 |
Ki = 54 nM
|
|
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CP0195775
|
(2,6-Dimethyl-phenyl)-[4'-methyl-4-(4-trifluoromethoxy-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C28H35F3N2O2
|
1
|
| 1 |
Ki = 55 nM
|
|
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CP0241291
|
4-[(4-Bromophenyl)methyl]-1'-(2,6-dimethylbenzoyl)-4'-methyl-1,4'-bipiperidine
Show/Hide
|
C27H35BrN2O
|
1
|
| 1 |
Ki = 58 nM
|
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CP0149009
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[4-[4-[1-(4-bromophenyl)ethyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C28H37BrN2O
|
1
|
| 1 |
Ki = 62 nM
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CP0460158
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-(2-hydroxyethoxy)carbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C29H38BrN3O3
|
1
|
| 1 |
Ki = 62 nM
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CP0466335
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[4-[4-[(3-bromophenyl)methyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C27H35BrN2O
|
1
|
| 1 |
Ki = 67 nM
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CP0328099
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4-[(4-Chlorophenyl)methyl]-1'-(2,6-dimethylbenzoyl)-4'-methyl-1,4'-bipiperidine
Show/Hide
|
C27H35ClN2O
|
1
|
| 1 |
Ki = 68 nM
|
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CP0922332
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{4-[(4-Bromo-phenyl)-hydroxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-(2,6-dimethyl-phenyl)-methanone
Show/Hide
|
C27H34BrN3O2
|
1
|
| 1 |
Ki = 78 nM
|
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CP0104983
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(2,6-Dimethyl-phenyl)-[4'-methyl-4-(4-methylsulfanyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C28H38N2OS
|
1
|
| 1 |
Ki = 86 nM
|
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CP0215833
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(2,6-Dimethyl-phenyl)-[4'-methyl-4-(4-methyl-benzyl)-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C28H38N2O
|
1
|
| 1 |
Ki = 113 nM
|
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CP0163569
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(2,6-Dimethyl-phenyl)-[4-(4-methoxy-benzyl)-4'-methyl-[1,4']bipiperidinyl-1'-yl]-methanone
Show/Hide
|
C28H38N2O2
|
1
|
| 1 |
Ki = 155 nM
|
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CP0363343
|
[4-[4-[(4-bromophenyl)-hydroxymethyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C27H35BrN2O2
|
1
|
| 1 |
Ki = 190 nM
|
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CP0538919
|
(4-Benzyl-4'-methyl-[1,4']bipiperidinyl-1'-yl)-(2,6-dimethyl-phenyl)-methanone
Show/Hide
|
C27H36N2O
|
1
|
| 1 |
Ki = 282 nM
|
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|
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CP0308132
|
(4-Biphenyl-4-ylmethyl-4'-methyl-[1,4']bipiperidinyl-1'-yl)-(2,6-dimethyl-phenyl)-methanone
Show/Hide
|
C33H40N2O
|
1
|
| 1 |
Ki = 363 nM
|
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CP0100506
|
1-{4-[1'-(2,6-Dimethyl-benzoyl)-4'-methyl-[1,4']bipiperidinyl-4-ylmethyl]-phenyl}-ethanone
Show/Hide
|
C29H38N2O2
|
1
|
| 1 |
Ki = 596 nM
|
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CP0184640
|
(4-Fluoro-naphthalen-1-yl)-{4-[4-(4-methoxy-benzenesulfonyl)-benzyl]-[1,4']bipiperidinyl-1'-yl}-methanone
Show/Hide
|
C35H37FN2O4S
|
1
|
| 1 |
Ki = 1000 nM
|
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CP0406507
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-ethoxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-pyridin-3-ylmethanone
Show/Hide
|
C26H33BrN4O2
|
1
|
| 1 |
Ki > 30 nM
|
|
|
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CP0448878
|
3-[4-[4-[(Z)-C-(4-bromophenyl)-N-ethoxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidine-1-carbonyl]-4-methyl-1H-pyridin-2-one
Show/Hide
|
C27H35BrN4O3
|
1
|
| 1 |
Ki > 30 nM
|
|
|
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CP0466320
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-phenoxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C33H38BrN3O2
|
1
|
| 1 |
Ki > 30 nM
|
|
|
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CP0879148
|
{4-[(4-Bromo-phenyl)-ethoxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-(1-oxy-pyridin-3-yl)-methanone
Show/Hide
|
C26H33BrN4O3
|
1
|
| 1 |
Ki > 30 nM
|
|
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CP0894627
|
{4-[(4-Bromo-phenyl)-ethoxyimino-methyl]-4'-methyl-[1,4']bipiperidinyl-1'-yl}-(2-methyl-1-oxy-pyridin-3-yl)-methanone
Show/Hide
|
C27H35BrN4O3
|
1
|
| 1 |
Ki > 30 nM
|
|
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CP0465705
|
[4-[4-[(Z)-C-(4-bromophenyl)-N-phenylmethoxycarbonimidoyl]piperidin-1-yl]-4-methylpiperidin-1-yl]-(2,6-dimethylphenyl)methanone
Show/Hide
|
C34H40BrN3O2
|
1
|
| 1 |
Ki > 500 nM
|
|
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