| Compound ID |
Compound Name |
Compound Formula |
|
CP0340520
|
N-[2-methyl-5-[5-(trifluoromethyl)-1H-imidazol-2-yl]phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C24H19F3N4O2
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
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CP0210678
|
N-[2-methyl-5-(5-methyl-1H-imidazol-2-yl)phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C24H22N4O2
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
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CP0290958
|
N-[5-(1H-benzimidazol-2-yl)-2-methylphenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C27H22N4O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
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CP0290960
|
N-[2-methyl-5-(1-methylimidazol-4-yl)phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C24H22N4O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0290959
|
N-[5-(1,5-dimethylimidazol-2-yl)-2-methylphenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C25H24N4O2
|
1
|
| 1 |
IC50 < 6 nM
|
|
|
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CP0228021
|
N-[2-methyl-5-(2-methyl-1H-imidazol-5-yl)phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C24H22N4O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
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CP0247151
|
N-[2-methyl-5-(5-methyl-1H-imidazol-4-yl)phenyl]-4-(pyridin-2-ylmethoxy)benzamide
Show/Hide
|
C24H22N4O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
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CP0306855
|
N-[2-methyl-5-[5-(trifluoromethyl)-1H-pyrazol-3-yl]phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C24H19F3N4O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0119723
|
N-[5-(1H-imidazol-2-yl)-2-methylphenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C23H20N4O2
|
1
|
| 1 |
IC50 < 12 nM
|
|
|
|
CP0278929
|
N-[2-methyl-5-(1,3,5-trimethylpyrazol-4-yl)phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C26H26N4O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0262749
|
N-[2-methyl-5-(1-methylimidazol-2-yl)phenyl]-4-(pyridin-2-ylmethoxy)benzamide
Show/Hide
|
C24H22N4O2
|
1
|
| 1 |
IC50 < 16 nM
|
|
|
|
CP0247152
|
N-[5-(6-aminopyridazin-3-yl)-2-methylphenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C24H21N5O2
|
1
|
| 1 |
IC50 < 19 nM
|
|
|
|
CP0210673
|
N-(2-methyl-5-pyridin-2-ylphenyl)-4-(pyridin-2-ylmethoxy)benzamide
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|
C25H21N3O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0358355
|
N-[5-(1,2-dimethylimidazol-4-yl)-2-methylphenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C25H24N4O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0068085
|
2-chloro-N-(4-chloro-3-(pyridin-2-yl)phenyl)-4-(methylsulfonyl)benzamide
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|
C19H14Cl2N2O3S
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0236876
|
N-[5-(1H-imidazol-5-yl)-2-methylphenyl]-4-(pyridin-2-ylmethoxy)benzamide
Show/Hide
|
C23H20N4O2
|
1
|
| 1 |
IC50 < 40 nM
|
|
|
|
CP0340521
|
N-[2-methyl-5-[5-(morpholin-4-ylmethyl)-1,3-thiazol-2-yl]phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C28H28N4O3S
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0278930
|
N-[2-methyl-5-(1,3-thiazol-2-yl)phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C23H19N3O2S
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0340522
|
N-[2-methyl-5-(7H-purin-6-yl)phenyl]-4-(pyridin-2-ylmethoxy)benzamide
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|
C25H20N6O2
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0443136
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-(3-fluorophenyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C25H22ClFN6O
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0562124
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-pyridin-3-yl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C24H22ClN7O
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0401533
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-pyridin-2-yl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C24H22ClN7O
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0401534
|
cyclopropylmethyl 7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxylate
Show/Hide
|
C23H24ClN5O2
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0559120
|
[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
Show/Hide
|
C23H25ClN6O
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0567426
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-phenyl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C25H23ClN6O
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0487209
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-(2-fluorophenyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C25H22ClFN6O
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0572499
|
propan-2-yl 7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxylate
Show/Hide
|
C22H24ClN5O2
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0443137
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-(3,4-difluorophenyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C25H21ClF2N6O
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0481374
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-(4-fluorophenyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C25H22ClFN6O
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0149569
|
4-methyl-1-[3-(1,4-oxazinan-4-yl)phenylcarboxamido]-3-[4-(2-pyridylmethoxy)phenylcarboxamido]benzene
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|
C31H30N4O4
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
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CP0278927
|
3-Fluoro-N-{4-methyl-3-[4-(pyridin-2-ylmethoxy)-benzoylamino]-phenyl}-5-pyrrolidin-1-yl-benzamide
Show/Hide
|
C31H29FN4O3
|
2
|
| 1 |
IC50 = 450 nM
|
|
|
| 2 |
IC50 > 30000 nM
|
|
|
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CP0499374
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-(cyclopropylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C23H25ClN6O
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0558117
|
[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methanone
Show/Hide
|
C25H29ClN6O2
|
1
|
| 1 |
IC50 = 550 nM
|
|
|
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CP0552750
|
N-[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-2-methoxyacetamide
Show/Hide
|
C21H23ClN6O2
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
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CP0499371
|
ethyl 7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxylate
Show/Hide
|
C21H22ClN5O2
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
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CP0572500
|
cyclopentyl 7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxylate
Show/Hide
|
C24H26ClN5O2
|
1
|
| 1 |
IC50 = 740 nM
|
|
|
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CP0473874
|
[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-morpholin-4-ylmethanone
Show/Hide
|
C23H25ClN6O2
|
1
|
| 1 |
IC50 = 790 nM
|
|
|
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CP0562125
|
N-[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]propanamide
Show/Hide
|
C21H23ClN6O
|
1
|
| 1 |
IC50 = 890 nM
|
|
|
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CP0473877
|
4-[[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]methyl]morpholine
Show/Hide
|
C23H27ClN6O
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
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CP0559121
|
phenyl 7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxylate
Show/Hide
|
C25H22ClN5O2
|
1
|
| 1 |
IC50 = 960 nM
|
|
|
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CP0316558
|
1-(3-dimethylaminophenylcarboxamido)-4-methyl-3-[4-(2-pyridylmethoxy)phenylcarboxamido]benzene
Show/Hide
|
C29H28N4O3
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
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CP0499375
|
[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-(4-hydroxypiperidin-1-yl)methanone
Show/Hide
|
C24H27ClN6O2
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
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CP0499373
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-ethyl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C21H23ClN6O
|
1
|
| 1 |
IC50 = 1300 nM
|
|
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CP0401532
|
[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-(3,5-dimethylpiperazin-1-yl)methanone
Show/Hide
|
C25H30ClN7O
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
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CP0499376
|
N-[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-2,2,2-trifluoroacetamide
Show/Hide
|
C20H18ClF3N6O
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
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CP0412779
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-methyl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C20H21ClN6O
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
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CP0202855
|
1-(3-dimethylaminophenylcarboxamido)-3-(4-isopropoxyphenylcarboxamido)-4-methylbenzene
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|
C26H29N3O3
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
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CP0473873
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-N-(2-hydroxyethyl)-N-methyl-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxamide
Show/Hide
|
C22H25ClN6O2
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
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CP0487211
|
[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]methanol
Show/Hide
|
C19H20ClN5O
|
1
|
| 1 |
IC50 = 4100 nM
|
|
|
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CP0487208
|
[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-(3-hydroxypyrrolidin-1-yl)methanone
Show/Hide
|
C23H25ClN6O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0562122
|
7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-2-carboxylic acid
Show/Hide
|
C19H18ClN5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0567425
|
[7-[5-chloro-4-(3,5-dimethylpyridin-2-yl)pyridin-2-yl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazin-2-yl]-(3-hydroxyazetidin-1-yl)methanone
Show/Hide
|
C22H23ClN6O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0227981
|
N-(2-methyl-5-pyridin-4-ylphenyl)-4-(pyridin-2-ylmethoxy)benzamide
Show/Hide
|
C25H21N3O2
|
1
|
| 1 |
IC50 > 400 nM
|
|
|
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CP0458251
|
N-(2-methyl-5-pyridin-3-ylphenyl)-4-(pyridin-2-ylmethoxy)benzamide
Show/Hide
|
C25H21N3O2
|
1
|
| 1 |
IC50 > 450 nM
|
|
|
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CP0150961
|
4-methyl-1-[3-(1,4-oxazinan-4-yl)phenylcarboxamido]-3-[4-(1,3-thiazol-4-ylmethoxy)phenylcarboxamido]benzene
Show/Hide
|
C29H28N4O4S
|
1
|
| 1 |
IC50 > 3000 nM
|
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|
