| Compound ID |
Compound Name |
Compound Formula |
|
CP0400231
|
N-(4-tert-butyl-2-fluoro-5-hydroxyphenyl)-4-oxo-1H-quinoline-3-carboxamide
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|
C20H19FN2O3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0088272
|
CHEBI:66901
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|
C24H28N2O3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0388845
|
N-(4-tert-butyl-3-hydroxyphenyl)-4-oxo-1H-quinoline-3-carboxamide
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|
C20H20N2O3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0490597
|
N-[4-tert-butyl-5-hydroxy-2-(trifluoromethyl)phenyl]-4-oxo-1H-quinoline-3-carboxamide
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|
C21H19F3N2O3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0387052
|
N-(3-tert-butyl-1H-indol-6-yl)-4-oxo-1H-quinoline-3-carboxamide
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|
C22H21N3O2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0494401
|
N-(5-tert-butyl-1H-indol-6-yl)-4-oxo-1H-quinoline-3-carboxamide
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|
C22H21N3O2
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0494402
|
N-(5-ethyl-1H-indol-6-yl)-4-oxo-1H-quinoline-3-carboxamide
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|
C20H17N3O2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0955289
|
2-(2-tert-butyl-5-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-6-fluoro-1H-indol-1-yl)-N,N,N-trimethylethanaminium
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|
C28H33F3N3O3+
|
1
|
| 1 |
EC50 = 38.1 nM
|
|
|
|
CP0408924
|
US10022352, Compound 319
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|
C28H36N2O4
|
1
|
| 1 |
EC50 = 39.05 nM
|
|
|
|
CP0525601
|
US10022352, Compound 310
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|
C26H29FN2O5
|
1
|
| 1 |
EC50 = 65.95 nM
|
|
|
|
CP0522810
|
US10022352, Compound 311
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|
C27H29F3N2O6
|
1
|
| 1 |
EC50 = 81.75 nM
|
|
|
|
CP0272151
|
N-(1H-indol-6-yl)-4-oxo-1H-quinoline-3-carboxamide
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|
C18H13N3O2
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0388846
|
N-(3-ethyl-1H-indol-6-yl)-4-oxo-1H-quinoline-3-carboxamide
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|
C20H17N3O2
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0397731
|
N-(4-tert-butyl-3-fluorophenyl)-4-oxo-1H-quinoline-3-carboxamide
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|
C20H19FN2O2
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0418616
|
N-(3-amino-4-tert-butylphenyl)-4-oxo-1H-quinoline-3-carboxamide
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|
C20H21N3O2
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0498138
|
N-(4-tert-butylphenyl)-4-oxo-1H-quinoline-3-carboxamide
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|
C20H20N2O2
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0523193
|
N-[4-tert-butyl-3-(hydroxymethyl)phenyl]-4-oxo-1H-quinoline-3-carboxamide
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|
C21H22N2O3
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0551665
|
US10022352, Compound 312
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|
C26H25F2N3O4
|
1
|
| 1 |
EC50 = 181 nM
|
|
|
|
CP0387018
|
N-(2-ethylphenyl)-4-oxo-1H-quinoline-3-carboxamide
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|
C18H16N2O2
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0387053
|
4-oxo-N-(4-propan-2-ylphenyl)-1H-quinoline-3-carboxamide
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|
C19H18N2O2
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0445051
|
4-oxo-N-(2-propan-2-ylphenyl)-1H-quinoline-3-carboxamide
Show/Hide
|
C19H18N2O2
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0408925
|
US10022352, Compound 314
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|
C24H21F3N2O3
|
1
|
| 1 |
EC50 = 228.5 nM
|
|
|
|
CP0408926
|
US10022352, Compound 315
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|
C26H27F3N2O6
|
1
|
| 1 |
EC50 = 272 nM
|
|
|
|
CP0525600
|
US10022352, Compound 313
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|
C24H21F2N3O3
|
1
|
| 1 |
EC50 = 283.5 nM
|
|
|
|
CP0921723
|
(S)-1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-(2-(4-(2,3-dihydroxypropoxy)-2-methylbutan-2-yl)-6-fluoro-1H-indol-5-yl)cyclopropanecarboxamide
Show/Hide
|
C27H29F3N2O6
|
1
|
| 1 |
EC50 = 285 nM
|
|
|
|
CP0523194
|
N-(3-amino-4-propan-2-ylphenyl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0417059
|
N-(3-amino-4-propylphenyl)-4-oxo-1H-quinoline-3-carboxamide
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|
C19H19N3O2
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0445050
|
N-(2,3-dihydro-1H-indol-6-yl)-4-oxo-1H-quinoline-3-carboxamide
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|
C18H15N3O2
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0400233
|
N-naphthalen-2-yl-4-oxo-1H-quinoline-3-carboxamide
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|
C20H14N2O2
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0487794
|
N-(4-ethylphenyl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C18H16N2O2
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0522808
|
US10022352, Compound 307
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|
C28H34N2O3
|
1
|
| 1 |
EC50 = 981 nM
|
|
|
|
CP0398461
|
4-oxo-N-phenyl-1H-quinoline-3-carboxamide
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|
C16H12N2O2
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0418619
|
N-(2,6-diethylphenyl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C20H20N2O2
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0555911
|
N-(3-amino-4-ethylphenyl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C18H17N3O2
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0942361
|
(R)-N-(2-tert-butyl-1-(2,3-dihydroxypropyl)-1H-indol-5-yl)-1-(3,4-dihydroxyphenyl)cyclopropanecarboxamide
Show/Hide
|
C25H30N2O5
|
1
|
| 1 |
EC50 = 1810 nM
|
|
|
|
CP0295398
|
N,N-dibenzyl-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C24H20N2O2
|
1
|
| 1 |
EC50 = 2100 nM
|
|
|
|
CP0445474
|
US10022352, Compound 308
Show/Hide
|
C30H35F3N2O8
|
1
|
| 1 |
EC50 = 3095 nM
|
|
|
|
CP0411631
|
N,N-dibenzyl-1-hydroxynaphthalene-2-carboxamide
Show/Hide
|
C25H21NO2
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0417058
|
methyl N-[2-tert-butyl-5-[(4-oxo-1H-quinoline-3-carbonyl)amino]phenyl]carbamate
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|
C22H23N3O4
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0530774
|
US10022352, Compound 320
Show/Hide
|
C23H21F3N2O4
|
1
|
| 1 |
EC50 = 4315 nM
|
|
|
|
CP0942360
|
N-(2-tert-butyl-1H-indol-5-yl)-1-(4-methoxyphenyl)-2,2-dimethylcyclopropanecarboxamide
Show/Hide
|
C25H30N2O2
|
1
|
| 1 |
EC50 = 4525 nM
|
|
|
|
CP0523192
|
N-(4-tert-butyl-3-sulfamoylphenyl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C20H21N3O4S
|
1
|
| 1 |
EC50 = 5100 nM
|
|
|
|
CP0400232
|
N-(1H-indazol-6-yl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C17H12N4O2
|
1
|
| 1 |
EC50 = 5600 nM
|
|
|
|
CP0504636
|
N-(3-amino-4-methylphenyl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C17H15N3O2
|
1
|
| 1 |
EC50 = 6000 nM
|
|
|
|
CP0411592
|
N-(1H-indol-5-yl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C18H13N3O2
|
1
|
| 1 |
EC50 = 6100 nM
|
|
|
|
CP0511173
|
N-(1-methylindol-6-yl)-4-oxo-1H-quinoline-3-carboxamide
Show/Hide
|
C19H15N3O2
|
1
|
| 1 |
EC50 = 6400 nM
|
|
|
|
CP0418617
|
N-(3-aminophenyl)-4-oxo-1H-quinoline-3-carboxamide
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|
C16H13N3O2
|
1
|
| 1 |
EC50 = 6900 nM
|
|
|
|
CP0557217
|
N-[2-(cyanomethyl)phenyl]-4-oxo-1H-quinoline-3-carboxamide
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|
C18H13N3O2
|
1
|
| 1 |
EC50 = 8500 nM
|
|
|
|
CP0400234
|
N,N-dibenzylquinoline-3-carboxamide
Show/Hide
|
C24H20N2O
|
1
|
| 1 |
EC50 = 16000 nM
|
|
|
