| Compound ID |
Compound Name |
Compound Formula |
|
CP0055808
|
3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-methylpropan-1-amine
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|
C18H22N2
|
4
|
| 1 |
IC50 = 0.93 nM
|
|
|
| 2 |
IC50 = 1.5 nM
|
|
|
| 3 |
IC50 = 3.9 nM
|
|
|
| 4 |
Ki = 0.92 nM
|
|
|
|
CP0051283
|
ATOMOXETINE
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|
C17H21NO
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0196465
|
(R)-2-((R)-(2-ethoxyphenoxy)(phenyl)methyl)morpholine
Show/Hide
|
C19H23NO3
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0008168
|
CAS_136434-34-9
Show/Hide
|
C18H19NOS
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0411809
|
2-[3-[[(1R,5S)-8-azabicyclo[3.2.1]octan-3-yl]oxy]phenyl]benzonitrile
Show/Hide
|
C20H20N2O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0478141
|
US9120771, KHG26767
Show/Hide
|
C16H15Cl2NO
|
1
|
| 1 |
IC50 = 5.5 nM
|
|
|
|
CP0101880
|
3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine
Show/Hide
|
C17H21NO2
|
3
|
| 1 |
IC50 = 6 nM
|
|
|
| 2 |
IC50 = 7.943 nM
|
|
|
| 3 |
IC50 = 8.3 nM
|
|
|
|
CP0434278
|
(R)-1-(1-(3,5-difluorophenyl)-3-(methylamino)propyl)-7-fluoro-3,3-dimethylindolin-2-one
Show/Hide
|
C20H21F3N2O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0375016
|
(R)-1-(1-(3-chlorophenyl)-3-(methylamino)propyl)-7-fluoro-3,3-dimethylindolin-2-one
Show/Hide
|
C20H22ClFN2O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0428136
|
(R)-3,3-dimethyl-1-(3-(methylamino)-1-phenylpropyl)indolin-2-one
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|
C20H24N2O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0281531
|
2-[6-[[(1S,5R)-8-azabicyclo[3.2.1]octan-3-yl]oxy]pyridin-2-yl]benzonitrile
Show/Hide
|
C19H19N3O
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0394661
|
(1S,5R)-3-(3-iodophenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C13H16INO
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0503544
|
CHEMBL1644610
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|
C20H18N4O
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0520033
|
CHEMBL1644476
Show/Hide
|
C13H16BrNO
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0405570
|
N-methyl-3-naphthalen-2-yl-3-(tetrazol-2-yl)propan-1-amine
Show/Hide
|
C15H17N5
|
1
|
| 1 |
IC50 = 13.3 nM
|
|
|
|
CP0434276
|
(R)-7-fluoro-1-(1-(3-fluorophenyl)-3-(methylamino)propyl)-3,3-dimethylindolin-2-one
Show/Hide
|
C20H22F2N2O
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0387636
|
(3aS,6aR)-3a-naphthalen-2-yl-2,3,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole
Show/Hide
|
C17H19N
|
1
|
| 1 |
IC50 = 14.13 nM
|
|
|
|
CP0487891
|
(S)-3-(5-(2H-1,2,3-triazol-2-yl)-2H-tetrazol-2-yl)-3-(3,4-dichlorophenyl)-N-methylpropan-1-amine
Show/Hide
|
C13H14Cl2N8
|
1
|
| 1 |
IC50 = 14.7 nM
|
|
|
|
CP0504293
|
(R)-1-(1-(3-chloro-5-fluorophenyl)-3-(methylamino)propyl)-7-fluoro-3,3-dimethylindolin-2-one
Show/Hide
|
C20H21ClF2N2O
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0503541
|
CHEMBL1644474
Show/Hide
|
C13H16ClNO
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0089865
|
(S)-3-(3,4-dichlorophenyl)-N-methyl-3-(5-methyl-2H-tetrazol-2-yl)propan-1-amine
Show/Hide
|
C12H15Cl2N5
|
1
|
| 1 |
IC50 = 19.8 nM
|
|
|
|
CP0426647
|
(3aR,6aS)-3a-(3,4-dichlorophenyl)-2-methyl-1,3,4,5,6,6a-hexahydrocyclopenta[c]pyrrole
Show/Hide
|
C14H17Cl2N
|
1
|
| 1 |
IC50 = 22.39 nM
|
|
|
|
CP0089680
|
(1S,2R)-1-(1H-indol-1-yl)-3-(methylamino)-1-phenylpropan-2-ol
Show/Hide
|
C18H20N2O
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0443740
|
US9120771, KHG26774
Show/Hide
|
C17H17Cl2NO
|
1
|
| 1 |
IC50 = 25.8 nM
|
|
|
|
CP0428137
|
1'-[(1R)-1-(3-fluorophenyl)-3-(methylamino)propyl]-1',2'-dihydrospiro[cyclohexane-1,3'-indole]-2'-one
Show/Hide
|
C23H27FN2O
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0083154
|
2-[(2S,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]ethanamine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0108780
|
(1S,5R)-3-(6-phenylpyridin-2-yl)oxy-8-azabicyclo[3.2.1]octane
Show/Hide
|
C18H20N2O
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0387630
|
(3aS,7aR)-7a-(3,4-dichlorophenyl)-2-ethyl-3,3a,4,5,6,7-hexahydro-1H-isoindole
Show/Hide
|
C16H21Cl2N
|
1
|
| 1 |
IC50 = 26.92 nM
|
|
|
|
CP0083152
|
(2R,4S)-4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C17H17Cl2N
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0435090
|
US9120771, KHG26776
Show/Hide
|
C17H17Cl2NO
|
1
|
| 1 |
IC50 = 27.1 nM
|
|
|
|
CP0411740
|
[(2S,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]methanamine
Show/Hide
|
C17H17Cl2N
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0515004
|
US9120771, KHG26775
Show/Hide
|
C17H17Cl2NO
|
1
|
| 1 |
IC50 = 28.4 nM
|
|
|
|
CP0407622
|
(1S,5R)-3-(3-chloro-5-phenylphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C19H20ClNO
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0394664
|
3-[3-[[(1S,5R)-8-azabicyclo[3.2.1]octan-3-yl]oxy]phenyl]benzonitrile
Show/Hide
|
C20H20N2O
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0429536
|
(3aR,7aS)-7a-(3,4-dichlorophenyl)-2-ethyl-3,3a,4,5,6,7-hexahydro-1H-isoindole
Show/Hide
|
C16H21Cl2N
|
1
|
| 1 |
IC50 = 38.02 nM
|
|
|
|
CP0049225
|
(2S,4S)-4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C17H17Cl2N
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0374268
|
3-(1H-indol-1-yl)-N-methyl-3-phenylpropan-1-amine
Show/Hide
|
C18H20N2
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0417752
|
1'-[(1R)-3-(methylamino)-1-phenylpropyl]-1',2'-dihydrospiro[cyclohexane-1,3'-indole]-2'-one
Show/Hide
|
C23H28N2O
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0394673
|
(1S,5R)-3-phenoxy-8-azabicyclo[3.2.1]octane
Show/Hide
|
C13H17NO
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0451981
|
(3aS,7aR)-7a-(3,4-dichlorophenyl)-2-methyl-3,3a,4,5,6,7-hexahydro-1H-isoindole
Show/Hide
|
C15H19Cl2N
|
1
|
| 1 |
IC50 = 56.23 nM
|
|
|
|
CP0394663
|
4-[3-[[(1R,5S)-8-azabicyclo[3.2.1]octan-3-yl]oxy]phenyl]benzonitrile
Show/Hide
|
C20H20N2O
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0387639
|
(3aR,6aS)-3a-naphthalen-2-yl-2,3,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole
Show/Hide
|
C17H19N
|
1
|
| 1 |
IC50 = 60.26 nM
|
|
|
|
CP0066127
|
3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11-yl)-N,N-dimethyl-propan-1-amine;hydrochloride
Show/Hide
|
C19H23ClN2
|
1
|
| 1 |
IC50 = 64.6 nM
|
|
|
|
CP0407692
|
(1S,5R)-3-(3-fluorophenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C13H16FNO
|
1
|
| 1 |
IC50 = 67 nM
|
|
|
|
CP0417119
|
3-(3,4-dichlorophenyl)-N-methyl-3-(tetrazol-2-yl)propan-1-amine
Show/Hide
|
C11H13Cl2N5
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0083153
|
1-[(2R,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]-N-methylmethanamine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0048099
|
1-(3,4-dichlorophenyl)-3-aza-bicyclo[3.1.0]hexane
Show/Hide
|
C11H11Cl2N
|
1
|
| 1 |
IC50 = 72.4 nM
|
|
|
|
CP0116683
|
(2R,4R)-4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C17H17Cl2N
|
1
|
| 1 |
IC50 = 73 nM
|
|
|
|
CP0394670
|
(1R,5S)-3-(3-fluoro-5-phenylphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C19H20FNO
|
1
|
| 1 |
IC50 = 85 nM
|
|
|
|
CP0503579
|
(1R,5S)-8-methyl-3-phenoxy-8-azabicyclo[3.2.1]octane
Show/Hide
|
C14H19NO
|
1
|
| 1 |
IC50 = 86 nM
|
|
|
|
CP0336186
|
2-[[(1R,5S)-8-azabicyclo[3.2.1]octan-3-yl]oxy]-6-phenylpyridine-4-carbonitrile
Show/Hide
|
C19H19N3O
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0490758
|
US9120771, KHG26766
Show/Hide
|
C16H16ClNO
|
1
|
| 1 |
IC50 = 90.2 nM
|
|
|
|
CP0407623
|
(1S,5R)-3-(3-nitrophenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C13H16N2O3
|
1
|
| 1 |
IC50 = 91 nM
|
|
|
|
CP0501296
|
[(2R,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]methanamine
Show/Hide
|
C17H17Cl2N
|
1
|
| 1 |
IC50 = 92 nM
|
|
|
|
CP0439420
|
(1S,5R)-3-(3-methylphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C14H19NO
|
1
|
| 1 |
IC50 = 92 nM
|
|
|
|
CP0477235
|
US9120771, KHG26770
Show/Hide
|
C17H17Cl2NO
|
1
|
| 1 |
IC50 = 93.1 nM
|
|
|
|
CP0394707
|
(2R,4R)-4-(3,4-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 98 nM
|
|
|
|
CP0046806
|
(3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-fluorophenyl)piperidine
Show/Hide
|
C19H20FNO3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0376794
|
(3aR,6aS)-3a-(3,4-dichlorophenyl)-2,3,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole
Show/Hide
|
C13H15Cl2N
|
1
|
| 1 |
IC50 = 107.15 nM
|
|
|
|
CP0081549
|
(1S,2R)-1-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C17H17Cl2N
|
1
|
| 1 |
IC50 = 112 nM
|
|
|
|
CP0285130
|
(2S,4R)-4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C17H17Cl2N
|
1
|
| 1 |
IC50 = 117 nM
|
|
|
|
CP0468239
|
(2R,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C16H15Cl2N
|
1
|
| 1 |
IC50 = 124 nM
|
|
|
|
CP0083159
|
1-[(2S,4R)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]-N-methylmethanamine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 126 nM
|
|
|
|
CP0499117
|
3-[[(1R,5S)-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile
Show/Hide
|
C14H16N2O
|
1
|
| 1 |
IC50 = 126 nM
|
|
|
|
CP0394667
|
(1R,5S)-3-[3-(trifluoromethyl)phenoxy]-8-azabicyclo[3.2.1]octane
Show/Hide
|
C14H16F3NO
|
1
|
| 1 |
IC50 = 128 nM
|
|
|
|
CP0503543
|
CHEMBL1644601
Show/Hide
|
C19H20BrNO
|
1
|
| 1 |
IC50 = 132 nM
|
|
|
|
CP0387632
|
(3aR,7aS)-7a-(3,4-dichlorophenyl)-2-methyl-3,3a,4,5,6,7-hexahydro-1H-isoindole
Show/Hide
|
C15H19Cl2N
|
1
|
| 1 |
IC50 = 141.25 nM
|
|
|
|
CP0499118
|
3-[[(1S,5R)-8-azabicyclo[3.2.1]octan-3-yl]oxy]-5-phenylbenzonitrile
Show/Hide
|
C20H20N2O
|
1
|
| 1 |
IC50 = 148 nM
|
|
|
|
CP0419304
|
US9120771, KHG26757
Show/Hide
|
C12H15Cl2NO
|
1
|
| 1 |
IC50 = 153 nM
|
|
|
|
CP0049223
|
2-[(2R,4R)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]ethanamine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 158 nM
|
|
|
|
CP0394706
|
(2S,4S)-4-(3,4-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0501295
|
(2R,4S)-4-(3,4-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 167 nM
|
|
|
|
CP0411739
|
(2S,4R)-4-(3,4-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 174 nM
|
|
|
|
CP0503883
|
(2R,4R)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C16H15Cl2N
|
1
|
| 1 |
IC50 = 174 nM
|
|
|
|
CP0489375
|
(R)-7-fluoro-3,3-dimethyl-1-(3-(methylamino)-1-phenylpropyl)indolin-2-one
Show/Hide
|
C20H23FN2O
|
1
|
| 1 |
IC50 = 175 nM
|
|
|
|
CP0407691
|
(1R,5S)-3-(2-chlorophenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C13H16ClNO
|
1
|
| 1 |
IC50 = 188 nM
|
|
|
|
CP0429868
|
(3aR,6aS)-2-methyl-3a-naphthalen-2-yl-1,3,4,5,6,6a-hexahydrocyclopenta[c]pyrrole
Show/Hide
|
C18H21N
|
1
|
| 1 |
IC50 = 190.55 nM
|
|
|
|
CP0376793
|
(3aS,7aR)-7a-(3,4-dichlorophenyl)-1,2,3,3a,4,5,6,7-octahydroisoindole
Show/Hide
|
C14H17Cl2N
|
1
|
| 1 |
IC50 = 204.17 nM
|
|
|
|
CP0851839
|
cis-(3aR,7aS)-2-methyl-3a-(naphthalen-1-yl)octahydro-1H-isoindole
Show/Hide
|
C19H23N
|
1
|
| 1 |
IC50 = 204.17 nM
|
|
|
|
CP0387635
|
(3aS,6aR)-3a-(3,4-dichlorophenyl)-2,3,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole
Show/Hide
|
C13H15Cl2N
|
1
|
| 1 |
IC50 = 208.93 nM
|
|
|
|
CP0141444
|
1-[(2S,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]-N-methylmethanamine
Show/Hide
|
C18H19Cl2N
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0481163
|
US9120771, KHG26773
Show/Hide
|
C17H15Cl2NO2
|
1
|
| 1 |
IC50 = 214 nM
|
|
|
|
CP0394668
|
(1R,5S)-3-(3-methoxyphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C14H19NO2
|
1
|
| 1 |
IC50 = 222 nM
|
|
|
|
CP0374564
|
3-(3,4-dichlorophenyl)-N,N-dimethyl-3-(tetrazol-2-yl)propan-1-amine
Show/Hide
|
C12H15Cl2N5
|
1
|
| 1 |
IC50 = 234 nM
|
|
|
|
CP0394734
|
[(2R,4R)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]methanamine
Show/Hide
|
C17H17Cl2N
|
1
|
| 1 |
IC50 = 257 nM
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CP0377167
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N,N-dimethyl-3-naphthalen-2-yl-3-(tetrazol-2-yl)propan-1-amine
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C16H19N5
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1
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| 1 |
IC50 = 264 nM
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CP0394731
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1-[(2R,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]-N,N-dimethylmethanamine
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C19H21Cl2N
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1
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| 1 |
IC50 = 309 nM
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CP0425515
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US9120771, KHG26756
Show/Hide
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C11H13Cl2NO
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1
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| 1 |
IC50 = 339 nM
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CP0499508
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(1S,5R)-3-(4-chlorophenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
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C13H16ClNO
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1
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| 1 |
IC50 = 347 nM
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CP0411738
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[(2S,4R)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]methanamine
Show/Hide
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C17H17Cl2N
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1
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| 1 |
IC50 = 371 nM
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CP0394730
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1-[(2R,4R)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]-N-methylmethanamine
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C18H19Cl2N
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1
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| 1 |
IC50 = 372 nM
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CP0391998
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3-(3-chlorophenyl)-4-(3,4-dichlorophenyl)pyrrolidin-2-one
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C16H12Cl3NO
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1
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| 1 |
IC50 = 384.2 nM
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CP0379676
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4-(3,4-dichlorophenyl)-3-naphthalen-2-ylpyrrolidin-2-one
Show/Hide
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C20H15Cl2NO
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1
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| 1 |
IC50 = 482.9 nM
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CP0391999
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3-(2-chlorophenyl)-4-(3,4-dichlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H12Cl3NO
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1
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| 1 |
IC50 = 509.5 nM
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CP0387633
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(3aS,7aR)-2-methyl-7a-naphthalen-2-yl-3,3a,4,5,6,7-hexahydro-1H-isoindole
Show/Hide
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C19H23N
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1
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| 1 |
IC50 = 537.03 nM
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CP0851835
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Cis-rac-(3aS,7aR)-2-methyl-3a-phenyloctahydro-1H-isoindole
Show/Hide
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C15H21N
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1
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| 1 |
IC50 = 562.34 nM
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CP0035258
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N-methyl-3-phenyl-3-[4-(trifluoromethyl)phenoxy]propan-1-amine
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C17H18F3NO
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2
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| 1 |
IC50 = 563 nM
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| 2 |
IC50 = 2535 nM
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CP0394736
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1-[(2S,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl]-N,N-dimethylmethanamine
Show/Hide
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C19H21Cl2N
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1
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| 1 |
IC50 = 565 nM
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CP0054778
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CAS_93413-69-5
Show/Hide
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C17H27NO2
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1
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| 1 |
IC50 = 581 nM
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CP0499847
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US9120771, KHG26754
Show/Hide
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C12H16ClNO
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1
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| 1 |
IC50 = 666 nM
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CP0394733
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(2S,4R)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
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C16H15Cl2N
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1
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| 1 |
IC50 = 731 nM
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CP0223721
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(1S,2S)-1-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
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C17H17Cl2N
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1
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| 1 |
IC50 = 766 nM
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CP0035683
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(1S,4S)-4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine;hydrochloride
Show/Hide
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C17H17Cl2N
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1
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| 1 |
IC50 = 825 nM
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CP0498485
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(2S,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
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C16H15Cl2N
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1
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| 1 |
IC50 = 855 nM
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CP0404045
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4-(3,4-dichlorophenyl)-3-phenylpyrrolidin-2-one
Show/Hide
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C16H13Cl2NO
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1
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| 1 |
IC50 = 865.7 nM
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CP0520034
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CHEMBL1644600
Show/Hide
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C20H20F3NO
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1
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| 1 |
IC50 = 891 nM
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CP0872272
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Cis-rac-(3aS,7aR)-3a-(2,4-dichlorophenyl)-2-methyloctahydro-1H-isoindole
Show/Hide
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C15H19Cl2N
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1
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| 1 |
IC50 = 912.01 nM
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CP0404046
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3,4-bis(3,4-dichlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H11Cl4NO
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1
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| 1 |
IC50 = 990.3 nM
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CP0408473
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4-(4-chlorophenyl)-3-naphthalen-2-ylpyrrolidin-2-one
Show/Hide
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C20H16ClNO
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1
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| 1 |
IC50 = 1187 nM
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CP0435089
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US9120771, KHG26769
Show/Hide
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C17H18ClNO
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1
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| 1 |
IC50 = 1344 nM
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CP0404042
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4-(2-chlorophenyl)-3-naphthalen-2-ylpyrrolidin-2-one
Show/Hide
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C20H16ClNO
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1
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| 1 |
IC50 = 1376 nM
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CP0049224
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(1R,2R)-1-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
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C17H17Cl2N
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1
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| 1 |
IC50 = 1642 nM
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CP0425516
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US9120771, KHG26765
Show/Hide
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C12H17NO
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1
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| 1 |
IC50 = 1660 nM
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CP0379668
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4-(3-chlorophenyl)-3-(4-chlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H13Cl2NO
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1
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| 1 |
IC50 = 1662 nM
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CP0379669
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4-(4-chlorophenyl)-3-(3,4-dichlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H12Cl3NO
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1
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| 1 |
IC50 = 1900 nM
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CP0379670
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3-(4-chlorophenyl)-4-(3,4-dichlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H12Cl3NO
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1
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| 1 |
IC50 = 2033 nM
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CP0478142
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US9120771, KHG26768
Show/Hide
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C17H19NO
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1
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| 1 |
IC50 = 2299 nM
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CP0851836
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Cis-rac-(3aS,7aR)-3a-(3,4-difluorophenyl)-2-methyloctahydro-1H-isoindole
Show/Hide
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C15H19F2N
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1
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| 1 |
IC50 = 2344.23 nM
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CP0872268
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Cis-rac-(3aS,7aR)-3a-(3-methoxyphenyl)-2-methyloctahydro-1H-isoindole
Show/Hide
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C16H23NO
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1
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| 1 |
IC50 = 2454.71 nM
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CP0379744
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4-(2-chlorophenyl)-3-(3,4-dichlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H12Cl3NO
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1
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| 1 |
IC50 = 2521 nM
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CP0391997
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4-(3-chlorophenyl)-3-(3,4-dichlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H12Cl3NO
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1
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| 1 |
IC50 = 2745 nM
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CP0872278
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(3aS,7aS)-3a-(3,4-dichlorobenzyl)octahydro-1H-isoindole
Show/Hide
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C15H19Cl2N
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1
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| 1 |
IC50 = 2951.21 nM
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CP0443830
|
US9120771, KHG26772
Show/Hide
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C17H16ClNO2
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1
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| 1 |
IC50 = 3475 nM
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CP0379743
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3-(2-chlorophenyl)-4-(4-chlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H13Cl2NO
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1
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| 1 |
IC50 = 3570 nM
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CP0851840
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rac-(3aS,7aS)-3a-(3,4-dichlorobenzyl)-2-methyloctahydro-1H-isoindole
Show/Hide
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C16H21Cl2N
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1
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| 1 |
IC50 = 3801.89 nM
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CP0403777
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3-(3-chlorophenyl)-4-(4-chlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H13Cl2NO
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1
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| 1 |
IC50 = 3825 nM
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CP0916858
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cis-rac-(3aS,6aR)-3a-(3,5-dichlorophenyl)-2-methyloctahydrocyclopenta[c]pyrrole
Show/Hide
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C14H17Cl2N
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1
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| 1 |
IC50 = 4265.8 nM
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CP0917254
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rac-(3aR,7aR)-3a-(3,4-dichlorobenzyl)-2-methyloctahydro-1H-isoindole
Show/Hide
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C16H21Cl2N
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1
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| 1 |
IC50 = 4466.84 nM
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CP0391963
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3,4-bis(4-chlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H13Cl2NO
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1
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| 1 |
IC50 = 5176 nM
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CP0923145
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(3aR,7aR)-3a-(3,4-dichlorobenzyl)octahydro-1H-isoindole
Show/Hide
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C15H19Cl2N
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1
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| 1 |
IC50 = 5370.32 nM
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CP0888363
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Cis-rac-(3aS,7aR)-3a-(3,4-dimethoxyphenyl)-2-methyloctahydro-1H-isoindole
Show/Hide
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C17H25NO2
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1
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| 1 |
IC50 = 5888.44 nM
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CP0871340
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cis-rac-(3aS,6aR)-3a-(3,4-difluorophenyl)-2-methyloctahydrocyclopenta[c]pyrrole
Show/Hide
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C14H17F2N
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1
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| 1 |
IC50 = 6456.54 nM
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CP0166272
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(1R,2S)-1-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C17H17Cl2N
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1
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| 1 |
IC50 = 7262 nM
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CP0486949
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4-(2-chlorophenyl)-3-(4-chlorophenyl)pyrrolidin-2-one
Show/Hide
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C16H13Cl2NO
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1
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| 1 |
IC50 = 7619 nM
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CP0916857
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cis-rac-(3aS,6aR)-3a-(3-methoxyphenyl)-2-methyloctahydrocyclopenta[c]pyrrole
Show/Hide
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C15H21NO
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1
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| 1 |
IC50 > 10000 nM
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CP0940723
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cis-rac-(3aS,6aR)-3a-(4-methoxyphenyl)-2-methyloctahydrocyclopenta[c]pyrrole
Show/Hide
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C15H21NO
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1
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| 1 |
IC50 > 10000 nM
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CP0851838
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Cis-rac-(3aS,7aR)-3a-(4-methoxyphenyl)-2-methyloctahydro-1H-isoindole
Show/Hide
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C16H23NO
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1
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| 1 |
IC50 = 14125.38 nM
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CP0375015
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1'-[(1S)-3-(methylamino)-1-phenylpropyl]-1',2'-dihydrospiro[cyclohexane-1,3'-indole]-2'-one
Show/Hide
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C23H28N2O
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1
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| 1 |
IC50 > 3000 nM
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CP0428142
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1'-[(1S)-1-(3-fluorophenyl)-3-(methylamino)propyl]-1',2'-dihydrospiro[cyclohexane-1,3'-indole]-2'-one
Show/Hide
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C23H27FN2O
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1
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| 1 |
IC50 > 3000 nM
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CP0434279
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(S)-3,3-dimethyl-1-(3-(methylamino)-1-phenylpropyl)indolin-2-one
Show/Hide
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C20H24N2O
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1
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| 1 |
IC50 > 3000 nM
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