| Compound ID |
Compound Name |
Compound Formula |
|
CP0472123
|
2-{6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]pyridin-3-yl}propan-2-ol
Show/Hide
|
C27H29N5O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0455389
|
1-{6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]pyridin-3-yl}1-methylethylamine
Show/Hide
|
C27H30N6
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0497372
|
1-{6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]pyridin-3-yl}cyclopropanol
Show/Hide
|
C27H27N5O
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0498345
|
6-[(R)-4-(4-Benzylphthalazin-1-yl)-2-methylpiperazin-1-yl]nicotinonitrile
Show/Hide
|
C26H24N6
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0502393
|
6-{4-[4-(4-Chlorobenzyl)phthalazin-1-yl]piperazin-1-yl}nicotinonitrile
Show/Hide
|
C25H21ClN6
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0455398
|
6-[(S)-4-(4-Benzylphthalazin-1-yl)-3-methylpiperazin-1-yl]nicotinonitrile
Show/Hide
|
C26H24N6
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0457490
|
6-{4-[4-(4-Cyanobenzyl)phthalazin-1-yl]piperazin-1-yl}nicotinonitrile
Show/Hide
|
C26H21N7
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0452552
|
(+/-)-2-{6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]pyridin-3-yl}propane-1,2-diol
Show/Hide
|
C27H29N5O2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0452558
|
6-{4-[4-(3-Chlorobenzyl)phthalazin-1-yl]piperazin-1-yl}nicotinonitrile
Show/Hide
|
C25H21ClN6
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0397016
|
1-{6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]pyridin-3-yl}ethanol
Show/Hide
|
C26H27N5O
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0422210
|
6-[(S)-4-(4-Benzylphthalazin-1-yl)-2-methylpiperazin-1-yl]nicotinonitrile
Show/Hide
|
C26H24N6
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0422211
|
6-{4-[4-(4-Fluorobenzyl)phthalazin-1-yl]piperazin-1-yl}nicotinonitrile
Show/Hide
|
C25H21FN6
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0457488
|
6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]nicotinonitrile
Show/Hide
|
C25H22N6
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0387836
|
1-Benzyl-4-[4-(5-trifluoromethylpyridin-2-yl)piperazin-1-yl]phthalazine
Show/Hide
|
C25H22F3N5
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0457489
|
6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]pyridine-3-sulfonicAcid Amide
Show/Hide
|
C24H24N6O2S
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0452554
|
N-[[6-[4-(4-benzylphthalazin-1-yl)piperazin-1-yl]pyridin-3-yl]methyl]acetamide
Show/Hide
|
C27H28N6O
|
1
|
| 1 |
IC50 = 96 nM
|
|
|
|
CP0374376
|
7-Benzyl-4-[4-(5-trifluoromethylpyridin-2-yl)piperazin-1-yl]furo[2,3-d]pyridazine
Show/Hide
|
C23H20F3N5O
|
1
|
| 1 |
IC50 = 139 nM
|
|
|
|
CP0474046
|
6-[4-(4-Benzylphthalazin-1-yl)[1,4]diazepan-1-yl]nicotinonitrile
Show/Hide
|
C26H24N6
|
1
|
| 1 |
IC50 = 153 nM
|
|
|
|
CP0407677
|
4-{4-[4-(5-Cyanopyridin-2-yl)piperazin-1-yl]phthalazin-1-ylmethyl}benzoic Acid Methyl Ester
Show/Hide
|
C27H24N6O2
|
1
|
| 1 |
IC50 = 165 nM
|
|
|
|
CP0497373
|
6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]nicotinamide
Show/Hide
|
C25H24N6O
|
1
|
| 1 |
IC50 = 173 nM
|
|
|
|
CP0387837
|
6-[(R)-4-(4-Benzylphthalazin-1-yl)-3-methylpiperazin-1-yl]nicotinonitrile
Show/Hide
|
C26H24N6
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0457491
|
[6-[4-(4-benzylphthalazin-1-yl)piperazin-1-yl]pyridin-3-yl]methanol
Show/Hide
|
C25H25N5O
|
1
|
| 1 |
IC50 = 187 nM
|
|
|
|
CP0374377
|
6-{4-[4-(4-Trifluoromethylbenzyl)phthalazin-1-yl]piperazin-1-yl}nicotinonitrile
Show/Hide
|
C26H21F3N6
|
1
|
| 1 |
IC50 = 226 nM
|
|
|
|
CP0374378
|
1-[6-[4-(4-benzylphthalazin-1-yl)piperazin-1-yl]pyridin-3-yl]-N,N-dimethylmethanamine
Show/Hide
|
C27H30N6
|
1
|
| 1 |
IC50 = 287 nM
|
|
|
|
CP0498346
|
4-(1-Benzyl-1H-indol-3-yl)-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-5'-carbonitrile
Show/Hide
|
C26H24N4
|
1
|
| 1 |
IC50 = 386 nM
|
|
|
|
CP0452555
|
1-Benzyl-4-(4-pyridin-2-yl-piperazin-1-yl)phthalazine
Show/Hide
|
C24H23N5
|
1
|
| 1 |
IC50 = 643 nM
|
|
|
|
CP0428583
|
1-Benzyl-4-(4-phenylpiperazin-1-yl)phthalazine
Show/Hide
|
C25H24N4
|
1
|
| 1 |
IC50 = 1095 nM
|
|
|
|
CP0387803
|
6-[4-(4-Benzylphthalazin-1-yl)piperazin-1-yl]nicotinic Acid
Show/Hide
|
C25H23N5O2
|
1
|
| 1 |
IC50 = 1644 nM
|
|
|
|
CP0428584
|
1-Pyridin-4-ylmethyl-4-(4-pyridin-2-ylpiperazin-1-yl)phthalazine
Show/Hide
|
C23H22N6
|
1
|
| 1 |
IC50 = 3690 nM
|
|
|
|
CP0387801
|
4-Benzyl-7-[4-(5-trifluoromethylpyridin-2-yl)piperazin-1-yl]furo[2,3-d]pyridazine
Show/Hide
|
C23H20F3N5O
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0387805
|
4-{4-[4-(5-Cyanopyridin-2-yl)piperazin-1-yl]phthalazin-1-ylmethyl}benzoic Acid
Show/Hide
|
C26H22N6O2
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0397036
|
4-[1-(4-Benzylphthalazin-1-yl)piperidin-4-yl]benzonitrile
Show/Hide
|
C27H24N4
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0397039
|
7-Benzyl-4-[4-(5-trifluoromethylpyridin-2-yl)piperazin-1-yl]-1Himidazo[4,5-d]pyridazine
Show/Hide
|
C22H20F3N7
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0431427
|
6-[4-(4-Benzylisoquinolin-1-yl)piperazin-1-yl]nicotinonitrile
Show/Hide
|
C26H23N5
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0455276
|
6-[4-(1-Benzylisoquinolin-4-yl)piperazin-1-yl]nicotinonitrile
Show/Hide
|
C26H23N5
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
