| Compound ID |
Compound Name |
Compound Formula |
|
CP0548822
|
4-[[(1R,6R)-6-amino-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide;hydrochloride
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C22H21Cl2F2N3O3S2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0549720
|
4-[[(1R,6R)-6-amino-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methylsulfanyl]-5-chloro-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide;hydrochloride
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|
C22H21Cl2F2N3O2S3
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0563654
|
5-chloro-4-[[(1S,6R)-6-(ethylamino)-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methylamino]-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide;hydrochloride
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|
C24H26Cl2F2N4O2S2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0559188
|
5-chloro-N-(4-chloro-1,3-thiazol-2-yl)-2-fluoro-4-[[(6S)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]benzenesulfonamide
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|
C21H18Cl2F2N4O2S2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0574527
|
5-chloro-2-fluoro-4-[[(6S)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]-N-(5-fluoro-1,3-thiazol-2-yl)benzenesulfonamide
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|
C21H18ClF3N4O2S2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0547311
|
5-chloro-4-[[(1R,6R)-6-(dimethylamino)-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
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|
C24H25Cl2F2N3O3S2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0315694
|
4-[[(1R,6R)-6-amino-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
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|
C22H20ClF2N3O3S2
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0010999
|
4-[2-(5-amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
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|
C18H12Cl2FN5O3S2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0508384
|
5-chloro-2-fluoro-4-[[(6S)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]-N-(1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C21H19ClF2N4O2S2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0529279
|
4-[[(1S,6R)-6-amino-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methylamino]-5-chloro-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide;hydrochloride
Show/Hide
|
C22H22Cl2F2N4O2S2
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0508385
|
5-chloro-4-[[(6S)-5-(4-chlorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C21H19Cl2FN4O2S2
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0574964
|
5-chloro-4-[[(1R,6R)-6-(ethylamino)-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methoxy]-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide;hydrochloride
Show/Hide
|
C24H25Cl2F2N3O3S2
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0472870
|
4-[[(1R,6R)-6-amino-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methylsulfanyl]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
Show/Hide
|
C22H21Cl2F2N3O2S3
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0566519
|
2,5-difluoro-4-[[(6S)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]-N-(1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C21H19F3N4O2S2
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0369849
|
4-[[(1S,6R)-6-amino-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methylamino]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
Show/Hide
|
C22H22Cl2F2N4O2S2
|
1
|
| 1 |
IC50 = 88 nM
|
|
|
|
CP0476408
|
5-chloro-2-fluoro-4-[[(6S)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H18ClF2N3O3S2
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0566520
|
3-chloro-4-[[(6S)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]-N-(1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C21H20ClFN4O2S2
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0567245
|
5-chloro-2-fluoro-4-[[(1R,6R)-2-(4-fluorophenyl)-6-(propan-2-ylamino)cyclohex-2-en-1-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
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|
C25H27Cl2F2N3O3S2
|
1
|
| 1 |
IC50 = 94 nM
|
|
|
|
CP0548823
|
5-chloro-4-[[(1R,6R)-6-(ethylamino)-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methylsulfanyl]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
Show/Hide
|
C24H25Cl2F2N3O2S3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0559187
|
5-chloro-2-fluoro-4-[[(6S)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H19ClF2N4O2S2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0566518
|
5-chloro-4-[[5-(2-chloro-4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H17Cl2F2N3O3S2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0552529
|
5-chloro-2-fluoro-4-[[(1R,6R)-2-(4-fluorophenyl)-6-(methylamino)cyclohex-2-en-1-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
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|
C23H23Cl2F2N3O3S2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0079810
|
2-(Dimethylamino)ethyl p-(butylamino)benzoate
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|
C15H24N2O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0513843
|
5-chloro-4-[[(1S,6R)-6-(ethylamino)-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methylamino]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
Show/Hide
|
C24H26Cl2F2N4O2S2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0566516
|
5-chloro-2-fluoro-4-[[5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H18ClF2N3O3S2
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0452115
|
5-chloro-2-fluoro-4-[[5-(3-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H18ClF2N3O3S2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0535790
|
2,5-difluoro-4-[[5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide
Show/Hide
|
C20H17F3N4O3S2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0567246
|
5-chloro-4-[[(1R,6R)-6-(diethylamino)-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
Show/Hide
|
C26H29Cl2F2N3O3S2
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
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CP0513398
|
5-chloro-4-[[5-(3,4-difluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H17ClF3N3O3S2
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0559186
|
5-chloro-2-fluoro-4-[[5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C21H18ClF2N3O3S2
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0566517
|
5-chloro-2-fluoro-4-[(5-phenyl-1,2,3,6-tetrahydropyridin-6-yl)methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H19ClFN3O3S2
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0468814
|
N-[(1R,2R)-2-[[2-chloro-5-fluoro-4-(1,3-thiazol-4-ylsulfamoyl)phenoxy]methyl]-3-(4-fluorophenyl)cyclohex-3-en-1-yl]acetamide
Show/Hide
|
C24H22ClF2N3O4S2
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
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CP0535791
|
5-chloro-4-[[5-(2-chloro-4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methylamino]-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C21H18Cl2F2N4O2S2
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
|
CP0567090
|
5-chloro-4-[[5-(3-chlorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H18Cl2FN3O3S2
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
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CP0508114
|
5-chloro-4-[[5-(5-chlorothiophen-2-yl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C19H16Cl2FN3O3S3
|
1
|
| 1 |
IC50 = 590 nM
|
|
|
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CP0535852
|
5-chloro-2-fluoro-4-[[5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(5-fluoropyridin-2-yl)benzenesulfonamide
Show/Hide
|
C23H19ClF3N3O3S
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
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CP0508382
|
5-chloro-2-fluoro-4-[[5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamide
Show/Hide
|
C20H17ClF2N4O3S2
|
1
|
| 1 |
IC50 = 700 nM
|
|
|
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CP0574963
|
5-chloro-2-fluoro-4-[[(1R,6R)-2-(4-fluorophenyl)-6-(1,2,4-triazol-4-yl)cyclohex-2-en-1-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C26H21ClF5N5O5S2
|
1
|
| 1 |
IC50 = 770 nM
|
|
|
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CP0574526
|
5-chloro-4-[[5-(4-chlorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H18Cl2FN3O3S2
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0567089
|
5-chloro-2-fluoro-4-[[5-(3-methoxyphenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C22H21ClFN3O4S2
|
1
|
| 1 |
IC50 = 1030 nM
|
|
|
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CP0472869
|
4-[[(1R,6R)-6-(azetidin-1-yl)-2-(4-fluorophenyl)cyclohex-2-en-1-yl]methoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide;hydrochloride
Show/Hide
|
C25H25Cl2F2N3O3S2
|
1
|
| 1 |
IC50 = 1150 nM
|
|
|
|
CP0535789
|
5-chloro-4-[[5-(2,4-difluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H17ClF3N3O3S2
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
|
CP0508381
|
5-chloro-2-fluoro-4-[[5-(furan-2-yl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C19H17ClFN3O4S2
|
1
|
| 1 |
IC50 = 1540 nM
|
|
|
|
CP0559184
|
5-chloro-2-fluoro-4-[[5-(4-methylphenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C22H21ClFN3O3S2
|
1
|
| 1 |
IC50 = 1670 nM
|
|
|
|
CP0547312
|
5-chloro-2-fluoro-4-[[(1R,6R)-2-(4-fluorophenyl)-6-imidazol-1-ylcyclohex-2-en-1-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide;2,2,2-trifluoroacetic acid
Show/Hide
|
C27H22ClF5N4O5S2
|
1
|
| 1 |
IC50 = 2340 nM
|
|
|
|
CP0508380
|
5-chloro-2-fluoro-4-[[5-(4-methoxyphenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C22H21ClFN3O4S2
|
1
|
| 1 |
IC50 = 3100 nM
|
|
|
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CP0448651
|
5-chloro-2-fluoro-4-[(5-pyridin-4-yl-1,2,3,6-tetrahydropyridin-6-yl)methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C20H18ClFN4O3S2
|
1
|
| 1 |
IC50 = 3920 nM
|
|
|
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CP0559185
|
5-chloro-4-[[5-(3,6-dihydro-2H-pyran-4-yl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C20H21ClFN3O4S2
|
1
|
| 1 |
IC50 = 3920 nM
|
|
|
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CP0508383
|
5-chloro-2-fluoro-4-[[5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(5-fluoropyrimidin-2-yl)benzenesulfonamide
Show/Hide
|
C22H18ClF3N4O3S
|
1
|
| 1 |
IC50 = 4800 nM
|
|
|
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CP0535851
|
5-chloro-2-fluoro-4-[[5-(1-methylpyrazol-4-yl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C19H19ClFN5O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0567194
|
5-chloro-2-fluoro-4-[[(6R)-5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C21H18ClF2N3O3S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
