Brief Information of the Compound and Protein
Compound Name
5-chloro-4-[[5-(4-chlorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
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PubChem ID
CID: 137640897
Canonical SMILES
Fc1cc(OCC2NCCC=C2c2ccc(Cl)cc2)c(Cl)cc1S(=O)(=O)Nc1cscn1
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Compound Formula C21H18Cl2FN3O3S2
Compound Structure
Protein Name
Sodium channel protein type 9 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q15858
Gene Name
SCN9A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 900 nM
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