Brief Information of the Compound and Protein
Compound Name
2,5-difluoro-4-[[5-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-6-yl]methoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide
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PubChem ID
CID: 137644331
Canonical SMILES
Fc1ccc(cc1)C1=CCCNC1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
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Compound Formula C20H17F3N4O3S2
Compound Structure
Protein Name
Sodium channel protein type 9 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q15858
Gene Name
SCN9A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 250 nM
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