Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT01348 , Dual specificity protein kinase TTK
Gene Name TTK
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P33981
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT01348
 
Compound ID Compound Name Compound Formula
CP0437416
US9512130, 2
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C27H24F5N5O3
 1
1
IC50 < 1 nM
   TI
   LI
   LO
   TS
CP0344042
JGS79C
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C33H39N7O2
 1
1
IC50 = 4.7 nM
   TI
   LI
   LO
   TS
CP0357567
N-(2,6-diethylphenyl)-2-[4-(4-methylpiperazin-1-yl)-2-(prop-2-enoylamino)anilino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide
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C35H40N8O2
 1
1
IC50 = 22.4 nM
   TI
   LI
   LO
   TS
CP0574217
N-(2,6-diethylphenyl)-2-[4-(4-methylpiperazin-1-yl)-2-(propanoylamino)anilino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide
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C35H42N8O2
 1
1
IC50 = 32.7 nM
   TI
   LI
   LO
   TS
CP0032521
9-cyclopentyl-2-[2-methoxy-4-(1-methylpiperidin-4-yl)oxyanilino]-7-methylpurin-8-one
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C24H32N6O3
 1
1
IC50 = 429 nM
   TI
   LI
   LO
   TS