Compound ID |
Compound Name |
Compound Formula |
CP0333594
|
methyl 2-[9-(4-amino-3-methoxyphenyl)-6-oxo-5,11-dihydrobenzo[b][1,4]benzodiazepin-3-yl]acetate
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|
C23H21N3O4
|
1
|
1 |
EC50 = 890 nM
|
|
|
CP0286129
|
3-(4-amino-3-methoxy-phenyl)-7-morpholin-4-yl-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one
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|
C24H24N4O3
|
2
|
1 |
EC50 = 2100 nM
|
|
|
2 |
EC50 = 46100 nM
|
|
|
CP0510897
|
4'-{6-[(trans-4-hydroxy-cyclohexylamino)-methyl]-1,4-dihydro-indeno[1,2-c]pyrazol-3-yl}-biphenyl-4-ol
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|
C29H29N3O2
|
1
|
1 |
EC50 = 2300 nM
|
|
|
CP0065182
|
2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-N,N-dimethylacetamide
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|
C24H24N4O3
|
1
|
1 |
EC50 = 2630 nM
|
|
|
CP0405447
|
4'-(6-{[(5-methyl-pyrazin-2-ylmethyl)-amino]-methyl}-1,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-biphenyl-4-ol
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|
C29H25N5O
|
1
|
1 |
EC50 = 4000 nM
|
|
|
CP0400040
|
4'-[6-(4-Hydroxy-cyclohexylmethyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl]-biphenyl-4-ol
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|
C28H27N3O2
|
1
|
1 |
EC50 = 4700 nM
|
|
|
CP0065184
|
8-(1,1-dioxo-1l6-isothiazolidin-2-yl)-3-(3-methoxy-4-nitrophenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one
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|
C23H22N4O4S
|
2
|
1 |
EC50 = 9000 nM
|
|
|
2 |
EC50 > 10000 nM
|
|
|
CP0020879
|
2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-2-methyl-N-(4-morpholin-4-ylphenyl)propanamide
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|
C34H35N5O4
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 > 59300 nM
|
|
|
CP0021747
|
2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-N-[4-(4-morpholinyl)phenyl]acetamide
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|
C32H31N5O4
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 > 59300 nM
|
|
|
CP0065181
|
3-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-N-(4-morpholin-4-ylphenyl)propanamide
Show/Hide
|
C33H33N5O4
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 > 59300 nM
|
|
|
CP0065183
|
3-(3-methoxy-4-nitrophenyl)-8-(2-oxopyrrolidin-1-yl)-5,10-dihydro-11H-dibenzo[b,e][1,4]diazepin-11-one
Show/Hide
|
C24H22N4O3
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 = 49500 nM
|
|
|
CP0185338
|
7-amino-3-(4-amino-3-methoxy-phenyl)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one
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|
C20H18N4O2
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 = 49900 nM
|
|
|
CP0195563
|
2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-7-yl]-2-methyl-N-(4-morpholin-4-ylphenyl)propanamide
Show/Hide
|
C34H35N5O4
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 > 59300 nM
|
|
|
CP0270494
|
8-methoxy-3-(3-methoxy-4-nitrophenyl)-5H-dibenzo[b,e][1,4]-diazepin-11(10H)-one
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|
C21H19N3O3
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 > 59300 nM
|
|
|
CP0333592
|
2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-7-yl]-N,N-dimethylacetamide
Show/Hide
|
C24H24N4O3
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 = 32500 nM
|
|
|
CP0333593
|
3-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5Hdibenzo[b,e][1,4]diazepin-8-yl]-N,N-dimethylpropanamide
Show/Hide
|
C25H26N4O3
|
2
|
1 |
EC50 > 10000 nM
|
|
|
2 |
EC50 = 51900 nM
|
|
|
CP0373581
|
[3-[4-(4-hydroxyphenyl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazol-6-yl]-(4-hydroxypiperidin-1-yl)methanone
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|
C28H25N3O3
|
1
|
1 |
EC50 = 25000 nM
|
|
|
CP0039009
|
3-(4'-HYDROXYBIPHENYL-4-YL)-N-(4-HYDROXYCYCLOHEXYL)-1,4-DIHYDROINDENO[1,2-C]PYRAZOLE-6-CARBOXAMIDE
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|
C29H27N3O3
|
1
|
1 |
EC50 > 59000 nM
|
|
|
CP0212707
|
3-(4'-hydroxy-biphenyl-4-yl)-1,4-dihydro-indeno[1,2-c]pyrazole-6-carboxylic acid (pyridin-4-ylmethyl)-amide
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|
C29H22N4O2
|
1
|
1 |
EC50 > 59000 nM
|
|
|
CP0295930
|
4-(6-(morpholinomethyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid
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|
C22H21N3O3
|
1
|
1 |
EC50 > 59000 nM
|
|
|
CP0373550
|
4-(6-(((1r,4r)-4-hydroxycyclohexyl)carbamoyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid
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|
C24H23N3O4
|
1
|
1 |
EC50 > 59000 nM
|
|
|
CP0374439
|
4-(6-((4-hydroxypiperidin-1-yl)methyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid
Show/Hide
|
C23H23N3O3
|
1
|
1 |
EC50 > 59000 nM
|
|
|
CP0464485
|
4-(6-(morpholinomethyl)-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzamide
Show/Hide
|
C22H22N4O2
|
1
|
1 |
EC50 > 59000 nM
|
|
|
CP0522247
|
4-{6-[(trans-4-hydroxy-cyclohexylamino)-methyl]-1,4-dihydro-indeno[1,2-c]pyrazol-3-yl}-benzoic acid
Show/Hide
|
C24H25N3O3
|
1
|
1 |
EC50 > 59000 nM
|
|
|
CP0213191
|
8-hydroxy-3-(3-methoxy-4-nitrophenyl)-5H-dibenzo[b,e][1,4]-diazepin-11(10H)-one
Show/Hide
|
C20H17N3O3
|
1
|
1 |
EC50 > 59300 nM
|
|
|