Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
 Cell Line Info 
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT03665 , Histamine H3 receptor
 Protein Info 
Gene Name HRH3
Organism Mus musculus, Mouse
Protein Classification Membrane receptor
Uniprot ID P58406
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006
 Cell Line Info 
 Protein ID: PT03665
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0041493
 Compound Info 
Clobenpropit
   Show/Hide
C14H17ClN4S
  2
1
EC50 = 1.7 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
Ki = 0.6 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0102830
 Compound Info 
3-methyl-2-(4-(3-(pyrrolidin-1-yl)propoxy)phenyl)quinazolin-4(3H)-one
   Show/Hide
C22H25N3O2
  2
1
EC50 = 9.6 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
Ki = 2.4 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0044460
 Compound Info 
N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
   Show/Hide
C15H24N4S
  2
1
EC50 = 11 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
Ki = 4.8 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0947399
 Compound Info 
3-([1,1,1-(3)H]methyl)-2-(4-{[3-(1-pyrrolidinyl)propyl]oxy}phenyl)-4(3H)-quinazolinone
   Show/Hide
C22H25N3O2
  1
1
Kd = 2.6 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0098027
 Compound Info 
2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide
   Show/Hide
C6H10N4S
  1
1
Ki = 2 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0061272
 Compound Info 
N(alpha)-Methylhistamine
   Show/Hide
C6H11N3
  1
1
Ki = 19 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0036920
 Compound Info 
2-(1H-imidazol-4-yl)ethan-1-amine
   Show/Hide
C5H9N3
  1
1
Ki = 68 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS