| Compound ID |
Compound Name |
Compound Formula |
|
CP0445349
|
(2S)-2-[[3-[[[4-(1-adamantyl)benzoyl]amino]methyl]-4-propoxyphenyl]methyl]-4-phenylbutanoic acid
Show/Hide
|
C38H45NO4
|
2
|
| 1 |
Activity = 50 nM
|
|
|
| 2 |
EC50 = 9.2 nM
|
|
|
|
CP0108032
|
(S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid
Show/Hide
|
C34H30N2O5
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0085946
|
CHEBI:79990
Show/Hide
|
C31H30N2O5
|
1
|
| 1 |
EC50 = 2.7 nM
|
|
|
|
CP0131144
|
(R)-2-Benzyl-3-(3-(((4-adamantan-1-yl)benzamido)-methyl)-4-propoxyphenyl)propanoic Acid
Show/Hide
|
C37H43NO4
|
1
|
| 1 |
EC50 = 3.6 nM
|
|
|
|
CP0064091
|
(2S,3S)-1-(4-tert-butylphenyl)-3-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C33H34N2O5
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0185954
|
2-[5-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonyl-3,6-dihydro-2H-pyridin-4-yl]acetic acid
Show/Hide
|
C32H30N2O6
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0098828
|
(5-{3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]benzyl}-2-phenyl-2H-1,2,3-triazol-4-yl)acetic acid
Show/Hide
|
C29H26N4O4
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0158747
|
2,4-dichloro-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide
Show/Hide
|
C21H12Cl4N2O3S
|
3
|
| 1 |
EC50 = 4 nM
|
|
|
| 2 |
EC50 = 150 nM
|
|
|
| 3 |
Ki = 10 nM
|
|
|
|
CP0256604
|
3-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-(2-methylpropoxycarbonyl)piperidine-4-carboxylic acid
Show/Hide
|
C30H36N2O6
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0185790
|
2-[5-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-(2-methylpropoxycarbonyl)-3,6-dihydro-2H-pyridin-4-yl]acetic acid
Show/Hide
|
C30H34N2O6
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0203503
|
2,4-dichloro-N-[3,5-dichloro-4-(5-chloropyridin-3-yl)oxyphenyl]benzenesulfonamide
Show/Hide
|
C17H9Cl5N2O3S
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0264542
|
5-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-propoxycarbonyl-3,4-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C29H32N2O6
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0159838
|
5-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-(2-methylpropoxycarbonyl)-3,4-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C30H34N2O6
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0410909
|
N-[3-acetyl-4-(5-chloropyridin-3-yl)oxyphenyl]-2,4-dichlorobenzenesulfonamide
Show/Hide
|
C19H13Cl3N2O4S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0005387
|
Avandamet
Show/Hide
|
C18H19N3O3S
|
24
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
EC50 = 35 nM
|
|
|
| 3 |
EC50 = 39 nM
|
|
|
| 4 |
EC50 = 40 nM
|
|
|
| 5 |
EC50 = 43 nM
|
|
|
| 6 |
EC50 = 45 nM
|
|
|
| 7 |
EC50 = 49 nM
|
|
|
| 8 |
EC50 = 76 nM
|
|
|
| 9 |
EC50 = 100 nM
|
|
|
| 10 |
EC50 = 120 nM
|
|
|
| 11 |
EC50 = 134 nM
|
|
|
| 12 |
EC50 = 156 nM
|
|
|
| 13 |
EC50 = 190 nM
|
|
|
| 14 |
EC50 = 260 nM
|
|
|
| 15 |
EC50 = 296.9 nM
|
|
|
| 16 |
EC50 = 300 nM
|
|
|
| 17 |
EC50 = 310 nM
|
|
|
| 18 |
EC50 = 480.6 nM
|
|
|
| 19 |
EC50 = 1100 nM
|
|
|
| 20 |
EC50 = 43710 nM
|
|
|
| 21 |
IC50 = 7.7 nM
|
|
|
| 22 |
IC50 = 88.4 nM
|
|
|
| 23 |
IC50 = 22000 nM
|
|
|
| 24 |
Kd = 47.6 nM
|
|
|
|
CP0239930
|
(3R,4S)-4-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
|
C30H28N2O6
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0484874
|
(2R)-2-[[3-[[[4-(1-adamantyl)benzoyl]amino]methyl]-4-propoxyphenyl]methyl]-3-cyclohexylpropanoic acid
Show/Hide
|
C37H49NO4
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0098837
|
2-(5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-2-phenyl-2H-1,2,3-triazol-4-yl)acetic acid
Show/Hide
|
C29H26N4O4
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0412338
|
(+/-)-2-{5-[(4-Adamantan-1-yl-benzoylamino)-methyl]-2-fluoro-4-propoxy-benzyl}-butyric acid
Show/Hide
|
C32H40FNO4
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0153538
|
5-[[4-bromo-2-(trifluoromethoxy)phenyl]sulfonylamino]-2-(5-chloropyridin-3-yl)oxy-N-ethylbenzamide
Show/Hide
|
C21H16BrClF3N3O5S
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0234393
|
2-(5-chloropyridin-3-yl)oxy-5-[(2,4-dichlorophenyl)sulfonylamino]-N-ethylbenzamide
Show/Hide
|
C20H16Cl3N3O4S
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0179484
|
5-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-phenylmethoxycarbonyl-3,4-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C33H32N2O6
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0091733
|
3-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-(2-methylpropoxycarbonyl)piperidine-4-carboxylic acid
Show/Hide
|
C30H36N2O6
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0137074
|
(2S,3S)-1-(4-methoxyphenyl)-3-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C30H28N2O6
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0142504
|
2,4-dichloro-N-[3-chloro-4-(5-chloropyridin-3-yl)oxy-5-fluorophenyl]benzenesulfonamide
Show/Hide
|
C17H9Cl4FN2O3S
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0367911
|
2-(5-chloropyridin-3-yl)oxy-5-[(3,4-dichlorophenyl)sulfonylamino]-N-ethylbenzamide
Show/Hide
|
C20H16Cl3N3O4S
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0126659
|
2-[(3R,4R)-1-ethoxycarbonyl-4-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]pyrrolidin-3-yl]acetic acid
Show/Hide
|
C27H30N2O6
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0417994
|
2-((3-((2-(4-tert-butylphenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C32H34N2O6
|
1
|
| 1 |
EC50 = 20.1 nM
|
|
|
|
CP0422713
|
(+/-)-2-{5-[(4-Adamantan-1-yl-2-fluoro-benzoylamino)-methyl]-4-ethoxy-2-fluoro-benzyl}-butyric acid
Show/Hide
|
C31H37F2NO4
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0380581
|
(S)-2-Benzyl-3-(3-(((4-adamantan-1-yl)benzamido)-methyl)-4-propoxyphenyl)propanoic Acid
Show/Hide
|
C37H43NO4
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0396452
|
(2S)-2-[[3-[[[4-(1-adamantyl)benzoyl]amino]methyl]-4-propoxyphenyl]methyl]-3-cyclohexylpropanoic acid
Show/Hide
|
C37H49NO4
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
|
CP0256519
|
5-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]-3,4-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C30H27F3N4O4
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0336617
|
3-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-pyrazole-4-carboxylic acid
Show/Hide
|
C29H25N3O4
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0422715
|
(+/-)-2-{5-[(4-Adamantan-1-yl-benzoylamino)-methyl]-4-ethoxy-2-fluoro-benzyl}-butyric acid
Show/Hide
|
C31H38FNO4
|
1
|
| 1 |
EC50 = 24 nM
|
|
|
|
CP0256606
|
5-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-(2-methylpropoxycarbonyl)-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C30H34N2O6
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0081394
|
1-(4-fluorophenyl)-3-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C29H25FN2O5
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0059868
|
2-(5-chloropyridin-3-yl)oxy-5-[(2,4-dichloro-5-methylphenyl)sulfonylamino]-N-ethylbenzamide
Show/Hide
|
C21H18Cl3N3O4S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0153539
|
N-[3-acetyl-5-chloro-4-(5-chloropyridin-3-yl)oxyphenyl]-2,4-dichlorobenzenesulfonamide
Show/Hide
|
C19H12Cl4N2O4S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0367910
|
2-(5-chloropyridin-3-yl)oxy-5-[[2-chloro-4-(trifluoromethyl)phenyl]sulfonylamino]-N-ethylbenzamide
Show/Hide
|
C21H16Cl2F3N3O4S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0507720
|
(S)-2-(4-(2-fluorophenylsulfonyl)piperazin-1-yl)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
|
C31H32FN3O6S
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0530887
|
(2R)-2-[[3-[[[4-(1-adamantyl)benzoyl]amino]methyl]-4-propoxyphenyl]methyl]-4-phenylbutanoic acid
Show/Hide
|
C38H45NO4
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0412337
|
(+/-)-2-{5-[(4-Adamantan-1-yl-2-fluoro-benzoylamino)-methyl]-2-fluoro-4-propoxy-benzyl}-butyric acid
Show/Hide
|
C32H39F2NO4
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0077847
|
((4-Methoxy-phenoxycarbonyl)-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzyl}-amino)-acetic acid
Show/Hide
|
C29H28N2O7
|
2
|
| 1 |
EC50 = 35 nM
|
|
|
| 2 |
EC50 = 1410 nM
|
|
|
|
CP0144349
|
2-((3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(naphthalen-1-ylmethyl)amino)acetic acid
Show/Hide
|
C32H30N2O4
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0422717
|
(+/-)-2-{5-[(4-Adamantan-1-yl-benzoylamino)-methyl]-2-fluoro-4-methoxy-benzyl}-butyric acid
Show/Hide
|
C30H36FNO4
|
1
|
| 1 |
EC50 = 36 nM
|
|
|
|
CP0503011
|
(S)-2-{5-[(4-Adamantan-1-yl-2-fluoro-benzoylamino)-methyl]-2-fluoro-4-propoxy-benzyl}-butyric acid
Show/Hide
|
C32H39F2NO4
|
1
|
| 1 |
EC50 = 38 nM
|
|
|
|
CP0064090
|
(2S,3S)-1-(4-tert-butylphenyl)-3-[[3-[2-[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C34H36N2O6
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0137086
|
(2S,3S)-1-(4-tert-butylphenyl)-3-[[3-[2-[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C34H36N2O6
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0256531
|
5-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-propoxycarbonyl-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C29H32N2O6
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0379502
|
(2S)-2-(4-propoxy-3-{[({4-[(3S,5S,7S)-tricyclo[3.3.1.1~3,7~]dec-1-yl]phenyl}carbonyl)amino]methyl}benzyl)butanoic acid
Show/Hide
|
C32H41NO4
|
2
|
| 1 |
EC50 = 41 nM
|
|
|
| 2 |
EC50 = 43 nM
|
|
|
|
CP0495873
|
2-((4-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C28H25ClN2O6
|
1
|
| 1 |
EC50 = 41.5 nM
|
|
|
|
CP0203701
|
3-[2-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]-1-(2-methylpropoxycarbonyl)piperidine-4-carboxylic acid
Show/Hide
|
C31H38N2O6
|
1
|
| 1 |
EC50 = 44 nM
|
|
|
|
CP0372723
|
2-[[3-[[[4-(1-adamantyl)benzoyl]amino]methyl]-4-ethoxyphenyl]methyl]butanoic acid
Show/Hide
|
C31H39NO4
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0417112
|
(2S,5S)-1-(4-methoxyphenoxy)carbonyl-5-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]pyrrolidine-2-carboxylic acid
Show/Hide
|
C31H30N2O7
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0144347
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(4-phenoxybenzyl)amino)acetic acid
Show/Hide
|
C34H32N2O5
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0457114
|
5-[[4-[2-[1,3-benzothiazol-2-yl(ethyl)amino]ethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C21H21N3O3S2
|
2
|
| 1 |
EC50 = 52 nM
|
|
|
| 2 |
IC50 = 25000 nM
|
|
|
|
CP0457112
|
(5Z)-5-[[4-[2-(1,3-benzothiazol-2-ylamino)ethoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C19H15N3O3S2
|
2
|
| 1 |
EC50 = 53 nM
|
|
|
| 2 |
IC50 = 14000 nM
|
|
|
|
CP0179303
|
5-[2-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]-1-(2-methylpropoxycarbonyl)-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C31H36N2O6
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0447381
|
5-[[4-[2-[1,3-benzothiazol-2-yl(methyl)amino]ethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C20H19N3O3S2
|
2
|
| 1 |
EC50 = 57 nM
|
|
|
| 2 |
IC50 = 20000 nM
|
|
|
|
CP0081395
|
(2S,3S)-1-(4-tert-butylphenyl)-3-[[3-[2-[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C33H33ClN2O5
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0177660
|
N-(3-acetyl-4-quinolin-3-yloxyphenyl)-2,4-dichlorobenzenesulfonamide
Show/Hide
|
C23H16Cl2N2O4S
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0287742
|
2-((3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(4-phenoxybenzyl)amino)acetic acid
Show/Hide
|
C34H32N2O5
|
1
|
| 1 |
EC50 = 67 nM
|
|
|
|
CP0169469
|
1-(6-methoxypyridin-3-yl)-3-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C29H27N3O6
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0845012
|
rac-2-{3-[(4-adamantan-1-yl-benzoylamino)-methyl]-4-propoxy-benzyl}-butyric acid
Show/Hide
|
C32H41NO4
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0181470
|
2,4-dichloro-N-(3,5-dichloro-4-quinolin-6-yloxyphenyl)benzenesulfonamide
Show/Hide
|
C21H12Cl4N2O3S
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0374297
|
2-((4-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)ethoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C29H27ClN2O6
|
1
|
| 1 |
EC50 = 75.4 nM
|
|
|
|
CP0233217
|
2,4-dichloro-N-[3,5-dichloro-4-(5-cyanopyridin-3-yl)oxyphenyl]benzenesulfonamide
Show/Hide
|
C18H9Cl4N3O3S
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0394908
|
(R)-2-{3-[(4-adamantan-1-yl-benzoylamino)-methyl]-4-propoxy-benzyl}-butyric acid
Show/Hide
|
C32H41NO4
|
1
|
| 1 |
EC50 = 83 nM
|
|
|
|
CP0203700
|
5-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C30H27F3N4O4
|
1
|
| 1 |
EC50 = 89 nM
|
|
|
|
CP0081392
|
(2S,3S)-1-(4-methoxyphenyl)-3-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C30H28N2O6
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0177663
|
2,4-dichloro-N-[3,5-dichloro-4-(5-methylpyridin-3-yl)oxyphenyl]benzenesulfonamide
Show/Hide
|
C18H12Cl4N2O3S
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0137069
|
(2S,3S)-1-(4-tert-butylphenyl)-3-[[3-[2-[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C33H33ClN2O5
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0153537
|
2,4-dichloro-N-(3-chloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide
Show/Hide
|
C21H13Cl3N2O3S
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0211451
|
2,4-dichloro-N-[4-(5-chloropyridin-3-yl)oxy-3,5-bis(trifluoromethyl)phenyl]benzenesulfonamide
Show/Hide
|
C19H9Cl3F6N2O3S
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0145814
|
2-((3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(phenethyl)amino)acetic acid
Show/Hide
|
C29H30N2O4
|
1
|
| 1 |
EC50 = 108 nM
|
|
|
|
CP0372719
|
(+/-)-2-{3-[(4-Adamantan-1-yl-benzoylamino)-methyl]-4-methoxy-benzyl}-butyric acid
Show/Hide
|
C30H37NO4
|
2
|
| 1 |
EC50 = 110 nM
|
|
|
| 2 |
EC50 = 120 nM
|
|
|
|
CP0081461
|
(2S,3S)-1-(4-tert-butylphenyl)-3-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C33H34N2O5
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0372717
|
2-[[3-[[[4-(1-adamantyl)benzoyl]amino]methyl]-4-methoxyphenyl]methyl]pentanoic acid
Show/Hide
|
C31H39NO4
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0137087
|
1-(4-chlorophenyl)-3-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C29H25ClN2O5
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0344270
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(heptyl)amino)acetic acid
Show/Hide
|
C28H36N2O4
|
1
|
| 1 |
EC50 = 136 nM
|
|
|
|
CP0412339
|
(+/-)-2-{3-[(4-Adamantan-1-yl-2-fluoro-benzoylamino)-methyl]-4-methoxy-benzyl}-butyric acid
Show/Hide
|
C30H36FNO4
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0440094
|
2-((3-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)ethoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C29H27ClN2O6
|
1
|
| 1 |
EC50 = 141.2 nM
|
|
|
|
CP0340032
|
4-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C29H25N3O4
|
1
|
| 1 |
EC50 = 156 nM
|
|
|
|
CP0384612
|
(R)-2-{5-[(4-Adamantan-1-yl-2-fluoro-benzoylamino)-methyl]-2-fluoro-4-propoxy-benzyl}-butyric acid
Show/Hide
|
C32H39F2NO4
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0239944
|
(3R,4S)-4-[2-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
|
C32H32N2O6
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0289417
|
2-[3-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonylpiperidin-4-yl]acetic acid
Show/Hide
|
C32H32N2O6
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0700372
|
3-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-(4-methoxyphenyl)-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C30H28N2O6
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
|
CP0492706
|
(+/-)-2-{3-[(4-Adamantan-1-yl-benzoylamino)-methyl]-5-fluoro-4-methoxy-benzyl}-butyric acid
Show/Hide
|
C30H36FNO4
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0177662
|
5-[2,6-dichloro-4-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]pyridine-3-carboxamide
Show/Hide
|
C18H11Cl4N3O4S
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0260226
|
2-(5-chloropyridin-3-yl)oxy-N-ethyl-5-[(4-iodophenyl)sulfonylamino]benzamide
Show/Hide
|
C20H17ClIN3O4S
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0447511
|
ethyl 5-[(4-chlorophenyl)sulfonylamino]-2-(5-chloropyridin-3-yl)oxybenzoate
Show/Hide
|
C20H16Cl2N2O5S
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0160819
|
3-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-(2-methylpropoxycarbonyl)piperidine-4-carboxylic acid
Show/Hide
|
C29H34N2O6
|
1
|
| 1 |
EC50 = 209 nM
|
|
|
|
CP0041219
|
Actos
Show/Hide
|
C19H20N2O3S
|
4
|
| 1 |
EC50 = 210 nM
|
|
|
| 2 |
EC50 = 800 nM
|
|
|
| 3 |
EC50 = 1100 nM
|
|
|
| 4 |
IC50 = 22000 nM
|
|
|
|
CP0372724
|
2-[[3-[[(4-cyclohexylbenzoyl)amino]methyl]-4-methoxyphenyl]methyl]butanoic acid
Show/Hide
|
C26H33NO4
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0177528
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(4-(benzyloxy)benzyl)amino)acetic acid
Show/Hide
|
C35H34N2O5
|
1
|
| 1 |
EC50 = 221 nM
|
|
|
|
CP0366486
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(pyridin-2-ylmethyl)amino)acetic acid
Show/Hide
|
C27H27N3O4
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0241222
|
5-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-(2-methylpropoxycarbonyl)-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C30H34N2O6
|
1
|
| 1 |
EC50 = 235 nM
|
|
|
|
CP0544330
|
2-[4-[(Z)-[6-(cyclopropylmethoxy)-3-oxo-1-benzofuran-2-ylidene]methyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C25H26O6
|
1
|
| 1 |
EC50 = 237 nM
|
|
|
|
CP0178968
|
(2S)-2-(4-[2-(3-[2,4-DIFLUOROPHENYL]-1-HEPTYLUREIDO)ETHYL]PHENOXY)-2-METHYLBUTYRIC ACID
Show/Hide
|
C27H36F2N2O4
|
2
|
| 1 |
EC50 = 243 nM
|
|
|
| 2 |
EC50 = 249 nM
|
|
|
|
CP0158748
|
2-chloro-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C22H12Cl3F3N2O3S
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0144346
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)((5-(2-chlorophenyl)furan-2-yl)methyl)amino)acetic acid
Show/Hide
|
C32H29ClN2O5
|
1
|
| 1 |
EC50 = 267 nM
|
|
|
|
CP0382082
|
3-[3-[[[4-(1-adamantyl)benzoyl]amino]methyl]-4-methoxyphenyl]-2-methylpropanoic acid
Show/Hide
|
C29H35NO4
|
1
|
| 1 |
EC50 = 280 nM
|
|
|
|
CP0417727
|
2-((3-((2-(4-isopropylphenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C31H32N2O6
|
1
|
| 1 |
EC50 = 284 nM
|
|
|
|
CP0418504
|
2-[4-[(Z)-(6-ethoxy-3-oxo-1-benzofuran-2-ylidene)methyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C23H24O6
|
1
|
| 1 |
EC50 = 285 nM
|
|
|
|
CP0118743
|
2-((3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(benzyl)amino)acetic acid
Show/Hide
|
C28H28N2O4
|
1
|
| 1 |
EC50 = 295 nM
|
|
|
|
CP0158750
|
2,4-dichloro-N-[4-(5-chloropyridin-3-yl)oxy-3-cyanophenyl]benzenesulfonamide
Show/Hide
|
C18H10Cl3N3O3S
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0301380
|
2,4-dichloro-N-[4-(5-chloropyridin-3-yl)oxy-3-(trifluoromethyl)phenyl]benzenesulfonamide
Show/Hide
|
C18H10Cl3F3N2O3S
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0435137
|
N-[4-(5-acetylpyridin-3-yl)oxy-3,5-dichlorophenyl]-2,4-dichlorobenzenesulfonamide
Show/Hide
|
C19H12Cl4N2O4S
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0294340
|
(3R,4S)-1-ethoxycarbonyl-4-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H30N2O6
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0177398
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(benzo[d][1,3]dioxol-5-ylmethyl)amino)acetic acid
Show/Hide
|
C29H28N2O6
|
1
|
| 1 |
EC50 = 307 nM
|
|
|
|
CP0447382
|
(5Z)-5-[[4-[2-[1,3-benzothiazol-2-yl(methyl)amino]ethoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C20H17N3O3S2
|
2
|
| 1 |
EC50 = 310 nM
|
|
|
| 2 |
IC50 = 13000 nM
|
|
|
|
CP0372058
|
2-[[4-methoxy-3-[[(4-phenylbenzoyl)amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
|
C26H27NO4
|
2
|
| 1 |
EC50 = 320 nM
|
|
|
| 2 |
EC50 = 340 nM
|
|
|
|
CP0533805
|
2-[4-[(Z)-(6-butoxy-3-oxo-1-benzofuran-2-ylidene)methyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C25H28O6
|
1
|
| 1 |
EC50 = 335 nM
|
|
|
|
CP0082410
|
2-((3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(3-phenoxybenzyl)amino)acetic acid
Show/Hide
|
C34H32N2O5
|
1
|
| 1 |
EC50 = 359 nM
|
|
|
|
CP0457113
|
(5Z)-5-[[4-[2-[ethyl(pyridin-2-yl)amino]ethoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C19H19N3O3S
|
2
|
| 1 |
EC50 = 360 nM
|
|
|
| 2 |
IC50 = 15000 nM
|
|
|
|
CP0064613
|
(2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)phenyl]ethoxy}phenyl)propanoic acid
Show/Hide
|
C20H24O7S
|
1
|
| 1 |
EC50 = 360 nM
|
|
|
|
CP0364778
|
2-((3-phenoxybenzyl)(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)amino)acetic acid
Show/Hide
|
C34H32N2O5
|
1
|
| 1 |
EC50 = 391 nM
|
|
|
|
CP0440095
|
2-((3-((2-(biphenyl-4-yl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C34H30N2O6
|
1
|
| 1 |
EC50 = 398 nM
|
|
|
|
CP0158752
|
2-(5-chloropyridin-3-yl)oxy-N-ethyl-5-[(4-nitrophenyl)sulfonylamino]benzamide
Show/Hide
|
C20H17ClN4O6S
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0447172
|
2,4-dichloro-N-[3-chloro-4-(5-chloropyridin-3-yl)oxyphenyl]benzenesulfonamide
Show/Hide
|
C17H10Cl4N2O3S
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0009053
|
(2S)-3-methyl-2-[(4-octoxybenzoyl)amino]butanoic acid
Show/Hide
|
C20H31NO4
|
6
|
| 1 |
EC50 = 400 nM
|
|
|
| 2 |
EC50 = 1184 nM
|
|
|
| 3 |
EC50 = 1484 nM
|
|
|
| 4 |
IC50 = 956.2 nM
|
|
|
| 5 |
IC50 = 2248 nM
|
|
|
| 6 |
Kd = 30.1 nM
|
|
|
|
CP0406521
|
2-methyl-2-{2-methyl-4-[({3-[4-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-5-yl}methyl)sulfanyl]phenoxy}propanoic acid
Show/Hide
|
C21H19F3N2O3S2
|
1
|
| 1 |
EC50 = 407 nM
|
|
|
|
CP0137072
|
(2R,3R)-1-(4-tert-butylphenyl)-3-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C33H34N2O5
|
1
|
| 1 |
EC50 = 410 nM
|
|
|
|
CP0082400
|
2-((3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(4-(benzyloxy)benzyl)amino)acetic acid
Show/Hide
|
C35H34N2O5
|
1
|
| 1 |
EC50 = 412 nM
|
|
|
|
CP0534402
|
2-[2,6-dimethyl-4-[(Z)-(3-oxo-6-propoxy-1-benzofuran-2-ylidene)methyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C24H26O6
|
1
|
| 1 |
EC50 = 412 nM
|
|
|
|
CP0188211
|
2-[[5-[[2-(4-tert-butylphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-2-fluorophenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
|
C26H29FN2O6
|
1
|
| 1 |
EC50 = 414 nM
|
|
|
|
CP0374298
|
2-((3-((5-methyl-2-(4-morpholinophenyl)oxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C32H33N3O7
|
1
|
| 1 |
EC50 = 417 nM
|
|
|
|
CP0117641
|
5-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-pyrazole-4-carboxylic acid
Show/Hide
|
C29H25N3O4
|
1
|
| 1 |
EC50 = 437 nM
|
|
|
|
CP0502606
|
2-[[4-methoxy-3-[[(4-phenylmethoxybenzoyl)amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
|
C27H29NO5
|
1
|
| 1 |
EC50 = 460 nM
|
|
|
|
CP0399671
|
2-methyl-2-[2-methyl-4-[2-[3-[4-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-5-yl]ethylsulfanyl]phenoxy]propanoic acid
Show/Hide
|
C22H21F3N2O3S2
|
1
|
| 1 |
EC50 = 465 nM
|
|
|
|
CP0203720
|
5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-pyrazole-4-carboxylic acid
Show/Hide
|
C29H25N3O4
|
1
|
| 1 |
EC50 = 490 nM
|
|
|
|
CP0170396
|
2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)amino}ethyl)phenyl]sulfanyl}-2-methylpropanoic acid
Show/Hide
|
C26H34F2N2O3S
|
1
|
| 1 |
EC50 = 500 nM
|
|
|
|
CP0137070
|
(2R,3R)-1-(4-tert-butylphenyl)-3-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C33H34N2O5
|
1
|
| 1 |
EC50 = 500 nM
|
|
|
|
CP0498489
|
2-(3-((2-fluoro-4-(trifluoromethyl)benzyl)carbamoyl)-4-methoxybenzyl)butanoic acid
Show/Hide
|
C21H21F4NO4
|
1
|
| 1 |
EC50 = 500 nM
|
|
|
|
CP0544331
|
2-[2,6-dimethyl-4-[(Z)-[6-(2-methylpropoxy)-3-oxo-1-benzofuran-2-ylidene]methyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C25H28O6
|
1
|
| 1 |
EC50 = 503 nM
|
|
|
|
CP0294480
|
2-((3-((2-(3-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C28H25ClN2O6
|
1
|
| 1 |
EC50 = 520 nM
|
|
|
|
CP0538991
|
5-[[4-[2-[1,3-benzothiazol-2-yl(propan-2-yl)amino]ethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C22H23N3O3S2
|
2
|
| 1 |
EC50 = 530 nM
|
|
|
| 2 |
IC50 = 20000 nM
|
|
|
|
CP0279977
|
(3R,4S)-1-ethoxycarbonyl-4-[2-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H32N2O6
|
1
|
| 1 |
EC50 = 540 nM
|
|
|
|
CP0544832
|
5-[[4-[2-[ethyl(pyridin-2-yl)amino]ethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C19H21N3O3S
|
2
|
| 1 |
EC50 = 540 nM
|
|
|
| 2 |
IC50 = 21000 nM
|
|
|
|
CP0090783
|
4-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-pyrrole-3-carboxylic acid
Show/Hide
|
C30H26N2O4
|
1
|
| 1 |
EC50 = 550 nM
|
|
|
|
CP0067563
|
2-(5-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-phenyl-2H-1,2,3-triazol-4-yl)acetic acid
Show/Hide
|
C28H24N4O4
|
1
|
| 1 |
EC50 = 560 nM
|
|
|
|
CP0430028
|
(S)-2-((1-(3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)phenyl)ethyl)(m-tolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C28H25ClN2O6
|
1
|
| 1 |
EC50 = 571 nM
|
|
|
|
CP0256533
|
2-[3-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-(2-methylpropoxycarbonyl)piperidin-4-yl]acetic acid
Show/Hide
|
C30H36N2O6
|
1
|
| 1 |
EC50 = 580 nM
|
|
|
|
CP0185199
|
(S)-3-{4-[3,3-Bis-(4-bromo-phenyl)-allyloxy]-phenyl}-2-ethoxy-propionic acid
Show/Hide
|
C26H24Br2O4
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2
|
| 1 |
EC50 = 590 nM
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|
|
| 2 |
EC50 = 900 nM
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CP0233214
|
2,4-dichloro-N-[4-(5-chloropyridin-3-yl)oxy-3-methylsulfonylphenyl]benzenesulfonamide
Show/Hide
|
C18H13Cl3N2O5S2
|
1
|
| 1 |
EC50 = 600 nM
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|
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CP0258699
|
2,4-dichloro-N-[4-(5-chloropyridin-3-yl)oxy-3-methylphenyl]benzenesulfonamide
Show/Hide
|
C18H13Cl3N2O3S
|
1
|
| 1 |
EC50 = 600 nM
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CP0372722
|
2-[[3-[[[4-(1-adamantyl)benzoyl]amino]methyl]-4-hexoxyphenyl]methyl]butanoic acid
Show/Hide
|
C35H47NO4
|
1
|
| 1 |
EC50 = 620 nM
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|
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CP0126661
|
(3R,4S)-4-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-(4-methylpyrimidin-2-yl)pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H30N4O4
|
1
|
| 1 |
EC50 = 630 nM
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|
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CP0279978
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(3R,4S)-4-[2-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
|
C32H32N2O6
|
1
|
| 1 |
EC50 = 630 nM
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|
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CP0531413
|
2-[4-[(Z)-(6-methoxy-3-oxo-1-benzofuran-2-ylidene)methyl]-2,6-dimethylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C22H22O6
|
1
|
| 1 |
EC50 = 634 nM
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|
|
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CP0449198
|
2-[4-[[3-[3-fluoro-4-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-5-yl]methylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C21H18F4N2O3S2
|
1
|
| 1 |
EC50 = 640 nM
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|
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CP0409665
|
2-{3-[(2-fluoro-4-trifluoromethylbenzoylamino)-methyl]-4-n-propoxyphenylmethyl}butyric acid
Show/Hide
|
C23H25F4NO4
|
1
|
| 1 |
EC50 = 650 nM
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|
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CP0399674
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2-[4-[[3-(3-chloro-4-methylphenyl)-1,2,4-thiadiazol-5-yl]methylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C21H21ClN2O3S2
|
1
|
| 1 |
EC50 = 669 nM
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|
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CP0271245
|
2-((3-((5-methyl-2-p-tolyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
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C29H28N2O6
|
1
|
| 1 |
EC50 = 684 nM
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|
|
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CP0447383
|
(5Z)-5-[[4-[2-[methyl(1,3-thiazol-2-yl)amino]ethoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
Show/Hide
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C16H15N3O3S2
|
2
|
| 1 |
EC50 = 700 nM
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|
|
| 2 |
IC50 = 42000 nM
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CP0224910
|
2-((3-((5-methyl-2-(4-(trifluoromethyl)phenyl)oxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C29H25F3N2O6
|
1
|
| 1 |
EC50 = 705 nM
|
|
|
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CP0495869
|
2-((3-((5-methyl-2-phenyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C28H26N2O6
|
1
|
| 1 |
EC50 = 705 nM
|
|
|
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CP0374280
|
(S)-2-((1-(3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)phenyl)ethyl)((2-fluoro-5-methylphenoxy)carbonyl)amino)acetic acid
Show/Hide
|
C28H24ClFN2O6
|
1
|
| 1 |
EC50 = 710 nM
|
|
|
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CP0502607
|
2-[[4-methoxy-3-[[(3-phenylbenzoyl)amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
|
C26H27NO4
|
1
|
| 1 |
EC50 = 710 nM
|
|
|
|
CP0063974
|
(3R,4S)-1-ethoxycarbonyl-4-[2-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H32N2O6
|
1
|
| 1 |
EC50 = 710 nM
|
|
|
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CP0197728
|
3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-pyrazole-4-carboxylic acid
Show/Hide
|
C29H25N3O4
|
1
|
| 1 |
EC50 = 752 nM
|
|
|
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CP0364796
|
2-(((1H-indol-2-yl)methyl)(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)amino)acetic acid
Show/Hide
|
C30H29N3O4
|
1
|
| 1 |
EC50 = 759 nM
|
|
|
|
CP0550779
|
2-[2,6-dimethyl-4-[(Z)-[6-(3-methylbutoxy)-3-oxo-1-benzofuran-2-ylidene]methyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C26H30O6
|
1
|
| 1 |
EC50 = 764 nM
|
|
|
|
CP0501324
|
(S)-2-((1-(3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)phenyl)ethyl)((3-methoxyphenoxy)carbonyl)amino)acetic acid
Show/Hide
|
C28H25ClN2O7
|
1
|
| 1 |
EC50 = 772 nM
|
|
|
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CP0399822
|
2-[[4-methoxy-3-[[[4-(2-phenylethoxy)benzoyl]amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
|
C28H31NO5
|
1
|
| 1 |
EC50 = 780 nM
|
|
|
|
CP0398827
|
(R)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-2-methylphenoxy)acetic acid
Show/Hide
|
C26H24Cl2N2O4
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
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CP0397604
|
2-methyl-2-[4-[3-[4-[(E)-3-phenylprop-2-enoyl]phenoxy]propyl]phenoxy]propanoic acid
Show/Hide
|
C28H28O5
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0462373
|
2-methyl-2-[4-[(4-phenoxyphenoxy)methyl]phenoxy]propanoic acid
Show/Hide
|
C23H22O5
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0476895
|
2-methyl-2-[4-[3-[4-[(E)-2-phenylethenyl]phenoxy]propyl]phenoxy]propanoic acid
Show/Hide
|
C27H28O4
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0412456
|
2-[4-[2-[3-(3,4-dichlorophenyl)-1,2,4-thiadiazol-5-yl]ethylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C21H20Cl2N2O3S2
|
1
|
| 1 |
EC50 = 815 nM
|
|
|
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CP0002766
|
2-(4-methoxy-3-((4-phenoxybenzamido)methyl)benzyl)butanoic acid
Show/Hide
|
C26H27NO5
|
1
|
| 1 |
EC50 = 820 nM
|
|
|
|
CP0462196
|
(5Z)-5-[[4-[2-[1,3-benzothiazol-2-yl(ethyl)amino]ethoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C21H19N3O3S2
|
2
|
| 1 |
EC50 = 820 nM
|
|
|
| 2 |
IC50 = 17000 nM
|
|
|
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CP0479940
|
2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)((cyclopropylmethoxy)carbonyl)amino)acetic acid
Show/Hide
|
C25H25ClN2O6
|
1
|
| 1 |
EC50 = 826 nM
|
|
|
|
CP0476772
|
(S)-2-(3-((4-(4-Chlorophenoxy)benzamido)methyl)-4-methoxybenzyl)butanoic acid
Show/Hide
|
C26H26ClNO5
|
1
|
| 1 |
EC50 = 830 nM
|
|
|
|
CP0340825
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(naphthalen-1-ylmethyl)amino)acetic acid
Show/Hide
|
C32H30N2O4
|
1
|
| 1 |
EC50 = 840 nM
|
|
|
|
CP0081393
|
(2R,3R)-1-(4-methoxyphenyl)-3-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-4-oxoazetidine-2-carboxylic acid
Show/Hide
|
C30H28N2O6
|
1
|
| 1 |
EC50 = 840 nM
|
|
|
|
CP0400030
|
2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(cyclohexyloxycarbonyl)amino)acetic acid
Show/Hide
|
C27H29ClN2O6
|
1
|
| 1 |
EC50 = 843 nM
|
|
|
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CP0551956
|
2-methyl-2-(3-pentadecylphenoxy)propanoic acid
Show/Hide
|
C25H42O3
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0344271
|
2-((3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(3-phenylpropyl)amino)acetic acid
Show/Hide
|
C30H32N2O4
|
1
|
| 1 |
EC50 = 901 nM
|
|
|
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CP0374299
|
2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(cyclobutoxycarbonyl)amino)acetic acid
Show/Hide
|
C25H25ClN2O6
|
1
|
| 1 |
EC50 = 905 nM
|
|
|
|
CP0523476
|
ethyl 2-methyl-2-[4-(6-nitro-2-oxochromene-3-carbonyl)phenoxy]propanoate
Show/Hide
|
C22H19NO8
|
1
|
| 1 |
EC50 = 910 nM
|
|
|
|
CP0372059
|
(S)-2-(3-((4-(4-Fluorophenoxy)benzamido)methyl)-4-methoxybenzyl)butanoic acid
Show/Hide
|
C26H26FNO5
|
1
|
| 1 |
EC50 = 920 nM
|
|
|
|
CP0271243
|
2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(p-tolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C28H25ClN2O6
|
2
|
| 1 |
EC50 = 963 nM
|
|
|
| 2 |
EC50 = 1321 nM
|
|
|
|
CP0373362
|
(S)-2-((1-(3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)phenyl)ethyl)((4-methoxyphenoxy)carbonyl)amino)acetic acid
Show/Hide
|
C28H25ClN2O7
|
1
|
| 1 |
EC50 = 970 nM
|
|
|
|
CP0494397
|
(S)-2-(3-((4-(4-bromophenoxy)benzamido)methyl)-4-methoxybenzyl)butanoic acid
Show/Hide
|
C26H26BrNO5
|
1
|
| 1 |
EC50 = 990 nM
|
|
|
|
CP0436763
|
2-{4-n-butoxy-3-[(2-fluoro-4-trifluoromethylbenzoylamino)methyl]phenylmethyl}pentanoic acid
Show/Hide
|
C23H25F4NO4
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0522258
|
2-(4-butoxy-3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)benzyl)pentanoic acid
Show/Hide
|
C25H29F4NO4
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0188352
|
2,4-dichloro-N-[4-(5-chloropyridin-3-yl)oxy-3-fluorophenyl]benzenesulfonamide
Show/Hide
|
C17H10Cl3FN2O3S
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0128750
|
2-((3-((2-(4-fluorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C28H25FN2O6
|
1
|
| 1 |
EC50 = 1007 nM
|
|
|
|
CP0071776
|
(3R,4S)-4-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-pyrimidin-2-ylpyrrolidine-3-carboxylic acid
Show/Hide
|
C28H28N4O4
|
1
|
| 1 |
EC50 = 1060 nM
|
|
|
|
CP0564979
|
2-[4-[(Z)-[6-(cyclopropylmethoxy)-3-oxo-1-benzofuran-2-ylidene]methyl]-2,6-dimethylphenoxy]acetic acid
Show/Hide
|
C23H22O6
|
1
|
| 1 |
EC50 = 1063 nM
|
|
|
|
CP0329281
|
2-[[5-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-2-fluorophenyl]methyl-(4-methoxyphenoxy)carbonylamino]acetic acid
Show/Hide
|
C28H24ClFN2O7
|
1
|
| 1 |
EC50 = 1087 nM
|
|
|
|
CP0425692
|
(2S)-2-{4-butoxy-3-[({[2-fluoro-4-(trifluoromethyl)phenyl]carbonyl}amino)methyl]benzyl}butanoic acid
Show/Hide
|
C24H27F4NO4
|
2
|
| 1 |
EC50 = 1100 nM
|
|
|
| 2 |
EC50 = 1400 nM
|
|
|
|
CP0075347
|
2-((3-((2-(2-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C28H25ClN2O6
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0522916
|
(+/-)-2-(2-fluoro-4-methoxy-5-((4-(trifluoromethyl)benzamido)methyl)benzyl)butanoic acid
Show/Hide
|
C21H21F4NO4
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0128749
|
2-((3-((2-(4-methoxyphenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C29H28N2O7
|
1
|
| 1 |
EC50 = 1124 nM
|
|
|
|
CP0506232
|
(S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-m-tolylpiperazin-1-yl)propanoic acid
Show/Hide
|
C32H35N3O4
|
1
|
| 1 |
EC50 = 1140 nM
|
|
|
|
CP0177584
|
(3R,4R)-4-[2-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
|
C32H32N2O6
|
1
|
| 1 |
EC50 = 1170 nM
|
|
|
|
CP0082408
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(2-(benzyloxy)ethyl)amino)acetic acid
Show/Hide
|
C30H32N2O5
|
1
|
| 1 |
EC50 = 1180 nM
|
|
|
|
CP0082407
|
2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(naphthalen-2-ylmethyl)amino)acetic acid
Show/Hide
|
C32H30N2O4
|
1
|
| 1 |
EC50 = 1210 nM
|
|
|
|
CP0420717
|
2-[butoxycarbonyl-[[5-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-2-fluorophenyl]methyl]amino]acetic acid
Show/Hide
|
C25H26ClFN2O6
|
1
|
| 1 |
EC50 = 1235 nM
|
|
|
|
CP0188212
|
2-[[5-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-2-fluorophenyl]methyl-(4-methylphenoxy)carbonylamino]acetic acid
Show/Hide
|
C28H24ClFN2O6
|
1
|
| 1 |
EC50 = 1255 nM
|
|
|
|
CP0504517
|
2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(propoxycarbonyl)amino)acetic acid
Show/Hide
|
C24H25ClN2O6
|
1
|
| 1 |
EC50 = 1257 nM
|
|
|
|
CP0461769
|
2-{4-n-butoxy-3-[(4-trifluoromethylbenzoylamino)methyl]phenylmethyl}butyric acid
Show/Hide
|
C24H28F3NO4
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0483816
|
2-{4-n-propoxy-3-[(4-trifluoromethylbenzoylamino)methyl]phenylmethyl}butyric acid
Show/Hide
|
C23H26F3NO4
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0561914
|
2-[4-[(Z)-(6-ethoxy-3-oxo-1-benzofuran-2-ylidene)methyl]-2,6-dimethylphenoxy]acetic acid
Show/Hide
|
C21H20O6
|
1
|
| 1 |
EC50 = 1323 nM
|
|
|
|
CP0157749
|
2-((3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(naphthalen-2-ylmethyl)amino)acetic acid
Show/Hide
|
C32H30N2O4
|
1
|
| 1 |
EC50 = 1390 nM
|
|
|
|
CP0461765
|
2-(4-butoxy-3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)benzyl)butanoic acid
Show/Hide
|
C24H27F4NO4
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0470919
|
2-methyl-2-[4-[2-(4-phenyldiazenylphenoxy)ethyl]phenoxy]propanoic acid
Show/Hide
|
C24H24N2O4
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0095457
|
2-((3-((2-(4-chlorophenyl)-4-methylthiazol-5-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
|
C28H25ClN2O5S
|
1
|
| 1 |
EC50 = 1411 nM
|
|
|
|
CP0444128
|
2-[(3S)-6-[3-(3-chlorophenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
|
C19H19ClO5
|
1
|
| 1 |
EC50 = 1430 nM
|
|
|
|
CP0402264
|
(S)-2-((1-(3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)phenyl)ethyl)((4-fluoro-3-methoxyphenoxy)carbonyl)amino)acetic acid
Show/Hide
|
C28H24ClFN2O7
|
1
|
| 1 |
EC50 = 1444 nM
|
|
|
|
CP0479939
|
2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(cyclopentyloxycarbonyl)amino)acetic acid
Show/Hide
|
C26H27ClN2O6
|
1
|
| 1 |
EC50 = 1482 nM
|
|
|
|
CP0526677
|
2-{4-methoxy-3-[(2-fluoro-4-trifluoromethylbenzoylamino)methyl]phenylmethyl}pentanoic acid
Show/Hide
|
C22H23F4NO4
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0230128
|
2-[[5-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-2-fluorophenyl]methyl-(2-methylpropoxycarbonyl)amino]acetic acid
Show/Hide
|
C25H26ClFN2O6
|
1
|
| 1 |
EC50 = 1504 nM
|
|
|
|
CP0421259
|
2-[4-[3-(3-chlorophenoxy)propoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C18H19ClO5
|
1
|
| 1 |
EC50 = 1540 nM
|
|
|
|
CP0340038
|
1-methyl-4-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1H-pyrrole-3-carboxylic acid
Show/Hide
|
C25H24N2O4
|
1
|
| 1 |
EC50 = 1570 nM
|
|
|
|
CP0547789
|
2-[4-[(Z)-(6-methoxy-3-oxo-1-benzofuran-2-ylidene)methyl]-2,6-dimethylphenoxy]acetic acid
Show/Hide
|
C20H18O6
|
1
|
| 1 |
EC50 = 1579 nM
|
|
|
|
CP0394696
|
2-(3-((3-fluoro-4-(trifluoromethyl)benzyl)carbamoyl)-4-methoxybenzyl)butanoic acid
Show/Hide
|
C21H21F4NO4
|
1
|
| 1 |
EC50 = 1600 nM
|
|
|
|
CP0538992
|
(5Z)-5-[[4-[2-[methyl(naphthalen-2-yl)amino]ethoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C23H20N2O3S
|
2
|
| 1 |
EC50 = 1600 nM
|
|
|
| 2 |
IC50 = 40000 nM
|
|
|
|
CP0411699
|
2-[6-[3-(3-bromophenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
|
C19H19BrO5
|
1
|
| 1 |
EC50 = 1670 nM
|
|
|
|
CP0476755
|
2-[6-[3-(3-chlorophenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C19H19ClO5
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1
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| 1 |
EC50 = 1690 nM
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CP0501323
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(S)-2-((1-(3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)phenyl)ethyl)(phenoxycarbonyl)amino)acetic acid
Show/Hide
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C27H23ClN2O6
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1
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| 1 |
EC50 = 1692 nM
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CP0518698
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(3R,8S,9Z)-8-[[(1R,4aR,7R,8aR)-7-(2-hydroxypropan-2-yl)-1,4a-dimethyl-2,3,4,5,6,7,8,8a-octahydronaphthalen-1-yl]oxy]heptadeca-1,9-dien-4,6-diyn-3-ol
Show/Hide
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C32H50O3
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1
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| 1 |
EC50 = 1700 nM
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CP0518699
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(1R)-1-ethenyl-9-[(Z,3S)-3-hydroxydodec-4-en-1-ynyl]-6-methoxy-1,3-dihydrobenzo[f][2]benzofuran-7-ol
Show/Hide
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C27H32O4
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1
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| 1 |
EC50 = 1700 nM
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CP0547788
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2-[2,6-dimethyl-4-[(Z)-[6-(2-methylpropoxy)-3-oxo-1-benzofuran-2-ylidene]methyl]phenoxy]acetic acid
Show/Hide
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C23H24O6
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1
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| 1 |
EC50 = 1745 nM
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CP0411710
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2-[6-[3-(3-methylphenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C20H22O5
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1
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| 1 |
EC50 = 1750 nM
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CP0457743
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2-[6-[3-(3-tert-butylphenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C23H28O5
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1
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| 1 |
EC50 = 1750 nM
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CP0551958
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2-methyl-2-[3-[(Z)-pentadec-8-enyl]phenoxy]propanoic acid
Show/Hide
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C25H40O3
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1
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| 1 |
EC50 = 1780 nM
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CP0145812
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2-((4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)(2-ethylbutyl)amino)acetic acid
Show/Hide
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C27H34N2O4
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1
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| 1 |
EC50 = 1800 nM
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CP0436765
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2-{4-ethoxy-3-[(4-trifluoromethylbenzoylamino)-methyl]phenylmethyl}butyric acid
Show/Hide
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C22H24F3NO4
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1
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| 1 |
EC50 = 1800 nM
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CP0457744
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2-[6-[3-(4-methylphenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C20H22O5
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1
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| 1 |
EC50 = 1810 nM
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CP0444806
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4-hexoxy-N-[(2S)-1-(hydroxyamino)-3-methyl-1-oxobutan-2-yl]benzamide
Show/Hide
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C18H28N2O4
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2
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| 1 |
EC50 = 1840 nM
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| 2 |
Kd = 123 nM
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CP0455779
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2-[6-[3-(3-phenylphenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C25H24O5
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1
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| 1 |
EC50 = 1850 nM
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CP0394697
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(2S)-2-{3-[({[2-fluoro-4-(trifluoromethyl)phenyl]carbonyl}amino)methyl]-4-methoxybenzyl}butanoic acid
Show/Hide
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C21H21F4NO4
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1
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| 1 |
EC50 = 1900 nM
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CP0488001
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(3R,8S,9Z)-3-[[(1R,4aR,7R,8aR)-7-(2-hydroxypropan-2-yl)-1,4a-dimethyl-2,3,4,5,6,7,8,8a-octahydronaphthalen-1-yl]oxy]heptadeca-1,9-dien-4,6-diyn-8-ol
Show/Hide
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C32H50O3
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1
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| 1 |
EC50 = 1900 nM
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CP0945997
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3-(4-(3-(3-chlorophenoxy)propoxy)phenyl)propanoic-2,2-d2 acid
Show/Hide
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C18H19ClO4
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1
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| 1 |
EC50 = 1920 nM
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CP0528437
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(2S)-2-[(4-hexoxybenzoyl)amino]-3-methylbutanoic acid
Show/Hide
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C18H27NO4
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2
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| 1 |
EC50 = 1940 nM
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| 2 |
Kd = 94 nM
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CP0008515
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(+/-)-2-(4-methoxy-3-((4-(trifluoromethyl)benzamido)methyl)benzyl)butanoic acid
Show/Hide
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C21H22F3NO4
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2
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| 1 |
EC50 = 2000 nM
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| 2 |
EC50 = 2600 nM
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CP0158749
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2-(5-chloropyridin-3-yl)oxy-N-ethyl-5-[(4-methoxyphenyl)sulfonylamino]benzamide
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C21H20ClN3O5S
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1
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| 1 |
EC50 = 2000 nM
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CP0481491
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2,4-dichloro-N-(3-chloro-4-naphthalen-2-yloxyphenyl)benzenesulfonamide
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C22H14Cl3NO3S
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1
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| 1 |
EC50 = 2000 nM
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CP0398169
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(1R,2S,4aR,5R,8R,8aS)-8-[(3R,8S,9Z)-8-hydroxyheptadeca-1,9-dien-4,6-diyn-3-yl]oxy-4a,8-dimethyl-2-propan-2-yl-1,2,3,4,5,6,7,8a-octahydronaphthalene-1,5-diol
Show/Hide
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C32H50O4
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1
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| 1 |
EC50 = 2000 nM
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CP0190238
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2-[[5-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-2-fluorophenyl]methyl-propoxycarbonylamino]acetic acid
Show/Hide
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C24H24ClFN2O6
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1
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| 1 |
EC50 = 2013 nM
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CP0476754
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2-[6-[3-(2-methylphenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C20H22O5
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1
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| 1 |
EC50 = 2020 nM
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CP0411709
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2-[6-[2-(3-tert-butylphenoxy)ethoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C22H26O5
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1
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| 1 |
EC50 = 2030 nM
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CP0307236
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2-[[2-fluoro-5-[[5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]methoxy]phenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
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C23H20F4N2O6
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1
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| 1 |
EC50 = 2062 nM
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CP0177586
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(3R,4S)-1-(1,3-benzoxazol-2-yl)-4-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]pyrrolidine-3-carboxylic acid
Show/Hide
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C31H29N3O5
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1
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| 1 |
EC50 = 2080 nM
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CP0469063
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(S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-(2-nitrophenylsulfonyl)piperazin-1-yl)propanoic acid
Show/Hide
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C31H32N4O8S
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1
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| 1 |
EC50 = 2160 nM
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CP0202689
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2-[[2-fluoro-5-[[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methoxy]phenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
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C23H23FN2O6
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1
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| 1 |
EC50 = 2182 nM
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CP0117642
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5-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-phenyl-2H-1,2,3-triazole-4-carboxylic acid
Show/Hide
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C27H22N4O4
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1
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| 1 |
EC50 = 2190 nM
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CP0412340
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(+/-)-2-(3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)-4-methoxybenzyl)butanoic acid
Show/Hide
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C21H21F4NO4
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2
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| 1 |
EC50 = 2200 nM
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| 2 |
EC50 = 2600 nM
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CP0382083
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2-[[3-[[(4-tert-butylbenzoyl)amino]methyl]-4-methoxyphenyl]methyl]butanoic acid
Show/Hide
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C24H31NO4
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1
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| 1 |
EC50 = 2300 nM
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CP0467104
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2-{4-n-hexyloxy-3-[(4-trifluoromethylbenzoylamino)methyl]phenylmethyl}butyric acid
Show/Hide
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C26H32F3NO4
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1
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| 1 |
EC50 = 2300 nM
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CP0003371
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[(3R,8S,9Z)-3-hydroxyheptadeca-1,9-dien-4,6-diyn-8-yl] (E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enoate
Show/Hide
|
C27H32O5
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1
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| 1 |
EC50 = 2300 nM
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CP0117566
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1-methyl-4-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1H-pyrrole-3-carboxylic acid
Show/Hide
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C25H24N2O4
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1
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| 1 |
EC50 = 2370 nM
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CP0181463
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2-[[2-fluoro-5-[[5-methyl-2-[4-(trifluoromethoxy)phenyl]-1,3-oxazol-4-yl]methoxy]phenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
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C23H20F4N2O7
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1
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| 1 |
EC50 = 2384 nM
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CP0492987
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2-{4-methoxy-3-[(4-trifluoromethylbenzoylamino)-methyl]phenylmethyl}hexanoic aci
Show/Hide
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C23H26F3NO4
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1
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| 1 |
EC50 = 2400 nM
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CP0224906
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2-((3-((2-(4-chlorophenyl)-5-methylthiazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
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C28H25ClN2O5S
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1
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| 1 |
EC50 = 2500 nM
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CP0071775
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(3R,4S)-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
Show/Hide
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C29H27F3N4O4
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1
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| 1 |
EC50 = 2500 nM
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CP0421260
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2-[6-[3-(2-fluorophenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C19H19FO5
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1
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| 1 |
EC50 = 2670 nM
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CP0111046
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2-[4-[[1-[(2,4-dichlorophenyl)carbamoyl]-3,4-dihydro-1H-isoquinolin-2-yl]methyl]-2-methylphenoxy]acetic acid
Show/Hide
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C26H24Cl2N2O4
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1
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| 1 |
EC50 = 2700 nM
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CP0514008
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(S)-2-(4-(4-fluorophenylsulfonyl)piperazin-1-yl)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
|
C31H32FN3O6S
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1
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| 1 |
EC50 = 2810 nM
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CP0329280
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2-[[3-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-5-fluorophenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
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C22H20ClFN2O6
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1
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| 1 |
EC50 = 2819 nM
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CP0068929
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(3R,4R)-1-ethoxycarbonyl-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]pyrrolidine-3-carboxylic acid
Show/Hide
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C27H30N2O6
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1
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| 1 |
EC50 = 2850 nM
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CP0230127
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2-[[(1S)-1-[3-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]phenyl]ethyl]-methoxycarbonylamino]acetic acid
Show/Hide
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C23H23ClN2O6
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1
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| 1 |
EC50 = 2857 nM
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CP0294479
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2-((3-((2-(4-chlorophenyl)-4-methyloxazol-5-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
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C28H25ClN2O6
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1
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| 1 |
EC50 = 2901 nM
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CP0411698
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2-[6-[3-(4-phenylphenoxy)propoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C25H24O5
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1
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| 1 |
EC50 = 2970 nM
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CP0000253
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2-(3-((4-(trifluoromethyl)benzyl)carbamoyl)-4-methoxybenzyl)butanoic acid
Show/Hide
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C21H22F3NO4
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1
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| 1 |
EC50 = 3000 nM
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CP0438102
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2-[4-[3-(3-chlorophenoxy)propoxy]-2-fluorophenoxy]acetic acid
Show/Hide
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C17H16ClFO5
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1
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| 1 |
EC50 = 3170 nM
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CP0387723
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(2S)-2-[[4-[2-[4-(1,3-dioxoisoindol-2-yl)-2-ethoxyphenyl]ethyl]phenyl]methyl]butanoic acid
Show/Hide
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C29H29NO5
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1
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| 1 |
EC50 = 3200 nM
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CP0508117
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(5Z)-5-[[4-[2-[1H-benzimidazol-2-yl(methyl)amino]ethoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
Show/Hide
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C20H18N4O3S
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2
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| 1 |
EC50 = 3400 nM
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| 2 |
IC50 = 38000 nM
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CP0374281
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2-(methoxycarbonyl(3-((2-(4-(trifluoromethyl)phenyl)thiazol-4-yl)methoxy)benzyl)amino)acetic acid
Show/Hide
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C22H19F3N2O5S
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1
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| 1 |
EC50 = 3443 nM
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CP0325274
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2-((3-((2-(4-cyanophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(ptolyloxycarbonyl)amino)acetic acid
Show/Hide
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C29H25N3O6
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1
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| 1 |
EC50 = 3445 nM
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CP0049844
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(Benzyl-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzyl}-amino)-acetic acid
Show/Hide
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C28H28N2O4
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1
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| 1 |
EC50 = 3600 nM
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CP0436764
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2-{4-methoxy-3-[(4-trifluoromethylbenzoylamino)-methyl]phenylmethyl}pentanoic acid
Show/Hide
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C22H24F3NO4
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1
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| 1 |
EC50 = 3600 nM
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CP0465977
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2-methyl-2-[4-(2-oxochromene-3-carbonyl)phenoxy]propanoic acid
Show/Hide
|
C20H16O6
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1
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| 1 |
EC50 = 3670 nM
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CP0461700
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3-(4-(2-((4-(trifluoromethyl)benzyl)(benzo[d]thiazol-2-yl)amino)ethoxy)phenyl)propanoic acid
Show/Hide
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C26H23F3N2O3S
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1
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| 1 |
EC50 = 3690 nM
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CP0551957
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2-(3-pentadecylphenoxy)acetic acid
Show/Hide
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C23H38O3
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1
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| 1 |
EC50 = 3700 nM
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CP0203721
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5-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-2-phenyl-2H-1,2,3-triazole-4-carboxylic acid
Show/Hide
|
C28H24N4O4
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1
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| 1 |
EC50 = 3790 nM
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CP0201620
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2-(5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-phenyl-2H-1,2,3-triazol-4-yl)acetic acid
Show/Hide
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C28H24N4O4
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1
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| 1 |
EC50 = 3860 nM
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CP0551954
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ethyl 2-methyl-2-(3-pentadecylphenoxy)propanoate
Show/Hide
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C27H46O3
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1
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| 1 |
EC50 = 3900 nM
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CP0076831
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Elafibranor
Show/Hide
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C22H24O4S
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1
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| 1 |
EC50 = 3962 nM
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CP0548288
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2-[2,6-dimethyl-4-[(Z)-(3-oxo-6-propoxy-1-benzofuran-2-ylidene)methyl]phenoxy]acetic acid
Show/Hide
|
C22H22O6
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1
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| 1 |
EC50 = 3962 nM
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CP0150880
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2-{[(3-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)methyl](methoxycarbonyl)amino}acetic acid
Show/Hide
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C22H21ClN2O6
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2
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| 1 |
EC50 = 4017 nM
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| 2 |
EC50 = 4100 nM
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CP0390607
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2-((3-((2-(3-chlorophenyl)thiazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid
Show/Hide
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C21H19ClN2O5S
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1
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| 1 |
EC50 = 4018 nM
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CP0072253
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(3R,4R)-4-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
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C30H28N2O6
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1
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| 1 |
EC50 = 4180 nM
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CP0239931
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2-[(3R,4R)-4-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonylpyrrolidin-3-yl]acetic acid
Show/Hide
|
C31H30N2O6
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1
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| 1 |
EC50 = 4180 nM
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CP0098834
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4-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-pyrrole-3-carboxylic acid
Show/Hide
|
C30H26N2O4
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1
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| 1 |
EC50 = 4200 nM
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CP0222162
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2-[[5-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-2-fluorophenyl]methyl-ethoxycarbonylamino]acetic acid
Show/Hide
|
C23H22ClFN2O6
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1
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| 1 |
EC50 = 4273 nM
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CP0427896
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2-[[5-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-2-fluorophenyl]methyl-(3-fluoropropoxycarbonyl)amino]acetic acid
Show/Hide
|
C24H23ClF2N2O6
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1
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| 1 |
EC50 = 4383 nM
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CP0459406
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2-[[4-methoxy-3-[[[4-(trifluoromethoxy)benzoyl]amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
|
C21H22F3NO5
|
1
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| 1 |
EC50 = 4400 nM
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CP0196069
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2-[(2R,4R)-1-[4-[[4-(2-fluoro-5-methoxyphenyl)-2-methylphenyl]methyl]phenyl]-4-(trifluoromethyl)pyrrolidin-2-yl]acetic acid
Show/Hide
|
C28H27F4NO3
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1
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| 1 |
EC50 = 4400 nM
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CP0111137
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2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}-2-fluorophenyl)methyl](methoxycarbonyl)amino}acetic acid
Show/Hide
|
C22H20ClFN2O6
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1
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| 1 |
EC50 = 4511 nM
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CP0411700
|
2-[2-methyl-4-[3-(4-phenylphenoxy)propoxy]phenoxy]acetic acid
Show/Hide
|
C24H24O5
|
1
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| 1 |
EC50 = 4560 nM
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CP0391103
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2-[[4-methoxy-3-[[(3-phenoxybenzoyl)amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
|
C26H27NO5
|
1
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| 1 |
EC50 = 4600 nM
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CP0417677
|
2-((3-((2-(4-chlorophenyl)thiazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid
Show/Hide
|
C21H19ClN2O5S
|
1
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| 1 |
EC50 = 4692 nM
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CP0068984
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2-[(3R,4R)-4-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonylpyrrolidin-3-yl]acetic acid
Show/Hide
|
C31H30N2O6
|
1
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| 1 |
EC50 = 4800 nM
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CP0501325
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2-(methoxycarbonyl(3-((2-(4-(trifluoromethyl)phenyl)oxazol-4-yl)methoxy)benzyl)amino)acetic acid
Show/Hide
|
C22H19F3N2O6
|
1
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| 1 |
EC50 = 4815 nM
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CP0442236
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(S)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)methyl)-4-methoxybenzyl)butanoic acid
Show/Hide
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C21H21F4NO4
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1
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| 1 |
EC50 = 4900 nM
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CP0349034
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5-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-phenylmethoxycarbonyl-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
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C33H32N2O6
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1
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| 1 |
EC50 = 4920 nM
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CP0504263
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2-((3-((2-(2-chlorophenyl)thiazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid
Show/Hide
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C21H19ClN2O5S
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1
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| 1 |
EC50 = 5036 nM
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CP0513847
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ethyl 2-methyl-2-[4-(2-oxochromene-3-carbonyl)phenoxy]propanoate
Show/Hide
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C22H20O6
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1
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| 1 |
EC50 = 5190 nM
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CP0377699
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(2S)-2-[[4-[2-[4-(1,3-dioxoisoindol-2-yl)-2-propoxyphenyl]ethyl]phenyl]methyl]butanoic acid
Show/Hide
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C30H31NO5
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1
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| 1 |
EC50 = 5200 nM
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CP0457742
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2-[6-(3-phenoxypropoxy)-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C19H20O5
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1
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| 1 |
EC50 = 5260 nM
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CP0396558
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2-[4-[(4-benzoylphenoxy)methyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C24H22O5
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1
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| 1 |
EC50 = 5400 nM
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CP0205708
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5-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-(2-methylpropoxycarbonyl)-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
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C29H32N2O6
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1
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| 1 |
EC50 = 5570 nM
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CP0053195
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(3R,4R)-4-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
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C30H28N2O6
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1
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| 1 |
EC50 = 5650 nM
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CP0279413
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4-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-1,2,3-triazole-5-carboxylic acid
Show/Hide
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C28H24N4O4
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1
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| 1 |
EC50 = 5800 nM
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CP0520653
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2-[4-[3-(4-benzoylphenoxy)propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C26H26O5
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1
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| 1 |
EC50 = 5800 nM
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CP0459171
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2-methyl-2-[4-[2-[4-[(E)-3-phenylprop-2-enoyl]phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
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C27H26O5
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1
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| 1 |
EC50 = 5900 nM
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CP0436681
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2-methyl-2-[4-[[4-[(E)-2-phenylethenyl]phenoxy]methyl]phenoxy]propanoic acid
Show/Hide
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C25H24O4
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1
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| 1 |
EC50 = 6000 nM
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CP0248079
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(3R,4R)-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
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C31H30N2O6
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1
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| 1 |
EC50 = 6170 nM
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CP0436762
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2-{4-benzyloxy-3-[(4-trifluoromethylbenzoylamino)methyl]benzyl}butyric acid
Show/Hide
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C27H26F3NO4
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1
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| 1 |
EC50 = 6200 nM
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CP0485323
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3-(4-(2-((4-tert-butylbenzyl)(benzo[d]thiazol-2-yl)amino)ethoxy)phenyl)propanoic acid
Show/Hide
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C29H32N2O3S
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1
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| 1 |
EC50 = 6340 nM
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CP0402268
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2-((3-((2-(3-chloro-4-fluorophenyl)oxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid
Show/Hide
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C21H18ClFN2O6
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1
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| 1 |
EC50 = 6386 nM
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CP0424859
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(2R)-2-[[4-[2-[4-(1,3-dioxoisoindol-2-yl)-2-ethoxyphenyl]ethyl]phenyl]methyl]butanoic acid
Show/Hide
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C29H29NO5
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1
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| 1 |
EC50 = 6900 nM
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CP0848635
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rac-2-(4-{2-[4-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-propoxyphenyl]ethyl}benzyl)butyric acid
Show/Hide
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C30H31NO5
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1
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| 1 |
EC50 = 6900 nM
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CP0386786
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2-methyl-2-[4-[2-(4-phenoxyphenoxy)ethyl]phenoxy]propanoic acid
Show/Hide
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C24H24O5
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1
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| 1 |
EC50 = 6900 nM
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CP0436761
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(R)-2-(4-butoxy-3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)benzyl)butanoic acid
Show/Hide
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C24H27F4NO4
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1
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| 1 |
EC50 = 7000 nM
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CP0389555
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(2S)-2-[[4-[2-[4-(1,3-dioxoisoindol-2-yl)-2-methoxyphenyl]ethyl]phenyl]methyl]butanoic acid
Show/Hide
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C28H27NO5
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1
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| 1 |
EC50 = 7100 nM
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CP0263537
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5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-phenyl-2H-1,2,3-triazole-4-carboxylic acid
Show/Hide
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C27H22N4O4
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1
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| 1 |
EC50 = 7330 nM
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CP0466657
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2-[6-(2-phenoxyethoxy)-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
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C18H18O5
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1
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| 1 |
EC50 = 7750 nM
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CP0067562
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5-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-1,2,3-triazole-4-carboxylic acid
Show/Hide
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C28H24N4O4
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1
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| 1 |
EC50 = 7900 nM
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CP0390076
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2-[[4-[2-[2-butoxy-4-(1,3-dioxoisoindol-2-yl)phenyl]ethyl]phenyl]methyl]butanoic acid
Show/Hide
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C31H33NO5
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1
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| 1 |
EC50 = 7900 nM
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CP0476896
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2-[4-[3-(1,3-benzothiazol-2-yloxy)propyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C20H21NO4S
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1
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| 1 |
EC50 = 7900 nM
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CP0551959
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2-methoxy-4-pentadecylbenzoic acid
Show/Hide
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C23H38O3
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1
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| 1 |
EC50 = 8100 nM
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CP0853045
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rac-2-(4-{2-[4-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-methoxyphenyl]ethyl}benzyl)butyric acid
Show/Hide
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C28H27NO5
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1
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| 1 |
EC50 = 8500 nM
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CP0039118
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2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy}acetic acid
Show/Hide
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C21H18F3NO3S2
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2
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| 1 |
EC50 = 8600 nM
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| 2 |
EC50 > 10000 nM
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CP0217233
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2-[[2-fluoro-5-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methoxy]phenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
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C22H21FN2O6
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1
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| 1 |
EC50 = 8607 nM
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CP0190237
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2-[[3-[[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]-4-fluorophenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
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C22H20ClFN2O6
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1
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| 1 |
EC50 = 9168 nM
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CP0417670
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2-((3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid
Show/Hide
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C21H19ClN2O6
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1
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| 1 |
EC50 = 9193 nM
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CP0071145
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4-(3-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-1,2,3-triazole-5-carboxylic acid
Show/Hide
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C28H24N4O4
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1
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| 1 |
EC50 = 9270 nM
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CP0263463
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5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-2-phenyl-2H-1,2,3-triazole-4-carboxylic acid
Show/Hide
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C28H24N4O4
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1
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| 1 |
EC50 = 9270 nM
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CP0417834
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2-(methoxycarbonyl(3-((2-p-tolylthiazol-4-yl)methoxy)benzyl)amino)acetic acid
Show/Hide
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C22H22N2O5S
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1
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| 1 |
EC50 = 9288 nM
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CP0851852
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rac-2-(4-{2-[4-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-ethoxyphenyl]ethyl}benzyl)butyric acid
Show/Hide
|
C29H29NO5
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1
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| 1 |
EC50 = 9300 nM
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CP0372720
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2-[[4-methoxy-3-[[(4-methylbenzoyl)amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
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C21H25NO4
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2
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| 1 |
EC50 = 9400 nM
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| 2 |
EC50 = 9600 nM
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CP0068987
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2-[(3R,4S)-1-ethoxycarbonyl-4-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]pyrrolidin-3-yl]acetic acid
Show/Hide
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C27H30N2O6
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1
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| 1 |
EC50 = 9680 nM
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CP0454151
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(R)-2-(2-(1-ethyl-3-(4-(trifluoromethoxy)phenyl)ureido)-2,3-dihydro-1H-inden-5-ylthio)-2-methylpropanoic acid
Show/Hide
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C23H25F3N2O4S
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1
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| 1 |
EC50 > 10000 nM
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CP0378994
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3-{3-[3,3-bis-(4-bromo-phenyl)-allyloxy]-phenyl}-acetic acid
Show/Hide
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C23H18Br2O3
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1
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| 1 |
EC50 > 10000 nM
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CP0398893
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2-[4-[3,3-bis(4-bromophenyl)prop-2-enylsulfanyl]-2-methylphenoxy]acetic acid
Show/Hide
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C24H20Br2O3S
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1
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| 1 |
EC50 > 10000 nM
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CP0425014
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2-[4-[3,3-bis(4-bromophenyl)prop-2-enylsulfanyl]-2-chlorophenoxy]acetic acid
Show/Hide
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C23H17Br2ClO3S
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1
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| 1 |
EC50 > 10000 nM
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CP0000252
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3-(4-methoxy-3-((4-(trifluoromethyl)benzamido)methyl)phenyl)-2-methylpropanoic acid
Show/Hide
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C20H20F3NO4
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1
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| 1 |
EC50 > 10000 nM
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CP0007838
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3-(4-methoxy-3-((4-(trifluoromethyl)benzamido)methyl)phenyl)propanoic acid
Show/Hide
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C19H18F3NO4
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1
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| 1 |
EC50 > 10000 nM
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CP0378766
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(R)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)methyl)-4-methoxybenzyl)butanoic acid
Show/Hide
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C21H21F4NO4
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1
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| 1 |
EC50 > 10000 nM
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CP0394694
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2-(3-((4-fluoro-3-(trifluoromethyl)benzamido)methyl)-4-methoxybenzyl)butanoic acid
Show/Hide
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C21H21F4NO4
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1
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| 1 |
EC50 > 10000 nM
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CP0422716
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(+/-)-2-(3-fluoro-4-methoxy-5-((4-(trifluoromethyl)benzamido)methyl)benzyl)butanoic acid
Show/Hide
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C21H21F4NO4
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1
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| 1 |
EC50 > 10000 nM
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CP0035660
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4-(((6-((3-(2,6-dichlorophenyl)-5-isopropylisoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid
Show/Hide
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C28H24Cl2F3N3O4
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1
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| 1 |
EC50 > 10000 nM
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CP0195439
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4-(((6-((5-cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid
Show/Hide
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C28H22Cl2F3N3O4
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1
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| 1 |
EC50 > 10000 nM
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CP0372721
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2-[[3-(benzamidomethyl)-4-methoxyphenyl]methyl]butanoic acid
Show/Hide
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C20H23NO4
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1
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| 1 |
EC50 > 10000 nM
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CP0377776
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2-[[4-methoxy-3-[[(2-phenylbenzoyl)amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
|
C26H27NO4
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1
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| 1 |
EC50 > 10000 nM
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CP0470324
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2-[[4-methoxy-3-[[(2-phenoxybenzoyl)amino]methyl]phenyl]methyl]butanoic acid
Show/Hide
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C26H27NO5
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1
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| 1 |
EC50 > 10000 nM
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CP0462062
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2-methyl-2-[4-[3-(4-phenyldiazenylphenoxy)propyl]phenoxy]propanoic acid
Show/Hide
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C25H26N2O4
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1
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| 1 |
EC50 = 10000 nM
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CP0063973
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2-[(3R,4R)-1-ethoxycarbonyl-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]pyrrolidin-3-yl]acetic acid
Show/Hide
|
C28H32N2O6
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1
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| 1 |
EC50 > 10000 nM
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CP0069349
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(3S,4R)-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-phenylpyrrolidine-3-carboxylic acid
Show/Hide
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C30H30N2O4
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1
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| 1 |
EC50 > 10000 nM
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CP0069351
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(3R,4R)-1-ethoxycarbonyl-4-[2-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H32N2O6
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1
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| 1 |
EC50 > 10000 nM
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CP0089192
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(3S,4R)-1-ethoxycarbonyl-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H30N2O6
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1
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| 1 |
EC50 > 10000 nM
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CP0148317
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2-[(3R,4S)-1-ethoxycarbonyl-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]pyrrolidin-3-yl]acetic acid
Show/Hide
|
C28H32N2O6
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1
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| 1 |
EC50 > 10000 nM
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CP0156178
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(3R,4R)-4-[2-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]ethyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
|
C32H32N2O6
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1
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| 1 |
EC50 > 10000 nM
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CP0239943
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(3S,4R)-4-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H27F3N4O4
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1
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| 1 |
EC50 > 10000 nM
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CP0271881
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2-[(3R,4R)-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-phenoxycarbonylpyrrolidin-3-yl]acetic acid
Show/Hide
|
C32H32N2O6
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1
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| 1 |
EC50 > 10000 nM
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CP0294341
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(3S,4R)-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
Show/Hide
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C29H27F3N4O4
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1
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| 1 |
EC50 > 10000 nM
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CP0377039
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2-[(1S)-5-(3-phenoxypropoxy)-2,3-dihydro-1H-inden-1-yl]acetic acid
Show/Hide
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C20H22O4
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1
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| 1 |
EC50 > 10000 nM
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CP0489509
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2-[4-[3-(3-chlorophenoxy)propoxy]phenyl]sulfonylacetic acid
Show/Hide
|
C17H17ClO6S
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1
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| 1 |
EC50 > 10000 nM
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CP0479824
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2-[(3S)-6-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
|
C22H18F3NO4S
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1
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| 1 |
EC50 > 10000 nM
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CP0190267
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2-[[2-fluoro-5-[[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy]phenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
|
C22H20F2N2O6
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1
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| 1 |
EC50 = 10010 nM
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CP0417991
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(S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-phenylpiperazin-1-yl)propanoic acid
Show/Hide
|
C31H33N3O4
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1
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| 1 |
EC50 = 10560 nM
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CP0377004
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2-[[4-[2-[4-(1,3-dioxoisoindol-2-yl)phenyl]ethyl]phenyl]methyl]butanoic acid
Show/Hide
|
C27H25NO4
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1
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| 1 |
EC50 = 11000 nM
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CP0387725
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4-[4-[2-[4-(1,3-dioxoisoindol-2-yl)phenyl]ethyl]phenoxy]butanoic acid
Show/Hide
|
C26H23NO5
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1
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| 1 |
EC50 = 12000 nM
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CP0424868
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(2R)-2-[[4-[2-[4-(1,3-dioxoisoindol-2-yl)-2-methoxyphenyl]ethyl]phenyl]methyl]butanoic acid
Show/Hide
|
C28H27NO5
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1
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| 1 |
EC50 = 12000 nM
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CP0551952
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2-acetyloxy-6-pentadecylbenzoic acid
Show/Hide
|
C24H38O4
|
1
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| 1 |
EC50 = 12000 nM
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CP0462063
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2-methyl-2-[4-[2-[4-[(E)-2-phenylethenyl]phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
|
C26H26O4
|
1
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| 1 |
EC50 = 12600 nM
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CP0322290
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(3S,4R)-4-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-phenoxycarbonylpyrrolidine-3-carboxylic acid
Show/Hide
|
C31H30N2O6
|
1
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| 1 |
EC50 = 13300 nM
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CP0279422
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5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzyl)-1-phenyl-1H-1,2,3-triazole-4-carboxylic acid
Show/Hide
|
C28H24N4O4
|
1
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| 1 |
EC50 = 13600 nM
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CP0152704
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2-[(3R,4S)-4-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-1-phenoxycarbonylpyrrolidin-3-yl]acetic acid
Show/Hide
|
C31H30N2O6
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1
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| 1 |
EC50 = 14600 nM
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CP0406287
|
4'-fluoro-7-hydroxyisoflavone
Show/Hide
|
C15H9FO3
|
1
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| 1 |
EC50 = 15380 nM
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CP0417676
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2-(methoxycarbonyl(3-((2-p-tolyloxazol-4-yl)methoxy)benzyl)amino)acetic acid
Show/Hide
|
C22H22N2O6
|
1
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| 1 |
EC50 = 15580 nM
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CP0376856
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2-[[4-[2-[4-(1,3-dioxoisoindol-2-yl)-2-hydroxyphenyl]ethyl]phenyl]methyl]butanoic acid
Show/Hide
|
C27H25NO5
|
1
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| 1 |
EC50 = 17000 nM
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|
|
|
CP0331637
|
2-[(2S)-1-[4-[(2,4-dichlorophenyl)methoxy]phenyl]pyrrolidin-2-yl]acetic acid
Show/Hide
|
C19H19Cl2NO3
|
1
|
| 1 |
EC50 = 17000 nM
|
|
|
|
CP0057581
|
2-Hydroxy-6-pentadecyl-benzoic acid
Show/Hide
|
C22H36O3
|
1
|
| 1 |
EC50 = 17000 nM
|
|
|
|
CP0437190
|
2-ethoxy-3-[4-(4-phenylmethoxyphenoxy)phenyl]propanoic acid
Show/Hide
|
C24H24O5
|
1
|
| 1 |
EC50 = 18000 nM
|
|
|
|
CP0373846
|
(3',5'-dimethoxy-7-hydroxyisoflavone)
Show/Hide
|
C17H14O5
|
1
|
| 1 |
EC50 = 18860 nM
|
|
|
|
CP0346384
|
(S)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-2-methylphenoxy)acetic acid
Show/Hide
|
C26H24Cl2N2O4
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0373358
|
(S)-2-(methoxycarbonyl(1-(3-((2-p-tolyloxazol-4-yl)methoxy)phenyl)ethyl)amino)acetic acid
Show/Hide
|
C23H24N2O6
|
1
|
| 1 |
EC50 = 20690 nM
|
|
|
|
CP0488451
|
2-methyl-2-[4-[(4-phenyldiazenylphenoxy)methyl]phenoxy]propanoic acid
Show/Hide
|
C23H22N2O4
|
1
|
| 1 |
EC50 = 21000 nM
|
|
|
|
CP0391822
|
3'-methoxy-7-hydroxyisoflavone
Show/Hide
|
C16H12O4
|
1
|
| 1 |
EC50 = 22290 nM
|
|
|
|
CP0294881
|
(3R,4R)-1-ethoxycarbonyl-4-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C26H28N2O6
|
1
|
| 1 |
EC50 = 24000 nM
|
|
|
|
CP0479958
|
2-(methoxycarbonyl(3-((2-phenylthiazol-4-yl)methoxy)benzyl)amino)acetic acid
Show/Hide
|
C21H20N2O5S
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0494053
|
2-(methoxycarbonyl(3-((2-phenyloxazol-4-yl)methoxy)benzyl)amino)acetic acid
Show/Hide
|
C21H20N2O6
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0501326
|
2-((3-((2-(2,4-difluorophenyl)oxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid
Show/Hide
|
C21H18F2N2O6
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0504258
|
2-(methoxycarbonyl(3-((2-m-tolyloxazol-4-yl)methoxy)benzyl)amino)acetic acid
Show/Hide
|
C22H22N2O6
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0522279
|
2-((3-((2-(4-fluorophenyl)oxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid
Show/Hide
|
C21H19FN2O6
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0518302
|
2-[[2-fluoro-5-[[5-methyl-2-(4-methylsulfonylphenyl)-1,3-oxazol-4-yl]methoxy]phenyl]methyl-methoxycarbonylamino]acetic acid
Show/Hide
|
C23H23FN2O8S
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0385191
|
3-(benzo[d][1,3]dioxol-5-yl)-7-hydroxy-4H-chromen-4-one
Show/Hide
|
C16H10O5
|
1
|
| 1 |
EC50 = 26940 nM
|
|
|
|
CP0551953
|
ethyl 2-(3-pentadecylphenoxy)acetate
Show/Hide
|
C25H42O3
|
1
|
| 1 |
EC50 = 29000 nM
|
|
|
|
CP0476092
|
2-[4-[[1-[(2,4-dichlorophenyl)carbamoyl]-1,3-dihydroisoindol-2-yl]methyl]-2-methylphenoxy]acetic acid
Show/Hide
|
C25H22Cl2N2O4
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0376722
|
2-[4-(hydroxymethyl)phenoxy]-2-methylpropanoic acid
Show/Hide
|
C11H14O4
|
1
|
| 1 |
EC50 = 30000 nM
|
|
|
|
CP0115307
|
2-(5-chloropyridin-3-yl)oxy-5-[(2,4-dichlorophenyl)sulfonylamino]benzoic acid
Show/Hide
|
C18H11Cl3N2O5S
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0115308
|
2-(5-chloropyridin-3-yl)oxy-N-ethyl-5-[(4-methylsulfonylphenyl)sulfonylamino]benzamide
Show/Hide
|
C21H20ClN3O6S2
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0174399
|
2,4-dichloro-N-[4-(5-chloropyridin-3-yl)oxy-3-methoxyphenyl]benzenesulfonamide
Show/Hide
|
C18H13Cl3N2O4S
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0258698
|
2,4-dichloro-N-[4-(5-chloropyridin-3-yl)oxyphenyl]benzenesulfonamide
Show/Hide
|
C17H11Cl3N2O3S
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0284391
|
5-[(4-tert-butylphenyl)sulfonylamino]-2-(5-chloropyridin-3-yl)oxy-N-ethylbenzamide
Show/Hide
|
C24H26ClN3O4S
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0063975
|
(3R,4R)-4-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H27F3N4O4
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0068924
|
(3R,4S)-4-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)-1,3-oxazol-2-yl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H26F3N3O5
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0260610
|
(3S,4S)-4-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H27F3N4O4
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0488121
|
2-[4-(1,3-benzothiazol-2-yloxymethyl)phenoxy]-2-methylpropanoic acid
Show/Hide
|
C18H17NO4S
|
1
|
| 1 |
EC50 = 32000 nM
|
|
|
|
CP0069347
|
(3R,4S)-1-ethoxycarbonyl-4-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C26H28N2O6
|
1
|
| 1 |
EC50 > 32000 nM
|
|
|
|
CP0183097
|
(3R,4R)-1-ethoxycarbonyl-4-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C26H28N2O6
|
1
|
| 1 |
EC50 > 32000 nM
|
|
|
|
CP0389252
|
2-[(2S)-1-[4-(2-methylphenoxy)phenyl]pyrrolidin-2-yl]acetic acid
Show/Hide
|
C19H21NO3
|
1
|
| 1 |
EC50 = 32000 nM
|
|
|
|
CP0386785
|
2-[4-[2-(1,3-benzothiazol-2-yloxy)ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C19H19NO4S
|
1
|
| 1 |
EC50 = 39300 nM
|
|
|
|
CP0517710
|
ethyl 2-methyl-2-[4-(2-oxo-3,4-dihydrochromene-3-carbonyl)phenoxy]propanoate
Show/Hide
|
C22H22O6
|
1
|
| 1 |
EC50 = 39670 nM
|
|
|
|
CP0545451
|
6-[2-[5-cyclopropyl-3-(3,5-dichloropyridin-4-yl)-1,2-oxazol-4-yl]-7-azaspiro[3.5]non-2-en-7-yl]-4-(trifluoromethyl)quinoline-2-carboxylic acid
Show/Hide
|
C30H23Cl2F3N4O3
|
1
|
| 1 |
EC50 > 40000 nM
|
|
|
|
CP0509610
|
(S)-2-(4-(3-chlorophenyl)piperazin-1-yl)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)propanoic acid
Show/Hide
|
C31H32ClN3O4
|
1
|
| 1 |
EC50 = 45230 nM
|
|
|
|
CP0551951
|
2-[3-[(Z)-pentadec-8-enyl]phenoxy]acetic acid
Show/Hide
|
C23H36O3
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0564509
|
ethyl 2-[3-[(Z)-pentadec-8-enyl]phenoxy]acetate
Show/Hide
|
C25H40O3
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0568253
|
ethyl 2-methyl-2-[3-[(Z)-pentadec-8-enyl]phenoxy]propanoate
Show/Hide
|
C27H44O3
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0479948
|
(S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-p-tolylpiperazin-1-yl)propanoic acid
Show/Hide
|
C32H35N3O4
|
1
|
| 1 |
EC50 = 50220 nM
|
|
|
|
CP0123421
|
CHEBI:30813
Show/Hide
|
C10H20O2
|
1
|
| 1 |
EC50 = 54000 nM
|
|
|
|
CP0386787
|
2-[4-[2-(4-benzoylphenoxy)ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C25H24O5
|
1
|
| 1 |
EC50 = 54600 nM
|
|
|
|
CP0457237
|
2-methyl-2-[4-(3-oxobenzo[f]chromene-2-carbonyl)phenoxy]propanoic acid
Show/Hide
|
C24H18O6
|
1
|
| 1 |
EC50 = 56710 nM
|
|
|
|
CP0015504
|
2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-2-methylpropanoic acid
Show/Hide
|
C19H20ClNO4
|
1
|
| 1 |
EC50 = 70360 nM
|
|
|
|
CP0495586
|
2-methyl-2-[4-[3-(4-phenoxyphenoxy)propyl]phenoxy]propanoic acid
Show/Hide
|
C25H26O5
|
1
|
| 1 |
EC50 = 75200 nM
|
|
|
|
CP0372957
|
(S)-3-(3-bromo-4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)phenyl)-2-(4-phenylpiperazin-1-yl)propanoic acid
Show/Hide
|
C31H32BrN3O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0091843
|
2-methyl-2-{2-methyl-4-[({3-[4-(trifluoromethoxy)phenyl]-1,2,4-thiadiazol-5-yl}methyl)sulfanyl]phenoxy}propanoic acid
Show/Hide
|
C21H19F3N2O4S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0158609
|
2-[4-[[3-(3,4-dichlorophenyl)-1,2,4-thiadiazol-5-yl]methylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C20H18Cl2N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0373602
|
2-methyl-2-[2-methyl-4-({3-[4-(trifluoromethoxy)phenyl]-1,2,4-thiadiazol-5-yl}methoxy)phenoxy]propanoic acid
Show/Hide
|
C21H19F3N2O5S
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0373603
|
2-methyl-2-{2-methyl-4-[({5-[4-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-3-yl}methyl)sulfanyl]phenoxy}propanoic acid
Show/Hide
|
C21H19F3N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0394580
|
2-methyl-2-[2-methyl-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-5-yl}methoxy)phenoxy]propanoic acid
Show/Hide
|
C21H19F3N2O4S
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0399666
|
2-[4-({[3-(4-chlorophenyl)-1,2,4-thiadiazol-5-yl]methyl}sulfanyl)-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C20H19ClN2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0399668
|
1-{2-methyl-4-[({3-[4-(trifluoromethoxy)phenyl]-1,2,4-thiadiazol-5-yl}methyl)sulfanyl]phenoxy}cyclopentane-1-carboxylic acid
Show/Hide
|
C23H21F3N2O4S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0399669
|
2-[4-[[3-[4-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-5-yl]methylsulfanyl]phenoxy]propanoic acid
Show/Hide
|
C19H15F3N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0399670
|
2-[4-[[3-[3-chloro-4-(trifluoromethoxy)phenyl]-1,2,4-thiadiazol-5-yl]methoxy]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C21H18ClF3N2O5S
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0399675
|
2-[4-[[3-(2,4-dichlorophenyl)-1,2,4-thiadiazol-5-yl]methylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C20H18Cl2N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0399676
|
2-[4-[[3-(3,4-dichlorophenyl)-1,2,4-thiadiazol-5-yl]methoxy]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C20H18Cl2N2O4S
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0412455
|
2-[4-[[3-(3,4-dimethylphenyl)-1,2,4-thiadiazol-5-yl]methoxy]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C22H24N2O4S
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0412457
|
2-methyl-2-{2-methyl-4-[({5-[4-(trifluoromethoxy)phenyl]-1,2,4-thiadiazol-3-yl}methyl)sulfanyl]phenoxy}propanoic acid
Show/Hide
|
C21H19F3N2O4S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0412459
|
2-[4-[[3-(3-chloro-4-methylphenyl)-1,2,4-thiadiazol-5-yl]methoxy]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C21H21ClN2O4S
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0412461
|
2-[4-[[5-(4-chlorophenyl)-1,2,4-thiadiazol-3-yl]methylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C20H19ClN2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0435125
|
2-[4-[[3-(3,4-dimethylphenyl)-1,2,4-thiadiazol-5-yl]methylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C22H24N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0435129
|
2-[4-[[3-[3-chloro-4-(trifluoromethoxy)phenyl]-1,2,4-thiadiazol-5-yl]methylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C21H18ClF3N2O4S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0449197
|
2-[4-[[5-(3,4-dichlorophenyl)-1,2,4-thiadiazol-3-yl]methylsulfanyl]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C20H18Cl2N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0459945
|
2-[4-[[3-[3-fluoro-4-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-5-yl]methoxy]-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C21H18F4N2O4S
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0510612
|
1-[4-[[3-(3,4-dichlorophenyl)-1,2,4-thiadiazol-5-yl]methylsulfanyl]-2-methylphenoxy]cyclopentane-1-carboxylic acid
Show/Hide
|
C22H20Cl2N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0399672
|
2-{2-methyl-4-[({3-[4-(trifluoromethyl)phenyl]-1,2,4-thiadiazol-5-yl}methyl)sulfanyl]phenoxy}acetic acid
Show/Hide
|
C19H15F3N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0427483
|
2-[4-({[3-(4-tert-butylphenyl)-1,2,4-thiadiazol-5-yl]methyl}sulfanyl)-2-methylphenoxy]-2-methylpropanoic acid
Show/Hide
|
C24H28N2O3S2
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0256605
|
1-benzyl-5-[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C31H30N2O4
|
1
|
| 1 |
EC50 > 7500 nM
|
|
|
|
CP0504306
|
(S)-2-((1-(3-((2-(4-chlorophenyl)oxazol-4-yl)methoxy)phenyl)ethyl)(methoxycarbonyl)amino)acetic acid
Show/Hide
|
C22H21ClN2O6
|
1
|
| 1 |
EC50 > 8300 nM
|
|
|
|
CP0689324
|
2-((4-methoxyphenoxy)carbonyl)acetic acid
Show/Hide
|
C29H29ClN2O7
|
1
|
| 1 |
IC50 = 1410 nM
|
|
|
|
CP0251631
|
2-[[4-[2-[2-(4-hydroxyphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy]phenyl]methyl-(4-methoxyphenoxy)carbonylamino]acetic acid
Show/Hide
|
C29H28N2O8
|
1
|
| 1 |
IC50 = 19800 nM
|
|
|
|
CP0109177
|
2-[(4-hydroxyphenyl)methyl-(4-methoxyphenoxy)carbonylamino]acetic acid
Show/Hide
|
C17H17NO6
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0109178
|
2-[[4-(3-benzamido-3-oxopropoxy)phenyl]methyl-(4-methoxyphenoxy)carbonylamino]acetic acid
Show/Hide
|
C27H26N2O8
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0117760
|
2-[[4-[2-[5-(hydroxymethyl)-2-phenyl-1,3-oxazol-4-yl]ethoxy]phenyl]methyl-(4-hydroxyphenoxy)carbonylamino]acetic acid
Show/Hide
|
C28H26N2O8
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0160752
|
2-[[4-[2-[5-(hydroxymethyl)-2-phenyl-1,3-oxazol-4-yl]ethoxy]phenyl]methyl-(4-methoxyphenoxy)carbonylamino]acetic acid
Show/Hide
|
C29H28N2O8
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0208813
|
2-[[4-[3-[acetyl(benzoyl)amino]-3-oxopropoxy]phenyl]methyl-(4-methoxyphenoxy)carbonylamino]acetic acid
Show/Hide
|
C29H28N2O9
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0337173
|
2-[(4-hydroxyphenoxy)carbonyl-[[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]acetic acid
Show/Hide
|
C28H26N2O7
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
