Brief Information of the Compound and Protein
Compound Name
methyl 14-benzyl-5-[4-(trifluoromethyl)phenyl]-2,3,7-triazatricyclo[7.5.0.02,6]tetradeca-1(9),3,5,7-tetraene-14-carboxylate
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PubChem ID
CID: 118720410
Canonical SMILES
COC(=O)C1(Cc2ccccc2)CCCCc2cnc3c(cnn3c12)-c1ccc(cc1)C(F)(F)F
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Compound Formula C27H24F3N3O2
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 74 nM
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